TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Clinical Research Institute Of Montreal
Curated by ChEMBL
Clinical Research Institute Of Montreal
Curated by ChEMBL
Affinity DataKi: 0.0869nMAssay Description:Binding affinity was measured on opioid receptor kappa 1More data for this Ligand-Target Pair
TargetMu-type opioid receptor(GUINEA PIG)
Clinical Research Institute of Montreal
Curated by PDSP Ki Database
Clinical Research Institute of Montreal
Curated by PDSP Ki Database
TargetMu-type opioid receptor(GUINEA PIG)
Clinical Research Institute of Montreal
Curated by PDSP Ki Database
Clinical Research Institute of Montreal
Curated by PDSP Ki Database
TargetMu-type opioid receptor(GUINEA PIG)
Clinical Research Institute of Montreal
Curated by PDSP Ki Database
Clinical Research Institute of Montreal
Curated by PDSP Ki Database
TargetMu-type opioid receptor(GUINEA PIG)
Clinical Research Institute of Montreal
Curated by PDSP Ki Database
Clinical Research Institute of Montreal
Curated by PDSP Ki Database
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montreal
Curated by ChEMBL
Clinical Research Institute Of Montreal
Curated by ChEMBL
Affinity DataKi: 0.248nMAssay Description:Displacement of [3H]DSLET from delta opioid receptor in rat brain membraneMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Clinical Research Institute Of Montreal
Curated by ChEMBL
Clinical Research Institute Of Montreal
Curated by ChEMBL
Affinity DataKi: 0.322nMAssay Description:Binding affinity was measured on opioid receptor kappa 1More data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montreal
Curated by ChEMBL
Clinical Research Institute Of Montreal
Curated by ChEMBL
Affinity DataKi: 0.369nMAssay Description:Displacement of [3H]DSLET from delta opioid receptor in rat brain membrane after 2 hrsMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(GUINEA PIG)
Clinical Research Institute of Montreal
Curated by PDSP Ki Database
Clinical Research Institute of Montreal
Curated by PDSP Ki Database
Affinity DataKi: 0.435nMAssay Description:Binding affinity was measured on mu opioid receptorMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montr£Al
Curated by ChEMBL
Clinical Research Institute Of Montr£Al
Curated by ChEMBL
Affinity DataKi: 0.467nMAssay Description:Binding affinity was determined by displacement of [3H]- DSLET at Opioid receptor delta 1 in rat brain membrane homogenatesMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montreal
Curated by ChEMBL
Clinical Research Institute Of Montreal
Curated by ChEMBL
Affinity DataKi: 0.476nMAssay Description:Binding affinity was determined by displacement of [3H]- DAMGO at Opioid receptor mu 1 in rat brain membrane homogenatesMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montreal
Curated by ChEMBL
Clinical Research Institute Of Montreal
Curated by ChEMBL
Affinity DataKi: 0.501nMAssay Description:Displacement of [3H]DSLET from delta opioid receptor in rat brain membraneMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montreal
Curated by ChEMBL
Clinical Research Institute Of Montreal
Curated by ChEMBL
Affinity DataKi: 0.536nMAssay Description:Displacement of [3H]DSLET from delta opioid receptor in rat brain membraneMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montr£Al
Curated by ChEMBL
Clinical Research Institute Of Montr£Al
Curated by ChEMBL
Affinity DataKi: 0.550nMAssay Description:Displacement of [3H]DAMGO from rat brain mu opioid receptorMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montreal
Curated by ChEMBL
Clinical Research Institute Of Montreal
Curated by ChEMBL
Affinity DataKi: 0.605nMAssay Description:Displacement of [3H]DSLET from delta opioid receptor in rat brain membraneMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montr£Al
Curated by ChEMBL
Clinical Research Institute Of Montr£Al
Curated by ChEMBL
Affinity DataKi: 0.616nMAssay Description:Displacement of [3H]DAMGO from rat brain mu opioid receptorMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montreal
Curated by ChEMBL
Clinical Research Institute Of Montreal
Curated by ChEMBL
Affinity DataKi: 0.646nMAssay Description:Displacement of [3H]DSLET from delta opioid receptor in rat brain membraneMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(GUINEA PIG)
Clinical Research Institute of Montreal
Curated by PDSP Ki Database
Clinical Research Institute of Montreal
Curated by PDSP Ki Database
Affinity DataKi: 0.653nMAssay Description:Binding affinity was measured on mu opioid receptorMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montreal
Curated by ChEMBL
Clinical Research Institute Of Montreal
Curated by ChEMBL
Affinity DataKi: 0.783nMAssay Description:Displacement of [3H]DSLET from delta opioid receptor in rat brain membraneMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(GUINEA PIG)
Clinical Research Institute of Montreal
Curated by PDSP Ki Database
Clinical Research Institute of Montreal
Curated by PDSP Ki Database
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Clinical Research Institute Of Montreal
Curated by ChEMBL
Clinical Research Institute Of Montreal
Curated by ChEMBL
Affinity DataKi: 0.810nMAssay Description:Binding affinity was measured on opioid receptor kappa 1More data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montreal
Curated by ChEMBL
Clinical Research Institute Of Montreal
Curated by ChEMBL
Affinity DataKi: 0.822nMAssay Description:Displacement of [3H]DSLET from rat brain delta opioid receptorMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Clinical Research Institute Of Montreal
Curated by ChEMBL
Clinical Research Institute Of Montreal
Curated by ChEMBL
Affinity DataKi: 0.823nMAssay Description:Binding affinity was measured on opioid receptor kappa 1More data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montreal
Curated by ChEMBL
Clinical Research Institute Of Montreal
Curated by ChEMBL
Affinity DataKi: 0.825nMAssay Description:Displacement of [3H]DSLET from delta opioid receptor in rat brain membraneMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montreal
Curated by ChEMBL
Clinical Research Institute Of Montreal
Curated by ChEMBL
Affinity DataKi: 0.978nMAssay Description:Displacement of [3H]DSLET from delta opioid receptor in rat brain membrane after 2 hrsMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(GUINEA PIG)
Clinical Research Institute of Montreal
Curated by PDSP Ki Database
Clinical Research Institute of Montreal
Curated by PDSP Ki Database
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montreal
Curated by ChEMBL
Clinical Research Institute Of Montreal
Curated by ChEMBL
Affinity DataKi: 1.01nMAssay Description:Displacement of [3H]DSLET from delta opioid receptor in rat brain membrane after 2 hrsMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montr£Al
Curated by ChEMBL
Clinical Research Institute Of Montr£Al
Curated by ChEMBL
Affinity DataKi: 1.05nMAssay Description:Displacement of [3H]DAMGO from rat brain mu opioid receptorMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montr£Al
Curated by ChEMBL
Clinical Research Institute Of Montr£Al
Curated by ChEMBL
Affinity DataKi: 1.17nMAssay Description:Displacement of [3H]DAMGO from rat brain mu opioid receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.18nMAssay Description:Binding affinity was measured on delta opioid receptorMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montreal
Curated by ChEMBL
Clinical Research Institute Of Montreal
Curated by ChEMBL
Affinity DataKi: 1.22nMAssay Description:Displacement of [3H]DSLET from delta opioid receptor in rat brain membraneMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montreal
Curated by ChEMBL
Clinical Research Institute Of Montreal
Curated by ChEMBL
Affinity DataKi: 1.25nMAssay Description:Displacement of [3H]DSLET from rat brain delta opioid receptorMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montreal
Curated by ChEMBL
Clinical Research Institute Of Montreal
Curated by ChEMBL
Affinity DataKi: 1.54nMAssay Description:Displacement of [3H]DSLET from delta opioid receptor in rat brain membrane after 2 hrsMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montreal
Curated by ChEMBL
Clinical Research Institute Of Montreal
Curated by ChEMBL
Affinity DataKi: 1.61nMAssay Description:Displacement of [3H]DSLET from rat brain delta opioid receptorMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montreal
Curated by ChEMBL
Clinical Research Institute Of Montreal
Curated by ChEMBL
Affinity DataKi: 1.65nMAssay Description:Displacement of [3H]DSLET from delta opioid receptor in rat brain membrane after 2 hrsMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(GUINEA PIG)
Clinical Research Institute of Montreal
Curated by PDSP Ki Database
Clinical Research Institute of Montreal
Curated by PDSP Ki Database
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montr£Al
Curated by ChEMBL
Clinical Research Institute Of Montr£Al
Curated by ChEMBL
Affinity DataKi: 1.74nMAssay Description:Displacement of [3H]DAMGO from rat brain mu opioid receptorMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(GUINEA PIG)
Clinical Research Institute of Montreal
Curated by PDSP Ki Database
Clinical Research Institute of Montreal
Curated by PDSP Ki Database
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montreal
Curated by ChEMBL
Clinical Research Institute Of Montreal
Curated by ChEMBL
Affinity DataKi: 1.84nMAssay Description:Displacement of [3H]DSLET from delta opioid receptor in rat brain membrane after 2 hrsMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montreal
Curated by ChEMBL
Clinical Research Institute Of Montreal
Curated by ChEMBL
Affinity DataKi: 1.84nMAssay Description:Displacement of [3H]DSLET from delta opioid receptor in rat brain membraneMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montreal
Curated by ChEMBL
Clinical Research Institute Of Montreal
Curated by ChEMBL
Affinity DataKi: 1.92nMAssay Description:Displacement of [3H]DSLET from rat brain delta opioid receptorMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montreal
Curated by ChEMBL
Clinical Research Institute Of Montreal
Curated by ChEMBL
Affinity DataKi: 2nMAssay Description:Displacement of [3H]DSLET from delta opioid receptor in rat brain membraneMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(GUINEA PIG)
Clinical Research Institute of Montreal
Curated by PDSP Ki Database
Clinical Research Institute of Montreal
Curated by PDSP Ki Database
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montr£Al
Curated by ChEMBL
Clinical Research Institute Of Montr£Al
Curated by ChEMBL
Affinity DataKi: 2.27nMAssay Description:Displacement of [3H]DAMGO from rat brain mu opioid receptorMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montr£Al
Curated by ChEMBL
Clinical Research Institute Of Montr£Al
Curated by ChEMBL
Affinity DataKi: 2.34nMAssay Description:Displacement of [3H]DAMGO from rat brain mu opioid receptorMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montr£Al
Curated by ChEMBL
Clinical Research Institute Of Montr£Al
Curated by ChEMBL
Affinity DataKi: 2.40nMAssay Description:Displacement of [3H]DAMGO from rat brain mu opioid receptorMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Clinical Research Institute Of Montreal
Curated by ChEMBL
Clinical Research Institute Of Montreal
Curated by ChEMBL
Affinity DataKi: 2.47nMAssay Description:Binding affinity was measured on opioid receptor kappa 1More data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montreal
Curated by ChEMBL
Clinical Research Institute Of Montreal
Curated by ChEMBL
Affinity DataKi: 2.72nMAssay Description:Displacement of [3H]DSLET from delta opioid receptor in rat brain membrane after 2 hrsMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montreal
Curated by ChEMBL
Clinical Research Institute Of Montreal
Curated by ChEMBL
Affinity DataKi: 3.31nMAssay Description:Displacement of [3H]DSLET from delta opioid receptor in rat brain membraneMore data for this Ligand-Target Pair