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Found 550 with Last Name = 'azak' and Initial = 'h'
TargetCarbonic anhydrase 2(Homo sapiens (Human))
Karamanoglu Mehmetbey University

Curated by ChEMBL
LigandPNGBDBM50428480(CHEMBL2335176)
Affinity DataKi:  170nMAssay Description:Inhibition of human carbonic anhydrase 2 using 4-nitrophenylacetate as substrate after 3 mins by spectrophotometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
Karamanoglu Mehmetbey University

Curated by ChEMBL
LigandPNGBDBM50428479(CHEMBL2335177)
Affinity DataKi:  250nMAssay Description:Inhibition of human carbonic anhydrase 2 using 4-nitrophenylacetate as substrate after 3 mins by spectrophotometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
Karamanoglu Mehmetbey University

Curated by ChEMBL
LigandPNGBDBM50428478(CHEMBL2335178)
Affinity DataKi:  290nMAssay Description:Inhibition of human carbonic anhydrase 2 using 4-nitrophenylacetate as substrate after 3 mins by spectrophotometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 1(Homo sapiens (Human))
Karamanoglu Mehmetbey University

Curated by ChEMBL
LigandPNGBDBM50428479(CHEMBL2335177)
Affinity DataKi:  3.93E+4nMAssay Description:Inhibition of human carbonic anhydrase 1 using 4-nitrophenylacetate as substrate after 3 mins by spectrophotometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 1(Homo sapiens (Human))
Karamanoglu Mehmetbey University

Curated by ChEMBL
LigandPNGBDBM50428478(CHEMBL2335178)
Affinity DataKi:  4.17E+4nMAssay Description:Inhibition of human carbonic anhydrase 1 using 4-nitrophenylacetate as substrate after 3 mins by spectrophotometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 1(Homo sapiens (Human))
Karamanoglu Mehmetbey University

Curated by ChEMBL
LigandPNGBDBM50428480(CHEMBL2335176)
Affinity DataKi:  4.26E+4nMAssay Description:Inhibition of human carbonic anhydrase 1 using 4-nitrophenylacetate as substrate after 3 mins by spectrophotometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExtracellular calcium-sensing receptor(Rattus norvegicus)
Mitsubishi Tanabe Pharma

Curated by ChEMBL
LigandPNGBDBM50272596(CHEMBL4126450)
Affinity DataIC50:  0.470nMAssay Description:Agonist activity at CaSR in rat parathyroid cells assessed as inhibition of PTH (1 to 84 residues) production in presence of Cacl2 by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol O-acyltransferase 2(Homo sapiens (Human))
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50429605(CHEMBL2334538)
Affinity DataIC50:  0.800nMAssay Description:Inhibition of ACAT2 (unknown origin) expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol O-acyltransferase 2(Homo sapiens (Human))
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50429604(CHEMBL2334539)
Affinity DataIC50:  0.900nMAssay Description:Inhibition of ACAT2 (unknown origin) expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol O-acyltransferase 2(Homo sapiens (Human))
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50429610(CHEMBL2334222)
Affinity DataIC50:  0.900nMAssay Description:Inhibition of ACAT2 (unknown origin) expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol O-acyltransferase 2(Homo sapiens (Human))
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50429604(CHEMBL2334539)
Affinity DataIC50:  0.900nMAssay Description:Inhibition of ACAT2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol O-acyltransferase 2(Homo sapiens (Human))
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50429603(CHEMBL2334540)
Affinity DataIC50:  0.900nMAssay Description:Inhibition of ACAT2 (unknown origin) expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExtracellular calcium-sensing receptor(Rattus norvegicus)
Mitsubishi Tanabe Pharma

Curated by ChEMBL
LigandPNGBDBM50272602(CHEMBL4126877)
Affinity DataIC50:  0.910nMAssay Description:Agonist activity at CaSR in rat parathyroid cells assessed as inhibition of PTH (1 to 84 residues) production in presence of Cacl2 by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol O-acyltransferase 2(Homo sapiens (Human))
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50429602(CHEMBL2334541)
Affinity DataIC50:  1nMAssay Description:Inhibition of ACAT2 (unknown origin) expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol O-acyltransferase 2(Homo sapiens (Human))
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50429601(CHEMBL2333808)
Affinity DataIC50:  1nMAssay Description:Inhibition of ACAT2 (unknown origin) expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol O-acyltransferase 2(Homo sapiens (Human))
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50429600(CHEMBL2333809)
Affinity DataIC50:  1.20nMAssay Description:Inhibition of ACAT2 (unknown origin) expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExtracellular calcium-sensing receptor(Rattus norvegicus)
Mitsubishi Tanabe Pharma

