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Found 31 with Last Name = 'athmani' and Initial = 's'
TargetHistamine H3 receptor(Rattus norvegicus (rat))
University College London

Curated by ChEMBL
LigandPNGBDBM50053297(1-{4-[2-(1H-Imidazol-4-yl)-ethoxy]-phenyl}-propan-...)
Affinity DataKi:  3.70nMAssay Description:Rat Histamine H3 receptor antagonism determined by [K+] - evoked depolarization-induced release of [3H]-histamine from rat cerebral cortex synaptosom...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
University College London

Curated by ChEMBL
LigandPNGBDBM22914(CHEMBL260374 | N-cyclohexyl-4-(1H-imidazol-5-yl)pi...)
Affinity DataKi:  4nMAssay Description:Rat Histamine H3 receptor antagonism determined by [K+] - evoked depolarization-induced release of [3H]-histamine from rat cerebral cortex synaptosom...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
University College London

Curated by ChEMBL
LigandPNGBDBM50033042(2-[2-(1H-Imidazol-4-yl)-ethylsulfanyl]-5-nitro-pyr...)
Affinity DataKi:  4.80nMAssay Description:Rat Histamine H3 receptor antagonism determined by [K+] - evoked depolarization-induced release of [3H]-histamine from rat cerebral cortex synaptosom...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
University College London

Curated by ChEMBL
LigandPNGBDBM50053275(4-[2-(1H-Imidazol-4-yl)-ethoxy]-benzoic acid methy...)
Affinity DataKi:  5.10nMAssay Description:Rat Histamine H3 receptor antagonism determined by [K+] - evoked depolarization-induced release of [3H]-histamine from rat cerebral cortex synaptosom...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
University College London

Curated by ChEMBL
LigandPNGBDBM50053281(4-[2-(1H-Imidazol-4-yl)-ethoxy]-benzoic acid ethyl...)
Affinity DataKi:  6nMAssay Description:Rat Histamine H3 receptor antagonism determined by [K+] - evoked depolarization-induced release of [3H]-histamine from rat cerebral cortex synaptosom...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
University College London

Curated by ChEMBL
LigandPNGBDBM50053289(4-[2-(1H-Imidazol-4-yl)-ethoxy]-benzonitrile | CHE...)
Affinity DataKi:  9nMAssay Description:Rat Histamine H3 receptor antagonism determined by [K+] - evoked depolarization-induced release of [3H]-histamine from rat cerebral cortex synaptosom...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
University College London

Curated by ChEMBL
LigandPNGBDBM50053273(4-[2-(4-Nitro-phenylsulfanyl)-ethyl]-1H-imidazole ...)
Affinity DataKi:  9nMAssay Description:Rat Histamine H3 receptor antagonism determined by [K+] - evoked depolarization-induced release of [3H]-histamine from rat cerebral cortex synaptosom...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
University College London

Curated by ChEMBL
LigandPNGBDBM50053274(4-[3-(4-Fluoro-phenoxy)-propyl]-1H-imidazole | CHE...)
Affinity DataKi:  11nMAssay Description:Rat Histamine H3 receptor antagonism determined by [K+] - evoked depolarization-induced release of [3H]-histamine from rat cerebral cortex synaptosom...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
University College London

Curated by ChEMBL
LigandPNGBDBM50053278(4-[3-(1H-Imidazol-4-yl)-propoxy]-benzonitrile | 4-...)
Affinity DataKi:  12nMAssay Description:Rat Histamine H3 receptor antagonism determined by [K+] - evoked depolarization-induced release of [3H]-histamine from rat cerebral cortex synaptosom...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
University College London

Curated by ChEMBL
LigandPNGBDBM50053290(4-[2-(3-Nitro-phenoxy)-ethyl]-1H-imidazole | CHEMB...)
Affinity DataKi:  12nMAssay Description:Rat Histamine H3 receptor antagonism determined by [K+] - evoked depolarization-induced release of [3H]-histamine from rat cerebral cortex synaptosom...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
University College London

