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Found 289 with Last Name = 'banerjee' and Initial = 'd'
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Biogen

Curated by ChEMBL
LigandPNGBDBM50105928(CHEMBL3598047)
Affinity DataIC50:  3nMAssay Description:Binding affinity to GST-tagged RORgamma LBD (unknown origin) assessed as inhibition of interaction with co-activatior peptide TRAP220 preincubated fo...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Biogen

Curated by ChEMBL
LigandPNGBDBM50108775(CHEMBL3596638)
Affinity DataIC50:  3nMAssay Description:Inverse agonist activity at human recombinant GST-tagged RORgammat ligand binding domain assessed as effect on receptor-biotin tagged TRAP220 co-acti...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Biogen

Curated by ChEMBL
LigandPNGBDBM50108782(CHEMBL3596639)
Affinity DataIC50:  3nMAssay Description:Inverse agonist activity at human recombinant GST-tagged RORgammat ligand binding domain assessed as effect on receptor-biotin tagged TRAP220 co-acti...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Biogen

Curated by ChEMBL
LigandPNGBDBM50106011(CHEMBL3598077)
Affinity DataIC50:  3.20nMAssay Description:Binding affinity to GST-tagged RORgamma LBD (unknown origin) assessed as inhibition of interaction with co-activatior peptide TRAP220 preincubated fo...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Biogen

Curated by ChEMBL
LigandPNGBDBM50105992(CHEMBL3598061)
Affinity DataIC50:  3.30nMAssay Description:Binding affinity to GST-tagged RORgamma LBD (unknown origin) assessed as inhibition of interaction with co-activatior peptide TRAP220 preincubated fo...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Biogen

Curated by ChEMBL
LigandPNGBDBM50105981(CHEMBL3598052)
Affinity DataIC50:  3.40nMAssay Description:Binding affinity to GST-tagged RORgamma LBD (unknown origin) assessed as inhibition of interaction with co-activatior peptide TRAP220 preincubated fo...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Biogen

Curated by ChEMBL
LigandPNGBDBM50105930(CHEMBL3598049)
Affinity DataIC50:  3.80nMAssay Description:Binding affinity to GST-tagged RORgamma LBD (unknown origin) assessed as inhibition of interaction with co-activatior peptide TRAP220 preincubated fo...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Biogen

Curated by ChEMBL
LigandPNGBDBM50105982(CHEMBL3598053)
Affinity DataIC50:  4.80nMAssay Description:Binding affinity to GST-tagged RORgamma LBD (unknown origin) assessed as inhibition of interaction with co-activatior peptide TRAP220 preincubated fo...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Biogen

Curated by ChEMBL
LigandPNGBDBM50105988(CHEMBL3598056)
Affinity DataIC50:  4.90nMAssay Description:Binding affinity to GST-tagged RORgamma LBD (unknown origin) assessed as inhibition of interaction with co-activatior peptide TRAP220 preincubated fo...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Biogen

Curated by ChEMBL
LigandPNGBDBM50105985(CHEMBL3598055)
Affinity DataIC50:  4.90nMAssay Description:Binding affinity to GST-tagged RORgamma LBD (unknown origin) assessed as inhibition of interaction with co-activatior peptide TRAP220 preincubated fo...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Biogen

Curated by ChEMBL
LigandPNGBDBM50105933(CHEMBL3598051)
Affinity DataIC50:  4.90nMAssay Description:Binding affinity to GST-tagged RORgamma LBD (unknown origin) assessed as inhibition of interaction with co-activatior peptide TRAP220 preincubated fo...More data for this Ligand-Target Pair
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Biogen

Curated by ChEMBL
LigandPNGBDBM50105990(CHEMBL3598057)
Affinity DataIC50:  5nMAssay Description:Binding affinity to GST-tagged RORgamma LBD (unknown origin) assessed as inhibition of interaction with co-activatior peptide TRAP220 preincubated fo...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Biogen

Curated by ChEMBL
LigandPNGBDBM50106002(CHEMBL3598070)
Affinity DataIC50:  5.10nMAssay Description:Binding affinity to GST-tagged RORgamma LBD (unknown origin) assessed as inhibition of interaction with co-activatior peptide TRAP220 preincubated fo...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Biogen

Curated by ChEMBL
LigandPNGBDBM50106003(CHEMBL3598071)
Affinity DataIC50:  5.20nMAssay Description:Binding affinity to GST-tagged RORgamma LBD (unknown origin) assessed as inhibition of interaction with co-activatior peptide TRAP220 preincubated fo...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Biogen

Curated by ChEMBL
LigandPNGBDBM50105995(CHEMBL3598063)
Affinity DataIC50:  6nMAssay Description:Binding affinity to GST-tagged RORgamma LBD (unknown origin) assessed as inhibition of interaction with co-activatior peptide TRAP220 preincubated fo...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Biogen

Curated by ChEMBL
LigandPNGBDBM50106009(CHEMBL3598076)
Affinity DataIC50:  6.20nMAssay Description:Binding affinity to GST-tagged RORgamma LBD (unknown origin) assessed as inhibition of interaction with co-activatior peptide TRAP220 preincubated fo...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Biogen

Curated by ChEMBL
LigandPNGBDBM50106007(CHEMBL3598074)
Affinity DataIC50:  6.40nMAssay Description:Binding affinity to GST-tagged RORgamma LBD (unknown origin) assessed as inhibition of interaction with co-activatior peptide TRAP220 preincubated fo...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Biogen

Curated by ChEMBL
LigandPNGBDBM50106008(CHEMBL3598075)
Affinity DataIC50:  8.40nMAssay Description:Binding affinity to GST-tagged RORgamma LBD (unknown origin) assessed as inhibition of interaction with co-activatior peptide TRAP220 preincubated fo...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Biogen

Curated by ChEMBL
LigandPNGBDBM50105929(CHEMBL3598048)
Affinity DataIC50:  8.60nMAssay Description:Binding affinity to GST-tagged RORgamma LBD (unknown origin) assessed as inhibition of interaction with co-activatior peptide TRAP220 preincubated fo...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Biogen

Curated by ChEMBL
LigandPNGBDBM50105984(CHEMBL3598054)
Affinity DataIC50:  9.20nMAssay Description:Binding affinity to GST-tagged RORgamma LBD (unknown origin) assessed as inhibition of interaction with co-activatior peptide TRAP220 preincubated fo...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Biogen

Curated by ChEMBL
LigandPNGBDBM50105998(CHEMBL3598065)
Affinity DataIC50:  9.40nMAssay Description:Binding affinity to GST-tagged RORgamma LBD (unknown origin) assessed as inhibition of interaction with co-activatior peptide TRAP220 preincubated fo...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Biogen

Curated by ChEMBL
LigandPNGBDBM50108770(CHEMBL3596635)
Affinity DataIC50:  10nMAssay Description:Inverse agonist activity at human recombinant GST-tagged RORgammat ligand binding domain assessed as effect on receptor-biotin tagged TRAP220 co-acti...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Biogen

Curated by ChEMBL
LigandPNGBDBM50161155(CHEMBL3793229)
Affinity DataIC50:  10nMAssay Description:Inverse agonist activity at recombinant human GST-tagged ROR-gamma receptor ligand binding domain assessed as inhibition of receptor and co-activator...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Biogen

Curated by ChEMBL
LigandPNGBDBM50108770(CHEMBL3596635)
Affinity DataIC50:  10nMAssay Description:Inverse agonist activity at human recombinant GST-tagged RORgammat ligand binding domain assessed as effect on receptor-biotin tagged TRAP220 co-acti...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Biogen

Curated by ChEMBL
LigandPNGBDBM50108898(CHEMBL3596629)
Affinity DataIC50:  11nMAssay Description:Inverse agonist activity at human recombinant GST-tagged RORgammat ligand binding domain assessed as effect on receptor-biotin tagged TRAP220 co-acti...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Biogen

Curated by ChEMBL
LigandPNGBDBM50108900(CHEMBL3596631)
Affinity DataIC50:  11nMAssay Description:Inverse agonist activity at human recombinant GST-tagged RORgammat ligand binding domain assessed as effect on receptor-biotin tagged TRAP220 co-acti...More data for this Ligand-Target Pair
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Biogen

Curated by ChEMBL
LigandPNGBDBM50105991(CHEMBL3598060)
Affinity DataIC50:  12nMAssay Description:Binding affinity to GST-tagged RORgamma LBD (unknown origin) assessed as inhibition of interaction with co-activatior peptide TRAP220 preincubated fo...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Biogen

Curated by ChEMBL
LigandPNGBDBM50105932(CHEMBL3598050)
Affinity DataIC50:  15nMAssay Description:Binding affinity to GST-tagged RORgamma LBD (unknown origin) assessed as inhibition of interaction with co-activatior peptide TRAP220 preincubated fo...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Biogen

Curated by ChEMBL
LigandPNGBDBM50106004(CHEMBL3598072)
Affinity DataIC50:  15nMAssay Description:Binding affinity to GST-tagged RORgamma LBD (unknown origin) assessed as inhibition of interaction with co-activatior peptide TRAP220 preincubated fo...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Biogen

Curated by ChEMBL
LigandPNGBDBM50105997(CHEMBL3598064)
Affinity DataIC50:  16nMAssay Description:Binding affinity to GST-tagged RORgamma LBD (unknown origin) assessed as inhibition of interaction with co-activatior peptide TRAP220 preincubated fo...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Biogen

Curated by ChEMBL
LigandPNGBDBM50106000(CHEMBL3598066)
Affinity DataIC50:  18nMAssay Description:Binding affinity to GST-tagged RORgamma LBD (unknown origin) assessed as inhibition of interaction with co-activatior peptide TRAP220 preincubated fo...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Biogen

Curated by ChEMBL
LigandPNGBDBM50105925(CHEMBL3598044)
Affinity DataIC50:  18nMAssay Description:Binding affinity to GST-tagged RORgamma LBD (unknown origin) assessed as inhibition of interaction with co-activatior peptide TRAP220 preincubated fo...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Biogen

Curated by ChEMBL
LigandPNGBDBM50108685(CHEMBL3596633)
Affinity DataIC50:  20nMAssay Description:Inverse agonist activity at human recombinant GST-tagged RORgammat ligand binding domain assessed as effect on receptor-biotin tagged TRAP220 co-acti...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Biogen

Curated by ChEMBL
LigandPNGBDBM50106001(CHEMBL3598068)
Affinity DataIC50:  21nMAssay Description:Binding affinity to GST-tagged RORgamma LBD (unknown origin) assessed as inhibition of interaction with co-activatior peptide TRAP220 preincubated fo...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Biogen

Curated by ChEMBL
LigandPNGBDBM50108899(CHEMBL3596630)
Affinity DataIC50:  22nMAssay Description:Inverse agonist activity at human recombinant GST-tagged RORgammat ligand binding domain assessed as effect on receptor-biotin tagged TRAP220 co-acti...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Biogen

Curated by ChEMBL
LigandPNGBDBM50105924(CHEMBL3598043)
Affinity DataIC50:  26nMAssay Description:Binding affinity to GST-tagged RORgamma LBD (unknown origin) assessed as inhibition of interaction with co-activatior peptide TRAP220 preincubated fo...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Biogen

Curated by ChEMBL
LigandPNGBDBM50105919(CHEMBL3596632)
Affinity DataIC50:  29nMAssay Description:Inverse agonist activity at human recombinant GST-tagged RORgammat ligand binding domain assessed as effect on receptor-biotin tagged TRAP220 co-acti...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Biogen

Curated by ChEMBL
LigandPNGBDBM50105919(CHEMBL3596632)
Affinity DataIC50:  29nMAssay Description:Binding affinity to GST-tagged RORgamma LBD (unknown origin) assessed as inhibition of interaction with co-activatior peptide TRAP220 preincubated fo...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Biogen

Curated by ChEMBL
LigandPNGBDBM50105922(CHEMBL3598041)
Affinity DataIC50:  38nMAssay Description:Binding affinity to GST-tagged RORgamma LBD (unknown origin) assessed as inhibition of interaction with co-activatior peptide TRAP220 preincubated fo...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Biogen

Curated by ChEMBL
LigandPNGBDBM50106005(CHEMBL3598073)
Affinity DataIC50:  40nMAssay Description:Binding affinity to GST-tagged RORgamma LBD (unknown origin) assessed as inhibition of interaction with co-activatior peptide TRAP220 preincubated fo...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Biogen

Curated by ChEMBL
LigandPNGBDBM50108896(CHEMBL3596627)
Affinity DataIC50:  50nMAssay Description:Inverse agonist activity at human recombinant GST-tagged RORgammat ligand binding domain assessed as effect on receptor-biotin tagged TRAP220 co-acti...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Biogen

Curated by ChEMBL
LigandPNGBDBM50108897(CHEMBL3596628)
Affinity DataIC50:  54nMAssay Description:Inverse agonist activity at human recombinant GST-tagged RORgammat ligand binding domain assessed as effect on receptor-biotin tagged TRAP220 co-acti...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Biogen

Curated by ChEMBL
LigandPNGBDBM50105927(CHEMBL3598046)
Affinity DataIC50:  54nMAssay Description:Binding affinity to GST-tagged RORgamma LBD (unknown origin) assessed as inhibition of interaction with co-activatior peptide TRAP220 preincubated fo...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Biogen

Curated by ChEMBL
LigandPNGBDBM50161156(CHEMBL3793914)
Affinity DataIC50:  56nMAssay Description:Inverse agonist activity at recombinant human GST-tagged ROR-gamma receptor ligand binding domain assessed as inhibition of receptor and co-activator...More data for this Ligand-Target Pair
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Biogen

Curated by ChEMBL
LigandPNGBDBM50105993(CHEMBL3598062)
Affinity DataIC50:  70nMAssay Description:Binding affinity to GST-tagged RORgamma LBD (unknown origin) assessed as inhibition of interaction with co-activatior peptide TRAP220 preincubated fo...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Biogen

Curated by ChEMBL
LigandPNGBDBM50161154(CHEMBL3793036)
Affinity DataIC50:  72nMAssay Description:Inverse agonist activity at recombinant human GST-tagged ROR-gamma receptor ligand binding domain assessed as inhibition of receptor and co-activator...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Biogen

Curated by ChEMBL
LigandPNGBDBM50161145(CHEMBL3793667)
Affinity DataIC50:  72nMAssay Description:Inverse agonist activity at recombinant human GST-tagged ROR-gamma receptor ligand binding domain assessed as inhibition of receptor and co-activator...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Biogen

Curated by ChEMBL
LigandPNGBDBM50105926(CHEMBL3598045)
Affinity DataIC50:  76nMAssay Description:Binding affinity to GST-tagged RORgamma LBD (unknown origin) assessed as inhibition of interaction with co-activatior peptide TRAP220 preincubated fo...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Biogen

Curated by ChEMBL
LigandPNGBDBM50108685(CHEMBL3596633)
Affinity DataIC50:  89nMAssay Description:Inverse agonist activity at human recombinant GST-tagged RORgammat ligand binding domain assessed as effect on receptor-biotin tagged TRAP220 co-acti...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Biogen

Curated by ChEMBL
LigandPNGBDBM50108884(CHEMBL3596600)
Affinity DataIC50:  100nMAssay Description:Inverse agonist activity at human recombinant GST-tagged RORgammat ligand binding domain assessed as effect on receptor-biotin tagged TRAP220 co-acti...More data for this Ligand-Target Pair
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