Curated by ChEMBL
LigandPNGBDBM50272605(CHEMBL4128542)
Affinity DataIC50:  1.40nMAssay Description:Agonist activity at CaSR in rat parathyroid cells assessed as inhibition of PTH (1 to 84 residues) production in presence of Cacl2 by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A/3B(Rattus norvegicus)
Dainippon Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM85330(CAS_68647 | NSC_68647 | ONDANSETRON | Ondansetron ...)
Affinity DataIC50:  1.40nMAssay Description:Binding affinity against 5-hydroxytryptamine 3 receptor in rat cortical membrane using [3H]GR-65630 as radioligandMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 3A/3B(Rattus norvegicus)
Dainippon Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50366571(CHEMBL1788261)
Affinity DataIC50:  1.5nMAssay Description:Binding affinity against 5-hydroxytryptamine 3 receptor in rat cortical membrane using [3H]GR-65630 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol O-acyltransferase 2(Homo sapiens (Human))
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50429599(CHEMBL2333810)
Affinity DataIC50:  1.70nMAssay Description:Inhibition of ACAT2 (unknown origin) expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A/3B(Rattus norvegicus)
Dainippon Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50069286(5-Chloro-4-ethylamino-N-(1-ethyl-4-methyl-[1,4]dia...)
Affinity DataIC50:  1.90nMAssay Description:Binding affinity against 5-hydroxytryptamine 3 receptor in rat cortical membrane using [3H]GR-65630 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol O-acyltransferase 2(Homo sapiens (Human))
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50429598(CHEMBL2333811)
Affinity DataIC50:  2nMAssay Description:Inhibition of ACAT2 (unknown origin) expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExtracellular calcium-sensing receptor(Rattus norvegicus)
Mitsubishi Tanabe Pharma

Curated by ChEMBL
LigandPNGBDBM50272606(CHEMBL4125917)
Affinity DataIC50:  2.10nMAssay Description:Agonist activity at CaSR in rat parathyroid cells assessed as inhibition of PTH (1 to 84 residues) production in presence of Cacl2 by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
Nippon Steel

Curated by ChEMBL
LigandPNGBDBM50064943((1-{3-[2-Fluoro-4-(imino-thiazolidin-3-yl-methyl)-...)
Affinity DataIC50:  2.30nMAssay Description:Binding affinity to human fibrinogen receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(GUINEA PIG)
Dainippon Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50112041(4-Amino-N-{1-[1-(2-amino-3-methyl-butyryl)-piperid...)
Affinity DataIC50:  2.5nMAssay Description:Inhibitory activity against 5-hydroxytryptamine 4 receptor of guinea pig striatum using [3H]-GR-113,808 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Dainippon Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50241107(1-(3-(4-(5-chloro-2-oxo-2,3-dihydrobenzo[d]imidazo...)
Affinity DataIC50:  2.5nMAssay Description:Binding affinity against dopamine D2 receptor in rat brain synaptic membrane using [3H]-spiperone as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(GUINEA PIG)
Dainippon Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50112039(4-Amino-N-{1-[1-(2-amino-pentanoyl)-piperidin-4-yl...)
Affinity DataIC50:  2.60nMAssay Description:Inhibitory activity against 5-hydroxytryptamine 4 receptor of guinea pig striatum using [3H]-GR-113,808 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(GUINEA PIG)
Dainippon Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50112038(4-Amino-N-{1-[1-(2-amino-2-methyl-propionyl)-piper...)
Affinity DataIC50:  2.60nMAssay Description:Inhibitory activity against 5-hydroxytryptamine 4 receptor of guinea pig striatum using [3H]-GR-113,808 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
Nippon Steel

Curated by ChEMBL
LigandPNGBDBM50064930(CHEMBL77113 | {1-[3-(4-Carbamimidoyl-benzoylamino)...)
Affinity DataIC50:  2.60nMAssay Description:Binding affinity to human fibrinogen receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol O-acyltransferase 2(Homo sapiens (Human))
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50429597(CHEMBL2333812)
Affinity DataIC50:  2.70nMAssay Description:Inhibition of ACAT2 (unknown origin) expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
Nippon Steel

Curated by ChEMBL
LigandPNGBDBM50064935(CHEMBL312368 | {1-[3-(4-Carbamimidoyl-2-fluoro-ben...)
Affinity DataIC50:  2.70nMAssay Description:Binding affinity to human fibrinogen receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
Nippon Steel

Curated by ChEMBL
LigandPNGBDBM50064941(CHEMBL78295 | {1-[3-(4-Carbamimidoyl-2-fluoro-benz...)
Affinity DataIC50:  2.70nMAssay Description:Binding affinity to human fibrinogen receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
Nippon Steel

Curated by ChEMBL
LigandPNGBDBM50064942(CHEMBL74908 | {1-[3-(4-Carbamimidoyl-benzoylamino)...)
Affinity DataIC50:  2.70nMAssay Description:Binding affinity to human fibrinogen receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A/3B(Rattus norvegicus)
Dainippon Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50070570(5-Chloro-N-((R)-1-ethyl-4-methyl-[1,4]diazepan-6-y...)
Affinity DataIC50:  2.90nMAssay Description:Binding affinity against 5-hydroxytryptamine 3 receptor in rat cortical membrane using [3H]GR-65630 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Dainippon Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50109771(3-{4-[(1-{2-[1-(Benzooxazole-2-carbonyl)-2-methyl-...)
Affinity DataIC50:  3.5nMAssay Description:In vitro inhibition of the human neutrophil elastase-catalyzed hydrolysis of the synthetic substrate Suc-Ala-Pro-Ala-MCAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
Nippon Steel

Curated by ChEMBL
LigandPNGBDBM50064922(CHEMBL432915 | {1-[3-(4-Carbamimidoyl-benzoylamino...)
Affinity DataIC50:  3.80nMAssay Description:Binding affinity to human fibrinogen receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(GUINEA PIG)
Dainippon Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50112046(4-Amino-N-{1-[1-(5-amino-pentanoyl)-piperidin-4-yl...)
Affinity DataIC50:  3.90nMAssay Description:Inhibitory activity against 5-hydroxytryptamine 4 receptor of guinea pig striatum using [3H]-GR-113,808 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(GUINEA PIG)
Dainippon Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50112042(4-Amino-N-{1-[1-(4-amino-butyryl)-piperidin-4-ylme...)
Affinity DataIC50:  4nMAssay Description:Inhibitory activity against 5-hydroxytryptamine 4 receptor of guinea pig striatum using [3H]-GR-113,808 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
Nippon Steel

Curated by ChEMBL
LigandPNGBDBM50064920((1-{3-[2-Fluoro-4-(imino-morpholin-4-yl-methyl)-be...)
Affinity DataIC50:  4nMAssay Description:Binding affinity to human fibrinogen receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol O-acyltransferase 2(Homo sapiens (Human))
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50429596(CHEMBL2333813)
Affinity DataIC50:  4nMAssay Description:Inhibition of ACAT2 (unknown origin) expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExtracellular calcium-sensing receptor(Rattus norvegicus)
Mitsubishi Tanabe Pharma

Curated by ChEMBL
LigandPNGBDBM50272607(CHEMBL4126057)
Affinity DataIC50:  4.30nMAssay Description:Agonist activity at CaSR in rat parathyroid cells assessed as inhibition of PTH (1 to 84 residues) production in presence of Cacl2 by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
Nippon Steel

Curated by ChEMBL
LigandPNGBDBM50064938(CHEMBL77635 | {1-[3-(4-Carbamimidoyl-2-fluoro-benz...)
Affinity DataIC50:  4.30nMAssay Description:Binding affinity to human fibrinogen receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Dainippon Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50366569(CHEMBL1788262)
Affinity DataIC50:  4.5nMAssay Description:Binding affinity against dopamine D2 receptor in rat brain synaptic membrane using [3H]-spiperone as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A/3B(Rattus norvegicus)
Dainippon Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50450877(CHEMBL2093035)
Affinity DataIC50:  4.5nMAssay Description:Binding affinity against 5-hydroxytryptamine 3 receptor in rat cortical membrane using [3H]GR-65630 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A/3B(Rattus norvegicus)
Dainippon Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50069288(5-Chloro-N-(1-ethyl-4-methyl-[1,4]diazepan-6-yl)-2...)
Affinity DataIC50:  4.80nMAssay Description:Binding affinity against 5-hydroxytryptamine 3 receptor in rat cortical membrane using [3H]GR-65630 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol O-acyltransferase 2(Homo sapiens (Human))
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50429595(CHEMBL2334194)
Affinity DataIC50:  5nMAssay Description:Inhibition of ACAT2 (unknown origin) expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
Nippon Steel

Curated by ChEMBL
LigandPNGBDBM50064926(CHEMBL77404 | {1-[3-(4-Carbamimidoyl-benzoylamino)...)
Affinity DataIC50:  5nMAssay Description:Binding affinity to human fibrinogen receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol O-acyltransferase 2(Homo sapiens (Human))
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50429577(CHEMBL2334212)
Affinity DataIC50:  5nMAssay Description:Inhibition of ACAT2 (unknown origin) expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol O-acyltransferase 2(Homo sapiens (Human))
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50429591(CHEMBL2334198)
Affinity DataIC50:  5nMAssay Description:Inhibition of ACAT2 (unknown origin) expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol O-acyltransferase 2(Homo sapiens (Human))
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50429593(CHEMBL2334196)
Affinity DataIC50:  5nMAssay Description:Inhibition of ACAT2 (unknown origin) expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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