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Found 10 with Last Name = 'augereau' and Initial = 'jm'
TargetVasopressin V1a receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50114031((2S)-1-[(2R,3S)-5-chloro-3-(2-chlorophenyl)-1-(3,4...)
Affinity DataKi:  2nMAssay Description:Binding affinity to vasopressin V1a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50029644(CHEMBL296908 | N-(3-(4-(4-(2-oxo-3,4-dihydroquinol...)
Affinity DataKi:  350nMAssay Description:Binding affinity to vasopressin V1a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C zeta type(Rattus norvegicus)
Sanofi Recherche

Curated by ChEMBL
LigandPNGBDBM50241867(((2R,3R,4R,5R,6R)-6-(3,4-dihydroxyphenethoxy)-5-hy...)
Affinity DataKi:  2.20E+4nMAssay Description:Displacement of [gamma32P]ATP from rat brain PKC by competitive Lineweaver-Burke plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C zeta type(Rattus norvegicus)
Sanofi Recherche

Curated by ChEMBL
LigandPNGBDBM50241867(((2R,3R,4R,5R,6R)-6-(3,4-dihydroxyphenethoxy)-5-hy...)
Affinity DataKi:  2.80E+4nMAssay Description:Inhibition of rat brain PKC using histone type 3-S as substrate by noncompetitive Lineweaver-Burke plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50292418(CHEMBL511334 | Khusimol)
Affinity DataKi:  4.10E+4nMAssay Description:Displacement of [3H]AVP from vasopressin V1a receptor in rat liver membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50292418(CHEMBL511334 | Khusimol)
Affinity DataKi:  5.30E+4nMAssay Description:Displacement of [3H]AVP from vasopressin V1a receptor in rat liver membrane by competitive displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C zeta type(Rattus norvegicus)
Sanofi Recherche

Curated by ChEMBL
LigandPNGBDBM50241867(((2R,3R,4R,5R,6R)-6-(3,4-dihydroxyphenethoxy)-5-hy...)
Affinity DataIC50:  68nMAssay Description:Displacement of [3H]PDBu from rat brain PKC by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C zeta type(Rattus norvegicus)
Sanofi Recherche

Curated by ChEMBL
LigandPNGBDBM50241867(((2R,3R,4R,5R,6R)-6-(3,4-dihydroxyphenethoxy)-5-hy...)
Affinity DataIC50:  2.10E+4nMAssay Description:Inhibition of rat brain PKC catalytic domain by mixed micellar assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C zeta type(Rattus norvegicus)
Sanofi Recherche

Curated by ChEMBL
LigandPNGBDBM50241867(((2R,3R,4R,5R,6R)-6-(3,4-dihydroxyphenethoxy)-5-hy...)
Affinity DataIC50:  2.50E+4nMAssay Description:Inhibition of rat brain PKC by mixed micellar assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50292418(CHEMBL511334 | Khusimol)
Affinity DataIC50:  1.25E+5nMAssay Description:Displacement of [3H]AVP from vasopressin V1a receptor in rat liver membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed