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Found 88 with Last Name = 'barnes' and Initial = 'g'
TargetCyclin-dependent kinase 1(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM27216((2R)-2-({6-[(3-chlorophenyl)amino]-9-(propan-2-yl)...)
Affinity DataIC50:  4nMAssay Description:Inhibition of human cdc2/cyclin B assessed as [32P] incorporation in histone H1 from [gamma32P]ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM7478(2-chloro-4-[(2-{[(1R)-1-(hydroxymethyl)-2-methylpr...)
Affinity DataIC50:  6nMAssay Description:Inhibition of human cdk5/p35More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM7478(2-chloro-4-[(2-{[(1R)-1-(hydroxymethyl)-2-methylpr...)
Affinity DataIC50:  6nMAssay Description:Inhibition of human cdk2/cyclin AMore data for this Ligand-Target Pair
TargetCyclin-dependent kinase 1(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM7478(2-chloro-4-[(2-{[(1R)-1-(hydroxymethyl)-2-methylpr...)
Affinity DataIC50:  6nMAssay Description:Inhibition of human cdc2/cyclin B assessed as [32P] incorporation in histone H1 from [gamma32P]ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM7478(2-chloro-4-[(2-{[(1R)-1-(hydroxymethyl)-2-methylpr...)
Affinity DataIC50:  9nMAssay Description:Inhibition of human cdk2/cyclin EMore data for this Ligand-Target Pair
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM27216((2R)-2-({6-[(3-chlorophenyl)amino]-9-(propan-2-yl)...)
Affinity DataIC50:  35nMAssay Description:Inhibition of human cdk2/cyclin EMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCdc2(Asterina pectinifera)
University Of California

Curated by ChEMBL
LigandPNGBDBM27216((2R)-2-({6-[(3-chlorophenyl)amino]-9-(propan-2-yl)...)
Affinity DataIC50:  40nMAssay Description:Inhibition of starfish cdc2/cyclin B assessed as [32P] incorporation in histone H1 from 150 M [gamma32P]ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCdc2(Asterina pectinifera)
University Of California

Curated by ChEMBL
LigandPNGBDBM7478(2-chloro-4-[(2-{[(1R)-1-(hydroxymethyl)-2-methylpr...)
Affinity DataIC50:  50nMAssay Description:Inhibition of starfish cdc2/cyclin B assessed as [32P] incorporation in histone H1 from 150 M [gamma32P]ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM27216((2R)-2-({6-[(3-chlorophenyl)amino]-9-(propan-2-yl)...)
Affinity DataIC50:  70nMAssay Description:Inhibition of human cdk2/cyclin AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM27216((2R)-2-({6-[(3-chlorophenyl)amino]-9-(propan-2-yl)...)
Affinity DataIC50:  75nMAssay Description:Inhibition of human cdk5/p35More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 1(Saccharomyces cerevisiae)
University Of California

Curated by ChEMBL
LigandPNGBDBM27216((2R)-2-({6-[(3-chlorophenyl)amino]-9-(propan-2-yl)...)
Affinity DataIC50:  80nMAssay Description:Inhibition of Saccharomyces cerevisiae cdc28More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCdc2(Asterina pectinifera)
University Of California

Curated by ChEMBL
LigandPNGBDBM7478(2-chloro-4-[(2-{[(1R)-1-(hydroxymethyl)-2-methylpr...)
Affinity DataIC50:  250nMAssay Description:Inhibition of starfish cdc2/cyclin B assessed as [32P] incorporation in histone H1 from 1.5 mM [gamma32P]ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 1(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50113707(2,6,9-Trisubstitute purine, 2 | 2-(2-hydroxyethyla...)
Affinity DataIC50:  340nMAssay Description:Inhibition of human cdc2/cyclin B assessed as [32P] incorporation in histone H1 from [gamma32P]ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCdc2(Asterina pectinifera)
University Of California

Curated by ChEMBL
LigandPNGBDBM27216((2R)-2-({6-[(3-chlorophenyl)amino]-9-(propan-2-yl)...)
Affinity DataIC50:  500nMAssay Description:Inhibition of starfish cdc2/cyclin B assessed as [32P] incorporation in histone H1 from 1.5 mM [gamma32P]ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 4(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM27216((2R)-2-({6-[(3-chlorophenyl)amino]-9-(propan-2-yl)...)
Affinity DataIC50:  850nMAssay Description:Inhibition of human cdk4/cyclin D1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 1(Saccharomyces cerevisiae)
University Of California

Curated by ChEMBL
LigandPNGBDBM7478(2-chloro-4-[(2-{[(1R)-1-(hydroxymethyl)-2-methylpr...)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibition of Saccharomyces cerevisiae cdc28More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent protein kinase PHO85(Saccharomyces cerevisiae)
University Of California

Curated by ChEMBL
LigandPNGBDBM50113707(2,6,9-Trisubstitute purine, 2 | 2-(2-hydroxyethyla...)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of yeast W303 Pho85 phosphorylation assessed as [32P] incorporation in histone H1 from [gamma32P]ATP by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInsulin receptor(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM7478(2-chloro-4-[(2-{[(1R)-1-(hydroxymethyl)-2-methylpr...)
Affinity DataIC50:  2.20E+3nMAssay Description:Inhibition of human insulin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 3(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM7478(2-chloro-4-[(2-{[(1R)-1-(hydroxymethyl)-2-methylpr...)
Affinity DataIC50:  3.33E+3nMAssay Description:Inhibition of human Erk1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInsulin receptor(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM27216((2R)-2-({6-[(3-chlorophenyl)amino]-9-(propan-2-yl)...)
Affinity DataIC50:  5.00E+3nMAssay Description:Inhibition of human insulin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
University Of Arkansas

Curated by ChEMBL
LigandPNGBDBM50013004(2-Acetylamino-4-methyl-pentanoic acid [1-(1-formyl...)
Affinity DataIC50:  5.20E+3nMAssay Description:Evaluated for the inhibition of trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen(Rattus norvegicus)
University Of Arkansas

Curated by ChEMBL
LigandPNGBDBM50013004(2-Acetylamino-4-methyl-pentanoic acid [1-(1-formyl...)
Affinity DataIC50:  5.20E+3nMAssay Description:Inhibition of plasminMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 1(Saccharomyces cerevisiae)
University Of California

Curated by ChEMBL
LigandPNGBDBM50113707(2,6,9-Trisubstitute purine, 2 | 2-(2-hydroxyethyla...)
Affinity DataIC50:  7.00E+3nMAssay Description:Inhibition of yeast W303 cdc28 phosphorylation assessed as [32P] incorporation in histone H1 from [gamma32P]ATP by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen(Rattus norvegicus)
University Of Arkansas

Curated by ChEMBL
LigandPNGBDBM50013003(CHEMBL3143639 | {1-[1-(5-Amino-1-formyl-pentylcarb...)
Affinity DataIC50:  8.90E+3nMAssay Description:Inhibition of plasminMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 3(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM27216((2R)-2-({6-[(3-chlorophenyl)amino]-9-(propan-2-yl)...)
Affinity DataIC50:  9.00E+3nMAssay Description:Inhibition of human Erk1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM27216((2R)-2-({6-[(3-chlorophenyl)amino]-9-(propan-2-yl)...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human GSK3-betaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 4(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM7478(2-chloro-4-[(2-{[(1R)-1-(hydroxymethyl)-2-methylpr...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human cdk4/cyclin D1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C gamma type(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM27216((2R)-2-({6-[(3-chlorophenyl)amino]-9-(propan-2-yl)...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human PKCgammaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C beta type(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM27216((2R)-2-({6-[(3-chlorophenyl)amino]-9-(propan-2-yl)...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human PKCbeta1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM27216((2R)-2-({6-[(3-chlorophenyl)amino]-9-(propan-2-yl)...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human PKCalphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C beta type(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM27216((2R)-2-({6-[(3-chlorophenyl)amino]-9-(propan-2-yl)...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human PKCbeta2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM7478(2-chloro-4-[(2-{[(1R)-1-(hydroxymethyl)-2-methylpr...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human GSK3-betaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen(Rattus norvegicus)
University Of Arkansas

Curated by ChEMBL
LigandPNGBDBM50228472(CHEMBL3143648)
Affinity DataIC50:  1.02E+4nMAssay Description:Inhibition of plasminMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-1(Homo sapiens (Human))
University Of Arkansas

Curated by ChEMBL
LigandPNGBDBM50013008(CHEMBL2371651 | {1-[1-(1-Formyl-4-guanidino-butylc...)
Affinity DataIC50:  1.12E+4nMAssay Description:Inhibition of Kallikrein proteolytic enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-1(Homo sapiens (Human))
University Of Arkansas

Curated by ChEMBL
LigandPNGBDBM50013001(CHEMBL3143646 | {1-[1-(4-Amino-1-formyl-butylcarba...)
Affinity DataIC50:  1.18E+4nMAssay Description:Inhibition of Kallikrein proteolytic enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-1(Homo sapiens (Human))
University Of Arkansas

Curated by ChEMBL
LigandPNGBDBM50012998(CHEMBL2371625 | {1-[1-(5-Amino-1-formyl-pentylcarb...)
Affinity DataIC50:  1.48E+4nMAssay Description:Inhibition of Kallikrein proteolytic enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-1(Homo sapiens (Human))
University Of Arkansas

Curated by ChEMBL
LigandPNGBDBM50013007(CHEMBL2371644 | {1-[1-(5-Amino-1-formyl-pentylcarb...)
Affinity DataIC50:  1.90E+4nMAssay Description:Inhibition of Kallikrein proteolytic enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-1(Homo sapiens (Human))
University Of Arkansas

Curated by ChEMBL
LigandPNGBDBM50013006(CHEMBL3143642 | {1-[1-(5-Amino-1-formyl-pentylcarb...)
Affinity DataIC50:  2.03E+4nMAssay Description:Inhibition of Kallikrein proteolytic enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-1(Homo sapiens (Human))
University Of Arkansas

Curated by ChEMBL
LigandPNGBDBM50013003(CHEMBL3143639 | {1-[1-(5-Amino-1-formyl-pentylcarb...)
Affinity DataIC50:  2.56E+4nMAssay Description:Inhibition of Kallikrein proteolytic enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-1(Homo sapiens (Human))
University Of Arkansas

Curated by ChEMBL
LigandPNGBDBM50228472(CHEMBL3143648)
Affinity DataIC50:  2.57E+4nMAssay Description:Inhibition of plasminMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-1(Homo sapiens (Human))
University Of Arkansas

Curated by ChEMBL
LigandPNGBDBM50012999(CHEMBL2371642 | {1-[1-(4-Amino-1-formyl-butylcarba...)
Affinity DataIC50:  2.93E+4nMAssay Description:Inhibition of Kallikrein proteolytic enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-1(Homo sapiens (Human))
University Of Arkansas

Curated by ChEMBL
LigandPNGBDBM50013004(2-Acetylamino-4-methyl-pentanoic acid [1-(1-formyl...)
Affinity DataIC50:  3.24E+4nMAssay Description:Inhibition of Kallikrein proteolytic enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-1(Homo sapiens (Human))
University Of Arkansas

Curated by ChEMBL
LigandPNGBDBM50228474(CHEMBL3143649)
Affinity DataIC50:  3.33E+4nMAssay Description:Inhibition of Kallikrein proteolytic enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-1(Homo sapiens (Human))
University Of Arkansas

Curated by ChEMBL
LigandPNGBDBM50228473(CHEMBL3143647)
Affinity DataIC50:  3.60E+4nMAssay Description:Evaluated for the inhibition of trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
University Of Arkansas

Curated by ChEMBL
LigandPNGBDBM50228472(CHEMBL3143648)
Affinity DataIC50:  4.59E+4nMAssay Description:Inhibition of Kallikrein proteolytic enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen(Rattus norvegicus)
University Of Arkansas

Curated by ChEMBL
LigandPNGBDBM50013006(CHEMBL3143642 | {1-[1-(5-Amino-1-formyl-pentylcarb...)
Affinity DataIC50:  4.70E+4nMAssay Description:Inhibition of plasminMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-1(Homo sapiens (Human))
University Of Arkansas

Curated by ChEMBL
LigandPNGBDBM50012996(CHEMBL2371655 | {1-[1-(4-Amino-1-formyl-butylcarba...)
Affinity DataIC50:  5.38E+4nMAssay Description:Inhibition of Kallikrein proteolytic enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen(Rattus norvegicus)
University Of Arkansas

Curated by ChEMBL
LigandPNGBDBM50228474(CHEMBL3143649)
Affinity DataIC50:  7.99E+4nMAssay Description:Evaluated for the inhibition of trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen(Rattus norvegicus)
University Of Arkansas

Curated by ChEMBL
LigandPNGBDBM50013008(CHEMBL2371651 | {1-[1-(1-Formyl-4-guanidino-butylc...)
Affinity DataIC50:  8.14E+4nMAssay Description:Inhibition of plasminMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
University Of Arkansas

Curated by ChEMBL
LigandPNGBDBM50013008(CHEMBL2371651 | {1-[1-(1-Formyl-4-guanidino-butylc...)
Affinity DataIC50:  8.14E+4nMAssay Description:Evaluated for the inhibition of trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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