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Found 12819 with Last Name = 'atteri' and Initial = 'e'
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM201((2S)-N-[(2S,3S)-4-[(2S)-N'-(cyclohexylmethyl)-2-ac...)
Affinity DataIC50:  9nMpH: 6.0Assay Description:In vitro inhibition of HIV-1 protease at pH 6 using 164 microM peptide substrateMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50281324(((S)-1-{N'-[(2S,3S)-3-((S)-2-Benzyloxycarbonylamin...)
Affinity DataIC50:  10nMpH: 6.0Assay Description:In vitro inhibition of HIV-1 protease at pH 6 using 164 microM peptide substrateMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50281333(CHEMBL97512 | {(S)-1-[N'-[(2S,3S)-3-((S)-2-Benzylo...)
Affinity DataIC50:  22nMpH: 6.0Assay Description:In vitro inhibition of HIV-1 protease at pH 6 using 164 microM peptide substrateMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50281332(CHEMBL95462 | {(S)-1-[N'-[(2S,3S)-3-((S)-2-Benzylo...)
Affinity DataIC50:  24nMpH: 6.0Assay Description:In vitro inhibition of HIV-1 protease at pH 6 using 164 microM peptide substrateMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50281328((S)-2-Acetylamino-N-{(1S,2S)-3-[N'-((S)-2-acetylam...)
Affinity DataIC50:  28nMpH: 6.0Assay Description:In vitro inhibition of HIV-1 protease at pH 6 using 164 microM peptide substrateMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50281330((S)-2-Acetylamino-N-{(1S,2S)-3-[N'-((R)-2-acetylam...)
Affinity DataIC50:  30nMpH: 6.0Assay Description:In vitro inhibition of HIV-1 protease at pH 6 using 164 microM peptide substrateMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50281335(((R)-1-{N'-Benzyl-N'-[(2S,3S)-3-((S)-2-benzyloxyca...)
Affinity DataIC50:  33nMpH: 6.0Assay Description:In vitro inhibition of HIV-1 protease at pH 6 using 164 microM peptide substrateMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50281327((S)-2-Acetylamino-N-{(1S,2S)-3-[N'-((S)-2-acetylam...)
Affinity DataIC50:  45nMpH: 6.0Assay Description:In vitro inhibition of HIV-1 protease at pH 6 using 164 microM peptide substrateMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50281337((S)-2-Acetylamino-N-{(1S,2S)-3-[N'-((S)-2-acetylam...)
Affinity DataIC50:  50nMpH: 6.0Assay Description:In vitro inhibition of HIV-1 protease at pH 6 using 164 microM peptide substrateMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50281329(CHEMBL97146 | quinoline-2-carboxylic acid {(S)-1-[...)
Affinity DataIC50:  65nMpH: 6.0Assay Description:In vitro inhibition of HIV-1 protease at pH 6 using 164 microM peptide substrateMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50281323(((S)-1-{N'-[(2S,3S)-3-((S)-2-Benzyloxycarbonylamin...)
Affinity DataIC50:  95nMpH: 6.0Assay Description:In vitro inhibition of HIV-1 protease at pH 6 using 164 microM peptide substrateMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50281334((S)-N-{(1S,2S)-1-Benzyl-3-[N-benzyl-N'-((R)-3-meth...)
Affinity DataIC50:  360nMpH: 6.0Assay Description:In vitro inhibition of HIV-1 protease at pH 6 using 164 microM peptide substrateMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50281338((S)-N-((1S,2S)-1-Benzyl-3-{N-benzyl-N'-[(R)-3-meth...)
Affinity DataIC50:  500nMpH: 6.0Assay Description:In vitro inhibition of HIV-1 protease at pH 6 using 164 microM peptide substrateMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGastricsin(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM201((2S)-N-[(2S,3S)-4-[(2S)-N'-(cyclohexylmethyl)-2-ac...)
Affinity DataIC50:  1.00E+3nMAssay Description:The compound was tested for its inhibitory activity against human gastricsinMore data for this Ligand-Target Pair
In DepthDetails Article
TargetPepsin A(Porcine)
TBA

Curated by ChEMBL
LigandPNGBDBM201((2S)-N-[(2S,3S)-4-[(2S)-N'-(cyclohexylmethyl)-2-ac...)
Affinity DataIC50:  1.00E+3nMAssay Description:The compound was tested for its inhibitory activity against human pepsinMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50281336(CHEMBL327985 | morpholine-4-carboxylic acid {(S)-1...)
Affinity DataIC50:  2.00E+3nMpH: 6.0Assay Description:In vitro inhibition of HIV-1 protease at pH 6 using 164 microM peptide substrateMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCathepsin E(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM201((2S)-N-[(2S,3S)-4-[(2S)-N'-(cyclohexylmethyl)-2-ac...)
Affinity DataIC50:  2.00E+3nMAssay Description:The compound was tested for its inhibitory activity against human cathepsin EMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCathepsin D(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM201((2S)-N-[(2S,3S)-4-[(2S)-N'-(cyclohexylmethyl)-2-ac...)
Affinity DataIC50:  7.50E+3nMAssay Description:The compound was tested for its inhibitory activity against human cathepsin DMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50281331(((R)-1-{N'-Benzyl-N'-[(2S,3S)-3-((S)-2-tert-butoxy...)
Affinity DataIC50:  5.20E+4nMpH: 6.0Assay Description:In vitro inhibition of HIV-1 protease at pH 6 using 164 microM peptide substrateMore data for this Ligand-Target Pair
In DepthDetails Article
TargetRenin(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM201((2S)-N-[(2S,3S)-4-[(2S)-N'-(cyclohexylmethyl)-2-ac...)
Affinity DataIC50: >5.80E+4nMAssay Description:The compound was tested for its inhibitory activity against human reninMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50281325(((S)-1-{N'-Benzyl-N'-[(2S,3S)-3-((R)-2-benzyloxyca...)
Affinity DataIC50: >1.00E+5nMpH: 6.0Assay Description:In vitro inhibition of HIV-1 protease at pH 6 using 164 microM peptide substrateMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50281326(2-Amino-N-{(S)-3-[N'-((R)-2-amino-3-methyl-butyryl...)
Affinity DataIC50: >1.00E+5nMpH: 6.0Assay Description:In vitro inhibition of HIV-1 protease at pH 6 using 164 microM peptide substrateMore data for this Ligand-Target Pair
In DepthDetails Article
TargetTyrosine-protein kinase ABL1 [201-500](Homo sapiens (Human))
Ambit

LigandPNGBDBM13530(4-[(4-methylpiperazin-1-yl)methyl]-N-[4-methyl-3-[...)
Affinity DataKd:  2nMpH: 7.4 T: 2°CAssay Description:Competition binding assay was used to measure the interaction between the phage-tagged kinase, immobilized competitive ligand, and unlinked test comp...More data for this Ligand-Target Pair
TargetTyrosine-protein kinase ABL1 [201-500,Q252H](Homo sapiens (Human))
Ambit

LigandPNGBDBM13530(4-[(4-methylpiperazin-1-yl)methyl]-N-[4-methyl-3-[...)
Affinity DataKd:  20nMpH: 7.4 T: 2°CAssay Description:Competition binding assay was used to measure the interaction between the phage-tagged kinase, immobilized competitive ligand, and unlinked test comp...More data for this Ligand-Target Pair
TargetTyrosine-protein kinase ABL1 [201-500,Y253F](Homo sapiens (Human))
Ambit

LigandPNGBDBM13530(4-[(4-methylpiperazin-1-yl)methyl]-N-[4-methyl-3-[...)
Affinity DataKd:  40nMpH: 7.4 T: 2°CAssay Description:Competition binding assay was used to measure the interaction between the phage-tagged kinase, immobilized competitive ligand, and unlinked test comp...More data for this Ligand-Target Pair
TargetTyrosine-protein kinase ABL1 [201-500,E255K](Homo sapiens (Human))
Ambit

LigandPNGBDBM13530(4-[(4-methylpiperazin-1-yl)methyl]-N-[4-methyl-3-[...)
Affinity DataKd:  100nMpH: 7.4 T: 2°CAssay Description:Competition binding assay was used to measure the interaction between the phage-tagged kinase, immobilized competitive ligand, and unlinked test comp...More data for this Ligand-Target Pair
TargetTyrosine-protein kinase ABL1 [201-500,M351T](Homo sapiens (Human))
Ambit

LigandPNGBDBM13530(4-[(4-methylpiperazin-1-yl)methyl]-N-[4-methyl-3-[...)
Affinity DataKd:  10nMpH: 7.4 T: 2°CAssay Description:Competition binding assay was used to measure the interaction between the phage-tagged kinase, immobilized competitive ligand, and unlinked test comp...More data for this Ligand-Target Pair
TargetTyrosine-protein kinase ABL1 [201-500,F359V](Homo sapiens (Human))
Ambit

LigandPNGBDBM13530(4-[(4-methylpiperazin-1-yl)methyl]-N-[4-methyl-3-[...)
Affinity DataKd:  20nMpH: 7.4 T: 2°CAssay Description:Competition binding assay was used to measure the interaction between the phage-tagged kinase, immobilized competitive ligand, and unlinked test comp...More data for this Ligand-Target Pair
TargetTyrosine-protein kinase ABL1 [201-500](Homo sapiens (Human))
Ambit

