Found 194 with Last Name = 'anton' and Initial = 'p' TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Duquesne University
Curated by ChEMBL
Duquesne University
Curated by ChEMBL
Affinity DataKi: 3.07E+3nMAssay Description:Displacement of [3H]WIN-35,428 from human DAT expressed in N2A cells after 15 mins by photoaffinity labelingMore data for this Ligand-Target Pair
Affinity DataIC50: 0.398nMAssay Description:Antagonist activity at human mGluR5 expressed in CHO cells assessed as increase in intracellular calcium level by FLIPRMore data for this Ligand-Target Pair
Affinity DataIC50: 0.398nMAssay Description:Antagonist activity at human mGluR5 expressed in CHO cells assessed as increase in intracellular calcium level by FLIPRMore data for this Ligand-Target Pair
Affinity DataIC50: 0.794nMAssay Description:Antagonist activity at human mGluR5 expressed in CHO cells assessed as increase in intracellular calcium level by FLIPRMore data for this Ligand-Target Pair
Affinity DataIC50: 0.910nMAssay Description:Displacement of [3H]LTD4 from CYSLT1 receptor in guinea pig lung membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:Displacement of [3H]LTD4 from CYSLT1 receptor in guinea pig lung membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 1.20nMAssay Description:Displacement of [3H]LTD4 from CYSLT1 receptor in guinea pig lung membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 1.20nMAssay Description:Displacement of [3H]LTD4 from CYSLT1 receptor in guinea pig lung membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 1.26nMAssay Description:Antagonist activity at human mGluR5 expressed in CHO cells assessed as increase in intracellular calcium level by FLIPRMore data for this Ligand-Target Pair
Affinity DataIC50: 1.30nMAssay Description:Displacement of [3H]LTD4 from CYSLT1 receptor in guinea pig lung membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 1.70nMAssay Description:Displacement of [3H]LTD4 from CYSLT1 receptor in guinea pig lung membraneMore data for this Ligand-Target Pair
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Technical University Dortmund
Curated by ChEMBL
Technical University Dortmund
Curated by ChEMBL
Affinity DataIC50: 2nMAssay Description:Inhibition of GSK3beta (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 2nMAssay Description:Antagonist activity at human recombinant GPR154 receptor expressed in HEK293 cells assessed as inhibition of neuropeptide S-induced increase of intra...More data for this Ligand-Target Pair
Affinity DataIC50: 2.5nMAssay Description:Displacement of [3H]LTD4 from CYSLT1 receptor in guinea pig lung membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 2.51nMAssay Description:Antagonist activity at human mGluR5 expressed in CHO cells assessed as increase in intracellular calcium level by FLIPRMore data for this Ligand-Target Pair
Affinity DataIC50: 3nMAssay Description:Displacement of [3H]LTD4 from CYSLT1 receptor in guinea pig lung membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 3.16nMAssay Description:Antagonist activity at human mGluR5 expressed in CHO cells assessed as increase in intracellular calcium level by FLIPRMore data for this Ligand-Target Pair
Affinity DataIC50: 3.16nMAssay Description:Antagonist activity at human mGluR5 expressed in CHO cells assessed as increase in intracellular calcium level by FLIPRMore data for this Ligand-Target Pair
Affinity DataIC50: 3.20nMAssay Description:Displacement of [3H]LTD4 from CYSLT1 receptor in guinea pig lung membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 3.40nMAssay Description:Displacement of [3H]LTD4 from CYSLT1 receptor in guinea pig lung membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 3.40nMAssay Description:Displacement of [3H]LTD4 from CYSLT1 receptor in guinea pig lung membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 4.10nMAssay Description:Displacement of [3H]LTD4 from CYSLT1 receptor in guinea pig lung membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 4.40nMAssay Description:Displacement of [3H]LTD4 from CYSLT1 receptor in guinea pig lung membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 4.5nMAssay Description:Displacement of [3H]LTD4 from CYSLT1 receptor in guinea pig lung membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 4.80nMAssay Description:Displacement of [3H]LTD4 from CYSLT1 receptor in guinea pig lung membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 4.90nMAssay Description:Displacement of [3H]LTD4 from CYSLT1 receptor in guinea pig lung membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 6.31nMAssay Description:Antagonist activity at human mGluR5 expressed in CHO cells assessed as increase in intracellular calcium level by FLIPRMore data for this Ligand-Target Pair
