Compile Data Set for Download or QSAR
maximum 50k data
Found 60 with Last Name = 'berkman' and Initial = 'ce'
TargetGamma-glutamyl hydrolase(Homo sapiens (Human))
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50070541((2S)-2-{[hydroxy(methyl)phosphoryl]amino}pentanedi...)
Affinity DataKi:  9.30E+5nMAssay Description:Compound was tested for inhibitory potency against gamma-Glutamyl Hydrolase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGamma-glutamyl hydrolase(Homo sapiens (Human))
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50070540((2S)-2-{[hydroxy(phenyl)phosphoryl]amino}pentanedi...)
Affinity DataKi:  9.50E+5nMAssay Description:Compound was tested for inhibitory potency against gamma-Glutamyl Hydrolase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate carboxypeptidase 2(Homo sapiens (Human))
Washington State University

Curated by ChEMBL
LigandPNGBDBM50358646(CHEMBL1921899)
Affinity DataIC50:  0.350nMAssay Description:Inhibition of PSMA using N-[4-(phenylazo)-benzoyl]-glutamyl-gamma-glutamic acid as substrate after 15 mins by HPLC analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate carboxypeptidase 2(Homo sapiens (Human))
Washington State University

Curated by ChEMBL
LigandPNGBDBM50358645(CHEMBL1921898)
Affinity DataIC50:  0.410nMAssay Description:Inhibition of PSMA using N-[4-(phenylazo)-benzoyl]-glutamyl-gamma-glutamic acid as substrate after 15 mins by HPLC analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate carboxypeptidase 2(Homo sapiens (Human))
Washington State University

Curated by ChEMBL
LigandPNGBDBM50331102(2-{[2-(4-Amino-4-carboxy-butyrylamino)-2-carboxyet...)
Affinity DataIC50:  0.550nMAssay Description:Inhibition of PSMA in human LNCaP cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate carboxypeptidase 2(Homo sapiens (Human))
Washington State University

Curated by ChEMBL
LigandPNGBDBM50222546(CHEMBL241779 | tetralithium (2S)-2-(phosphonatoami...)
Affinity DataIC50:  0.860nMAssay Description:Inhibition of PSMAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate carboxypeptidase 2(Homo sapiens (Human))
Washington State University

Curated by ChEMBL
LigandPNGBDBM50358647(CHEMBL1921900)
Affinity DataIC50:  1.93nMAssay Description:Inhibition of PSMA using N-[4-(phenylazo)-benzoyl]-glutamyl-gamma-glutamic acid as substrate after 15 mins by HPLC analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate carboxypeptidase 2(Homo sapiens (Human))
Washington State University

Curated by ChEMBL
LigandPNGBDBM50222549((S)-2-phosphonoamino-pentanedioic acid | CHEMBL238...)
Affinity DataIC50:  2.30nMAssay Description:Inhibition of PSMAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate carboxypeptidase 2(Homo sapiens (Human))
Washington State University

Curated by ChEMBL
LigandPNGBDBM50358644(CHEMBL1921897)
Affinity DataIC50:  14nMAssay Description:Inhibition of PSMA using N-[4-(phenylazo)-benzoyl]-glutamyl-gamma-glutamic acid as substrate after 15 mins by HPLC analysisMore data for this Ligand-Target Pair
TargetGlutamate carboxypeptidase 2(Homo sapiens (Human))
Washington State University

Curated by ChEMBL
LigandPNGBDBM50222551(CHEMBL241780 | tetralithium (2S)-2-(phosphonatooxy...)
Affinity DataIC50:  15nMAssay Description:Inhibition of PSMAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate carboxypeptidase 2(Homo sapiens (Human))
Washington State University

Curated by ChEMBL
LigandPNGBDBM50222550(CHEMBL239882 | tetrapotassium (3S,8S)-6-oxido-1-ox...)
Affinity DataIC50:  35nMAssay Description:Inhibition of PSMAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate carboxypeptidase 2(Homo sapiens (Human))
Washington State University

Curated by ChEMBL
LigandPNGBDBM50222542(CHEMBL238831 | tetrapotassium (3S,8S)-2-methyl-6-o...)
Affinity DataIC50:  55nMAssay Description:Inhibition of PSMAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate carboxypeptidase 2(Homo sapiens (Human))
Washington State University

Curated by ChEMBL
LigandPNGBDBM50372201(CHEMBL270610)
Affinity DataIC50:  125nMAssay Description:Inhibition of human PSMAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate carboxypeptidase 2(Homo sapiens (Human))
Washington State University

Curated by ChEMBL
LigandPNGBDBM50372204(CHEMBL402223)
Affinity DataIC50:  140nMAssay Description:Inhibition of human PSMAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate carboxypeptidase 2(Homo sapiens (Human))
Washington State University

Curated by ChEMBL
LigandPNGBDBM50331103((S)-2-carboxy-2-((S)-4-carboxy-4-(6-(2-(5-(3-ethyl...)
Affinity DataIC50:  144nMAssay Description:Inhibition of PSMA in human LNCaP cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate carboxypeptidase 2(Homo sapiens (Human))
Washington State University

