Affinity DataKi: 0.0780nMAssay Description:Compound was tested for inhibition of squalene synthase in rat liver.More data for this Ligand-Target Pair
Affinity DataKi: 0.0780nMAssay Description:Inhibitory activity against squalene synthase in rat liver squalene synthase (RLSS) enzyme assayMore data for this Ligand-Target Pair
Affinity DataKi: 0.0780nMAssay Description:Competitive inhibitory activity of the compound was evaluated against squalene synthase in rat liver.More data for this Ligand-Target Pair
Affinity DataKi: 0.100nMAssay Description:Displacement of [3H]-N-methyl scopolamine from muscarinic acetylcholine M2 receptor expressed in CHO cell membraneMore data for this Ligand-Target Pair
Affinity DataKi: 0.120nMAssay Description:Displacement of [3H]-N-methyl scopolamine from muscarinic acetylcholine M1 receptor expressed in CHO cell membraneMore data for this Ligand-Target Pair
Affinity DataKi: 0.160nMAssay Description:Displacement of [3H]-N-methyl scopolamine from muscarinic acetylcholine M3 receptor expressed in CHO cell membraneMore data for this Ligand-Target Pair
Affinity DataKi: 0.300nMAssay Description:Binding affinity towards Dopamine receptor D1 in rat striatal tissue by [3H]-SCH- 23390 displacement.More data for this Ligand-Target Pair
Affinity DataKi: 0.400nMAssay Description:In vitro affinity of compound towards dopamine (D1) receptor was determined by measuring their ability to displace [3H]-SCH-23,390 from rat striatal ...More data for this Ligand-Target Pair
Affinity DataKi: 1.90nMAssay Description:Inhibition of [3H]-SCH-23,390 binding to rat striatal homogenate dopamine receptor D1More data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Binding affinity towards Dopamine receptor D1 in rat striatal tissue by [3H]-SCH- 23390 displacement.More data for this Ligand-Target Pair
Affinity DataKi: 2.10nMAssay Description:Binding affinity towards Dopamine receptor D1 in rat striatal tissue by [3H]-SCH- 23390 displacement.More data for this Ligand-Target Pair
Affinity DataKi: 3.30nMAssay Description:Inhibition of [3H]-SCH-23,390 binding to rat striatal homogenate dopamine receptor D1More data for this Ligand-Target Pair
Affinity DataKi: 3.30nMAssay Description:Binding affinity towards Dopamine receptor D1 in rat striatal tissue by [3H]-SCH- 23390 displacement.More data for this Ligand-Target Pair
Affinity DataKi: 3.70nMAssay Description:Binding affinity towards Dopamine receptor D1 in rat striatal tissue by [3H]-SCH- 23390 displacement.More data for this Ligand-Target Pair
Affinity DataKi: 5.10nMAssay Description:Binding affinity towards Dopamine receptor D1 in rat striatal tissue by [3H]-SCH- 23390 displacement.More data for this Ligand-Target Pair
Affinity DataKi: 5.70nMAssay Description:Binding affinity towards Dopamine receptor D1 in rat striatal tissue by [3H]-SCH- 23390 displacement.More data for this Ligand-Target Pair
Affinity DataKi: 7.10nMAssay Description:Inhibition of [3H]-SCH-23,390 binding to rat striatal homogenate dopamine receptor D1More data for this Ligand-Target Pair
Affinity DataKi: 7.60nMAssay Description:Binding affinity towards Dopamine receptor D1 in rat striatal tissue by [3H]-SCH- 23390 displacement.More data for this Ligand-Target Pair
Affinity DataKi: 8.70nMAssay Description:Binding affinity towards Dopamine receptor D1 in rat striatal tissue by [3H]-SCH- 23390 displacement.More data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Binding affinity towards Dopamine receptor D1 in rat striatal tissue by [3H]-SCH- 23390 displacement.More data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:Binding affinity towards Dopamine receptor D1 in rat striatal tissue by [3H]-SCH- 23390 displacement.More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Schering-Plough
Curated by PDSP Ki Database
Schering-Plough
Curated by PDSP Ki Database
Affinity DataKi: 23nMAssay Description:Binding affinity towards Dopamine receptor D1 in rat striatal tissue by [3H]-SCH- 23390 displacement.More data for this Ligand-Target Pair
Affinity DataKi: 24nMAssay Description:Inhibition of [3H]-SCH-23,390 binding to rat striatal homogenate dopamine receptor D1More data for this Ligand-Target Pair
Affinity DataKi: 24nMAssay Description:Binding affinity towards Dopamine receptor D1 in rat striatal tissue by [3H]-SCH- 23390 displacement.More data for this Ligand-Target Pair
Affinity DataKi: 33nMAssay Description:Binding affinity towards Dopamine receptor D1 in rat striatal tissue by [3H]-SCH- 23390 displacement.More data for this Ligand-Target Pair
Affinity DataKi: 46nMAssay Description:Binding affinity towards Dopamine receptor D1 in rat striatal tissue by [3H]-SCH- 23390 displacement.More data for this Ligand-Target Pair
Affinity DataKi: 50nMAssay Description:Inhibition of human SERT expressed in HEK293 cells assessed as reduction in [3]5-HT uptakeMore data for this Ligand-Target Pair
Affinity DataKi: 68nMAssay Description:In vitro affinity of compound towards dopamine (D1) receptor was determined by measuring their ability to displace [3H]-SCH-23,390 from rat striatal ...More data for this Ligand-Target Pair
Affinity DataKi: 73nMAssay Description:Inhibition of [3H]-SCH-23,390 binding to rat striatal homogenate dopamine receptor D1More data for this Ligand-Target Pair
Affinity DataKi: 100nMAssay Description:Binding affinity towards Dopamine receptor D1 in rat striatal tissue by [3H]-SCH- 23390 displacement.More data for this Ligand-Target Pair
Affinity DataKi: 265nMAssay Description:Binding affinity towards Dopamine receptor D2 in rat striatal tissue by [3H]-spiperone displacement.More data for this Ligand-Target Pair
Affinity DataKi: 284nMAssay Description:Binding affinity towards Dopamine receptor D2 in rat striatal tissue by [3H]-spiperone displacement.More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Schering-Plough
Curated by PDSP Ki Database
Schering-Plough
Curated by PDSP Ki Database
Affinity DataKi: 474nMAssay Description:Inhibition of [3H]-SCH-23,390 binding to rat striatal homogenate dopamine receptor D1More data for this Ligand-Target Pair
Affinity DataKi: 513nMAssay Description:Displacement of [3H]-spiperone from rat striatal homogenate dopamine receptor D2More data for this Ligand-Target Pair
Affinity DataKi: 514nMAssay Description:Displacement of [3H]-spiperone from rat striatal homogenate dopamine receptor D2More data for this Ligand-Target Pair
Affinity DataKi: 531nMAssay Description:Inhibition of [3H]-SCH-23,390 binding to rat striatal homogenate dopamine receptor D1More data for this Ligand-Target Pair
Affinity DataKi: 581nMAssay Description:Binding affinity towards Dopamine receptor D2 in rat striatal tissue by [3H]-spiperone displacement.More data for this Ligand-Target Pair
Affinity DataKi: 626nMAssay Description:Binding affinity towards Dopamine receptor D2 in rat striatal tissue by [3H]-spiperone displacement.More data for this Ligand-Target Pair
Affinity DataKi: 648nMAssay Description:In vitro affinity of compound towards Dopamine receptor D2 was determined by measuring their ability to displace [3H]-spiperone from rat striatal hom...More data for this Ligand-Target Pair
Affinity DataKi: 760nMAssay Description:Binding affinity towards Dopamine receptor D2 in rat striatal tissue by [3H]-spiperone displacement.More data for this Ligand-Target Pair
Affinity DataKi: 800nMAssay Description:Inhibition of human SERT expressed in HEK293 cells assessed as reduction in [3]5-HT uptakeMore data for this Ligand-Target Pair
Affinity DataKi: 898nMAssay Description:Inhibition of [3H]-SCH-23,390 binding to rat striatal homogenate dopamine receptor D1More data for this Ligand-Target Pair
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity towards Dopamine receptor D1 in rat striatal tissue by [3H]-SCH- 23390 displacement.More data for this Ligand-Target Pair