Affinity DataIC50: 1.26nMAssay Description:Inhibition of JNK3 by high throughput screeningMore data for this Ligand-Target Pair
Affinity DataIC50: 3.98nMAssay Description:Inhibition of p38alpha by high throughput screeningMore data for this Ligand-Target Pair
Affinity DataIC50: 5nMAssay Description:Inhibition of catalytic activity of GSK3-beta by AlphaLISA assayMore data for this Ligand-Target Pair
Affinity DataIC50: 5.01nMAssay Description:Inhibition of human GSK3-beta expressed in baculovirus by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataIC50: 6.31nMAssay Description:Inhibition of human GSK3-beta expressed in baculovirus by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataIC50: 6.31nMAssay Description:Inhibition of JNK3 by high throughput screeningMore data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Inhibition of human GSK3-beta expressed in baculovirus by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Inhibition of human GSK3-beta expressed in baculovirus by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataIC50: 12.6nMAssay Description:Inhibition of human full length His-tagged GSK3-beta expressed in baculovirus by alphaLISA assayMore data for this Ligand-Target Pair
Affinity DataIC50: 12.6nMAssay Description:Inhibition of human GSK3-beta expressed in baculovirus by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataIC50: 13nMAssay Description:Inhibition of catalytic activity of GSK3-beta by AlphaLISA assayMore data for this Ligand-Target Pair
Affinity DataIC50: 19.9nMAssay Description:Inhibition of human full length His-tagged GSK3-beta expressed in baculovirus by alphaLISA assayMore data for this Ligand-Target Pair
Affinity DataIC50: 20nMAssay Description:Inhibition of catalytic activity of GSK3-beta by AlphaLISA assayMore data for this Ligand-Target Pair
Affinity DataIC50: 20nMAssay Description:Inhibition of catalytic activity of GSK3-beta by AlphaLISA assayMore data for this Ligand-Target Pair
Affinity DataIC50: 20nMAssay Description:Inhibition of catalytic activity of GSK3-beta by AlphaLISA assayMore data for this Ligand-Target Pair
Affinity DataIC50: 32nMAssay Description:Inhibition of catalytic activity of GSK3-beta by AlphaLISA assayMore data for this Ligand-Target Pair
Affinity DataIC50: 32nMAssay Description:Inhibition of catalytic activity of GSK3-beta by AlphaLISA assayMore data for this Ligand-Target Pair
Affinity DataIC50: 32nMAssay Description:Inhibition of catalytic activity of GSK3-beta by AlphaLISA assayMore data for this Ligand-Target Pair
Affinity DataIC50: 40nMAssay Description:Inhibition of Escherichia coli his-tagged DNA gyrase supercoiling activity using pBR322 DNA in presence of ATP incubated for 1 hr by H19 dye based hi...More data for this Ligand-Target Pair
Affinity DataIC50: 40nMAssay Description:Inhibition of catalytic activity of GSK3-beta by AlphaLISA assayMore data for this Ligand-Target Pair
Affinity DataIC50: 50.1nMAssay Description:Inhibition of N-terminal histidine-tagged human full length JNK3 by radiometric filter binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: 63nMAssay Description:Inhibition of catalytic activity of GSK3-beta by AlphaLISA assayMore data for this Ligand-Target Pair
Affinity DataIC50: 63.1nMAssay Description:Inhibition of human full length His-tagged GSK3-beta expressed in baculovirus by alphaLISA assayMore data for this Ligand-Target Pair
Affinity DataIC50: 79nMAssay Description:Inhibition of catalytic activity of GSK3-beta by AlphaLISA assayMore data for this Ligand-Target Pair
Affinity DataIC50: 79nMAssay Description:Inhibition of catalytic activity of GSK3-beta by AlphaLISA assayMore data for this Ligand-Target Pair
Affinity DataIC50: 79.4nMAssay Description:Inhibition of human flag-tagged GSK3-beta expressed in HEK-MSRII cells assessed as CRMP-2 phosphorylation by alphaLISA assayMore data for this Ligand-Target Pair
