Affinity DataKi: 0.900nMAssay Description:Compound was evaluated for its binding affinity by displacement of [3H]- DAMPGO from opioid receptor mu by using opioid radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 0.900nMAssay Description:Compound was evaluated for its binding affinity by displacement [3H]- DSLET from Opioid receptor delta 1 by using opioid radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 2.5nMAssay Description:Compound was evaluated for its binding affinity by displacement [3H]- DSLET from Opioid receptor delta 1 by using opioid radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 7nMAssay Description:Compound was evaluated for its binding affinity by displacement [3H]- DSLET from Opioid receptor delta 1 by using opioid radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 9.5nMAssay Description:Compound was evaluated for its binding affinity by displacement of [3H]- DAMPGO from opioid receptor mu by using opioid radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 11nMAssay Description:Compound was evaluated for its binding affinity by displacement of [3H]- DAMPGO from opioid receptor mu by using opioid radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 11nMAssay Description:Compound was evaluated for its binding affinity by displacement [3H]- DSLET from Opioid receptor delta 1 by using opioid radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 21nMAssay Description:Compound was evaluated for its binding affinity by displacement [3H]- DSLET from Opioid receptor delta 1 by using opioid radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 21nMAssay Description:Compound was evaluated for its binding affinity by displacement [3H]- DSLET from Opioid receptor delta 1 by using opioid radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 32nMAssay Description:Compound was evaluated for its binding affinity by displacement of [3H]- DAMPGO from opioid receptor mu by using opioid radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 32nMAssay Description:Dissociation rate constant of compound for mutant T46S Escherichia coli dihydrofolate reductaseMore data for this Ligand-Target Pair
Affinity DataKi: 45nMAssay Description:Compound was evaluated for its binding affinity by displacement [3H]- DSLET from Opioid receptor delta 1 by using opioid radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 45nMAssay Description:Compound was evaluated for its binding affinity by displacement [3H]- DSLET from Opioid receptor delta 1 by using opioid radioligand binding assayMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Georgetown University
Curated by PDSP Ki Database
Georgetown University
Curated by PDSP Ki Database
Affinity DataKi: 91nMAssay Description:Dissociation rate constant of compound for mutant T46A Escherichia coli dihydrofolate reductaseMore data for this Ligand-Target Pair
Affinity DataKi: 91nMAssay Description:Compound was evaluated for its binding affinity by displacement [3H]- DSLET from Opioid receptor delta 1 by using opioid radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 150nMAssay Description:Compound was evaluated for its binding affinity by displacement of [3H]- DAMPGO from opioid receptor mu by using opioid radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 150nMAssay Description:Compound was evaluated for its binding affinity by displacement of [3H]- DAMPGO from opioid receptor mu by using opioid radioligand binding assayMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Georgetown University
Curated by PDSP Ki Database
Georgetown University
Curated by PDSP Ki Database
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Georgetown University
Curated by PDSP Ki Database
Georgetown University
Curated by PDSP Ki Database
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Georgetown University
Curated by PDSP Ki Database
Georgetown University
Curated by PDSP Ki Database
Affinity DataKi: 700nMAssay Description:Compound was evaluated for its binding affinity by displacement of [3H]- DAMPGO from opioid receptor mu by using opioid radioligand binding assayMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Georgetown University
Curated by PDSP Ki Database
Georgetown University
Curated by PDSP Ki Database
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Georgetown University
Curated by PDSP Ki Database
Georgetown University
Curated by PDSP Ki Database
Affinity DataIC50: 0.460nMAssay Description:Binding affinity towards dopamine transporter in rat striatum using [3H]WIN-35 428 as radioligandMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Georgetown University
Curated by PDSP Ki Database
Georgetown University
Curated by PDSP Ki Database
Affinity DataIC50: 0.960nMAssay Description:Inhibition of 3[H] WIN-35 428 binding to Dopamine transporter (DAT)More data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Georgetown University
Curated by PDSP Ki Database
Georgetown University
Curated by PDSP Ki Database
Affinity DataIC50: 2.48nMAssay Description:Inhibition of uptake from dopamine transporter in rat striatum using [3H]DA as radioligandMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Georgetown University
Curated by PDSP Ki Database
Georgetown University
Curated by PDSP Ki Database
Affinity DataIC50: 2.96nMAssay Description:Inhibition of 3[H] WIN-35 428 binding to Dopamine transporter (DAT)More data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Georgetown University
Curated by PDSP Ki Database
Georgetown University
Curated by PDSP Ki Database
