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Found 98 with Last Name = 'balas' and Initial = 'l'
TargetCannabinoid receptor 1(Homo sapiens (Human))
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM22988((5Z,8Z,11Z,14Z)-N-(2-hydroxyethyl)icosa-5,8,11,14-...)
Affinity DataKi:  70nMAssay Description:Displacement of [3H]CP55-940 from human recombinant CB1 receptor expressed in COS cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM22988((5Z,8Z,11Z,14Z)-N-(2-hydroxyethyl)icosa-5,8,11,14-...)
Affinity DataKi:  70nMAssay Description:Displacement of [3H]CP55-940 from human recombinant CB1 receptor in COS cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Umr Cnrs 5074

Curated by ChEMBL
LigandPNGBDBM22988((5Z,8Z,11Z,14Z)-N-(2-hydroxyethyl)icosa-5,8,11,14-...)
Affinity DataKi:  90nMAssay Description:Binding affinity of the compound towards Cannabinoid receptor 1 in rat forebrain membranes using [3H]-CP-55,940 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM22988((5Z,8Z,11Z,14Z)-N-(2-hydroxyethyl)icosa-5,8,11,14-...)
Affinity DataKi:  180nMAssay Description:Displacement of [3H]CP55-940 from human recombinant CB2 receptor in COS cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM22988((5Z,8Z,11Z,14Z)-N-(2-hydroxyethyl)icosa-5,8,11,14-...)
Affinity DataKi:  180nMAssay Description:Displacement of [3H]CP55-940 from human recombinant CB2 receptor expressed in COS cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50186533((3Z,6Z,9Z,12Z)-17-((R)-1-hydroxypropan-2-ylamino)-...)
Affinity DataKi:  220nMAssay Description:Displacement of [3H]CP55-940 from human recombinant CB2 receptor in COS cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Umr Cnrs 5074

Curated by ChEMBL
LigandPNGBDBM50128915((8Z,11Z,14Z)-1-Hydroxy-tricosa-8,11,14,17-tetraen-...)
Affinity DataKi:  360nMAssay Description:Binding affinity of the compound towards Cannabinoid receptor 1 in rat forebrain membranes using [3H]-CP-55,940 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50186533((3Z,6Z,9Z,12Z)-17-((R)-1-hydroxypropan-2-ylamino)-...)
Affinity DataKi:  570nMAssay Description:Displacement of [3H]CP55-940 from human recombinant CB1 receptor in COS cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50292882((3Z,6Z,9Z,12Z)-17-((R)-1-hydroxypropan-2-ylamino)-...)
Affinity DataKi:  1.02E+3nMAssay Description:Displacement of [3H]CP55-940 from human recombinant CB2 receptor expressed in COS cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Umr Cnrs 5074

Curated by ChEMBL
LigandPNGBDBM50128914((12Z,15Z)-1-Hydroxy-henicosa-12,15-dien-4-one | CH...)
Affinity DataKi:  2.10E+3nMAssay Description:Binding affinity of the compound towards Cannabinoid receptor 1 in rat forebrain membranes using [3H]-CP-55,940 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Umr Cnrs 5074

Curated by ChEMBL
LigandPNGBDBM50128912((5Z,8Z,11Z)-2,2-Dimethyl-icosa-5,8,11,14-tetraenoi...)
Affinity DataKi:  2.10E+3nMAssay Description:Binding affinity of the compound towards Fatty-acid amide hydrolase (FAAH) in rat forebrain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50292882((3Z,6Z,9Z,12Z)-17-((R)-1-hydroxypropan-2-ylamino)-...)
Affinity DataKi:  2.80E+3nMAssay Description:Displacement of [3H]CP55-940 from human recombinant CB1 receptor expressed in COS cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Umr Cnrs 5074

Curated by ChEMBL
LigandPNGBDBM22988((5Z,8Z,11Z,14Z)-N-(2-hydroxyethyl)icosa-5,8,11,14-...)
Affinity DataKi:  3.00E+3nMAssay Description:Binding affinity of the compound towards Fatty-acid amide hydrolase (FAAH) in rat forebrain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Umr Cnrs 5074

Curated by ChEMBL
LigandPNGBDBM50128913((5Z,8Z,11Z)-Icosa-5,8,11,14-tetraenoic acid 2-hydr...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity of the compound towards Cannabinoid receptor 1 in rat forebrain membranes using [3H]-CP-55,940 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Umr Cnrs 5074

Curated by ChEMBL
LigandPNGBDBM50128912((5Z,8Z,11Z)-2,2-Dimethyl-icosa-5,8,11,14-tetraenoi...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity of the compound towards Cannabinoid receptor 1 in rat forebrain membranes using [3H]-CP-55,940 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Umr Cnrs 5074

