TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
University Of Belgrade
Curated by ChEMBL
University Of Belgrade
Curated by ChEMBL
Affinity DataIC50: <1nMAssay Description:Inhibition of HIV-1 reverse transcriptase preincubated for 45 mins followed by substrate addition by immunoassayMore data for this Ligand-Target Pair
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
University Of Belgrade
Curated by ChEMBL
University Of Belgrade
Curated by ChEMBL
Affinity DataIC50: 4.80nMAssay Description:Inhibition of wild-type HIV-1 reverse transcriptase by Picogreen assayMore data for this Ligand-Target Pair
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
University Of Belgrade
Curated by ChEMBL
University Of Belgrade
Curated by ChEMBL
Affinity DataIC50: 9.40nMAssay Description:Inhibition of HIV-1 reverse transcriptase using ABTS as substrate and RNA template primed with oligo(dT)12-18 in presence of digoxigenin/biotin-label...More data for this Ligand-Target Pair
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
University Of Belgrade
Curated by ChEMBL
University Of Belgrade
Curated by ChEMBL
Affinity DataIC50: 10nMAssay Description:Inhibition of HIV-1 LTR reverse transcriptase infected in human CEM cells using RNA template incubated for 1 hr by RT-PCR based cell-free assayMore data for this Ligand-Target Pair
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
University Of Belgrade
Curated by ChEMBL
University Of Belgrade
Curated by ChEMBL
Affinity DataIC50: 50nMAssay Description:Inhibition of HIV-1 LTR reverse transcriptase infected in human CEM cells using RNA template incubated for 1 hr by RT-PCR based cell-free assayMore data for this Ligand-Target Pair
Affinity DataIC50: 82nMAssay Description:Inhibition of human recombinant CYP3A4More data for this Ligand-Target Pair
Affinity DataIC50: 275nMAssay Description:Inhibition of human recombinant CYP3A4More data for this Ligand-Target Pair
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
University Of Belgrade
Curated by ChEMBL
University Of Belgrade
Curated by ChEMBL
Affinity DataIC50: 300nMAssay Description:Inhibition of HIV-1 reverse transcriptase preincubated for 45 mins followed by substrate addition by immunoassayMore data for this Ligand-Target Pair
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
University Of Belgrade
Curated by ChEMBL
University Of Belgrade
Curated by ChEMBL
Affinity DataIC50: 720nMAssay Description:Inhibition of HIV-1 reverse transcriptase using ABTS as substrate and RNA template primed with oligo(dT)12-18 in presence of digoxigenin/biotin-label...More data for this Ligand-Target Pair
Affinity DataIC50: 923nMAssay Description:Inhibition of human recombinant CYP3A4More data for this Ligand-Target Pair
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
University Of Belgrade
Curated by ChEMBL
University Of Belgrade
Curated by ChEMBL
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of HIV-1 LTR reverse transcriptase infected in human CEM cells using RNA template incubated for 1 hr by RT-PCR based cell-free assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.63E+3nMAssay Description:Inhibition of human recombinant CYP3A4More data for this Ligand-Target Pair
Affinity DataIC50: 2.35E+3nMAssay Description:Inhibition of human recombinant CYP3A4More data for this Ligand-Target Pair
Affinity DataIC50: 4.06E+3nMAssay Description:Inhibition of human recombinant CYP3A4More data for this Ligand-Target Pair
Affinity DataIC50: 4.65E+3nMAssay Description:Inhibition of recombinant HIV-1 subtype C integrase using double-stranded FITC-labelled target DNA as substrate pre-incubated for 45 mins followed by...More data for this Ligand-Target Pair
Affinity DataIC50: 1.83E+4nMAssay Description:Inhibition of recombinant HIV-1 subtype C integrase using double-stranded FITC-labelled target DNA as substrate pre-incubated for 45 mins followed by...More data for this Ligand-Target Pair
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
University Of Belgrade
Curated by ChEMBL
University Of Belgrade
Curated by ChEMBL
Affinity DataIC50: 7.41E+4nMAssay Description:Inhibition of recombinant HIV-1 reverse transcriptase using ABTS as substrate incubated for 1 hr by ELISAMore data for this Ligand-Target Pair
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
University Of Belgrade
Curated by ChEMBL
University Of Belgrade
Curated by ChEMBL
Affinity DataIC50: 2.79E+5nMAssay Description:Inhibition of recombinant HIV-1 reverse transcriptase using ABTS as substrate incubated for 1 hr by ELISAMore data for this Ligand-Target Pair
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
University Of Belgrade
Curated by ChEMBL
University Of Belgrade
Curated by ChEMBL
Affinity DataEC50: 120nMAssay Description:Inhibition of HIV-1 reverse transcriptase in virus infected human C8166 cells assessed as reduction in virus-induced cytopathic effect by MTT assayMore data for this Ligand-Target Pair
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
University Of Belgrade
Curated by ChEMBL
University Of Belgrade
Curated by ChEMBL
Affinity DataEC50: 120nMAssay Description:Inhibition of HIV-1 reverse transcriptase in virus infected human C8166 cells assessed as reduction in virus-induced cytopathic effect by MTT assayMore data for this Ligand-Target Pair
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
University Of Belgrade
Curated by ChEMBL
University Of Belgrade
Curated by ChEMBL
Affinity DataEC50: 120nMAssay Description:Inhibition of HIV-1 reverse transcriptase in virus infected human C8166 cells assessed as reduction in virus-induced cytopathic effect by MTT assayMore data for this Ligand-Target Pair
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
University Of Belgrade
Curated by ChEMBL
University Of Belgrade
Curated by ChEMBL
Affinity DataEC50: 120nMAssay Description:Inhibition of HIV-1 reverse transcriptase in virus infected human C8166 cells assessed as reduction in virus-induced cytopathic effect by MTT assayMore data for this Ligand-Target Pair
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
University Of Belgrade
Curated by ChEMBL
University Of Belgrade
Curated by ChEMBL
Affinity DataEC50: 120nMAssay Description:Inhibition of HIV-1 reverse transcriptase in virus infected human C8166 cells assessed as reduction in virus-induced cytopathic effect by MTT assayMore data for this Ligand-Target Pair
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
University Of Belgrade
Curated by ChEMBL
University Of Belgrade
Curated by ChEMBL
Affinity DataEC50: 120nMAssay Description:Inhibition of HIV-1 reverse transcriptase in virus infected human C8166 cells assessed as reduction in virus-induced cytopathic effect by MTT assayMore data for this Ligand-Target Pair
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
University Of Belgrade
Curated by ChEMBL
University Of Belgrade
Curated by ChEMBL
Affinity DataEC50: 120nMAssay Description:Inhibition of HIV-1 reverse transcriptase in virus infected human C8166 cells assessed as reduction in virus-induced cytopathic effect by MTT assayMore data for this Ligand-Target Pair
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
University Of Belgrade
Curated by ChEMBL
University Of Belgrade
Curated by ChEMBL
Affinity DataEC50: 120nMAssay Description:Inhibition of HIV-1 reverse transcriptase in virus infected human C8166 cells assessed as reduction in virus-induced cytopathic effect by MTT assayMore data for this Ligand-Target Pair
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
University Of Belgrade
Curated by ChEMBL
University Of Belgrade
Curated by ChEMBL
Affinity DataEC50: 120nMAssay Description:Inhibition of HIV-1 reverse transcriptase in virus infected human C8166 cells assessed as reduction in virus-induced cytopathic effect by MTT assayMore data for this Ligand-Target Pair
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
University Of Belgrade
Curated by ChEMBL
University Of Belgrade
Curated by ChEMBL
Affinity DataEC50: 120nMAssay Description:Inhibition of HIV-1 reverse transcriptase in virus infected human C8166 cells assessed as reduction in virus-induced cytopathic effect by MTT assayMore data for this Ligand-Target Pair
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
University Of Belgrade
Curated by ChEMBL
University Of Belgrade
Curated by ChEMBL
Affinity DataEC50: 90nMAssay Description:Inhibition of HIV-1 reverse transcriptase in virus infected human C8166 cells assessed as reduction in virus-induced cytopathic effect by MTT assayMore data for this Ligand-Target Pair
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
University Of Belgrade
Curated by ChEMBL
University Of Belgrade
Curated by ChEMBL
Affinity DataEC50: 90nMAssay Description:Inhibition of HIV-1 reverse transcriptase in virus infected human C8166 cells assessed as reduction in virus-induced cytopathic effect by MTT assayMore data for this Ligand-Target Pair
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
University Of Belgrade
Curated by ChEMBL
University Of Belgrade
Curated by ChEMBL
Affinity DataEC50: 90nMAssay Description:Inhibition of HIV-1 reverse transcriptase in virus infected human C8166 cells assessed as reduction in virus-induced cytopathic effect by MTT assayMore data for this Ligand-Target Pair
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
University Of Belgrade
Curated by ChEMBL
University Of Belgrade
Curated by ChEMBL
Affinity DataEC50: 90nMAssay Description:Inhibition of HIV-1 reverse transcriptase in virus infected human C8166 cells assessed as reduction in virus-induced cytopathic effect by MTT assayMore data for this Ligand-Target Pair
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
University Of Belgrade
Curated by ChEMBL
University Of Belgrade
Curated by ChEMBL
Affinity DataEC50: 9.72E+3nMAssay Description:Inhibition of HIV-1 reverse transcriptase in virus infected human C8166 cells assessed as reduction in virus-induced cytopathic effect by MTT assayMore data for this Ligand-Target Pair
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
University Of Belgrade
Curated by ChEMBL
University Of Belgrade
Curated by ChEMBL
Affinity DataEC50: 170nMAssay Description:Inhibition of HIV-1 reverse transcriptase in virus infected human C8166 cells assessed as reduction in virus-induced cytopathic effect by MTT assayMore data for this Ligand-Target Pair
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
University Of Belgrade
Curated by ChEMBL
University Of Belgrade
Curated by ChEMBL
Affinity DataEC50: 170nMAssay Description:Inhibition of HIV-1 reverse transcriptase in virus infected human C8166 cells assessed as reduction in virus-induced cytopathic effect by MTT assayMore data for this Ligand-Target Pair
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
University Of Belgrade
Curated by ChEMBL
University Of Belgrade
Curated by ChEMBL
Affinity DataEC50: 1.59E+3nMAssay Description:Inhibition of HIV-1 reverse transcriptase in virus infected human C8166 cells assessed as reduction in virus-induced cytopathic effect by MTT assayMore data for this Ligand-Target Pair
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
University Of Belgrade
Curated by ChEMBL
University Of Belgrade
Curated by ChEMBL
Affinity DataEC50: 170nMAssay Description:Inhibition of HIV-1 reverse transcriptase in virus infected human C8166 cells assessed as reduction in virus-induced cytopathic effect by MTT assayMore data for this Ligand-Target Pair
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
University Of Belgrade
Curated by ChEMBL
University Of Belgrade
Curated by ChEMBL
Affinity DataEC50: 170nMAssay Description:Inhibition of HIV-1 reverse transcriptase in virus infected human C8166 cells assessed as reduction in virus-induced cytopathic effect by MTT assayMore data for this Ligand-Target Pair
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
University Of Belgrade
Curated by ChEMBL
University Of Belgrade
Curated by ChEMBL
Affinity DataEC50: 170nMAssay Description:Inhibition of HIV-1 reverse transcriptase in virus infected human C8166 cells assessed as reduction in virus-induced cytopathic effect by MTT assayMore data for this Ligand-Target Pair
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
University Of Belgrade
Curated by ChEMBL
University Of Belgrade
Curated by ChEMBL
Affinity DataEC50: 170nMAssay Description:Inhibition of HIV-1 reverse transcriptase in virus infected human C8166 cells assessed as reduction in virus-induced cytopathic effect by MTT assayMore data for this Ligand-Target Pair
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
University Of Belgrade
Curated by ChEMBL
University Of Belgrade
Curated by ChEMBL
Affinity DataEC50: 170nMAssay Description:Inhibition of HIV-1 reverse transcriptase in virus infected human C8166 cells assessed as reduction in virus-induced cytopathic effect by MTT assayMore data for this Ligand-Target Pair
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
University Of Belgrade
Curated by ChEMBL
University Of Belgrade
Curated by ChEMBL
Affinity DataEC50: 1.87E+3nMAssay Description:Inhibition of HIV-1 reverse transcriptase in virus infected human C8166 cells assessed as reduction in virus-induced cytopathic effect by MTT assayMore data for this Ligand-Target Pair
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
University Of Belgrade
Curated by ChEMBL
University Of Belgrade
Curated by ChEMBL
Affinity DataEC50: 170nMAssay Description:Inhibition of HIV-1 reverse transcriptase in virus infected human C8166 cells assessed as reduction in virus-induced cytopathic effect by MTT assayMore data for this Ligand-Target Pair
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
University Of Belgrade
Curated by ChEMBL
University Of Belgrade
Curated by ChEMBL
Affinity DataEC50: 170nMAssay Description:Inhibition of HIV-1 reverse transcriptase in virus infected human C8166 cells assessed as reduction in virus-induced cytopathic effect by MTT assayMore data for this Ligand-Target Pair
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
University Of Belgrade
Curated by ChEMBL
University Of Belgrade
Curated by ChEMBL
Affinity DataEC50: 170nMAssay Description:Inhibition of HIV-1 reverse transcriptase in virus infected human C8166 cells assessed as reduction in virus-induced cytopathic effect by MTT assayMore data for this Ligand-Target Pair