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Found 169 with Last Name = 'berk' and Initial = 'b'
TargetDopamine beta-hydroxylase(Bos taurus)
TBA

Curated by ChEMBL
LigandPNGBDBM50014978(1-(3,5-Difluoro-4-hydroxy-benzyl)-1,3-dihydro-imid...)
Affinity DataKi:  5.70nMpH: 4.5Assay Description:Binding affinity towards Dopamine beta hydroxylase using tyramine substrate at pH 4.5 in the absence of fumarateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTissue alpha-L-fucosidase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50065258((2S,3R,4S,5R)-2-Methyl-piperidine-3,4,5-triol | (2...)
Affinity DataKi:  29nMAssay Description:Inhibition constant against Alpha-FucosidaseMore data for this Ligand-Target Pair
TargetDopamine beta-hydroxylase(Bos taurus)
TBA

Curated by ChEMBL
LigandPNGBDBM50014983(1-(3,5-Difluoro-benzyl)-1,3-dihydro-imidazole-2-th...)
Affinity DataKi:  41nMpH: 4.5Assay Description:Binding affinity towards Dopamine beta hydroxylase using tyramine substrate at pH 4.5 in the absence of fumarateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDopamine beta-hydroxylase(Bos taurus)
TBA

Curated by ChEMBL
LigandPNGBDBM50014968(1-(4-Hydroxy-benzyl)-1,3-dihydro-imidazole-2-thion...)
Affinity DataKi:  55nMpH: 4.5Assay Description:Binding affinity towards Dopamine beta hydroxylase using tyramine substrate at pH 4.5 in the absence of fumarateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDopamine beta-hydroxylase(Bos taurus)
TBA

Curated by ChEMBL
LigandPNGBDBM50014968(1-(4-Hydroxy-benzyl)-1,3-dihydro-imidazole-2-thion...)
Affinity DataKi:  55nMpH: 4.5Assay Description:Compound was evaluated for the inhibition of Dopamine beta hydroxylase at pH 4.5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDopamine beta-hydroxylase(Bos taurus)
TBA

Curated by ChEMBL
LigandPNGBDBM50000439(5-Butyl-pyridine-2-carboxylic acid | 5-Butyl-pyrid...)
Affinity DataKi:  149nMAssay Description:Compound was evaluated for the inhibition of Dopamine beta hydroxylase at pH 4.5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDopamine beta-hydroxylase(Bos taurus)
TBA

Curated by ChEMBL
LigandPNGBDBM50000439(5-Butyl-pyridine-2-carboxylic acid | 5-Butyl-pyrid...)
Affinity DataKi:  149nMpH: 4.5Assay Description:Binding affinity towards Dopamine beta hydroxylase using tyramine substrate at pH 4.5 in the absence of fumarateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDopamine beta-hydroxylase(Bos taurus)
TBA

Curated by ChEMBL
LigandPNGBDBM50014968(1-(4-Hydroxy-benzyl)-1,3-dihydro-imidazole-2-thion...)
Affinity DataKi:  344nMpH: 6.6Assay Description:Compound was evaluated for the inhibition of Dopamine beta hydroxylase at pH 6.6More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTissue alpha-L-fucosidase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50403111(CHEMBL1289015)
Affinity DataKi:  4.00E+3nMAssay Description:Inhibition constant against Alpha-FucosidaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetTissue alpha-L-fucosidase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50285247((2R,3R,4R,5R)-2-Methyl-piperidine-3,4,5-triol | CH...)
Affinity DataKi:  1.10E+4nMAssay Description:Inhibition constant against Alpha-FucosidaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetTissue alpha-L-fucosidase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50065259((2R,3R,4R,5R)-2-(Hydroxymethyl)piperidine-3,4,5-tr...)
Affinity DataKi:  3.00E+4nMAssay Description:Inhibition constant against Alpha-FucosidaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetDopamine beta-hydroxylase(Bos taurus)
TBA

Curated by ChEMBL
LigandPNGBDBM50241361(CHEMBL1515 | METHIMAZOLE | US9138393, Methimazole ...)
Affinity DataKi:  4.50E+4nMpH: 4.5Assay Description:Compound was evaluated for the inhibition of Dopamine beta hydroxylase at pH 6.6More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTissue alpha-L-fucosidase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50403112(CHEMBL2115566)
Affinity DataKi:  5.00E+4nMAssay Description:Inhibition constant against Alpha-FucosidaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetTissue alpha-L-fucosidase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50403114(CHEMBL1337303)
Affinity DataKi:  5.30E+4nMAssay Description:Inhibition constant against Alpha-FucosidaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetTissue alpha-L-fucosidase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50104411((R)-6-Methyl-tetrahydro-thiopyran-2,3,4,5-tetraol ...)
Affinity DataKi:  8.00E+4nMAssay Description:Inhibition constant against Alpha-FucosidaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetTissue alpha-L-fucosidase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50280035(1-(4-Hydroxy-2-methyl-3,4-dihydro-2H-pyran-3-yl)-e...)
Affinity DataKi:  9.00E+4nMAssay Description:Inhibition constant against Alpha-FucosidaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetTissue alpha-L-fucosidase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50242419(6-Deoxy-L-galactose | 6-deoxy-L-galactopyranoseL-f...)
Affinity DataKi:  3.00E+5nMAssay Description:Inhibition constant against Alpha-FucosidaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetDopamine beta-hydroxylase(Bos taurus)
TBA