Curated by ChEMBL
LigandPNGBDBM50185017((Z)-N-{(1R)-3-(2,6-dichlorobenzoyloxy)-1-[(4-hydro...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of [14C]anandamide hydrolysis in rat brain membrane in the absence of UV irradiationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Umr Cnrs 5074

Curated by ChEMBL
LigandPNGBDBM50185014((Z)-N-{(1S)-3-chloro-1-[(4-hydroxyphenyl)methyl]pr...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of [14C]anandamide hydrolysis in rat brain membrane in the absence of UV irradiationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Umr Cnrs 5074

Curated by ChEMBL
LigandPNGBDBM50185008((Z)-N-[(1S)-2-hydroxy-1-[(4-hydroxyphenyl)methyl]e...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of [14C]anandamide hydrolysis in rat brain membrane in the absence of UV irradiationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Umr Cnrs 5074

Curated by ChEMBL
LigandPNGBDBM50185015((Z)-N-{(1S)-3-(2,6-dichlorobenzoyloxy)-1-[(4-hydro...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of [14C]anandamide hydrolysis in rat brain membrane in the presence of UV irradiationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Umr Cnrs 5074

Curated by ChEMBL
LigandPNGBDBM50185020((Z)-N-{(1R)-3-chloro-1-[(4-hydroxyphenyl)methyl]pr...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of [14C]anandamide hydrolysis in rat brain membrane in the absence of UV irradiationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Umr Cnrs 5074

Curated by ChEMBL
LigandPNGBDBM50185017((Z)-N-{(1R)-3-(2,6-dichlorobenzoyloxy)-1-[(4-hydro...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of [14C]anandamide hydrolysis in rat brain membrane in the presence of UV irradiationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Umr Cnrs 5074

Curated by ChEMBL
LigandPNGBDBM50185020((Z)-N-{(1R)-3-chloro-1-[(4-hydroxyphenyl)methyl]pr...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of [14C]anandamide hydrolysis in rat brain membrane in the presence of UV irradiationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Umr Cnrs 5074

Curated by ChEMBL
LigandPNGBDBM50185013((Z)-N-{(1S)-3-iodo-1-[(4-hydroxyphenyl)methyl]prop...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of [14C]anandamide hydrolysis in rat brain membrane in the presence of UV irradiationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Umr Cnrs 5074

Curated by ChEMBL
LigandPNGBDBM50185013((Z)-N-{(1S)-3-iodo-1-[(4-hydroxyphenyl)methyl]prop...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of [14C]anandamide hydrolysis in rat brain membrane in the absence of UV irradiationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Umr Cnrs 5074

Curated by ChEMBL
LigandPNGBDBM50185012((Z)-N-{(1R)-3-iodo-1-[(4-hydroxyphenyl)methyl]prop...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of [14C]anandamide hydrolysis in rat brain membrane in the absence of UV irradiationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Umr Cnrs 5074

Curated by ChEMBL
LigandPNGBDBM50185011((Z)-N-[(1S)-2-hydroxy-1-[(4-hydroxyphenyl)methyl]e...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of [14C]anandamide hydrolysis in rat brain membrane in the absence of UV irradiationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Umr Cnrs 5074

Curated by ChEMBL
LigandPNGBDBM50185008((Z)-N-[(1S)-2-hydroxy-1-[(4-hydroxyphenyl)methyl]e...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of [14C]anandamide hydrolysis in rat brain membrane in the presence of UV irradiationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Umr Cnrs 5074

Curated by ChEMBL
LigandPNGBDBM50185014((Z)-N-{(1S)-3-chloro-1-[(4-hydroxyphenyl)methyl]pr...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of [14C]anandamide hydrolysis in rat brain membrane in the presence of UV irradiationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Umr Cnrs 5074

Curated by ChEMBL
LigandPNGBDBM50185012((Z)-N-{(1R)-3-iodo-1-[(4-hydroxyphenyl)methyl]prop...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of [14C]anandamide hydrolysis in rat brain membrane in the presence of UV irradiationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Umr Cnrs 5074

Curated by ChEMBL
LigandPNGBDBM50185011((Z)-N-[(1S)-2-hydroxy-1-[(4-hydroxyphenyl)methyl]e...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of [14C]anandamide hydrolysis in rat brain membrane in the presence of UV irradiationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Umr Cnrs 5074

Curated by ChEMBL
LigandPNGBDBM50185015((Z)-N-{(1S)-3-(2,6-dichlorobenzoyloxy)-1-[(4-hydro...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of [14C]anandamide hydrolysis in rat brain membrane in the absence of UV irradiationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(RAT)
Medical College Of Ohio

