Affinity DataIC50: 750nMAssay Description:To identify inhibitors of TMPRSS2 that may be used directly in clinical studies or as lead compounds to develop targeted drugs, we screened several c...More data for this Ligand-Target Pair
Affinity DataIC50: 930nMAssay Description:To identify inhibitors of TMPRSS2 that may be used directly in clinical studies or as lead compounds to develop targeted drugs, we screened several c...More data for this Ligand-Target Pair
Ligand InfoPurchase
Affinity DataIC50: 1.37E+3nMAssay Description:To identify inhibitors of TMPRSS2 that may be used directly in clinical studies or as lead compounds to develop targeted drugs, we screened several c...More data for this Ligand-Target Pair
Affinity DataIC50: 2.64E+3nMAssay Description:To identify inhibitors of TMPRSS2 that may be used directly in clinical studies or as lead compounds to develop targeted drugs, we screened several c...More data for this Ligand-Target Pair
Ligand InfoPurchase
Affinity DataIC50: 2.68E+3nMAssay Description:To identify inhibitors of TMPRSS2 that may be used directly in clinical studies or as lead compounds to develop targeted drugs, we screened several c...More data for this Ligand-Target Pair
Ligand InfoPurchase
TargetNAD-dependent protein deacetylase sirtuin-3, mitochondrial(Homo sapiens (Human))
Fred Hutchinson Cancer Research Center
Curated by ChEMBL
Fred Hutchinson Cancer Research Center
Curated by ChEMBL
Affinity DataIC50: 6.00E+3nMAssay Description:Inhibition of SIRT3 (unknown origin) by luminescence assayMore data for this Ligand-Target Pair
TargetNAD-dependent histone deacetylase SIR2(Saccharomyces cerevisiae)
Fred Hutchinson Cancer Research Center
Curated by ChEMBL
Fred Hutchinson Cancer Research Center
Curated by ChEMBL
Affinity DataIC50: 8.80E+3nMAssay Description:In vitro inhibition of sirtuin 2 was evaluated using yeast whole cell lysatesMore data for this Ligand-Target Pair
TargetNAD-dependent histone deacetylase SIR2(Saccharomyces cerevisiae)
Fred Hutchinson Cancer Research Center
Curated by ChEMBL
Fred Hutchinson Cancer Research Center
Curated by ChEMBL
Affinity DataIC50: 1.20E+4nMAssay Description:In vitro inhibition of sirtuin 2 was evaluated using yeast whole cell lysatesMore data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-2(Homo sapiens (Human))
Fred Hutchinson Cancer Research Center
Curated by ChEMBL
Fred Hutchinson Cancer Research Center
Curated by ChEMBL
Affinity DataIC50: 1.30E+4nMAssay Description:Inhibition of SIRT2 (unknown origin) by luminescence assayMore data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-1(Homo sapiens (Human))
Fred Hutchinson Cancer Research Center
Curated by ChEMBL
Fred Hutchinson Cancer Research Center
Curated by ChEMBL
Affinity DataIC50: 2.10E+4nMAssay Description:Inhibition of C-terminal His-6-tagged recombinant human SIRT1 expressed in Escherichia coli BL21(DE3) by luminescence assayMore data for this Ligand-Target Pair
TargetNAD-dependent histone deacetylase SIR2(Saccharomyces cerevisiae)
Fred Hutchinson Cancer Research Center
Curated by ChEMBL
Fred Hutchinson Cancer Research Center
Curated by ChEMBL
Affinity DataIC50: 2.50E+4nMAssay Description:In vitro inhibition of sirtuin 2 was evaluated using yeast whole cell lysatesMore data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-1(Homo sapiens (Human))
Fred Hutchinson Cancer Research Center
Curated by ChEMBL
Fred Hutchinson Cancer Research Center
Curated by ChEMBL
Affinity DataIC50: 2.60E+4nMAssay Description:Inhibition of C-terminal His-6-tagged recombinant human SIRT1 expressed in Escherichia coli BL21(DE3) by luminescence assayMore data for this Ligand-Target Pair
TargetNAD-dependent histone deacetylase SIR2(Saccharomyces cerevisiae)
Fred Hutchinson Cancer Research Center
Curated by ChEMBL
Fred Hutchinson Cancer Research Center
Curated by ChEMBL
Affinity DataIC50: 2.70E+4nMAssay Description:In vitro inhibition of sirtuin 2 was evaluated using yeast whole cell lysatesMore data for this Ligand-Target Pair
TargetNAD-dependent histone deacetylase SIR2(Saccharomyces cerevisiae)
Fred Hutchinson Cancer Research Center
Curated by ChEMBL
Fred Hutchinson Cancer Research Center
Curated by ChEMBL
Affinity DataIC50: 2.70E+4nMAssay Description:In vitro inhibition of sirtuin 2 was evaluated using yeast whole cell lysatesMore data for this Ligand-Target Pair
TargetNAD-dependent histone deacetylase SIR2(Saccharomyces cerevisiae)
Fred Hutchinson Cancer Research Center
Curated by ChEMBL
Fred Hutchinson Cancer Research Center
Curated by ChEMBL
Affinity DataIC50: 2.70E+4nMAssay Description:In vitro inhibition of sirtuin 2 was evaluated using yeast whole cell lysatesMore data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-2(Homo sapiens (Human))
Fred Hutchinson Cancer Research Center
Curated by ChEMBL
Fred Hutchinson Cancer Research Center
Curated by ChEMBL
Affinity DataIC50: 3.20E+4nMAssay Description:Inhibition of SIRT2 (unknown origin) by luminescence assayMore data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-1(Homo sapiens (Human))
Fred Hutchinson Cancer Research Center
Curated by ChEMBL
Fred Hutchinson Cancer Research Center
Curated by ChEMBL
Affinity DataIC50: 3.70E+4nMAssay Description:Inhibition of C-terminal His-6-tagged recombinant human SIRT1 expressed in Escherichia coli BL21(DE3) by luminescence assayMore data for this Ligand-Target Pair
TargetNAD-dependent histone deacetylase SIR2(Saccharomyces cerevisiae)
Fred Hutchinson Cancer Research Center
Curated by ChEMBL
Fred Hutchinson Cancer Research Center
Curated by ChEMBL
Affinity DataIC50: 3.90E+4nMAssay Description:In vitro inhibition of sirtuin 2 was evaluated using yeast whole cell lysatesMore data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-1(Homo sapiens (Human))
Fred Hutchinson Cancer Research Center
Curated by ChEMBL
Fred Hutchinson Cancer Research Center
Curated by ChEMBL
Affinity DataIC50: 4.10E+4nMAssay Description:Inhibition of C-terminal His-6-tagged recombinant human SIRT1 expressed in Escherichia coli BL21(DE3) by luminescence assayMore data for this Ligand-Target Pair
TargetNAD-dependent histone deacetylase SIR2(Saccharomyces cerevisiae)
Fred Hutchinson Cancer Research Center
Curated by ChEMBL
Fred Hutchinson Cancer Research Center
Curated by ChEMBL
Affinity DataIC50: 4.10E+4nMAssay Description:In vitro inhibition of sirtuin 2 was evaluated using yeast whole cell lysatesMore data for this Ligand-Target Pair
TargetNAD-dependent histone deacetylase SIR2(Saccharomyces cerevisiae)
Fred Hutchinson Cancer Research Center
Curated by ChEMBL
Fred Hutchinson Cancer Research Center
Curated by ChEMBL
Affinity DataIC50: 4.30E+4nMAssay Description:In vitro inhibition of sirtuin 2 was evaluated using yeast whole cell lysatesMore data for this Ligand-Target Pair
TargetNAD-dependent histone deacetylase SIR2(Saccharomyces cerevisiae)
Fred Hutchinson Cancer Research Center
Curated by ChEMBL
Fred Hutchinson Cancer Research Center
Curated by ChEMBL
Affinity DataIC50: 4.40E+4nMAssay Description:In vitro inhibition of sirtuin 2 was evaluated using yeast whole cell lysatesMore data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-2(Homo sapiens (Human))
Fred Hutchinson Cancer Research Center
Curated by ChEMBL
Fred Hutchinson Cancer Research Center
Curated by ChEMBL
Affinity DataIC50: 5.10E+4nMAssay Description:Inhibition of SIRT2 (unknown origin) by luminescence assayMore data for this Ligand-Target Pair
TargetNAD-dependent histone deacetylase SIR2(Saccharomyces cerevisiae)
Fred Hutchinson Cancer Research Center
Curated by ChEMBL
Fred Hutchinson Cancer Research Center
Curated by ChEMBL
Affinity DataIC50: 5.20E+4nMAssay Description:In vitro inhibition of sirtuin 2 was evaluated using yeast whole cell lysatesMore data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-1(Homo sapiens (Human))
Fred Hutchinson Cancer Research Center
Curated by ChEMBL
Fred Hutchinson Cancer Research Center
Curated by ChEMBL
Affinity DataIC50: 5.60E+4nMAssay Description:Inhibition of C-terminal His-6-tagged recombinant human SIRT1 expressed in Escherichia coli BL21(DE3) by luminescence assayMore data for this Ligand-Target Pair
TargetNAD-dependent histone deacetylase SIR2(Saccharomyces cerevisiae)
Fred Hutchinson Cancer Research Center
Curated by ChEMBL
Fred Hutchinson Cancer Research Center
Curated by ChEMBL
Affinity DataIC50: 5.90E+4nMAssay Description:In vitro inhibition of sirtuin 2 was evaluated using yeast whole cell lysatesMore data for this Ligand-Target Pair
TargetNAD-dependent histone deacetylase SIR2(Saccharomyces cerevisiae)
Fred Hutchinson Cancer Research Center
Curated by ChEMBL
Fred Hutchinson Cancer Research Center
Curated by ChEMBL
Affinity DataIC50: 6.50E+4nMAssay Description:In vitro inhibition of sirtuin 2 was evaluated using yeast whole cell lysatesMore data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-2(Homo sapiens (Human))
Fred Hutchinson Cancer Research Center
Curated by ChEMBL
Fred Hutchinson Cancer Research Center
Curated by ChEMBL
Affinity DataIC50: 6.80E+4nMAssay Description:Inhibition of SIRT2 (unknown origin) by luminescence assayMore data for this Ligand-Target Pair
TargetNAD-dependent histone deacetylase SIR2(Saccharomyces cerevisiae)
Fred Hutchinson Cancer Research Center
Curated by ChEMBL
Fred Hutchinson Cancer Research Center
Curated by ChEMBL
Affinity DataIC50: 7.00E+4nMAssay Description:In vitro inhibition of sirtuin 2 was evaluated using yeast whole cell lysatesMore data for this Ligand-Target Pair
TargetNAD-dependent histone deacetylase SIR2(Saccharomyces cerevisiae)
Fred Hutchinson Cancer Research Center
Curated by ChEMBL
Fred Hutchinson Cancer Research Center
Curated by ChEMBL
Affinity DataIC50: 7.30E+4nMAssay Description:In vitro inhibition of sirtuin 2 was evaluated using yeast whole cell lysatesMore data for this Ligand-Target Pair
TargetNAD-dependent histone deacetylase SIR2(Saccharomyces cerevisiae)
Fred Hutchinson Cancer Research Center
Curated by ChEMBL
Fred Hutchinson Cancer Research Center
Curated by ChEMBL
Affinity DataIC50: 7.40E+4nMAssay Description:In vitro inhibition of sirtuin 2 was evaluated using yeast whole cell lysatesMore data for this Ligand-Target Pair
TargetNAD-dependent histone deacetylase SIR2(Saccharomyces cerevisiae)
Fred Hutchinson Cancer Research Center
Curated by ChEMBL
Fred Hutchinson Cancer Research Center
Curated by ChEMBL
Affinity DataIC50: 8.10E+4nMAssay Description:In vitro inhibition of sirtuin 2 was evaluated using yeast whole cell lysatesMore data for this Ligand-Target Pair
TargetNAD-dependent histone deacetylase SIR2(Saccharomyces cerevisiae)
Fred Hutchinson Cancer Research Center
Curated by ChEMBL
Fred Hutchinson Cancer Research Center
Curated by ChEMBL
Affinity DataIC50: 8.60E+4nMAssay Description:In vitro inhibition of sirtuin 2 was evaluated using yeast whole cell lysatesMore data for this Ligand-Target Pair
TargetNAD-dependent histone deacetylase SIR2(Saccharomyces cerevisiae)
Fred Hutchinson Cancer Research Center
Curated by ChEMBL
Fred Hutchinson Cancer Research Center
Curated by ChEMBL
Affinity DataIC50: 8.60E+4nMAssay Description:In vitro inhibition of sirtuin 2 was evaluated using yeast whole cell lysatesMore data for this Ligand-Target Pair
TargetNAD-dependent histone deacetylase SIR2(Saccharomyces cerevisiae)
Fred Hutchinson Cancer Research Center
Curated by ChEMBL
Fred Hutchinson Cancer Research Center
Curated by ChEMBL
Affinity DataIC50: 8.90E+4nMAssay Description:In vitro inhibition of sirtuin 2 was evaluated using yeast whole cell lysatesMore data for this Ligand-Target Pair
TargetNAD-dependent histone deacetylase SIR2(Saccharomyces cerevisiae)
Fred Hutchinson Cancer Research Center
Curated by ChEMBL
Fred Hutchinson Cancer Research Center
Curated by ChEMBL
Affinity DataIC50: 9.70E+4nMAssay Description:In vitro inhibition of sirtuin 2 was evaluated using yeast whole cell lysatesMore data for this Ligand-Target Pair
TargetNAD-dependent histone deacetylase SIR2(Saccharomyces cerevisiae)
Fred Hutchinson Cancer Research Center
Curated by ChEMBL
Fred Hutchinson Cancer Research Center
Curated by ChEMBL
Affinity DataIC50: 1.11E+5nMAssay Description:In vitro inhibition of sirtuin 2 was evaluated using yeast whole cell lysatesMore data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-3, mitochondrial(Homo sapiens (Human))
Fred Hutchinson Cancer Research Center
Curated by ChEMBL
Fred Hutchinson Cancer Research Center
Curated by ChEMBL
Affinity DataIC50: 1.22E+5nMAssay Description:Inhibition of SIRT3 (unknown origin) by luminescence assayMore data for this Ligand-Target Pair
TargetNAD-dependent histone deacetylase SIR2(Saccharomyces cerevisiae)
Fred Hutchinson Cancer Research Center
Curated by ChEMBL
Fred Hutchinson Cancer Research Center
Curated by ChEMBL
Affinity DataIC50: 1.22E+5nMAssay Description:In vitro inhibition of sirtuin 2 was evaluated using yeast whole cell lysatesMore data for this Ligand-Target Pair
TargetNAD-dependent histone deacetylase SIR2(Saccharomyces cerevisiae)
Fred Hutchinson Cancer Research Center
Curated by ChEMBL
Fred Hutchinson Cancer Research Center
Curated by ChEMBL
Affinity DataIC50: 1.25E+5nMAssay Description:In vitro inhibition of sirtuin 2 was evaluated using yeast whole cell lysatesMore data for this Ligand-Target Pair
TargetNAD-dependent histone deacetylase SIR2(Saccharomyces cerevisiae)
Fred Hutchinson Cancer Research Center
Curated by ChEMBL
Fred Hutchinson Cancer Research Center
Curated by ChEMBL
Affinity DataIC50: 1.25E+5nMAssay Description:In vitro inhibition of sirtuin 2 was evaluated using yeast whole cell lysatesMore data for this Ligand-Target Pair
TargetNAD-dependent histone deacetylase SIR2(Saccharomyces cerevisiae)
Fred Hutchinson Cancer Research Center
Curated by ChEMBL
Fred Hutchinson Cancer Research Center
Curated by ChEMBL
Affinity DataIC50: 1.28E+5nMAssay Description:In vitro inhibition of sirtuin 2 was evaluated using yeast whole cell lysatesMore data for this Ligand-Target Pair
TargetNAD-dependent histone deacetylase SIR2(Saccharomyces cerevisiae)
Fred Hutchinson Cancer Research Center
Curated by ChEMBL
Fred Hutchinson Cancer Research Center
Curated by ChEMBL
Affinity DataIC50: 1.31E+5nMAssay Description:In vitro inhibition of sirtuin 2 was evaluated using yeast whole cell lysatesMore data for this Ligand-Target Pair
TargetNAD-dependent histone deacetylase SIR2(Saccharomyces cerevisiae)
Fred Hutchinson Cancer Research Center
Curated by ChEMBL
Fred Hutchinson Cancer Research Center
Curated by ChEMBL
Affinity DataIC50: 1.34E+5nMAssay Description:In vitro inhibition of sirtuin 2 was evaluated using yeast whole cell lysatesMore data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-3, mitochondrial(Homo sapiens (Human))
Fred Hutchinson Cancer Research Center
Curated by ChEMBL
Fred Hutchinson Cancer Research Center
Curated by ChEMBL
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of SIRT3 (unknown origin) by luminescence assayMore data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-3, mitochondrial(Homo sapiens (Human))
Fred Hutchinson Cancer Research Center
Curated by ChEMBL
Fred Hutchinson Cancer Research Center
Curated by ChEMBL
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of SIRT3 (unknown origin) by luminescence assayMore data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-1(Homo sapiens (Human))
Fred Hutchinson Cancer Research Center
Curated by ChEMBL
Fred Hutchinson Cancer Research Center
Curated by ChEMBL
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of C-terminal His-6-tagged recombinant human SIRT1 expressed in Escherichia coli BL21(DE3) by luminescence assayMore data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-3, mitochondrial(Homo sapiens (Human))
Fred Hutchinson Cancer Research Center
Curated by ChEMBL
Fred Hutchinson Cancer Research Center
Curated by ChEMBL
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of SIRT3 (unknown origin) by luminescence assayMore data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-2(Homo sapiens (Human))
Fred Hutchinson Cancer Research Center
Curated by ChEMBL
Fred Hutchinson Cancer Research Center
Curated by ChEMBL
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of SIRT2 (unknown origin) by luminescence assayMore data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-2(Homo sapiens (Human))
Fred Hutchinson Cancer Research Center
Curated by ChEMBL
Fred Hutchinson Cancer Research Center
Curated by ChEMBL
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of SIRT2 (unknown origin) by luminescence assayMore data for this Ligand-Target Pair