Affinity DataIC50: 7.5nMAssay Description:Displacement of [3H]LTD4 from CYSLT1 receptor in guinea pig lung membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 7.94nMAssay Description:Antagonist activity at human mGluR5 expressed in CHO cells assessed as increase in intracellular calcium level by FLIPRMore data for this Ligand-Target Pair
Affinity DataIC50: 9.30nMAssay Description:Displacement of [3H]LTD4 from CYSLT1 receptor in guinea pig lung membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Antagonist activity at human mGluR5 expressed in CHO cells assessed as increase in intracellular calcium level by FLIPRMore data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Antagonist activity at human mGluR5 expressed in CHO cells assessed as increase in intracellular calcium level by FLIPRMore data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Antagonist activity at human recombinant GPR154 receptor expressed in HEK293 cells assessed as inhibition of neuropeptide S-induced increase of intra...More data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Antagonist activity at human mGluR5 expressed in CHO cells assessed as increase in intracellular calcium level by FLIPRMore data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Antagonist activity at human mGluR5 expressed in CHO cells assessed as increase in intracellular calcium level by FLIPRMore data for this Ligand-Target Pair
Affinity DataIC50: 12nMAssay Description:Displacement of [3H]LTD4 from CYSLT1 receptor in guinea pig lung membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 12.6nMAssay Description:Antagonist activity at human mGluR5 expressed in CHO cells assessed as increase in intracellular calcium level by FLIPRMore data for this Ligand-Target Pair
Affinity DataIC50: 12.6nMAssay Description:Antagonist activity at human mGluR5 expressed in CHO cells assessed as increase in intracellular calcium level by FLIPRMore data for this Ligand-Target Pair
Affinity DataIC50: 14nMAssay Description:Displacement of [3H]LTD4 from CYSLT1 receptor in guinea pig lung membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 15nMAssay Description:Displacement of [3H]LTD4 from CYSLT1 receptor in guinea pig lung membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 15.8nMAssay Description:Antagonist activity at human mGluR5 expressed in CHO cells assessed as increase in intracellular calcium level by FLIPRMore data for this Ligand-Target Pair
Affinity DataIC50: 15.8nMAssay Description:Antagonist activity at human mGluR5 expressed in CHO cells assessed as increase in intracellular calcium level by FLIPRMore data for this Ligand-Target Pair
Affinity DataIC50: 15.8nMAssay Description:Antagonist activity at human mGluR5 expressed in CHO cells assessed as increase in intracellular calcium level by FLIPRMore data for this Ligand-Target Pair
Affinity DataIC50: 15.8nMAssay Description:Antagonist activity at human mGluR5 expressed in CHO cells assessed as increase in intracellular calcium level by FLIPRMore data for this Ligand-Target Pair
Affinity DataIC50: 16nMAssay Description:Displacement of [3H]LTD4 from CYSLT1 receptor in guinea pig lung membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 16nMAssay Description:Displacement of [3H]LTD4 from CYSLT1 receptor in guinea pig lung membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 16nMAssay Description:Displacement of [3H]LTD4 from CYSLT1 receptor in guinea pig lung membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 17nMAssay Description:Displacement of [3H]LTD4 from CYSLT1 receptor in guinea pig lung membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 19.9nMAssay Description:Antagonist activity at human mGluR5 expressed in CHO cells assessed as increase in intracellular calcium level by FLIPRMore data for this Ligand-Target Pair
Affinity DataIC50: 19.9nMAssay Description:Antagonist activity at human mGluR5 expressed in CHO cells assessed as increase in intracellular calcium level by FLIPRMore data for this Ligand-Target Pair
