Affinity DataKi: 2.44E+6nMAssay Description:Displacement of specific [125I]AB-MECA binding at human Adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 3.36E+6nMAssay Description:Displacement of specific [125I]AB-MECA binding at human Adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 3.47E+6nMAssay Description:Displacement of specific [125I]AB-MECA binding at human Adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 3.57E+6nMAssay Description:Displacement of specific [125I]AB-MECA binding at human Adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 3.69E+6nMAssay Description:Displacement of specific [125I]AB-MECA binding at human Adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 3.75E+6nMAssay Description:Displacement of specific [125I]AB-MECA binding at human Adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 4.08E+6nMAssay Description:Displacement of specific [125I]AB-MECA binding at human Adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 4.13E+6nMAssay Description:Displacement of specific [125I]AB-MECA binding at human Adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 4.33E+6nMAssay Description:Displacement of specific [125I]AB-MECA binding at human Adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 4.33E+6nMAssay Description:Displacement of specific [125I]AB-MECA binding at human Adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 4.34E+6nMAssay Description:Displacement of specific [125I]AB-MECA binding at human Adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 4.65E+6nMAssay Description:Displacement of specific [125I]AB-MECA binding at human Adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 4.79E+6nMAssay Description:Displacement of specific [125I]AB-MECA binding at human Adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 4.95E+6nMAssay Description:Displacement of specific [125I]AB-MECA binding at human Adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 5.32E+6nMAssay Description:Displacement of specific [125I]AB-MECA binding at human Adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 5.33E+6nMAssay Description:Displacement of specific [125I]AB-MECA binding at human Adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 6.22E+6nMAssay Description:Displacement of specific [125I]AB-MECA binding at human Adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetEnvelope glycoprotein gp160(Human immunodeficiency virus type 1 group M subtyp...)
Ibitecs, Cea
Curated by ChEMBL
Ibitecs, Cea
Curated by ChEMBL
Affinity DataIC50: 0.260nMAssay Description:Displacement of soluble CD4 from HIV1 SF162 gp120 after overnight incubation by ELISAMore data for this Ligand-Target Pair
TargetEnvelope glycoprotein gp160(Human immunodeficiency virus type 1 group M subtyp...)
Ibitecs, Cea
Curated by ChEMBL
Ibitecs, Cea
Curated by ChEMBL
Affinity DataIC50: 0.280nMAssay Description:Displacement of soluble CD4 from HIV1 SF162 gp120 after overnight incubation by ELISAMore data for this Ligand-Target Pair
TargetEnvelope glycoprotein gp160(Human immunodeficiency virus type 1 group M subtyp...)
Ibitecs, Cea
Curated by ChEMBL
Ibitecs, Cea
Curated by ChEMBL
Affinity DataIC50: 0.300nMAssay Description:Displacement of soluble CD4 from HIV1 SF162 gp120 after overnight incubation by ELISAMore data for this Ligand-Target Pair
TargetEnvelope glycoprotein gp160(Human immunodeficiency virus type 1 group M subtyp...)
Ibitecs, Cea
Curated by ChEMBL
Ibitecs, Cea
Curated by ChEMBL
Affinity DataIC50: 0.320nMAssay Description:Displacement of soluble CD4 from HIV1 SF162 gp120 after overnight incubation by ELISAMore data for this Ligand-Target Pair
TargetEnvelope glycoprotein gp160(Human immunodeficiency virus type 1 group M subtyp...)
Ibitecs, Cea
Curated by ChEMBL
Ibitecs, Cea
Curated by ChEMBL
Affinity DataIC50: 0.350nMAssay Description:Displacement of soluble CD4 from HIV1 SF162 gp120 after overnight incubation by ELISAMore data for this Ligand-Target Pair
TargetEnvelope glycoprotein gp160(Human immunodeficiency virus type 1 group M subtyp...)
Ibitecs, Cea
Curated by ChEMBL
Ibitecs, Cea
Curated by ChEMBL
Affinity DataIC50: 0.5nMAssay Description:Displacement of soluble CD4 from HIV1 SF162 gp120 after overnight incubation by ELISAMore data for this Ligand-Target Pair
TargetEnvelope glycoprotein gp160(Human immunodeficiency virus type 1 group M subtyp...)
Ibitecs, Cea
Curated by ChEMBL
Ibitecs, Cea
Curated by ChEMBL
Affinity DataIC50: 0.520nMAssay Description:Displacement of soluble CD4 from HIV1 SF162 gp120 after overnight incubation by ELISAMore data for this Ligand-Target Pair
TargetEnvelope glycoprotein gp160(Human immunodeficiency virus type 1 group M subtyp...)
Ibitecs, Cea
Curated by ChEMBL
Ibitecs, Cea
Curated by ChEMBL
Affinity DataIC50: 0.860nMAssay Description:Displacement of soluble CD4 from HIV1 SF162 gp120 after overnight incubation by ELISAMore data for this Ligand-Target Pair
TargetEnvelope glycoprotein gp160(Human immunodeficiency virus type 1 group M subtyp...)
Ibitecs, Cea
Curated by ChEMBL
Ibitecs, Cea
Curated by ChEMBL
Affinity DataIC50: 1.10nMAssay Description:Displacement of soluble CD4 from HIV1 SF162 gp120 after overnight incubation by ELISAMore data for this Ligand-Target Pair
TargetEnvelope glycoprotein gp160(Human immunodeficiency virus type 1 group M subtyp...)
Ibitecs, Cea
Curated by ChEMBL
Ibitecs, Cea
Curated by ChEMBL
Affinity DataIC50: 1.40nMAssay Description:Displacement of soluble CD4 from HIV1 SF162 gp120 after overnight incubation by ELISAMore data for this Ligand-Target Pair
TargetEnvelope glycoprotein gp160(Human immunodeficiency virus type 1 group M subtyp...)
Ibitecs, Cea
Curated by ChEMBL
Ibitecs, Cea
Curated by ChEMBL
Affinity DataIC50: 5.20nMAssay Description:Displacement of soluble CD4 from HIV1 SF162 gp120 after overnight incubation by ELISAMore data for this Ligand-Target Pair
TargetEnvelope glycoprotein gp160(Human immunodeficiency virus type 1 group M subtyp...)
Ibitecs, Cea
Curated by ChEMBL
Ibitecs, Cea
Curated by ChEMBL
Affinity DataIC50: 5.30nMAssay Description:Displacement of soluble CD4 from HIV1 SF162 gp120 after overnight incubation by ELISAMore data for this Ligand-Target Pair
TargetEnvelope glycoprotein gp160(Human immunodeficiency virus type 1 group M subtyp...)
Ibitecs, Cea
Curated by ChEMBL
Ibitecs, Cea
Curated by ChEMBL
Affinity DataIC50: 8.10nMAssay Description:Displacement of soluble CD4 from HIV1 SF162 gp120 after overnight incubation by ELISAMore data for this Ligand-Target Pair
TargetEnvelope glycoprotein gp160(Human immunodeficiency virus type 1 group M subtyp...)
Ibitecs, Cea
Curated by ChEMBL
Ibitecs, Cea
Curated by ChEMBL
Affinity DataIC50: 284nMAssay Description:Displacement of soluble CD4 from HIV1 SF162 gp120 after overnight incubation by ELISAMore data for this Ligand-Target Pair
TargetCyclin-dependent kinase 1/G2/mitotic-specific cyclin-B1/G2/mitotic-specific cyclin-B2/G2/mitotic-specific cyclin-B3(Homo sapiens (Human))
Vanderbilt University School Of Medicine
Curated by ChEMBL
Vanderbilt University School Of Medicine
Curated by ChEMBL
Affinity DataIC50: 400nMAssay Description:Inhibition of Cyclin-dependent kinase 1-cyclin B of M-phase Marthasterias glacialis oocytesMore data for this Ligand-Target Pair
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Vanderbilt University School Of Medicine
Curated by ChEMBL
Vanderbilt University School Of Medicine
Curated by ChEMBL
Affinity DataIC50: 800nMAssay Description:Inhibition of Cyclin-dependent kinase 5-p35nck5aMore data for this Ligand-Target Pair
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Vanderbilt University School Of Medicine
Curated by ChEMBL
Vanderbilt University School Of Medicine
Curated by ChEMBL
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of Cyclin-dependent kinase 5-p35nck5aMore data for this Ligand-Target Pair
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Vanderbilt University School Of Medicine
Curated by ChEMBL
Vanderbilt University School Of Medicine
Curated by ChEMBL
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of Cyclin-dependent kinase 5-p35nck5aMore data for this Ligand-Target Pair
TargetCyclin-dependent kinase 1/G2/mitotic-specific cyclin-B1/G2/mitotic-specific cyclin-B2/G2/mitotic-specific cyclin-B3(Homo sapiens (Human))
Vanderbilt University School Of Medicine
Curated by ChEMBL
Vanderbilt University School Of Medicine
Curated by ChEMBL
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of Cyclin-dependent kinase 1-cyclin B of M-phase Marthasterias glacialis oocytesMore data for this Ligand-Target Pair
TargetCyclin-dependent kinase 1/G2/mitotic-specific cyclin-B1/G2/mitotic-specific cyclin-B2/G2/mitotic-specific cyclin-B3(Homo sapiens (Human))
Vanderbilt University School Of Medicine
Curated by ChEMBL
Vanderbilt University School Of Medicine
Curated by ChEMBL
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of Cyclin-dependent kinase 1-cyclin B of M-phase Marthasterias glacialis oocytesMore data for this Ligand-Target Pair
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Vanderbilt University School Of Medicine
Curated by ChEMBL
Vanderbilt University School Of Medicine
Curated by ChEMBL
Affinity DataIC50: 1.90E+3nMAssay Description:Inhibition of Cyclin-dependent kinase 5-p35nck5aMore data for this Ligand-Target Pair
TargetEnvelope glycoprotein gp160(Human immunodeficiency virus type 1 group M subtyp...)
Ibitecs, Cea
Curated by ChEMBL
Ibitecs, Cea
Curated by ChEMBL
Affinity DataIC50: 2.03E+3nMAssay Description:Displacement of soluble CD4 from HIV1 SF162 gp120 after overnight incubation by ELISAMore data for this Ligand-Target Pair
TargetCyclin-dependent kinase 1/G2/mitotic-specific cyclin-B1/G2/mitotic-specific cyclin-B2/G2/mitotic-specific cyclin-B3(Homo sapiens (Human))
Vanderbilt University School Of Medicine
Curated by ChEMBL
Vanderbilt University School Of Medicine
Curated by ChEMBL
Affinity DataIC50: 2.10E+3nMAssay Description:Inhibition of Cyclin-dependent kinase 1-cyclin B of M-phase Marthasterias glacialis oocytesMore data for this Ligand-Target Pair
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Vanderbilt University School Of Medicine
Curated by ChEMBL
Vanderbilt University School Of Medicine
Curated by ChEMBL
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of Cyclin-dependent kinase 5-p35nck5aMore data for this Ligand-Target Pair
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Vanderbilt University School Of Medicine
Curated by ChEMBL
Vanderbilt University School Of Medicine
Curated by ChEMBL
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of Cyclin-dependent kinase 5-p35nck5aMore data for this Ligand-Target Pair
TargetCyclin-dependent kinase 1/G2/mitotic-specific cyclin-B1/G2/mitotic-specific cyclin-B2/G2/mitotic-specific cyclin-B3(Homo sapiens (Human))
Vanderbilt University School Of Medicine
Curated by ChEMBL
Vanderbilt University School Of Medicine
Curated by ChEMBL
Affinity DataIC50: 6.50E+3nMAssay Description:Inhibition of Cyclin-dependent kinase 1-cyclin B of M-phase Marthasterias glacialis oocytesMore data for this Ligand-Target Pair
Affinity DataIC50: 2.29E+4nMAssay Description:Inhibition of human DNA topoisomerase-1 using supercoiled pBAD-GFPuv plasmid DNA as substrate assessed as prevention of supercoiled DNA template from...More data for this Ligand-Target Pair
Affinity DataIC50: 2.54E+4nMAssay Description:Inhibition of human DNA topoisomerase-1 using supercoiled pBAD-GFPuv plasmid DNA as substrate assessed as prevention of supercoiled DNA template from...More data for this Ligand-Target Pair
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Vanderbilt University School Of Medicine
Curated by ChEMBL
Vanderbilt University School Of Medicine
Curated by ChEMBL
Affinity DataIC50: 2.60E+4nMAssay Description:Inhibition of Cyclin-dependent kinase 5-p35nck5aMore data for this Ligand-Target Pair
Affinity DataIC50: 2.89E+4nMAssay Description:Inhibition of human DNA topoisomerase-2 using supercoiled pBAD-GFPuv plasmid DNA as substrate assessed as prevention of supercoiled DNA template from...More data for this Ligand-Target Pair
Affinity DataIC50: >5.00E+4nMAssay Description:Binding affinity towards adenosine A1 receptor of rat brain membranes with 1 M NaCl by inhibition of [125-I]-labeled aminobenzyl adenosine binding More data for this Ligand-Target Pair
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of human DNA topoisomerase 1 using plasmid pBAD-GFPuv as substrate after 30 mins by agarose gel electrophoresisMore data for this Ligand-Target Pair
Affinity DataIC50: >5.00E+4nMAssay Description:Binding affinity to adenosine A1 receptor of rat brain membranes without NaCl by inhibition of [125-I]-labeled aminobenzyl adenosine bindingMore data for this Ligand-Target Pair