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Found 94 with Last Name = 'bernad' and Initial = 'n'
TargetGastrin-releasing peptide receptor(RAT)
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50005601(CHEMBL2369819)
Affinity DataKi: >0nMAssay Description:In vitro binding affinity against bombesin / GRP receptors on rat pancreatic acini.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(RAT)
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50408923(CHEMBL2114155)
Affinity DataKi: >0nMAssay Description:In vitro binding affinity against bombesin / GRP receptors on rat pancreatic acini.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(RAT)
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50089280(CHEMBL437655 | JMV 1535)
Affinity DataKi:  1.70nMAssay Description:In vitro binding affinity against bombesin / GRP receptors on rat pancreatic acini.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(RAT)
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50089284(CHEMBL265856 | JMV 1803)
Affinity DataKi:  1.80nMAssay Description:In vitro binding affinity against bombesin / GRP receptors on rat pancreatic acini.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(RAT)
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50089285(CHEMBL415110 | JMV 1799)
Affinity DataKi:  3.10nMAssay Description:In vitro binding affinity against bombesin / GRP receptors on rat pancreatic acini.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(RAT)
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50089282((D)Phe-Gln-Trp-Ala-Val-Gly-His-Leu-Leu-NH2 | CHEMB...)
Affinity DataKi:  3.20nMAssay Description:In vitro binding affinity against bombesin / GRP receptors on rat pancreatic acini.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(RAT)
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50089281(CHEMBL386480 | JMV 1802)
Affinity DataKi:  3.80nMAssay Description:In vitro binding affinity against bombesin / GRP receptors on rat pancreatic acini.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(RAT)
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50089291(CHEMBL415021 | JMV 1813)
Affinity DataKi:  5.20nMAssay Description:In vitro binding affinity against bombesin / GRP receptors on rat pancreatic acini.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(RAT)
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50089278(CHEMBL411016 | JMV 1801)
Affinity DataKi:  9nMAssay Description:In vitro binding affinity against bombesin / GRP receptors on rat pancreatic acini.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(RAT)
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50089279(CHEMBL406013 | JMV 1719)
Affinity DataKi:  13nMAssay Description:In vitro binding affinity against bombesin / GRP receptors on rat pancreatic acini.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(RAT)
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50089286(CHEMBL407022 | JMV 1693)
Affinity DataKi:  127nMAssay Description:In vitro binding affinity against bombesin / GRP receptors on rat pancreatic acini.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(RAT)
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50408922(CHEMBL2115179)
Affinity DataKi:  225nMAssay Description:In vitro binding affinity against bombesin / GRP receptors on rat pancreatic acini.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(RAT)
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50089288(Bombesin analogues | CHEMBL415022)
Affinity DataKi:  300nMAssay Description:In vitro binding affinity against bombesin / GRP receptors on rat pancreatic acini.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(RAT)
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50089292(Bombesin analogues | CHEMBL439440)
Affinity DataKi:  500nMAssay Description:In vitro binding affinity against bombesin / GRP receptors on rat pancreatic acini.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(RAT)
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50089290(Bombesin analogues | CHEMBL413938)
Affinity DataKi:  650nMAssay Description:In vitro binding affinity against bombesin / GRP receptors on rat pancreatic acini.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(RAT)
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50089293(Bombesin analogues | CHEMBL407481)
Affinity DataKi:  2.25E+3nMAssay Description:In vitro binding affinity against bombesin / GRP receptors on rat pancreatic acini.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(RAT)
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50089289(Bombesin analogues | CHEMBL384241)
Affinity DataKi: >1.00E+6nMAssay Description:In vitro binding affinity against bombesin / GRP receptors on rat pancreatic acini.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(RAT)
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50089287(Bombesin analogues | CHEMBL384242)
Affinity DataKi: >1.00E+6nMAssay Description:In vitro binding affinity against bombesin / GRP receptors on rat pancreatic acini.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(MOUSE)
Ccipe-Faculte De Pharmacie

Curated by ChEMBL
LigandPNGBDBM50451028(CHEMBL2062146 | PD-149164)
Affinity DataIC50:  0.0830nMAssay Description:Binding affinity towards Cholecystokinin type B receptor in mouse cortex membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Ep Cnrs 51

Curated by ChEMBL
LigandPNGBDBM50016425((S)-3-{(S)-2-[(S)-2-(2-{(S)-2-[(S)-2-tert-Butoxyca...)
Affinity DataIC50:  0.200nMAssay Description:Inhibition of [125I]-BH-CCK- binding to cholecystokinin type B receptor from jurkat TcellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Ep Cnrs 51

Curated by ChEMBL
LigandPNGBDBM50016425((S)-3-{(S)-2-[(S)-2-(2-{(S)-2-[(S)-2-tert-Butoxyca...)
Affinity DataIC50:  0.290nMAssay Description:Inhibition of [125I]-BH-CCK- binding to cholecystokinin type B receptor from guinea pig brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Ep Cnrs 51

Curated by ChEMBL
LigandPNGBDBM50016425((S)-3-{(S)-2-[(S)-2-(2-{(S)-2-[(S)-2-tert-Butoxyca...)
Affinity DataIC50:  0.290nMAssay Description:In vitro binding affinity against Cholecystokinin type B receptor in guinea pig brain membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetPancreatic alpha-amylase(Homo sapiens (Human))
Ep Cnrs 51

Curated by ChEMBL
LigandPNGBDBM50033631(2-{2-[2-(2-{2-[2-tert-Butoxycarbonylamino-3-(4-sul...)
Affinity DataIC50:  0.300nMAssay Description:Tested in vitro for inhibition of amylase release from rat pancreatic aciniMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(MOUSE)
Ccipe-Faculte De Pharmacie

Curated by ChEMBL
LigandPNGBDBM21147((3S)-3-[(2S)-2-[(2S)-2-{2-[(2S)-2-[(2S)-2-[(3S)-3-...)
Affinity DataIC50:  0.300nMAssay Description:Binding affinity towards Cholecystokinin type B receptor in mouse cortex membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPancreatic alpha-amylase(Homo sapiens (Human))
Ep Cnrs 51

Curated by ChEMBL
LigandPNGBDBM50033632(3-{2-[2-(2-{2-[2-tert-Butoxycarbonylamino-3-(4-sul...)
Affinity DataIC50:  0.5nMAssay Description:Tested in vitro for inhibition of amylase release from rat pancreatic aciniMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Ccipe-Faculte De Pharmacie

Curated by ChEMBL
LigandPNGBDBM21147((3S)-3-[(2S)-2-[(2S)-2-{2-[(2S)-2-[(2S)-2-[(3S)-3-...)
Affinity DataIC50:  1nMAssay Description:Compound was evaluated for the binding affinity towards rat pancreatic Cholecystokinin type A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPancreatic alpha-amylase(Homo sapiens (Human))
Ep Cnrs 51

Curated by ChEMBL
LigandPNGBDBM50033636(3-{2-[2-(2-{2-[2-tert-Butoxycarbonylamino-3-(4-sul...)
Affinity DataIC50:  1nMAssay Description:Tested in vitro for inhibition of amylase release from rat pancreatic aciniMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Ccipe-Faculte De Pharmacie

Curated by ChEMBL
LigandPNGBDBM50366632(PD-170292)
Affinity DataIC50:  1.20nMAssay Description:Compound was evaluated for the binding affinity towards rat pancreatic Cholecystokinin type A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Ep Cnrs 51

Curated by ChEMBL
LigandPNGBDBM50033640(2-{2-[2-(2-{2-[2-tert-Butoxycarbonylamino-3-(4-sul...)
Affinity DataIC50:  2nMAssay Description:Tested in vitro for inhibition of amylase release from rat pancreatic aciniMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Ep Cnrs 51

Curated by ChEMBL
LigandPNGBDBM50033640(2-{2-[2-(2-{2-[2-tert-Butoxycarbonylamino-3-(4-sul...)
Affinity DataIC50:  2nMAssay Description:Inhibition of [125I]-BH-CCK- binding to cholecystokinin type B receptor from jurkat TcellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(RAT)
Ep Cnrs 51

Curated by ChEMBL
LigandPNGBDBM50016425((S)-3-{(S)-2-[(S)-2-(2-{(S)-2-[(S)-2-tert-Butoxyca...)
Affinity DataIC50:  2.30nMAssay Description:Inhibition of [125I]-BH-CCK- binding to peripheral cholecystokinin type B receptor from rat pancreatic aciniMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(RAT)
Ep Cnrs 51

Curated by ChEMBL
LigandPNGBDBM50016425((S)-3-{(S)-2-[(S)-2-(2-{(S)-2-[(S)-2-tert-Butoxyca...)
Affinity DataIC50:  2.30nMAssay Description:In vitro binding affinity against Cholecystokinin type B receptor of rat pancreatic aciniMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGastrin/cholecystokinin type B receptor(RAT)
Ep Cnrs 51

Curated by ChEMBL
LigandPNGBDBM50033640(2-{2-[2-(2-{2-[2-tert-Butoxycarbonylamino-3-(4-sul...)
Affinity DataIC50:  3nMAssay Description:Inhibition of [125I]-BH-CCK- binding to peripheral cholecystokinin type B receptor from rat pancreatic aciniMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(MOUSE)
Ccipe-Faculte De Pharmacie

Curated by ChEMBL
LigandPNGBDBM50366632(PD-170292)
Affinity DataIC50:  6.70nMAssay Description:Binding affinity towards Cholecystokinin type B receptor in mouse cortex membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Ep Cnrs 51

Curated by ChEMBL
LigandPNGBDBM50033631(2-{2-[2-(2-{2-[2-tert-Butoxycarbonylamino-3-(4-sul...)
Affinity DataIC50:  7nMAssay Description:Inhibition of [125I]-BH-CCK- binding to cholecystokinin type B receptor from guinea pig brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPancreatic alpha-amylase(Homo sapiens (Human))
Ep Cnrs 51

Curated by ChEMBL
LigandPNGBDBM50033636(3-{2-[2-(2-{2-[2-tert-Butoxycarbonylamino-3-(4-sul...)
Affinity DataIC50:  8nMAssay Description:Inhibition of [125I]-BH-CCK- binding to cholecystokinin type B receptor from jurkat TcellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Ep Cnrs 51

Curated by ChEMBL
LigandPNGBDBM50281671((S)-3-{(S)-2-[(S)-2-(2-{(S)-2-[(S)-2-tert-Butoxyca...)
Affinity DataIC50:  10nMAssay Description:In vitro binding affinity against Cholecystokinin type B receptor in guinea pig brain membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Ep Cnrs 51

Curated by ChEMBL
LigandPNGBDBM50033629(3-{2-[2-(2-{2-[2-tert-Butoxycarbonylamino-3-(4-sul...)
Affinity DataIC50:  10nMAssay Description:Inhibition of [125I]-BH-CCK- binding to peripheral cholecystokinin type B receptor from rat pancreatic aciniMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Ep Cnrs 51

Curated by ChEMBL
LigandPNGBDBM50281671((S)-3-{(S)-2-[(S)-2-(2-{(S)-2-[(S)-2-tert-Butoxyca...)
Affinity DataIC50:  10nMAssay Description:In vitro binding affinity against Cholecystokinin type B receptor in guinea pig brain membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGastrin/cholecystokinin type B receptor(RAT)
Ep Cnrs 51

Curated by ChEMBL
LigandPNGBDBM50033633(3-{2-[2-(2-{2-[2-tert-Butoxycarbonylamino-3-(4-sul...)
Affinity DataIC50:  12nMAssay Description:Inhibition of [125I]-BH-CCK- binding to peripheral cholecystokinin type B receptor from rat pancreatic aciniMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Ep Cnrs 51

Curated by ChEMBL
LigandPNGBDBM50033629(3-{2-[2-(2-{2-[2-tert-Butoxycarbonylamino-3-(4-sul...)
Affinity DataIC50:  13nMAssay Description:Inhibition of [125I]-BH-CCK- binding to cholecystokinin type B receptor from jurkat TcellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(RAT)
Ep Cnrs 51

Curated by ChEMBL
LigandPNGBDBM50033634(3-{2-[2-(2-{2-[2-tert-Butoxycarbonylamino-3-(4-sul...)
Affinity DataIC50:  13nMAssay Description:Inhibition of [125I]-BH-CCK- binding to cholecystokinin type B receptor from jurkat TcellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(RAT)
Ep Cnrs 51

Curated by ChEMBL
LigandPNGBDBM50033632(3-{2-[2-(2-{2-[2-tert-Butoxycarbonylamino-3-(4-sul...)
Affinity DataIC50:  14nMAssay Description:Inhibition of [125I]-BH-CCK- binding to cholecystokinin type B receptor from jurkat TcellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(RAT)
Ep Cnrs 51

Curated by ChEMBL
LigandPNGBDBM50033633(3-{2-[2-(2-{2-[2-tert-Butoxycarbonylamino-3-(4-sul...)
Affinity DataIC50:  15nMAssay Description:Inhibition of [125I]-BH-CCK- binding to cholecystokinin type B receptor from guinea pig brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(RAT)
Ep Cnrs 51

Curated by ChEMBL
LigandPNGBDBM50033634(3-{2-[2-(2-{2-[2-tert-Butoxycarbonylamino-3-(4-sul...)
Affinity DataIC50:  16nMAssay Description:Inhibition of [125I]-BH-CCK- binding to peripheral cholecystokinin type B receptor from rat pancreatic aciniMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(RAT)
Ep Cnrs 51

Curated by ChEMBL
LigandPNGBDBM50033636(3-{2-[2-(2-{2-[2-tert-Butoxycarbonylamino-3-(4-sul...)
Affinity DataIC50:  18nMAssay Description:Inhibition of [125I]-BH-CCK- binding to cholecystokinin type B receptor from guinea pig brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(RAT)
Ep Cnrs 51

Curated by ChEMBL
LigandPNGBDBM50033632(3-{2-[2-(2-{2-[2-tert-Butoxycarbonylamino-3-(4-sul...)
Affinity DataIC50:  23nMAssay Description:Inhibition of [125I]-BH-CCK- binding to peripheral cholecystokinin type B receptor from rat pancreatic aciniMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(RAT)
Ep Cnrs 51

Curated by ChEMBL
LigandPNGBDBM50033629(3-{2-[2-(2-{2-[2-tert-Butoxycarbonylamino-3-(4-sul...)
Affinity DataIC50:  30nMAssay Description:Inhibition of [125I]-BH-CCK- binding to peripheral cholecystokinin type B receptor from rat pancreatic aciniMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(MOUSE)
Ccipe-Faculte De Pharmacie

Curated by ChEMBL
LigandPNGBDBM50289879(CHEMBL62205 | [(S)-2-(1H-Indol-3-yl)-1-methyl-1-ph...)
Affinity DataIC50:  32nMAssay Description:Binding affinity towards Cholecystokinin type B receptor in mouse cortex membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Ep Cnrs 51

Curated by ChEMBL
LigandPNGBDBM50033633(3-{2-[2-(2-{2-[2-tert-Butoxycarbonylamino-3-(4-sul...)
Affinity DataIC50:  32nMAssay Description:Inhibition of [125I]-BH-CCK- binding to cholecystokinin type B receptor from guinea pig brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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