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Found 969 with Last Name = 'aoki' and Initial = 'j'
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Nihon Schering K.K.

Curated by ChEMBL
LigandPNGBDBM50485592(CHEMBL350445)
Affinity DataKi:  400nMAssay Description:TP_TRANSPORTER: inhibition of Taxol transepithelial transport (basal to apical) in Caco-2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Mus musculus)
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50527415(CHEMBL4529959)
Affinity DataIC50:  3.30nMAssay Description:Inhibition of ATX in mouse plasma after 2 hrs by LC-MS/MS analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetProbable G-protein coupled receptor 174(Mus musculus)
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50601663(CHEMBL5208556)
Affinity DataIC50:  3.40nMAssay Description:Antagonist activity at mouse GPR174 transfected in human HEK293FT cells co-transfected with AP-TGFalpha assessed as inhibition of LysoPalloT-NH-C3-ph...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetProbable G-protein coupled receptor 174(Mus musculus)
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50601663(CHEMBL5208556)
Affinity DataIC50:  3.40nMAssay Description:Antagonist activity at mouse GPR174 transfected in human HEK293FT cells co-transfected with AP-TGFalpha assessed as inhibition of LysoPalloT-NH-C3-ph...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetProbable G-protein coupled receptor 174(Mus musculus)
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50601671(CHEMBL5180950)
Affinity DataIC50:  3.80nMAssay Description:Antagonist activity at mouse GPR174 transfected in human HEK293FT cells co-transfected with AP-TGFalpha assessed as inhibition of LysoPalloT-NH-C3-ph...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetProbable G-protein coupled receptor 174(Mus musculus)
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50601671(CHEMBL5180950)
Affinity DataIC50:  3.80nMAssay Description:Antagonist activity at mouse GPR174 transfected in human HEK293FT cells co-transfected with AP-TGFalpha assessed as inhibition of LysoPalloT-NH-C3-ph...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50527415(CHEMBL4529959)
Affinity DataIC50:  4.20nMAssay Description:Inhibition of ATX (unknown origin) expressed in human HEK293 cells using TG-mTMP as substrate after 2 hrs by fluorescence based plate reader assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetProbable G-protein coupled receptor 174(Mus musculus)
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50601668(CHEMBL5187227)
Affinity DataIC50:  4.70nMAssay Description:Antagonist activity at mouse GPR174 transfected in human HEK293FT cells co-transfected with AP-TGFalpha assessed as inhibition of LysoPalloT-NH-C3-ph...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetProbable G-protein coupled receptor 174(Mus musculus)
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50601668(CHEMBL5187227)
Affinity DataIC50:  4.80nMAssay Description:Antagonist activity at mouse GPR174 transfected in human HEK293FT cells co-transfected with AP-TGFalpha assessed as inhibition of LysoPalloT-NH-C3-ph...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetProbable G-protein coupled receptor 174(Mus musculus)
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50601664(CHEMBL5196983)
Affinity DataIC50:  5.40nMAssay Description:Antagonist activity at mouse GPR174 transfected in human HEK293FT cells co-transfected with AP-TGFalpha assessed as inhibition of LysoPalloT-NH-C3-ph...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetProbable G-protein coupled receptor 174(Mus musculus)
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50601664(CHEMBL5196983)
Affinity DataIC50:  5.5nMAssay Description:Antagonist activity at mouse GPR174 transfected in human HEK293FT cells co-transfected with AP-TGFalpha assessed as inhibition of LysoPalloT-NH-C3-ph...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetProbable G-protein coupled receptor 174(Mus musculus)
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50601682(CHEMBL5173365)
Affinity DataIC50:  5.60nMAssay Description:Inverse agonist activity at mouse GPR174 transfected in human HEK293FT cells co-transfected with AP-TGFalpha assessed as inhibition of LysoPalloT-NH-...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetProbable G-protein coupled receptor 174(Mus musculus)
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50601682(CHEMBL5173365)
Affinity DataIC50:  5.60nMAssay Description:Inverse agonist activity at mouse GPR174 transfected in human HEK293FT cells co-transfected with AP-TGFalpha assessed as inhibition of LysoPalloT-NH-...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetProbable G-protein coupled receptor 174(Mus musculus)
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50601670(CHEMBL5202805)
Affinity DataIC50:  6.60nMAssay Description:Antagonist activity at mouse GPR174 transfected in human HEK293FT cells co-transfected with AP-TGFalpha assessed as inhibition of LysoPalloT-NH-C3-ph...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetProbable G-protein coupled receptor 174(Mus musculus)
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50601670(CHEMBL5202805)
Affinity DataIC50:  6.70nMAssay Description:Antagonist activity at mouse GPR174 transfected in human HEK293FT cells co-transfected with AP-TGFalpha assessed as inhibition of LysoPalloT-NH-C3-ph...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Mus musculus)
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50527451(CHEMBL4515130)
Affinity DataIC50:  9.40nMAssay Description:Inhibition of ATX in mouse plasma after 2 hrs by LC-MS/MS analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Mus musculus)
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50527434(CHEMBL4466454)
Affinity DataIC50:  9.90nMAssay Description:Inhibition of ATX in mouse plasma after 2 hrs by LC-MS/MS analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEctonucleotide pyrophosphatase/phosphodiesterase 2(Danio rerio)
The University of Tokyo

LigandPNGBDBM103570(ATX inhibitor 18)
Affinity DataIC50:  10nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Mus musculus)
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50527442(CHEMBL4465067)
Affinity DataIC50:  11nMAssay Description:Inhibition of ATX in mouse plasma after 2 hrs by LC-MS/MS analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM103575(ATX inhibitor 10 analogue 5 | US8551988, 65)
Affinity DataIC50:  13nMAssay Description:Inhibition of ATX (unknown origin) expressed in human HEK293 cells using TG-mTMP as substrate after 2 hrs by fluorescence based plate reader assayMore data for this Ligand-Target Pair
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Mus musculus)
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM103575(ATX inhibitor 10 analogue 5 | US8551988, 65)
Affinity DataIC50:  13nMMore data for this Ligand-Target Pair
TargetProbable G-protein coupled receptor 174(Mus musculus)
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50601669(CHEMBL5198736)
Affinity DataIC50:  13nMAssay Description:Antagonist activity at mouse GPR174 transfected in human HEK293FT cells co-transfected with AP-TGFalpha assessed as inhibition of LysoPalloT-NH-C3-ph...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetProbable G-protein coupled receptor 174(Mus musculus)
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50601669(CHEMBL5198736)
Affinity DataIC50:  13nMAssay Description:Antagonist activity at mouse GPR174 transfected in human HEK293FT cells co-transfected with AP-TGFalpha assessed as inhibition of LysoPalloT-NH-C3-ph...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Mus musculus)
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50527449(CHEMBL4442653)
Affinity DataIC50:  13nMAssay Description:Inhibition of ATX in mouse plasma after 2 hrs by LC-MS/MS analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Mus musculus)
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50527429(CHEMBL4593078)
Affinity DataIC50:  14nMAssay Description:Inhibition of ATX in mouse plasma after 2 hrs by LC-MS/MS analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Mus musculus)
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50527459(CHEMBL4581989)
Affinity DataIC50:  15nMAssay Description:Inhibition of ATX in mouse plasma after 2 hrs by LC-MS/MS analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Mus musculus)
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50527435(CHEMBL4474913)
Affinity DataIC50:  16nMAssay Description:Inhibition of ATX in mouse plasma after 2 hrs by LC-MS/MS analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Mus musculus)
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50527445(CHEMBL4453366)
Affinity DataIC50:  19nMAssay Description:Inhibition of ATX in mouse plasma after 2 hrs by LC-MS/MS analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Mus musculus)
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50527452(CHEMBL4451331)
Affinity DataIC50:  21nMAssay Description:Inhibition of ATX in mouse plasma after 2 hrs by LC-MS/MS analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Mus musculus)
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM103576(ATX inhibitor 10 analogue 6)
Affinity DataIC50:  22nMMore data for this Ligand-Target Pair
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Mus musculus)
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50527412(CHEMBL4482895)
Affinity DataIC50:  23nMAssay Description:Inhibition of ATX in mouse plasma after 2 hrs by LC-MS/MS analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Mus musculus)
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM103577(ATX inhibitor 10 analogue 7)
Affinity DataIC50:  25nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Mus musculus)
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50527440(CHEMBL4469815)
