TargetSynaptic vesicle glycoprotein 2A(Homo sapiens)
Jagiellonian University Medical College
Curated by ChEMBL
Jagiellonian University Medical College
Curated by ChEMBL
Affinity DataKi: >2.50E+5nMAssay Description:Binding affinity to human SV2A in presence of levetiracetam by radioligand binding assayMore data for this Ligand-Target Pair
TargetSynaptic vesicle glycoprotein 2A(Mus musculus)
Jagiellonian University Medical College
Curated by ChEMBL
Jagiellonian University Medical College
Curated by ChEMBL
Affinity DataKi: >2.50E+5nMAssay Description:Binding affinity to mouse SV2A in presence of levetiracetam by radioligand binding assayMore data for this Ligand-Target Pair
TargetSynaptic vesicle glycoprotein 2A(Mus musculus)
Jagiellonian University Medical College
Curated by ChEMBL
Jagiellonian University Medical College
Curated by ChEMBL
Affinity DataKi: >2.50E+5nMAssay Description:Binding affinity to mouse SV2A in presence of levetiracetam by radioligand binding assayMore data for this Ligand-Target Pair
TargetSynaptic vesicle glycoprotein 2A(Homo sapiens)
Jagiellonian University Medical College
Curated by ChEMBL
Jagiellonian University Medical College
Curated by ChEMBL
Affinity DataKi: >2.50E+5nMAssay Description:Binding affinity to human SV2A in presence of levetiracetam by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: <5.00E+7nMAssay Description:Inhibition of CYP3A4More data for this Ligand-Target Pair
Affinity DataKi: <5.00E+7nMAssay Description:Inhibition of CYP3A4More data for this Ligand-Target Pair
Affinity DataKi: <5.00E+7nMAssay Description:Inhibition of CYP3A4More data for this Ligand-Target Pair
Affinity DataKi: <5.00E+7nMAssay Description:Inhibition of CYP3A4More data for this Ligand-Target Pair
Affinity DataKi: <5.00E+7nMAssay Description:Inhibition of CYP3A4More data for this Ligand-Target Pair
Affinity DataKi: <5.00E+7nMAssay Description:Inhibition of CYP3A4More data for this Ligand-Target Pair
Affinity DataKi: <5.00E+7nMAssay Description:Inhibition of CYP3A4More data for this Ligand-Target Pair
Affinity DataKi: <5.00E+7nMAssay Description:Inhibition of CYP3A4More data for this Ligand-Target Pair
TargetDual specificity protein phosphatase 1(Homo sapiens (Human))
University Of Pittsburgh
Curated by ChEMBL
University Of Pittsburgh
Curated by ChEMBL
Affinity DataIC50: 1.15E+4nMAssay Description:Inhibition of Myc-tagged human Dusp1 expressed in TPA-induced human HeLa cells asssessed as decrease in dephosphorylation of pERK measured by immunos...More data for this Ligand-Target Pair
TargetDual specificity protein phosphatase 6(Homo sapiens (Human))
University Of Pittsburgh
Curated by ChEMBL
University Of Pittsburgh
Curated by ChEMBL
Affinity DataIC50: 1.23E+4nMAssay Description:Inhibition of Myc-tagged human Dusp6 expressed in TPA-induced human HeLa cells asssessed as decrease in dephosphorylation of pERK measured by immunos...More data for this Ligand-Target Pair
TargetExcitatory amino acid transporter 2(Homo sapiens (Human))
Jagiellonian University Medical College
Curated by ChEMBL
Jagiellonian University Medical College
Curated by ChEMBL
Affinity DataEC50: 11nMAssay Description:Activation of human EAAT2 transfected in COS7 cells assessed as glutamate uptakeMore data for this Ligand-Target Pair
TargetExcitatory amino acid transporter 2(Homo sapiens (Human))
Jagiellonian University Medical College
Curated by ChEMBL
Jagiellonian University Medical College
Curated by ChEMBL
Affinity DataEC50: 20nMAssay Description:Activation of human EAAT2 transfected in COS7 cells assessed as glutamate uptakeMore data for this Ligand-Target Pair
TargetExcitatory amino acid transporter 2(Homo sapiens (Human))
Jagiellonian University Medical College
Curated by ChEMBL
Jagiellonian University Medical College
Curated by ChEMBL
Affinity DataEC50: 25nMAssay Description:Activation of human EAAT2 transfected in Glial cells assessed as glutamate uptakeMore data for this Ligand-Target Pair
TargetExcitatory amino acid transporter 2(Homo sapiens (Human))
Jagiellonian University Medical College
Curated by ChEMBL
Jagiellonian University Medical College
Curated by ChEMBL
Affinity DataEC50: 0.100nMAssay Description:Activation of human EAAT2 transfected in Glial cells assessed as glutamate uptakeMore data for this Ligand-Target Pair
Affinity DataKd: 1.97E+6nMAssay Description:Binding affinity to human serum albumin assessed as dissociation constant by LC/MS analysisMore data for this Ligand-Target Pair