Curated by ChEMBL
LigandPNGBDBM50241361(CHEMBL1515 | METHIMAZOLE | US9138393, Methimazole ...)
Affinity DataKi:  7.16E+5nMpH: 6.6Assay Description:Compound was evaluated for the inhibition of Dopamine beta hydroxylase at pH 4.5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTissue alpha-L-fucosidase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50037814(2,5-Bis-hydroxymethyl-pyrrolidine-3,4-diol | CHEMB...)
Affinity DataKi:  9.10E+5nMAssay Description:Inhibition constant against Alpha-FucosidaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetTissue alpha-L-fucosidase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50403113(CHEMBL2115524)
Affinity DataKi:  1.00E+6nMAssay Description:Inhibition constant against Alpha-FucosidaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetTissue alpha-L-fucosidase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50280032((2R,3R,4R,5S)-2-Methyl-piperidine-3,4,5-triol | 1,...)
Affinity DataKi:  1.70E+6nMAssay Description:Inhibition constant against Alpha-FucosidaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetTissue alpha-L-fucosidase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50076963((3R,5R)-2-Hydroxymethyl-1-methyl-piperidine-3,4,5-...)
Affinity DataKi:  5.30E+6nMAssay Description:Inhibition constant against Alpha-FucosidaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetTissue alpha-L-fucosidase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50179480((2R,3S,4R,5S)-2-methylpiperidine-3,4,5-triol | CHE...)
Affinity DataKi:  7.90E+6nMAssay Description:Inhibition constant against Alpha-FucosidaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetTissue alpha-L-fucosidase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50280035(1-(4-Hydroxy-2-methyl-3,4-dihydro-2H-pyran-3-yl)-e...)
Affinity DataKi:  2.60E+7nMAssay Description:Inhibition constant against Alpha-FucosidaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetTissue alpha-L-fucosidase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50163440((2R,3S,4R,5S)-2-(hydroxymethyl)piperidine-3,4,5-tr...)
Affinity DataKi:  3.40E+7nMAssay Description:Inhibition constant against Alpha-FucosidaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetTissue alpha-L-fucosidase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50403109(CHEMBL2115527)
Affinity DataKi:  3.50E+7nMAssay Description:Inhibition constant against Alpha-Fucosidase; Uncompetitive inhibitionMore data for this Ligand-Target Pair
In DepthDetails Article
TargetTissue alpha-L-fucosidase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50403109(CHEMBL2115527)
Affinity DataKi:  3.50E+7nMAssay Description:Inhibition constant against Alpha-Fucosidase; Uncompetitive inhibitionMore data for this Ligand-Target Pair
In DepthDetails Article
TargetTissue alpha-L-fucosidase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50280039(2-Phenyl-3,4-dihydro-2H-pyran-3,4-diol | CHEMBL120...)
Affinity DataKi:  8.30E+7nMAssay Description:Inhibition constant against Alpha-Fucosidase; Uncompetitive inhibitionMore data for this Ligand-Target Pair
In DepthDetails Article
TargetTissue alpha-L-fucosidase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50280039(2-Phenyl-3,4-dihydro-2H-pyran-3,4-diol | CHEMBL120...)
Affinity DataKi:  8.30E+7nMAssay Description:Inhibition constant against Alpha-Fucosidase; Uncompetitive inhibitionMore data for this Ligand-Target Pair
In DepthDetails Article
TargetTissue alpha-L-fucosidase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50403110(CHEMBL179085)
Affinity DataKi:  9.00E+7nMAssay Description:Inhibition constant against Alpha-FucosidaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetTissue alpha-L-fucosidase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50280034(1-(4-Hydroxy-2-phenyl-3,4-dihydro-2H-pyran-3-yl)-e...)
Affinity DataKi: >1.00E+8nMAssay Description:Inhibition constant against Alpha-FucosidaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetTissue alpha-L-fucosidase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM18351((2R,3R,4R,5S)-2-(Hydroxymethyl)piperidine-3,4,5-tr...)
Affinity DataKi: >1.00E+8nMAssay Description:Inhibition constant against Alpha-FucosidaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetTissue alpha-L-fucosidase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50280038(3,5-Dimethyl-2-phenyl-3,4-dihydro-2H-pyran-4-ol | ...)
Affinity DataKi: >1.00E+8nMAssay Description:Inhibition constant against Alpha-FucosidaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetTissue alpha-L-fucosidase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50280037(3-Benzyloxy-2-phenyl-3,4-dihydro-2H-pyran-4-ol | C...)
Affinity DataKi: >1.00E+8nMAssay Description:Inhibition constant against Alpha-FucosidaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetTissue alpha-L-fucosidase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50280036(2-Phenyl-3,4-dihydro-2H-pyran-4-ol | CHEMBL333105)
Affinity DataKi: >1.00E+8nMAssay Description:Inhibition constant against Alpha-FucosidaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetTissue alpha-L-fucosidase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50280038(3,5-Dimethyl-2-phenyl-3,4-dihydro-2H-pyran-4-ol | ...)
Affinity DataKi: >1.00E+8nMAssay Description:Inhibition constant against Alpha-FucosidaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetAromatase(Homo sapiens (Human))
Istanbul Medipol University

Curated by ChEMBL
LigandPNGBDBM50460601(CHEMBL4227385)
Affinity DataIC50:  0.420nMAssay Description:Inhibition of aromatase (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Istanbul Medipol University

Curated by ChEMBL
LigandPNGBDBM10015(2-[3-(1-cyano-1-methylethyl)-5-(1H-1,2,4-triazol-1...)
Affinity DataIC50:  1.5nMAssay Description:Inhibition of aromatase (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetAromatase(Homo sapiens (Human))
Istanbul Medipol University

Curated by ChEMBL
LigandPNGBDBM50460600(CHEMBL118266)
Affinity DataIC50:  4nMAssay Description:Inhibition of aromatase (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCation-independent mannose-6-phosphate receptor(Homo sapiens (Human))
University Of Nebraska

Curated by ChEMBL
LigandPNGBDBM50373067(CHEMBL1162089)
Affinity DataIC50:  90nMAssay Description:Displacement of pentamannosyl phosphate bovine serum albumin from M6P/IGF2RMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Istanbul Medipol University

Curated by ChEMBL
LigandPNGBDBM50460621(CHEMBL4228753)
Affinity DataIC50:  177nMAssay Description:Inhibition of aromatase (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Istanbul Medipol University

Curated by ChEMBL
LigandPNGBDBM50361943(CHEMBL1939366)
Affinity DataIC50:  240nMAssay Description:Inhibition of aromatase (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4B(Homo sapiens (Human))
Istanbul Medipol University

Curated by ChEMBL
LigandPNGBDBM14361((R,S)-Rolipram | 4-(3-cyclopentyloxy-4-methoxy-phe...)
Affinity DataIC50:  320nMAssay Description:Inhibition of recombinant human PDE4B using 5'-cGMP as substrate measured after 90 mins by colorimetric assayMore data for this Ligand-Target Pair
TargetDopamine beta-hydroxylase(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50000439(5-Butyl-pyridine-2-carboxylic acid | 5-Butyl-pyrid...)
Affinity DataIC50:  700nMAssay Description:Inhibition of Dopamine beta hydroxylase in spontaneously hypertensive rats; Value ranges from 0.4-1.1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Istanbul Medipol University

Curated by ChEMBL
LigandPNGBDBM50460610(CHEMBL4227458)
Affinity DataIC50:  935nMAssay Description:Inhibition of aromatase (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Istanbul Medipol University

Curated by ChEMBL
LigandPNGBDBM8610(1-[4-(4-{[(2R,4S)-2-(2,4-dichlorophenyl)-2-(1H-imi...)
Affinity DataIC50:  951nMAssay Description:Inhibition of aromatase (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4B(Homo sapiens (Human))
Istanbul Medipol University

Curated by ChEMBL
LigandPNGBDBM50557181(CHEMBL4765150)
Affinity DataIC50:  970nMAssay Description:Inhibition of recombinant human PDE4B using 5'-cGMP as substrate measured after 90 mins by colorimetric assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Istanbul Medipol University

Curated by ChEMBL
LigandPNGBDBM50460613(CHEMBL4228244)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of aromatase (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Istanbul Medipol University

Curated by ChEMBL
LigandPNGBDBM50460602(CHEMBL4225521)
Affinity DataIC50:  1.09E+3nMAssay Description:Inhibition of aromatase (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Istanbul Medipol University

Curated by ChEMBL
LigandPNGBDBM50460607(CHEMBL4224728)
Affinity DataIC50:  1.18E+3nMAssay Description:Inhibition of aromatase (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
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