TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Nri Institute Of Pharmacy
Curated by ChEMBL
Nri Institute Of Pharmacy
Curated by ChEMBL
Affinity DataKi: 5nMAssay Description:Inhibition of PIM1 (unknown origin) up to 120 mins by Michaelis-Menten plot analysisMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Nri Institute Of Pharmacy
Curated by ChEMBL
Nri Institute Of Pharmacy
Curated by ChEMBL
Affinity DataKi: 7.70nMAssay Description:Inhibition of N-terminal GST-tagged recombinant human full length Pim-1 expressed in Escherichia coli cellsMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Nri Institute Of Pharmacy
Curated by ChEMBL
Nri Institute Of Pharmacy
Curated by ChEMBL
Affinity DataKi: 12nMAssay Description:Inhibition of PIM1 (unknown origin) up to 120 mins by Michaelis-Menten plot analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 0.350nMAssay Description:Inhibition of human SGLT2More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 6.5nMAssay Description:Inhibitory activity against FAAH in Wistar rat brain homogenateMore data for this Ligand-Target Pair
Affinity DataIC50: 7.20nMAssay Description:Inhibitory activity against FAAH in Wistar rat brain homogenateMore data for this Ligand-Target Pair
Affinity DataIC50: 8nMAssay Description:Inhibitory activity against FAAH in Wistar rat brain homogenateMore data for this Ligand-Target Pair
Affinity DataIC50: 8nMAssay Description:Inhibitory activity against FAAH in Wistar rat brain homogenateMore data for this Ligand-Target Pair
Affinity DataIC50: 9.70nMAssay Description:Inhibitory activity against FAAH in Wistar rat brain homogenateMore data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Inhibitory activity against FAAH in Wistar rat brain homogenateMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Nri Institute Of Pharmacy
Curated by ChEMBL
Nri Institute Of Pharmacy
Curated by ChEMBL
Affinity DataIC50: 60nMAssay Description:Inhibition of human PIM1 by ELISAMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Nri Institute Of Pharmacy
Curated by ChEMBL
Nri Institute Of Pharmacy
Curated by ChEMBL
Affinity DataIC50: 80nMAssay Description:Inhibition of human PIM1 by ELISAMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Nri Institute Of Pharmacy
Curated by ChEMBL
Nri Institute Of Pharmacy
Curated by ChEMBL
Affinity DataIC50: 111nMAssay Description:Inhibition of PIM1 (unknown origin)More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Nri Institute Of Pharmacy
Curated by ChEMBL
Nri Institute Of Pharmacy
Curated by ChEMBL
Affinity DataIC50: <150nMAssay Description:Inhibition of PIM1 (unknown origin)More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Nri Institute Of Pharmacy
Curated by ChEMBL
Nri Institute Of Pharmacy
Curated by ChEMBL
Affinity DataIC50: <150nMAssay Description:Inhibition of PIM1 (unknown origin)More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Nri Institute Of Pharmacy
Curated by ChEMBL
Nri Institute Of Pharmacy
Curated by ChEMBL
Affinity DataIC50: 434nMAssay Description:Inhibition of PIM1 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 1.57E+3nMAssay Description:Inhibitory activity against FAAH in Wistar rat brain homogenateMore data for this Ligand-Target Pair
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Guru Ghasidas Vishwavidyalaya (A Central University)
Curated by ChEMBL
Guru Ghasidas Vishwavidyalaya (A Central University)
Curated by ChEMBL
Affinity DataIC50: 2.49E+3nMAssay Description:Competitive inhibition of PTP1B (unknown origin) using p-nitrophenyl phosphate as substrateMore data for this Ligand-Target Pair
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Guru Ghasidas Vishwavidyalaya (A Central University)
Curated by ChEMBL
Guru Ghasidas Vishwavidyalaya (A Central University)
Curated by ChEMBL
Affinity DataIC50: 2.90E+3nMAssay Description:Competitive inhibition of PTP1B (unknown origin) using p-nitrophenyl phosphate as substrateMore data for this Ligand-Target Pair
Affinity DataIC50: 4.18E+3nMAssay Description:Inhibitory activity against FAAH in Wistar rat brain homogenateMore data for this Ligand-Target Pair
Affinity DataIC50: 5.83E+3nMAssay Description:Inhibitory activity against FAAH in Wistar rat brain homogenateMore data for this Ligand-Target Pair
TargetPlasmepsin II(Plasmodium falciparum)
Guru Ghasidas Vishwavidyalaya (A Central University)
Curated by ChEMBL
Guru Ghasidas Vishwavidyalaya (A Central University)
Curated by ChEMBL
Affinity DataIC50: 6.00E+3nMAssay Description:Inhibition of Plasmodium falciparum plasmepsin 2More data for this Ligand-Target Pair
TargetPlasmepsin II(Plasmodium falciparum)
Guru Ghasidas Vishwavidyalaya (A Central University)
Curated by ChEMBL
Guru Ghasidas Vishwavidyalaya (A Central University)
Curated by ChEMBL
Affinity DataIC50: 6.00E+3nMAssay Description:Inhibition of Plasmodium falciparum plasmepsin 2More data for this Ligand-Target Pair
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Guru Ghasidas Vishwavidyalaya (A Central University)
Curated by ChEMBL
Guru Ghasidas Vishwavidyalaya (A Central University)
Curated by ChEMBL
Affinity DataIC50: 2.15E+4nMAssay Description:Inhibition of PTP1B (unknown origin)More data for this Ligand-Target Pair