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Found 180 with Last Name = 'archer' and Initial = 's'
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
TBA

Curated by ChEMBL
LigandPNGBDBM50290071(CHEMBL542149 | N-[(S)-1-(3-Amino-phenyl)-2-pyrroli...)
Affinity DataKi:  0.0592nMAssay Description:Compound was evaluated for the inhibition of Opioid receptor kappa1 binding to guinea pig brain membranes, using 1 nM [3H]- U69,593 as radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
TBA

Curated by ChEMBL
LigandPNGBDBM50290076(CHEMBL558596 | N-[(S)-1-(3-Acetylamino-phenyl)-2-p...)
Affinity DataKi:  0.0855nMAssay Description:Compound was evaluated for the inhibition of Opioid receptor kappa1 binding to guinea pig brain membranes, using 1 nM [3H]- U69,593 as radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
TargetMu-type opioid receptor(CALF)
University of Rochester

Curated by PDSP Ki Database
LigandPNGBDBM85393(14β-(p-chlorocinnamoylamino)-7,8-dihydrocodei...)
Affinity DataKi:  0.120nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMu-type opioid receptor(CALF)
University of Rochester

Curated by PDSP Ki Database
LigandPNGBDBM85396(CACO)
Affinity DataKi:  0.460nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetOpioid receptor delta 1(Bos taurus)
University of Rochester

Curated by PDSP Ki Database
LigandPNGBDBM85393(14β-(p-chlorocinnamoylamino)-7,8-dihydrocodei...)
Affinity DataKi:  0.75nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMu-type opioid receptor(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50001707(10,17-dihydroxy-4-methyl-(13R,17S)-12-oxa-4-azapen...)
Affinity DataKi:  0.780nMAssay Description:Inhibitory binding constant in guinea pig brain homogenate was reported at mu site at a temperature 25 degree Centigrade labeled with [3H](D-Ala2-MeP...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50290072(5-{3-[3-((S)-1-{[2-(3,4-Dichloro-phenyl)-acetyl]-m...)
Affinity DataKi:  0.898nMAssay Description:Compound was evaluated for the inhibition of Opioid receptor delta 1 binding to guinea pig brain membranes, using 0.2 nM [3H]-naltrindole as radiolig...More data for this Ligand-Target Pair
In DepthDetails Article
TargetMu-type opioid receptor(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM60212((4R,4aS,7aR,12bS)-3-(cyclopropylmethyl)-4a,9-bis(o...)
Affinity DataKi:  1.10nMAssay Description:Inhibitory binding constant in guinea pig brain homogenate was reported at mu site at a temperature 25 degree Centigrade labeled with [3H](D-Ala2-MeP...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(CALF)
University of Rochester

Curated by PDSP Ki Database
LigandPNGBDBM85394(N-CPM-CACO)
Affinity DataKi:  1.10nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetKappa-type opioid receptor(CALF)
University of Rochester

Curated by PDSP Ki Database
LigandPNGBDBM85393(14β-(p-chlorocinnamoylamino)-7,8-dihydrocodei...)
Affinity DataKi:  1.10nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMu-type opioid receptor(CALF)
University of Rochester

Curated by PDSP Ki Database
LigandPNGBDBM85395(MC-CAM)
Affinity DataKi:  1.40nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
TBA

Curated by ChEMBL
LigandPNGBDBM50290072(5-{3-[3-((S)-1-{[2-(3,4-Dichloro-phenyl)-acetyl]-m...)
Affinity DataKi:  1.40nMAssay Description:Compound was evaluated for the inhibition of Opioid receptor kappa1 binding to guinea pig brain membranes, using 1 nM [3H]- U69,593 as radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
TargetDelta-type opioid receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50290070(5-{3-[3-(1-{[2-(3,4-Dichloro-phenyl)-acetyl]-methy...)
Affinity DataKi:  1.80nMAssay Description:Compound was evaluated for the inhibition of Opioid receptor delta 1 binding to guinea pig brain membranes, using 0.2 nM [3H]-naltrindole as radiolig...More data for this Ligand-Target Pair
In DepthDetails Article
TargetDelta-type opioid receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM60212((4R,4aS,7aR,12bS)-3-(cyclopropylmethyl)-4a,9-bis(o...)
Affinity DataKi:  6.60nMAssay Description:Inhibitory binding constant in guinea pig brain homogenate was reported at Opioid receptor delta 1 at a a temperature 25 degree Celsius labeled with ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetMu-type opioid receptor(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50290071(CHEMBL542149 | N-[(S)-1-(3-Amino-phenyl)-2-pyrroli...)
Affinity DataKi:  7.70nMAssay Description:Compound was evaluated for the inhibition of Opioid receptor mu 1 binding to guinea pig brain membranes, using [3H]- DAMGO as radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
TargetDelta-type opioid receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50290071(CHEMBL542149 | N-[(S)-1-(3-Amino-phenyl)-2-pyrroli...)
Affinity DataKi:  7.80nMAssay Description:Compound was evaluated for the inhibition of Opioid receptor delta 1 binding to guinea pig brain membranes, using 0.2 nM [3H]-naltrindole as radiolig...More data for this Ligand-Target Pair
In DepthDetails Article
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
TBA

Curated by ChEMBL
LigandPNGBDBM50290070(5-{3-[3-(1-{[2-(3,4-Dichloro-phenyl)-acetyl]-methy...)
Affinity DataKi:  8.20nMAssay Description:Compound was evaluated for the inhibition of Opioid receptor kappa1 binding to guinea pig brain membranes, using 1 nM [3H]- U69,593 as radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
TargetMu-type opioid receptor(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50290076(CHEMBL558596 | N-[(S)-1-(3-Acetylamino-phenyl)-2-p...)
Affinity DataKi:  8.40nMAssay Description:Compound was evaluated for the inhibition of Opioid receptor mu 1 binding to guinea pig brain membranes, using [3H]- DAMGO as radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
TBA

Curated by ChEMBL
LigandPNGBDBM60212((4R,4aS,7aR,12bS)-3-(cyclopropylmethyl)-4a,9-bis(o...)
Affinity DataKi:  8.5nMAssay Description:Inhibitory binding constant in guinea pig brain homogenate was reported at Opioid receptor kappa 1 at temperature 25 degree Celsius labeled with (-)-...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(CALF)
University of Rochester

Curated by PDSP Ki Database
LigandPNGBDBM85394(N-CPM-CACO)
Affinity DataKi:  9.80nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetOpioid receptor delta 1(Bos taurus)
University of Rochester

Curated by PDSP Ki Database
LigandPNGBDBM85395(MC-CAM)
Affinity DataKi:  12nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50290076(CHEMBL558596 | N-[(S)-1-(3-Acetylamino-phenyl)-2-p...)
Affinity DataKi:  14nMAssay Description:Compound was evaluated for the inhibition of Opioid receptor delta 1 binding to guinea pig brain membranes, using 0.2 nM [3H]-naltrindole as radiolig...More data for this Ligand-Target Pair
In DepthDetails Article
TargetKappa-type opioid receptor(CALF)
University of Rochester

Curated by PDSP Ki Database
LigandPNGBDBM85395(MC-CAM)
Affinity DataKi:  14nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
TBA

Curated by ChEMBL
LigandPNGBDBM50290074(CHEMBL558597 | N-[(R)-1-(3-Amino-phenyl)-2-pyrroli...)
Affinity DataKi:  15nMAssay Description:Compound was evaluated for the inhibition of Opioid receptor kappa1 binding to guinea pig brain membranes, using 1 nM [3H]- U69,593 as radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
TargetOpioid receptor delta 1(Bos taurus)
University of Rochester

Curated by PDSP Ki Database
LigandPNGBDBM85394(N-CPM-CACO)
Affinity DataKi:  16nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
TBA

Curated by ChEMBL
LigandPNGBDBM50290075(CHEMBL542403 | N-[(R)-1-(3-Acetylamino-phenyl)-2-p...)
Affinity DataKi:  18nMAssay Description:Compound was evaluated for the inhibition of Opioid receptor kappa1 binding to guinea pig brain membranes, using 1 nM [3H]- U69,593 as radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
TargetKappa-type opioid receptor(CALF)
University of Rochester

Curated by PDSP Ki Database
LigandPNGBDBM85396(CACO)
Affinity DataKi:  19nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMu-type opioid receptor(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50016086(4-cyclopropylmethyl-10,17-dihydroxy-(13R,17S)-12-o...)
Affinity DataKi:  31nMAssay Description:Inhibitory binding constant in guinea pig brain homogenate was reported at mu site at a temperature 25 degree Centigrade labeled with [3H](D-Ala2-MeP...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50001707(10,17-dihydroxy-4-methyl-(13R,17S)-12-oxa-4-azapen...)
Affinity DataKi:  50nMAssay Description:Inhibitory binding constant in guinea pig brain homogenate was reported at Opioid receptor delta 1 at a a temperature 25 degree Celsius labeled with ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetDelta-type opioid receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50290073(5-{3-[3-((R)-1-{[2-(3,4-Dichloro-phenyl)-acetyl]-m...)
Affinity DataKi:  86nMAssay Description:Compound was evaluated for the inhibition of Opioid receptor delta 1 binding to guinea pig brain membranes, using 0.2 nM [3H]-naltrindole as radiolig...More data for this Ligand-Target Pair
In DepthDetails Article
TargetMu-type opioid receptor(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50290072(5-{3-[3-((S)-1-{[2-(3,4-Dichloro-phenyl)-acetyl]-m...)
Affinity DataKi:  98nMAssay Description:Compound was evaluated for the inhibition of Opioid receptor mu 1 binding to guinea pig brain membranes, using [3H]- DAMGO as radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
TBA

Curated by ChEMBL
LigandPNGBDBM50016086(4-cyclopropylmethyl-10,17-dihydroxy-(13R,17S)-12-o...)
Affinity DataKi:  102nMAssay Description:Inhibitory binding constant in guinea pig brain homogenate was reported at Opioid receptor kappa 1 at temperature 25 degree Celsius labeled with (-)-...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
TBA

Curated by ChEMBL
LigandPNGBDBM50001707(10,17-dihydroxy-4-methyl-(13R,17S)-12-oxa-4-azapen...)
Affinity DataKi:  137nMAssay Description:Inhibitory binding constant in guinea pig brain homogenate was reported at Opioid receptor kappa 1 at temperature 25 degree Celsius labeled with (-)-...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
TBA

Curated by ChEMBL
LigandPNGBDBM50290073(5-{3-[3-((R)-1-{[2-(3,4-Dichloro-phenyl)-acetyl]-m...)
Affinity DataKi:  139nMAssay Description:Compound was evaluated for the inhibition of Opioid receptor kappa1 binding to guinea pig brain membranes, using 1 nM [3H]- U69,593 as radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
TargetMu-type opioid receptor(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50290070(5-{3-[3-(1-{[2-(3,4-Dichloro-phenyl)-acetyl]-methy...)
Affinity DataKi:  176nMAssay Description:Compound was evaluated for the inhibition of Opioid receptor mu 1 binding to guinea pig brain membranes, using [3H]- DAMGO as radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
TargetDelta-type opioid receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50016086(4-cyclopropylmethyl-10,17-dihydroxy-(13R,17S)-12-o...)
Affinity DataKi:  281nMAssay Description:Inhibitory binding constant in guinea pig brain homogenate was reported at Opioid receptor delta 1 at a temperature 25 degree Celsius labeled with [3...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50290075(CHEMBL542403 | N-[(R)-1-(3-Acetylamino-phenyl)-2-p...)
Affinity DataKi:  1.04E+3nMAssay Description:Compound was evaluated for the inhibition of Opioid receptor mu 1 binding to guinea pig brain membranes, using [3H]- DAMGO as radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
TargetMu-type opioid receptor(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50290073(5-{3-[3-((R)-1-{[2-(3,4-Dichloro-phenyl)-acetyl]-m...)
Affinity DataKi:  1.19E+3nMAssay Description:Compound was evaluated for the inhibition of Opioid receptor mu 1 binding to guinea pig brain membranes, using [3H]- DAMGO as radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
TargetMu-type opioid receptor(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50290074(CHEMBL558597 | N-[(R)-1-(3-Amino-phenyl)-2-pyrroli...)
Affinity DataKi:  1.38E+3nMAssay Description:Compound was evaluated for the inhibition of Opioid receptor mu 1 binding to guinea pig brain membranes, using [3H]- DAMGO as radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
TargetDelta-type opioid receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50290074(CHEMBL558597 | N-[(R)-1-(3-Amino-phenyl)-2-pyrroli...)
Affinity DataKi:  1.85E+3nMAssay Description:Compound was evaluated for the inhibition of Opioid receptor delta 1 binding to guinea pig brain membranes, using 0.2 nM [3H]-naltrindole as radiolig...More data for this Ligand-Target Pair
In DepthDetails Article
TargetDelta-type opioid receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50290075(CHEMBL542403 | N-[(R)-1-(3-Acetylamino-phenyl)-2-p...)
Affinity DataKi:  3.07E+3nMAssay Description:Compound was evaluated for the inhibition of Opioid receptor delta 1 binding to guinea pig brain membranes, using 0.2 nM [3H]-naltrindole as radiolig...More data for this Ligand-Target Pair
In DepthDetails Article
TargetMu-type opioid receptor(CALF)
University of Rochester

Curated by PDSP Ki Database
LigandPNGBDBM50287332(1N-[4-cyclopropylmethyl-10-hydroxy-(13R,14R)-12-ox...)
Affinity DataIC50:  0.210nMAssay Description:Compound was tested for Inhibition of [3H]-DAMGO (0.25 nM) binding to mu receptor from bovine striatal membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetMu-type opioid receptor(CALF)
University of Rochester

Curated by PDSP Ki Database
LigandPNGBDBM50456193(CHEMBL607068)
Affinity DataIC50:  0.280nMAssay Description:Binding affinity against mu opioid receptor from calf frontal cortex.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(CALF)
University of Rochester

Curated by PDSP Ki Database
LigandPNGBDBM50033645(1N-[10-hydroxy-4,13-dimethyl-14-oxo-(13R,17S)-12-o...)
Affinity DataIC50:  0.330nMAssay Description:Binding affinity against mu opioid receptor from calf frontal cortex.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(CALF)
University of Rochester

Curated by PDSP Ki Database
LigandPNGBDBM50030143(CHEMBL41098 | bis-(1N-[10-hydroxy-4-methyl-14-oxo-...)
Affinity DataIC50:  0.400nMAssay Description:Evaluation for the inhibition of mu opioid binding to bovine striatal membranes by the affinity ligand 0.25 nM [3H]DAMGO radiolabeled opioidMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(CALF)
University of Rochester

Curated by PDSP Ki Database
LigandPNGBDBM50030143(CHEMBL41098 | bis-(1N-[10-hydroxy-4-methyl-14-oxo-...)
Affinity DataIC50:  0.400nMAssay Description:Inhibitory activity of the compound against Opioid receptor mu 1 binding to bovine striatal membraneMore data for this Ligand-Target Pair
In DepthDetails Article
TargetMu-type opioid receptor(CALF)
University of Rochester

Curated by PDSP Ki Database
LigandPNGBDBM50033654(1N-[10-methoxy-4-methyl-14-oxo-(13R,17S)-12-oxa-4-...)
Affinity DataIC50:  0.440nMAssay Description:Binding affinity against mu opioid receptor from calf frontal cortex.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(CALF)
University of Rochester

Curated by PDSP Ki Database
LigandPNGBDBM50033647(1N-[4-cyclopropylmethyl-10-hydroxy-13-methyl-14-ox...)
Affinity DataIC50:  0.520nMAssay Description:Binding affinity against mu opioid receptor from calf frontal cortex.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287332(1N-[4-cyclopropylmethyl-10-hydroxy-(13R,14R)-12-ox...)
Affinity DataIC50:  0.530nMAssay Description:Compound was tested for Inhibition of 9 (1nM) binding to Opioid receptor delta 1 from bovine striatal MembranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetMu-type opioid receptor(CALF)
University of Rochester

Curated by PDSP Ki Database
LigandPNGBDBM50287331(1N-[10-hydroxy-4-methyl-(13R,14R)-12-oxa-4-azapent...)
Affinity DataIC50:  0.560nMAssay Description:Compound was tested for Inhibition of [3H]-DAMGO (0.25 nM) binding to mu receptor from bovine striatal membranesMore data for this Ligand-Target Pair
In DepthDetails Article
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