Curated by ChEMBL
LigandPNGBDBM50222545(CHEMBL394011 | tripotassium (2S)-2-{[(4-phenylbuto...)
Affinity DataIC50:  180nMAssay Description:Inhibition of human PSMAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate carboxypeptidase 2(Homo sapiens (Human))
Washington State University

Curated by ChEMBL
LigandPNGBDBM50222545(CHEMBL394011 | tripotassium (2S)-2-{[(4-phenylbuto...)
Affinity DataIC50:  180nMAssay Description:Inhibition of PSMAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate carboxypeptidase 2(Homo sapiens (Human))
Washington State University

Curated by ChEMBL
LigandPNGBDBM50222552(CHEMBL239041 | tripotassium (2S)-2-[({2-[benzoyl(m...)
Affinity DataIC50:  280nMAssay Description:Inhibition of PSMAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate carboxypeptidase 2(Homo sapiens (Human))
Washington State University

Curated by ChEMBL
LigandPNGBDBM50088185(CHEMBL3427435)
Affinity DataIC50:  400nMAssay Description:Inhibition of PSMA (unknown origin) incubated for 15 mins using PABGgG substrate by HPLC methodMore data for this Ligand-Target Pair
TargetGlutamate carboxypeptidase 2(Homo sapiens (Human))
Washington State University

Curated by ChEMBL
LigandPNGBDBM50372203(CHEMBL270594)
Affinity DataIC50:  435nMAssay Description:Inhibition of human PSMAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate carboxypeptidase 2(Homo sapiens (Human))
Washington State University

Curated by ChEMBL
LigandPNGBDBM50372205(CHEMBL270824)
Affinity DataIC50:  438nMAssay Description:Inhibition of human PSMAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate carboxypeptidase 2(Homo sapiens (Human))
Washington State University

Curated by ChEMBL
LigandPNGBDBM50372202(CHEMBL437209)
Affinity DataIC50:  569nMAssay Description:Inhibition of human PSMAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate carboxypeptidase 2(Homo sapiens (Human))
Washington State University

Curated by ChEMBL
LigandPNGBDBM50372206(CHEMBL402033)
Affinity DataIC50:  572nMAssay Description:Inhibition of human PSMAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInsulin-like growth factor 1 receptor(Homo sapiens (Human))
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50212958(4-(4-(3,4-dihydroxyphenyl)butyl)benzene-1,2-diol |...)
Affinity DataIC50:  600nMAssay Description:Inhibition of IGF1RMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate carboxypeptidase 2(Homo sapiens (Human))
Washington State University

Curated by ChEMBL
LigandPNGBDBM50222543(CHEMBL239465 | tetrapotassium (3R,8S)-6-oxido-1-ox...)
Affinity DataIC50:  700nMAssay Description:Inhibition of PSMAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate carboxypeptidase 2(Homo sapiens (Human))
Washington State University

Curated by ChEMBL
LigandPNGBDBM50222548(CHEMBL391840 | tetrapotassium (2S)-2-{[(2-carboxyl...)
Affinity DataIC50:  790nMAssay Description:Inhibition of PSMAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInsulin-like growth factor 1 receptor(Homo sapiens (Human))
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50212959(4-(4-p-tolylbutyl)benzene-1,2-diol | CHEMBL245942)
Affinity DataIC50:  800nMAssay Description:Inhibition of IGF1RMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInsulin-like growth factor 1 receptor(Homo sapiens (Human))
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50212960(4-(4-(4-chlorophenyl)butyl)benzene-1,2-diol | CHEM...)
Affinity DataIC50:  800nMAssay Description:Inhibition of IGF1RMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInsulin-like growth factor 1 receptor(Homo sapiens (Human))
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50212956(4-(4-phenylbutyl)benzene-1,2-diol | CHEMBL442420)
Affinity DataIC50:  800nMAssay Description:Inhibition of IGF1RMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInsulin-like growth factor 1 receptor(Homo sapiens (Human))
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM22372(4-[(2R,3S)-4-(3,4-dihydroxyphenyl)-2,3-dimethylbut...)
Affinity DataIC50:  900nMAssay Description:Inhibition of IGF1RMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInsulin-like growth factor 1 receptor(Homo sapiens (Human))
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50212961(5-phenyl-5,6,7,8-tetrahydronaphthalene-2,3-diol | ...)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of IGF1RMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInsulin-like growth factor 1 receptor(Homo sapiens (Human))
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50212955(4-(4-(4-hydroxyphenyl)butyl)benzene-1,2-diol | CHE...)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of IGF1RMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInsulin-like growth factor 1 receptor(Homo sapiens (Human))
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50212957(4-(4-(3,4-dichlorophenyl)butyl)benzene-1,2-diol | ...)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of IGF1RMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInsulin-like growth factor 1 receptor(Homo sapiens (Human))
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50212962(4-(4-(4-methoxyphenyl)butyl)benzene-1,2-diol | CHE...)
Affinity DataIC50:  1.10E+3nMAssay Description:Inhibition of IGF1RMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate carboxypeptidase 2(Homo sapiens (Human))
Washington State University