Curated by ChEMBL
LigandPNGBDBM50053298(4-[3-(4-Trifluoromethyl-phenoxy)-propyl]-1H-imidaz...)
Affinity DataKi:  14nMAssay Description:Rat Histamine H3 receptor antagonism determined by [K+] - evoked depolarization-induced release of [3H]-histamine from rat cerebral cortex synaptosom...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
University College London

Curated by ChEMBL
LigandPNGBDBM50053288(4-[2-(4-Propyl-phenoxy)-ethyl]-1H-imidazole | CHEM...)
Affinity DataKi:  19nMAssay Description:Rat Histamine H3 receptor antagonism determined by [K+] - evoked depolarization-induced release of [3H]-histamine from rat cerebral cortex synaptosom...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
University College London

Curated by ChEMBL
LigandPNGBDBM50033036(CHEMBL419574 | [2-(1H-Imidazol-4-yl)-ethyl]-(5-nit...)
Affinity DataKi:  20nMAssay Description:Rat Histamine H3 receptor antagonism determined by [K+] - evoked depolarization-induced release of [3H]-histamine from rat cerebral cortex synaptosom...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
University College London

Curated by ChEMBL
LigandPNGBDBM50053294(4-[2-(4-Chloro-phenoxy)-ethyl]-1H-imidazole | CHEM...)
Affinity DataKi:  21nMAssay Description:Rat Histamine H3 receptor antagonism determined by [K+] - evoked depolarization-induced release of [3H]-histamine from rat cerebral cortex synaptosom...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
University College London

Curated by ChEMBL
LigandPNGBDBM50053292(1-{4-[2-(1H-Imidazol-4-yl)-ethoxy]-phenyl}-ethanon...)
Affinity DataKi:  23nMAssay Description:Rat Histamine H3 receptor antagonism determined by [K+] - evoked depolarization-induced release of [3H]-histamine from rat cerebral cortex synaptosom...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
University College London

Curated by ChEMBL
LigandPNGBDBM50053280(CHEMBL435383 | [2-(1H-Imidazol-4-yl)-ethyl]-(4-nit...)
Affinity DataKi:  23nMAssay Description:Rat Histamine H3 receptor antagonism determined by [K+] - evoked depolarization-induced release of [3H]-histamine from rat cerebral cortex synaptosom...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
University College London

Curated by ChEMBL
LigandPNGBDBM50053277(4-[2-(4-Bromo-phenoxy)-ethyl]-1H-imidazole | CHEMB...)
Affinity DataKi:  24nMAssay Description:Rat Histamine H3 receptor antagonism determined by [K+] - evoked depolarization-induced release of [3H]-histamine from rat cerebral cortex synaptosom...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
University College London

Curated by ChEMBL
LigandPNGBDBM50053279(4-[2-(4-Nitro-phenoxy)-ethyl]-1H-imidazole | CHEMB...)
Affinity DataKi:  35nMAssay Description:Rat Histamine H3 receptor antagonism determined by [K+] - evoked depolarization-induced release of [3H]-histamine from rat cerebral cortex synaptosom...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
University College London

Curated by ChEMBL
LigandPNGBDBM50053271(4-[2-(4-Methoxy-phenoxy)-ethyl]-1H-imidazole | CHE...)
Affinity DataKi:  38nMAssay Description:Rat Histamine H3 receptor antagonism determined by [K+] - evoked depolarization-induced release of [3H]-histamine from rat cerebral cortex synaptosom...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
University College London

Curated by ChEMBL
LigandPNGBDBM50053282(3-[2-(1H-Imidazol-4-yl)-ethoxy]-benzonitrile | CHE...)
Affinity DataKi:  39nMAssay Description:Rat Histamine H3 receptor antagonism determined by [K+] - evoked depolarization-induced release of [3H]-histamine from rat cerebral cortex synaptosom...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
University College London

Curated by ChEMBL
LigandPNGBDBM50053295(CHEMBL125751 | {4-[2-(1H-Imidazol-4-yl)-ethoxy]-ph...)
Affinity DataKi:  54nMAssay Description:Rat Histamine H3 receptor antagonism determined by [K+] - evoked depolarization-induced release of [3H]-histamine from rat cerebral cortex synaptosom...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
University College London

Curated by ChEMBL
LigandPNGBDBM50053272(4-(2-p-Tolyloxy-ethyl)-1H-imidazole | CHEMBL125947)
Affinity DataKi:  56nMAssay Description:Rat Histamine H3 receptor antagonism determined by [K+] - evoked depolarization-induced release of [3H]-histamine from rat cerebral cortex synaptosom...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
University College London

Curated by ChEMBL
LigandPNGBDBM50053284(4-[2-(4-Trifluoromethyl-phenoxy)-ethyl]-1H-imidazo...)
Affinity DataKi:  68nMAssay Description:Rat Histamine H3 receptor antagonism determined by [K+] - evoked depolarization-induced release of [3H]-histamine from rat cerebral cortex synaptosom...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
University College London

Curated by ChEMBL
LigandPNGBDBM50053285(4-[2-(4-Ethyl-phenoxy)-ethyl]-1H-imidazole | CHEMB...)
Affinity DataKi:  80nMAssay Description:Rat Histamine H3 receptor antagonism determined by [K+] - evoked depolarization-induced release of [3H]-histamine from rat cerebral cortex synaptosom...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
University College London

Curated by ChEMBL
LigandPNGBDBM50053276(4-[2-(Naphthalen-2-yloxy)-ethyl]-1H-imidazole | CH...)
Affinity DataKi:  90nMAssay Description:Rat Histamine H3 receptor antagonism determined by [K+] - evoked depolarization-induced release of [3H]-histamine from rat cerebral cortex synaptosom...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
University College London

Curated by ChEMBL
LigandPNGBDBM50053296(4-[2-(Naphthalen-1-yloxy)-ethyl]-1H-imidazole | CH...)
Affinity DataKi:  137nMAssay Description:Rat Histamine H3 receptor antagonism determined by [K+] - evoked depolarization-induced release of [3H]-histamine from rat cerebral cortex synaptosom...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
University College London

Curated by ChEMBL
LigandPNGBDBM50053287(4-(4-Nitro-benzylsulfanylmethyl)-1H-imidazole | CH...)
Affinity DataKi:  313nMAssay Description:Rat Histamine H3 receptor antagonism determined by [K+] - evoked depolarization-induced release of [3H]-histamine from rat cerebral cortex synaptosom...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
University College London

Curated by ChEMBL
LigandPNGBDBM50053293(CHEMBL339606 | {4-[2-(1H-Imidazol-4-yl)-ethoxy]-ph...)
Affinity DataKi:  338nMAssay Description:Rat Histamine H3 receptor antagonism determined by [K+] - evoked depolarization-induced release of [3H]-histamine from rat cerebral cortex synaptosom...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
University College London

Curated by ChEMBL
LigandPNGBDBM50053283(2-[2-(1H-Imidazol-4-yl)-ethoxy]-benzonitrile | CHE...)
Affinity DataKi:  483nMAssay Description:Rat Histamine H3 receptor antagonism determined by [K+] - evoked depolarization-induced release of [3H]-histamine from rat cerebral cortex synaptosom...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
University College London

Curated by ChEMBL
LigandPNGBDBM50053286(4-(2-Pentafluorophenyloxy-ethyl)-1H-imidazole | CH...)
Affinity DataKi: >500nMAssay Description:Rat Histamine H3 receptor antagonism determined by [K+] - evoked depolarization-induced release of [3H]-histamine from rat cerebral cortex synaptosom...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
University College London

Curated by ChEMBL
LigandPNGBDBM50053291(4-[2-(3,5-Dichloro-phenoxy)-ethyl]-1H-imidazole | ...)
Affinity DataKi: >500nMAssay Description:Rat Histamine H3 receptor antagonism determined by [K+] - evoked depolarization-induced release of [3H]-histamine from rat cerebral cortex synaptosom...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed