Affinity DataKi: 2nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from mouse histamine H3 receptor after 30 mins by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from mouse histamine H3 receptor after 30 mins by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 3nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from mouse histamine H3 receptor after 30 mins by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 3nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from mouse histamine H3 receptor after 30 mins by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 3nMAssay Description:Compound was evaluated for its binding affinity against Histamine H3 receptor of guinea pig brain membraneMore data for this Ligand-Target Pair
Affinity DataKi: 3nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from mouse histamine H3 receptor after 30 mins by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:Compound was evaluated for its binding affinity against Histamine H3 receptor of guinea pig brain membraneMore data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from mouse histamine H3 receptor after 30 mins by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from mouse histamine H3 receptor after 30 mins by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from mouse histamine H3 receptor after 30 mins by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from mouse histamine H3 receptor after 30 mins by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 5nMAssay Description:Compound was evaluated for its binding affinity against Histamine H3 receptor of guinea pig brain membraneMore data for this Ligand-Target Pair
Affinity DataKi: 5nMAssay Description:Compound was evaluated for its binding affinity against Histamine H3 receptor of guinea pig brain membraneMore data for this Ligand-Target Pair
Affinity DataKi: 6nMAssay Description:Compound was evaluated for its binding affinity against Histamine H3 receptor of guinea pig brain membraneMore data for this Ligand-Target Pair
Affinity DataKi: 7nMAssay Description:Compound was evaluated for its binding affinity against Histamine H3 receptor of guinea pig brain membraneMore data for this Ligand-Target Pair
Affinity DataKi: 7nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from mouse histamine H3 receptor after 30 mins by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 7nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from mouse histamine H3 receptor after 30 mins by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 7nMAssay Description:Compound was evaluated for its binding affinity against Histamine H3 receptor of guinea pig brain membraneMore data for this Ligand-Target Pair
Affinity DataKi: 9nMAssay Description:Compound was evaluated for its binding affinity against Histamine H3 receptor of guinea pig brain membraneMore data for this Ligand-Target Pair
Affinity DataKi: 15nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from mouse histamine H3 receptor after 30 mins by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 16nMAssay Description:Compound was evaluated for its binding affinity against Histamine H3 receptor of guinea pig brain membraneMore data for this Ligand-Target Pair
Affinity DataKi: 16nMAssay Description:Compound was evaluated for its binding affinity against Histamine H3 receptor of guinea pig brain membraneMore data for this Ligand-Target Pair
Affinity DataKi: 18nMAssay Description:Compound was evaluated for its binding affinity against Histamine H3 receptor of guinea pig brain membraneMore data for this Ligand-Target Pair
Affinity DataKi: 18nMAssay Description:Compound was evaluated for its binding affinity against Histamine H3 receptor of guinea pig brain membraneMore data for this Ligand-Target Pair
Affinity DataKi: 21nMAssay Description:Compound was evaluated for its binding affinity against Histamine H3 receptor of guinea pig brain membraneMore data for this Ligand-Target Pair
Affinity DataKi: 22nMAssay Description:Compound was evaluated for its binding affinity against Histamine H3 receptor of guinea pig brain membraneMore data for this Ligand-Target Pair
Affinity DataKi: 25nMAssay Description:Compound was evaluated for its binding affinity against Histamine H3 receptor of guinea pig brain membraneMore data for this Ligand-Target Pair
Affinity DataKi: 26nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from mouse histamine H3 receptor after 30 mins by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 32nMAssay Description:Compound was evaluated for its binding affinity against Histamine H3 receptor of guinea pig brain membraneMore data for this Ligand-Target Pair
Affinity DataKi: 37nMAssay Description:Compound was evaluated for its binding affinity against Histamine H3 receptor of guinea pig brain membraneMore data for this Ligand-Target Pair
Affinity DataKi: 44nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from mouse histamine H3 receptor after 30 mins by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 46nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from mouse histamine H3 receptor after 30 mins by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 51nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from mouse histamine H3 receptor after 30 mins by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 70nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from mouse histamine H3 receptor after 30 mins by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 90nMAssay Description:Compound was evaluated for its binding affinity against Histamine H3 receptor of guinea pig brain membraneMore data for this Ligand-Target Pair
Affinity DataKi: 115nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from mouse histamine H3 receptor after 30 mins by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 120nMAssay Description:Compound was evaluated for its binding affinity against Histamine H3 receptor of guinea pig brain membraneMore data for this Ligand-Target Pair
Affinity DataKi: 270nMAssay Description:Compound was evaluated for its binding affinity against Histamine H3 receptor of guinea pig brain membraneMore data for this Ligand-Target Pair
Affinity DataKi: 370nMAssay Description:Compound was evaluated for its binding affinity against Histamine H3 receptor of guinea pig brain membraneMore data for this Ligand-Target Pair
Affinity DataKi: 430nMAssay Description:Compound was evaluated for its binding affinity against Histamine H3 receptor of guinea pig brain membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 300nMAssay Description:Inhibition of CYP2D6 in human liver microsomesMore data for this Ligand-Target Pair
Affinity DataIC50: 4.00E+3nMAssay Description:Inhibition of CYP2C9 in human liver microsomesMore data for this Ligand-Target Pair
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of CYP2D6 in human liver microsomesMore data for this Ligand-Target Pair
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of CYP2C9 in human liver microsomesMore data for this Ligand-Target Pair
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of CYP2C9 in human liver microsomesMore data for this Ligand-Target Pair
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of CYP2C9 in human liver microsomesMore data for this Ligand-Target Pair
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of CYP2C9 in human liver microsomesMore data for this Ligand-Target Pair
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of CYP2C9 in human liver microsomesMore data for this Ligand-Target Pair
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of CYP2C9 in human liver microsomesMore data for this Ligand-Target Pair
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of CYP2C9 in human liver microsomesMore data for this Ligand-Target Pair