Curated by ChEMBL
LigandPNGBDBM50088192(CHEMBL3427442)
Affinity DataIC50:  1.30E+3nMAssay Description:Inhibition of PSMA (unknown origin) incubated for 15 mins using PABGgG substrate by HPLC methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate carboxypeptidase 2(Homo sapiens (Human))
Washington State University

Curated by ChEMBL
LigandPNGBDBM50088182(CHEMBL3427434)
Affinity DataIC50:  1.30E+3nMAssay Description:Inhibition of PSMA (unknown origin) incubated for 15 mins using PABGgG substrate by HPLC methodMore data for this Ligand-Target Pair
TargetGlutamate carboxypeptidase 2(Homo sapiens (Human))
Washington State University

Curated by ChEMBL
LigandPNGBDBM50222547(CHEMBL400842 | tripotassium (2S)-2-({[2-(benzoylam...)
Affinity DataIC50:  1.80E+3nMAssay Description:Inhibition of PSMAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate carboxypeptidase 2(Homo sapiens (Human))
Washington State University

Curated by ChEMBL
LigandPNGBDBM50088190(CHEMBL3427440)
Affinity DataIC50:  2.60E+3nMAssay Description:Inhibition of PSMA (unknown origin) incubated for 15 mins using PABGgG substrate by HPLC methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate carboxypeptidase 2(Homo sapiens (Human))
Washington State University

Curated by ChEMBL
LigandPNGBDBM50088191(CHEMBL3427441)
Affinity DataIC50:  3.00E+3nMAssay Description:Inhibition of PSMA (unknown origin) incubated for 15 mins using PABGgG substrate by HPLC methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyunsaturated fatty acid lipoxygenase ALOX15(Homo sapiens (Human))
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM22372(4-[(2R,3S)-4-(3,4-dihydroxyphenyl)-2,3-dimethylbut...)
Affinity DataIC50:  3.80E+3nMAssay Description:Inhibition of 15 LOXMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyunsaturated fatty acid lipoxygenase ALOX15(Homo sapiens (Human))
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50212958(4-(4-(3,4-dihydroxyphenyl)butyl)benzene-1,2-diol |...)
Affinity DataIC50:  3.90E+3nMAssay Description:Inhibition of 15 LOXMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate carboxypeptidase 2(Homo sapiens (Human))
Washington State University

Curated by ChEMBL
LigandPNGBDBM50222544(CHEMBL391138 | tetrapotassium (2S)-2-{[(3-oxido-3-...)
Affinity DataIC50:  4.10E+3nMAssay Description:Inhibition of PSMAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate carboxypeptidase 2(Homo sapiens (Human))
Washington State University

Curated by ChEMBL
LigandPNGBDBM50331104(6-(2-(-5-(3-ethyl-1,1-dimethyl-6,8-disulfo-1H-benz...)
Affinity DataIC50:  6.10E+3nMAssay Description:Inhibition of PSMA in human LNCaP cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyunsaturated fatty acid lipoxygenase ALOX15(Homo sapiens (Human))
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50212956(4-(4-phenylbutyl)benzene-1,2-diol | CHEMBL442420)
Affinity DataIC50:  7.30E+3nMAssay Description:Inhibition of 15 LOXMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyunsaturated fatty acid lipoxygenase ALOX15(Homo sapiens (Human))
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50212955(4-(4-(4-hydroxyphenyl)butyl)benzene-1,2-diol | CHE...)
Affinity DataIC50:  9.40E+3nMAssay Description:Inhibition of 15 LOXMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate carboxypeptidase 2(Homo sapiens (Human))
Washington State University

Curated by ChEMBL
LigandPNGBDBM50088193(CHEMBL3427443)
Affinity DataIC50:  1.10E+4nMAssay Description:Inhibition of PSMA (unknown origin) incubated for 15 mins using PABGgG substrate by HPLC methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyunsaturated fatty acid lipoxygenase ALOX15(Homo sapiens (Human))
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50212962(4-(4-(4-methoxyphenyl)butyl)benzene-1,2-diol | CHE...)
Affinity DataIC50:  1.50E+4nMAssay Description:Inhibition of 15 LOXMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyunsaturated fatty acid lipoxygenase ALOX15(Homo sapiens (Human))
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50212960(4-(4-(4-chlorophenyl)butyl)benzene-1,2-diol | CHEM...)
Affinity DataIC50:  1.50E+4nMAssay Description:Inhibition of 15 LOXMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate carboxypeptidase 2(Homo sapiens (Human))
Washington State University

Curated by ChEMBL
LigandPNGBDBM50088183(CHEMBL3427433)
Affinity DataIC50:  1.90E+4nMAssay Description:Inhibition of PSMA (unknown origin) incubated for 15 mins using PABGgG substrate by HPLC methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyunsaturated fatty acid lipoxygenase ALOX15(Homo sapiens (Human))
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50212959(4-(4-p-tolylbutyl)benzene-1,2-diol | CHEMBL245942)
Affinity DataIC50:  2.16E+4nMAssay Description:Inhibition of 15 LOXMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Displayed 1 to 50 (of 60 total ) | Next | Last >>
Jump to: