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Found 6 Enz. Inhib. hit(s) with Target = 'Gastrin/cholecystokinin type B receptor' and Ligand = 'BDBM50033634'
TargetGastrin/cholecystokinin type B receptor(RAT)
Ep Cnrs 51

Curated by ChEMBL
LigandPNGBDBM50033634(3-{2-[2-(2-{2-[2-tert-Butoxycarbonylamino-3-(4-sul...)
Affinity DataIC50:  13nMAssay Description:Inhibition of [125I]-BH-CCK- binding to cholecystokinin type B receptor from jurkat TcellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(RAT)
Ep Cnrs 51

Curated by ChEMBL
LigandPNGBDBM50033634(3-{2-[2-(2-{2-[2-tert-Butoxycarbonylamino-3-(4-sul...)
Affinity DataIC50:  16nMAssay Description:Inhibition of [125I]-BH-CCK- binding to peripheral cholecystokinin type B receptor from rat pancreatic aciniMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Ep Cnrs 51

Curated by ChEMBL
LigandPNGBDBM50033634(3-{2-[2-(2-{2-[2-tert-Butoxycarbonylamino-3-(4-sul...)
Affinity DataIC50:  57nMAssay Description:Inhibition of [125I]-BH-CCK- binding to cholecystokinin type B receptor from guinea pig brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Ep Cnrs 51

Curated by ChEMBL
LigandPNGBDBM50033634(3-{2-[2-(2-{2-[2-tert-Butoxycarbonylamino-3-(4-sul...)
Affinity DataIC50:  65nMAssay Description:Tested in vitro for amylase release from rat pancreatic acini (% of amylase secretion at 1 mM)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Ep Cnrs 51

Curated by ChEMBL
LigandPNGBDBM50033634(3-{2-[2-(2-{2-[2-tert-Butoxycarbonylamino-3-(4-sul...)
Affinity DataIC50:  200nMAssay Description:Inhibition of [125I]-BH-CCK- binding to cholecystokinin type B receptor from jurkat TcellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Ep Cnrs 51

Curated by ChEMBL
LigandPNGBDBM50033634(3-{2-[2-(2-{2-[2-tert-Butoxycarbonylamino-3-(4-sul...)
Affinity DataIC50:  250nMAssay Description:Inhibition of [125I]-BH-CCK- binding to cholecystokinin type B receptor from jurkat TcellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed