Reaction Details Report a problem with these data
Target
Norepinephrine transporter
Ligand
BDBM86206
Substrate
n/a
Ki
90±n/a nM
Comments
PDSP_3054
Citation
 Kozikowski, AP; Johnson, KM; Deschaux, O; Bandyopadhyay, BC; Araldi, GL; Carmona, G; Munzar, P; Smith, MP; Balster, RL; Beardsley, PM; Tella, SR Mixed cocaine agonist/antagonist properties of (+)-methyl 4beta-(4-chlorophenyl)-1-methylpiperidine-3alpha-carboxylate, a piperidine-based analog of cocaine. J Pharmacol Exp Ther 305:143-50 (2003) [PubMed]  Article 
Target
Name:
Norepinephrine transporter
Synonyms:
n/a
Type:
Enzyme Catalytic Domain
Mol. Mass.:
2082.45
Organism:
RAT
Description:
Norepinephrine transporter 0 RAT::Q9JIA2
Residue:
19
Sequence:
MLLARMKPQVQPELGGADQ
  
Inhibitor
Name:
BDBM86206
Synonyms:
CAS_8268 | CPCA, + | NSC_8268
Type:
Small organic molecule
Emp. Form.:
C13H16ClNO2
Mol. Mass.:
253.725
SMILES:
CN1CCC([C@@H](C1)C(O)=O)c1ccc(Cl)cc1 |r|
Structure:
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