Curated by ChEMBL
LigandPNGBDBM50407339(CHEMBL1790307)
Affinity DataKd:  15nMAssay Description:In vitro anti-oxytocic activity with out Mg2+.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(RAT)
Medical College Of Ohio

Curated by ChEMBL
LigandPNGBDBM50407336(CHEMBL412616)
Affinity DataKd:  25nMAssay Description:In vitro activity was determinedfor the anti-oxytocic activity with 0.5 mM Mg2+.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(RAT)
Medical College Of Ohio

Curated by ChEMBL
LigandPNGBDBM50407346(CHEMBL408786)
Affinity DataKd:  214nMAssay Description:Compound was evaluated for the oxytocic activity with out Mg2+.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(RAT)
Medical College Of Ohio

Curated by ChEMBL
LigandPNGBDBM50407349(CHEMBL265357)
Affinity DataKd:  6.20nMAssay Description:In vitro activity was determinedfor the anti-oxytocic activity with 0.5 mM Mg2+.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(RAT)
Medical College Of Ohio

Curated by ChEMBL
LigandPNGBDBM50407350(CHEMBL263521)
Affinity DataKd:  3nMAssay Description:In vitro antioxycic activity with out Mg2+.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Rattus norvegicus (Rat))
Medical College Of Ohio

Curated by ChEMBL
LigandPNGBDBM50407343(CHEMBL412806)
Affinity DataKd: >501nMAssay Description:Antidiuretic activity at V2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(RAT)
Medical College Of Ohio

Curated by ChEMBL
LigandPNGBDBM50407343(CHEMBL412806)
Affinity DataKd:  5.10nMAssay Description:In vitro anti-oxytocic activity with out Mg2+.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(RAT)
Medical College Of Ohio

Curated by ChEMBL
LigandPNGBDBM50407333(CHEMBL412942)
Affinity DataKd:  4.80nMAssay Description:In vitro activity for the anti-oxytocic activity with out Mg2+.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(RAT)
Medical College Of Ohio

Curated by ChEMBL
LigandPNGBDBM50407344(CHEMBL261914)
Affinity DataKd:  22nMAssay Description:In vitro anti-oxytocic activity with out Mg2+.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(RAT)
Medical College Of Ohio

Curated by ChEMBL
LigandPNGBDBM50407332(CHEMBL405005)
Affinity DataKd:  13nMAssay Description:In vitro activity for the anti-oxytocic activity with out Mg2+.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(RAT)
Medical College Of Ohio

Curated by ChEMBL
LigandPNGBDBM50407335(CHEMBL428187)
Affinity DataKd:  17nMAssay Description:In vitro anti-oxytocic activity with out Mg2+.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(RAT)
Medical College Of Ohio

Curated by ChEMBL
LigandPNGBDBM50407342(CHEMBL415160)
Affinity DataKd:  7.40nMAssay Description:In vitro activity for the anti-oxytocic activity with out Mg2+More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(RAT)
Medical College Of Ohio

Curated by ChEMBL
LigandPNGBDBM50407334(CHEMBL1790313)
Affinity DataKd:  19nMAssay Description:In vitro anti-oxytocic activity with out Mg2+.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(RAT)
Medical College Of Ohio

Curated by ChEMBL
LigandPNGBDBM50407341(CHEMBL264449)
Affinity DataKd:  26nMAssay Description:In vitro activity for the anti-oxytocic activity with out Mg2+.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(RAT)
Medical College Of Ohio

Curated by ChEMBL
LigandPNGBDBM50407345(CHEMBL1790315)
Affinity DataKd:  23nMAssay Description:In vitro antioxycic activity with out Mg2+.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(RAT)
Medical College Of Ohio

Curated by ChEMBL
LigandPNGBDBM50407337(CHEMBL1790314)
Affinity DataKd:  13nMAssay Description:In vitro anti-oxytocic activity with out Mg2+.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(RAT)
Medical College Of Ohio

Curated by ChEMBL
LigandPNGBDBM50407348(CHEMBL1790312)
Affinity DataKd:  9.60nMAssay Description:In vitro anti-oxytocic activity with out Mg2+.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(RAT)
Medical College Of Ohio

Curated by ChEMBL
LigandPNGBDBM50407340(CHEMBL1790310)
Affinity DataKd:  11nMAssay Description:In vitro antioxycic activity with out Mg2+.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(RAT)
Medical College Of Ohio

Curated by ChEMBL
LigandPNGBDBM50407338(CHEMBL385062)
Affinity DataKd:  45nMAssay Description:In vitro activity for the anti-oxytocic activity with out Mg2+.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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