Affinity DataIC50: 3.67nMAssay Description:In vitro binding affinity at dopamine transporter in rat striatum by [3H]WIN-35428 displacement.More data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Georgetown University
Curated by PDSP Ki Database
Georgetown University
Curated by PDSP Ki Database
Affinity DataIC50: 4.05nMAssay Description:Inhibition of uptake from dopamine transporter in rat striatum using [3H]DA as radioligandMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Georgetown University
Curated by PDSP Ki Database
Georgetown University
Curated by PDSP Ki Database
Affinity DataIC50: 4.10nMAssay Description:Inhibition of 3[H] WIN-35 428 binding to Dopamine transporter (DAT)More data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Georgetown University
Curated by PDSP Ki Database
Georgetown University
Curated by PDSP Ki Database
Affinity DataIC50: 4.5nMAssay Description:Inhibition of 3[H] WIN-35 428 binding to Dopamine transporter (DAT)More data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Georgetown University
Curated by PDSP Ki Database
Georgetown University
Curated by PDSP Ki Database
Affinity DataIC50: 4.5nMAssay Description:In vitro binding affinity at dopamine transporter in rat striatum by [3H]WIN-35428 displacement.More data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Georgetown University
Curated by PDSP Ki Database
Georgetown University
Curated by PDSP Ki Database
Affinity DataIC50: 6.63nMAssay Description:Inhibition of uptake from dopamine transporter in rat striatum using [3H]DA as radioligandMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Georgetown University
Curated by PDSP Ki Database
Georgetown University
Curated by PDSP Ki Database
Affinity DataIC50: 7nMAssay Description:In vitro binding affinity at dopamine transporter in rat striatum by [3H]WIN-35428 displacement.More data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Georgetown University
Curated by PDSP Ki Database
Georgetown University
Curated by PDSP Ki Database
Affinity DataIC50: 8.23nMAssay Description:Inhibition of 3[H] WIN-35 428 binding to Dopamine transporter (DAT)More data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Georgetown University
Curated by PDSP Ki Database
Georgetown University
Curated by PDSP Ki Database
Affinity DataIC50: 9.37nMAssay Description:In vitro binding affinity at dopamine transporter in rat striatum by [3H]WIN-35428 displacement.More data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Georgetown University
Curated by PDSP Ki Database
Georgetown University
Curated by PDSP Ki Database
Affinity DataIC50: 10.1nMAssay Description:Inhibition of uptake from dopamine transporter in rat striatum using [3H]DA as radioligandMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Georgetown University
Curated by PDSP Ki Database
Georgetown University
Curated by PDSP Ki Database
Affinity DataIC50: 10.1nMAssay Description:In vitro binding affinity at dopamine transporter in rat striatum by [3H]WIN-35428 displacement.More data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Georgetown University
Curated by PDSP Ki Database
Georgetown University
Curated by PDSP Ki Database
Affinity DataIC50: 10.6nMAssay Description:Inhibition of [3H]WIN-35428 binding to dopamine transporter of rat striatumMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Georgetown University
Curated by PDSP Ki Database
Georgetown University
Curated by PDSP Ki Database
Affinity DataIC50: 10.6nMAssay Description:In vitro binding affinity at dopamine transporter in rat striatum by [3H]WIN-35428 displacement.More data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Georgetown University
Curated by PDSP Ki Database
Georgetown University
Curated by PDSP Ki Database
Affinity DataIC50: 10.6nMAssay Description:Inhibition of binding of 3[H] WIN-35 428 to Dopamine transporter (DAT) of rat striatum.More data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Georgetown University
Curated by PDSP Ki Database
Georgetown University
Curated by PDSP Ki Database
Affinity DataIC50: 10.6nMAssay Description:Binding affinity towards dopamine transporter in rat striatum using [3H]WIN-35 428 as radioligandMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Georgetown University
Curated by PDSP Ki Database
Georgetown University
Curated by PDSP Ki Database
Affinity DataIC50: 11.2nMAssay Description:Inhibition of [3H]WIN-35428 binding to dopamine transporter of rat striatumMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Georgetown University
Curated by PDSP Ki Database
Georgetown University
Curated by PDSP Ki Database
Affinity DataIC50: 11.2nMAssay Description:Binding affinity towards dopamine transporter in rat striatum using [3H]WIN-35 428 as radioligandMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Georgetown University
Curated by PDSP Ki Database
Georgetown University
Curated by PDSP Ki Database
Affinity DataIC50: 11.6nMAssay Description:Inhibition of 3[H] WIN-35 428 binding to Dopamine transporter (DAT)More data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Georgetown University
Curated by PDSP Ki Database
Georgetown University
Curated by PDSP Ki Database
Affinity DataIC50: 14.3nMAssay Description:Inhibition of 3[H] WIN-35 428 binding to Dopamine transporter (DAT)More data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Georgetown University
Curated by PDSP Ki Database
Georgetown University
Curated by PDSP Ki Database
Affinity DataIC50: 17.2nMAssay Description:In vitro binding affinity at dopamine transporter in rat striatum by [3H]WIN-35428 displacement.More data for this Ligand-Target Pair