LigandPNGBDBM13216(BMS-354825 | CHEMBL1421 | DASATINIB | N-(2-Chloro-...)
Affinity DataKd:  0.5nMpH: 7.4 T: 2°CAssay Description:Competition binding assay was used to measure the interaction between the phage-tagged kinase, immobilized competitive ligand, and unlinked test comp...More data for this Ligand-Target Pair
TargetTyrosine-protein kinase ABL1 [201-500,Q252H](Homo sapiens (Human))
Ambit

LigandPNGBDBM13216(BMS-354825 | CHEMBL1421 | DASATINIB | N-(2-Chloro-...)
Affinity DataKd:  1nMpH: 7.4 T: 2°CAssay Description:Competition binding assay was used to measure the interaction between the phage-tagged kinase, immobilized competitive ligand, and unlinked test comp...More data for this Ligand-Target Pair
TargetTyrosine-protein kinase ABL1 [201-500,Y253F](Homo sapiens (Human))
Ambit

LigandPNGBDBM13216(BMS-354825 | CHEMBL1421 | DASATINIB | N-(2-Chloro-...)
Affinity DataKd:  1nMpH: 7.4 T: 2°CAssay Description:Competition binding assay was used to measure the interaction between the phage-tagged kinase, immobilized competitive ligand, and unlinked test comp...More data for this Ligand-Target Pair
TargetTyrosine-protein kinase ABL1 [201-500,E255K](Homo sapiens (Human))
Ambit

LigandPNGBDBM13216(BMS-354825 | CHEMBL1421 | DASATINIB | N-(2-Chloro-...)
Affinity DataKd:  2nMpH: 7.4 T: 2°CAssay Description:Competition binding assay was used to measure the interaction between the phage-tagged kinase, immobilized competitive ligand, and unlinked test comp...More data for this Ligand-Target Pair
TargetTyrosine-protein kinase ABL1 [201-500,M351T](Homo sapiens (Human))
Ambit

LigandPNGBDBM13216(BMS-354825 | CHEMBL1421 | DASATINIB | N-(2-Chloro-...)
Affinity DataKd:  0.700nMpH: 7.4 T: 2°CAssay Description:Competition binding assay was used to measure the interaction between the phage-tagged kinase, immobilized competitive ligand, and unlinked test comp...More data for this Ligand-Target Pair
TargetTyrosine-protein kinase ABL1 [201-500,F359V](Homo sapiens (Human))
Ambit

LigandPNGBDBM13216(BMS-354825 | CHEMBL1421 | DASATINIB | N-(2-Chloro-...)
Affinity DataKd:  0.300nMpH: 7.4 T: 2°CAssay Description:Competition binding assay was used to measure the interaction between the phage-tagged kinase, immobilized competitive ligand, and unlinked test comp...More data for this Ligand-Target Pair
TargetTyrosine-protein kinase ABL1 [201-500,H396P](Homo sapiens (Human))
Ambit

LigandPNGBDBM13530(4-[(4-methylpiperazin-1-yl)methyl]-N-[4-methyl-3-[...)
Affinity DataKd:  60nMAssay Description:Competition binding assay was used to measure the interaction between the phage-tagged kinase, immobilized competitive ligand, and unlinked test comp...More data for this Ligand-Target Pair
TargetTyrosine-protein kinase ABL1 [201-500,T315I](Homo sapiens (Human))
Ambit

LigandPNGBDBM13530(4-[(4-methylpiperazin-1-yl)methyl]-N-[4-methyl-3-[...)
Affinity DataKd:  6.00E+3nMAssay Description:Competition binding assay was used to measure the interaction between the phage-tagged kinase, immobilized competitive ligand, and unlinked test comp...More data for this Ligand-Target Pair
TargetTyrosine-protein kinase ABL1 [201-500,T315N](Homo sapiens (Human))
Ambit

LigandPNGBDBM13530(4-[(4-methylpiperazin-1-yl)methyl]-N-[4-methyl-3-[...)
Affinity DataKd: >1.00E+4nMAssay Description:Competition binding assay was used to measure the interaction between the phage-tagged kinase, immobilized competitive ligand, and unlinked test comp...More data for this Ligand-Target Pair
TargetMast/stem cell growth factor receptor Kit [N822K](Homo sapiens (Human))
Ambit

LigandPNGBDBM13530(4-[(4-methylpiperazin-1-yl)methyl]-N-[4-methyl-3-[...)
Affinity DataKd:  3nMAssay Description:Competition binding assay was used to measure the interaction between the phage-tagged kinase, immobilized competitive ligand, and unlinked test comp...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMast/stem cell growth factor receptor Kit [V559D](Homo sapiens (Human))
Ambit

LigandPNGBDBM13530(4-[(4-methylpiperazin-1-yl)methyl]-N-[4-methyl-3-[...)
Affinity DataKd:  20nMAssay Description:Competition binding assay was used to measure the interaction between the phage-tagged kinase, immobilized competitive ligand, and unlinked test comp...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM13530(4-[(4-methylpiperazin-1-yl)methyl]-N-[4-methyl-3-[...)
Affinity DataKd:  3.00E+3nMAssay Description:Competition binding assay was used to measure the interaction between the phage-tagged kinase, immobilized competitive ligand, and unlinked test comp...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1 [201-500,H396P](Homo sapiens (Human))
Ambit

LigandPNGBDBM13216(BMS-354825 | CHEMBL1421 | DASATINIB | N-(2-Chloro-...)
Affinity DataKd:  1nMAssay Description:Competition binding assay was used to measure the interaction between the phage-tagged kinase, immobilized competitive ligand, and unlinked test comp...More data for this Ligand-Target Pair
TargetTyrosine-protein kinase ABL1 [201-500,T315I](Homo sapiens (Human))
Ambit

LigandPNGBDBM13216(BMS-354825 | CHEMBL1421 | DASATINIB | N-(2-Chloro-...)
Affinity DataKd:  600nMAssay Description:Competition binding assay was used to measure the interaction between the phage-tagged kinase, immobilized competitive ligand, and unlinked test comp...More data for this Ligand-Target Pair
TargetTyrosine-protein kinase ABL1 [201-500,T315N](Homo sapiens (Human))
Ambit

LigandPNGBDBM13216(BMS-354825 | CHEMBL1421 | DASATINIB | N-(2-Chloro-...)
Affinity DataKd:  40nMAssay Description:Competition binding assay was used to measure the interaction between the phage-tagged kinase, immobilized competitive ligand, and unlinked test comp...More data for this Ligand-Target Pair
TargetMast/stem cell growth factor receptor Kit [N822K](Homo sapiens (Human))
Ambit

LigandPNGBDBM13216(BMS-354825 | CHEMBL1421 | DASATINIB | N-(2-Chloro-...)
Affinity DataKd:  0.400nMAssay Description:Competition binding assay was used to measure the interaction between the phage-tagged kinase, immobilized competitive ligand, and unlinked test comp...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMast/stem cell growth factor receptor Kit [V559D](Homo sapiens (Human))
Ambit

LigandPNGBDBM13216(BMS-354825 | CHEMBL1421 | DASATINIB | N-(2-Chloro-...)
Affinity DataKd:  0.700nMAssay Description:Competition binding assay was used to measure the interaction between the phage-tagged kinase, immobilized competitive ligand, and unlinked test comp...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM13216(BMS-354825 | CHEMBL1421 | DASATINIB | N-(2-Chloro-...)
Affinity DataKd: >1.00E+4nMAssay Description:Competition binding assay was used to measure the interaction between the phage-tagged kinase, immobilized competitive ligand, and unlinked test comp...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1 [201-500](Homo sapiens (Human))
Ambit

LigandPNGBDBM6572(6-(2,6-dichlorophenyl)-2-[(4-fluoro-3-methylphenyl...)
Affinity DataKd:  1nMAssay Description:Competition binding assay was used to measure the interaction between the phage-tagged kinase, immobilized competitive ligand, and unlinked test comp...More data for this Ligand-Target Pair
TargetTyrosine-protein kinase ABL1 [201-500,Q252H](Homo sapiens (Human))
Ambit

LigandPNGBDBM6572(6-(2,6-dichlorophenyl)-2-[(4-fluoro-3-methylphenyl...)
Affinity DataKd:  2nMAssay Description:Competition binding assay was used to measure the interaction between the phage-tagged kinase, immobilized competitive ligand, and unlinked test comp...More data for this Ligand-Target Pair
TargetTyrosine-protein kinase ABL1 [201-500,Y253F](Homo sapiens (Human))
Ambit

LigandPNGBDBM6572(6-(2,6-dichlorophenyl)-2-[(4-fluoro-3-methylphenyl...)
Affinity DataKd:  1nMAssay Description:Competition binding assay was used to measure the interaction between the phage-tagged kinase, immobilized competitive ligand, and unlinked test comp...More data for this Ligand-Target Pair
TargetTyrosine-protein kinase ABL1 [201-500,E255K](Homo sapiens (Human))
Ambit

LigandPNGBDBM6572(6-(2,6-dichlorophenyl)-2-[(4-fluoro-3-methylphenyl...)
Affinity DataKd:  4nMAssay Description:Competition binding assay was used to measure the interaction between the phage-tagged kinase, immobilized competitive ligand, and unlinked test comp...More data for this Ligand-Target Pair
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