Affinity DataIC50: 79.4nMAssay Description:Inhibition of JNK1 by high throughput screeningMore data for this Ligand-Target Pair
Affinity DataIC50: 100nMAssay Description:Inhibition of human CYP1A2 by fluorescence assayMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Glaxosmithkline
Curated by ChEMBL
Glaxosmithkline
Curated by ChEMBL
Affinity DataIC50: 100nMAssay Description:Inhibition of PI3Kdelta (unknown origin) using PIP2 as substrate pretreated for 15 mins followed by substrate addition measured after 1 hrMore data for this Ligand-Target Pair
Affinity DataIC50: 100nMAssay Description:Inhibition of catalytic activity of GSK3-beta by AlphaLISA assayMore data for this Ligand-Target Pair
Affinity DataIC50: 100nMAssay Description:Inhibitory activity against bovine mitochondrial F1F0-ATP synthaseMore data for this Ligand-Target Pair
Affinity DataIC50: 100nMAssay Description:Inhibition of human GSK3-beta expressed in baculovirus by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataIC50: 126nMAssay Description:Inhibition of human GSK3-beta expressed in baculovirus by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataIC50: 126nMAssay Description:Inhibition of human GSK3-beta expressed in baculovirus by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataIC50: 126nMAssay Description:Inhibition of N-terminal histidine-tagged human full length JNK3 by radiometric filter binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: 126nMAssay Description:Inhibition of human GSK3-beta expressed in baculovirus by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataIC50: 126nMAssay Description:Inhibition of PIM1 (unknown origin) using TAMRA-ERMRPRKRQGSVRRRV-NH2 as substrate pretreated for 30 mins followed by substrate addition measured afte...More data for this Ligand-Target Pair
Affinity DataIC50: 158nMAssay Description:Inhibition of recombinant CDK2 expressed in baculovirus using [gamma-32P]-ATP by 33-P leadseeker assayMore data for this Ligand-Target Pair
Affinity DataIC50: 158nMAssay Description:Inhibition of human full length His-tagged GSK3-beta expressed in baculovirus by alphaLISA assayMore data for this Ligand-Target Pair
Affinity DataIC50: 158nMAssay Description:Inhibition of human GSK3-beta expressed in baculovirus by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataIC50: 160nMAssay Description:Inhibition of Escherichia coli his-tagged DNA gyrase supercoiling activity using pBR322 DNA in presence of ATP incubated for 1 hr by H19 dye based hi...More data for this Ligand-Target Pair
Affinity DataIC50: 160nMAssay Description:Inhibition of Escherichia coli his-tagged DNA gyrase supercoiling activity using pBR322 DNA in presence of ATP incubated for 1 hr by H19 dye based hi...More data for this Ligand-Target Pair
Affinity DataIC50: 200nMAssay Description:Inhibition of recombinant CDK2 expressed in baculovirus using [gamma-32P]-ATP by 33-P leadseeker assayMore data for this Ligand-Target Pair
Affinity DataIC50: 200nMAssay Description:Inhibition of human CYP2C9 by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 200nMAssay Description:Inhibition of p38alpha by high throughput screeningMore data for this Ligand-Target Pair
Affinity DataIC50: 251nMAssay Description:Inhibition of GSK3-beta by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataIC50: 251nMAssay Description:Inhibition of GSK3-beta by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataIC50: 251nMAssay Description:Inhibition of human full length His-tagged GSK3-beta expressed in baculovirus by alphaLISA assayMore data for this Ligand-Target Pair
Affinity DataIC50: 251nMAssay Description:Inhibition of recombinant CDK2 expressed in baculovirus using [gamma-32P]-ATP by 33-P leadseeker assayMore data for this Ligand-Target Pair
Affinity DataIC50: 251nMAssay Description:Inhibition of N-terminal His(6)-tagged truncated human JNK3 transfected in baculovirus expression system by fluorescence anisotropyMore data for this Ligand-Target Pair