Affinity DataIC50:  26nMAssay Description:Inhibition of ATX in mouse plasma after 2 hrs by LC-MS/MS analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Mus musculus)
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM103568(ATX inhibitor 16 | Chicago Sky Blue)
Affinity DataIC50:  26nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50527434(CHEMBL4466454)
Affinity DataIC50:  30nMAssay Description:Inhibition of ATX (unknown origin)-mediated cell migration in human MDA-MB-231 cells assessed as reduction in cell motility after 3 hrs by Diff-Quick...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Mus musculus)
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50527444(CHEMBL4438238)
Affinity DataIC50:  30nMAssay Description:Inhibition of ATX in mouse plasma after 2 hrs by LC-MS/MS analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Mus musculus)
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50527439(CHEMBL4471030)
Affinity DataIC50:  31nMAssay Description:Inhibition of ATX in mouse plasma after 2 hrs by LC-MS/MS analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Mus musculus)
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50527427(CHEMBL4572641)
Affinity DataIC50:  31nMAssay Description:Inhibition of ATX in mouse plasma after 2 hrs by LC-MS/MS analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Mus musculus)
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50527443(CHEMBL4534048)
Affinity DataIC50:  37nMAssay Description:Inhibition of ATX in mouse plasma after 2 hrs by LC-MS/MS analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Mus musculus)
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50527433(CHEMBL4515759)
Affinity DataIC50:  40nMAssay Description:Inhibition of ATX in mouse plasma after 2 hrs by LC-MS/MS analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Mus musculus)
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50527432(CHEMBL4474496)
Affinity DataIC50:  44nMAssay Description:Inhibition of ATX in mouse plasma after 2 hrs by LC-MS/MS analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Mus musculus)
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM103980(Disubstituted aryl-Me ATX inhibitor 8)
Affinity DataIC50:  45nMAssay Description:Inhibitory activities of hit compounds towards ENPP1-5 were calculated using pNP-TMP, and the inhibitory activities of hit compounds towards ENPP6 an...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Mus musculus)
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50527458(CHEMBL4535941)
Affinity DataIC50:  49nMAssay Description:Inhibition of ATX in mouse plasma after 2 hrs by LC-MS/MS analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProbable G-protein coupled receptor 174(Mus musculus)
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50601678(CHEMBL5179787)
Affinity DataIC50:  51nMAssay Description:Antagonist activity at mouse GPR174 transfected in human HEK293FT cells co-transfected with AP-TGFalpha assessed as inhibition of LysoPalloT-NH-C3-ph...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetProbable G-protein coupled receptor 174(Mus musculus)
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50601678(CHEMBL5179787)
Affinity DataIC50:  51nMAssay Description:Antagonist activity at mouse GPR174 transfected in human HEK293FT cells co-transfected with AP-TGFalpha assessed as inhibition of LysoPalloT-NH-C3-ph...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Mus musculus)
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM103979(Disubstituted aryl-Me ATX inhibitor 7)
Affinity DataIC50:  53nMAssay Description:Inhibitory activities of hit compounds towards ENPP1-5 were calculated using pNP-TMP, and the inhibitory activities of hit compounds towards ENPP6 an...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Mus musculus)
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50527441(CHEMBL4538038)
Affinity DataIC50:  56nMAssay Description:Inhibition of ATX in mouse plasma after 2 hrs by LC-MS/MS analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Mus musculus)
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM103902(Disubstituted aryl-Me ATX inhibitor 9 | US8563583,...)
Affinity DataIC50:  57nMAssay Description:Inhibitory activities of hit compounds towards ENPP1-5 were calculated using pNP-TMP, and the inhibitory activities of hit compounds towards ENPP6 an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Mus musculus)
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50527436(CHEMBL4440388)
Affinity DataIC50:  57nMAssay Description:Inhibition of ATX in mouse plasma after 2 hrs by LC-MS/MS analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Mus musculus)
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50527431(CHEMBL4573110)
Affinity DataIC50:  71nMAssay Description:Inhibition of ATX in mouse plasma after 2 hrs by LC-MS/MS analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
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