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Found 156 with Last Name = 'bhan' and Initial = 'a'
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Affymax

Curated by ChEMBL
LigandPNGBDBM50171117(2-(4-(N-(3-bromo-4-(difluoro(phosphono)methyl)benz...)
Affinity DataKi:  13nMAssay Description:Inhibitory activity against protein tyrosine phosphatase 1B using O-methyl fluorescein monophosphateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Affymax

Curated by ChEMBL
LigandPNGBDBM50171106((4-{[(Benzyl-methyl-carbamoyl)-methyl]-[3-bromo-4-...)
Affinity DataKi:  14nMAssay Description:Inhibitory activity against protein tyrosine phosphatase 1B using O-methyl fluorescein monophosphateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Affymax

Curated by ChEMBL
LigandPNGBDBM50171096(CHEMBL371929 | {4-[[3-Bromo-4-(difluoro-phosphono-...)
Affinity DataKi:  53nMAssay Description:Inhibitory activity against protein tyrosine phosphatase 1B using O-methyl fluorescein monophosphateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Affymax

Curated by ChEMBL
LigandPNGBDBM50171100(CHEMBL198882 | {4-[[4-(Difluoro-phosphono-methyl)-...)
Affinity DataKi:  56nMAssay Description:Inhibitory activity against protein tyrosine phosphatase 1B using O-methyl fluorescein monophosphateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDihydrofolate reductase(Homo sapiens (Human))
Guru Nanak Dev University

Curated by ChEMBL
LigandPNGBDBM50515758(CHEMBL4453575)
Affinity DataKi:  92nMAssay Description:Inhibition of human dihydrofolate reductase assessed as inhibition constant by UV-Vis spectra based Benesi Hilebrand equation analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Affymax

Curated by ChEMBL
LigandPNGBDBM50171099((4-((N-(4-(1,2,3-thiadiazol-4-yl)benzyl)phenylsulf...)
Affinity DataKi:  98nMAssay Description:Inhibitory activity against protein tyrosine phosphatase 1B using O-methyl fluorescein monophosphateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Affymax

Curated by ChEMBL
LigandPNGBDBM50171118((4-{[(Benzyl-methyl-carbamoyl)-methyl]-[4-(difluor...)
Affinity DataKi:  590nMAssay Description:Inhibitory activity against protein tyrosine phosphatase 1B using O-methyl fluorescein monophosphateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Affymax

Curated by ChEMBL
LigandPNGBDBM50171112(({4-[(Benzenesulfonyl-benzyl-amino)-methyl]-phenyl...)
Affinity DataKi:  1.10E+3nMAssay Description:Inhibitory activity against protein tyrosine phosphatase 1B using O-methyl fluorescein monophosphateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDihydrofolate reductase(Homo sapiens (Human))
Guru Nanak Dev University

Curated by ChEMBL
LigandPNGBDBM50515763(CHEMBL4458303)
Affinity DataKi:  1.60E+3nMAssay Description:Inhibition of human dihydrofolate reductase assessed as inhibition constant by UV-Vis spectra based Benesi Hilebrand equation analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMannose-6-phosphate isomerase(Homo sapiens (Human))
Affymax Research Institute

Curated by ChEMBL
LigandPNGBDBM50071516(2-[4-(3,4-Dichloro-phenylsulfanyl)-butyrylamino]-i...)
Affinity DataKi:  4.00E+3nMAssay Description:Compound was tested for inhibition of human phosphomannose isomerase (PMI)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMannose-6-phosphate isomerase(Homo sapiens (Human))
Affymax Research Institute

Curated by ChEMBL
LigandPNGBDBM50071531(2-[4-(2,4-Dichloro-phenoxy)-butyrylamino]-indan-2-...)
Affinity DataKi:  4.00E+3nMAssay Description:Compound was tested for inhibition of yeast phosphomannose isomerase (PMI)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGuanine deaminase(Homo sapiens (Human))
University Of Maryland

Curated by ChEMBL
LigandPNGBDBM50193757(3-benzyl-4,5,7,8-tetrahydro-6-hydroxymethyl-6H-imi...)
Affinity DataKi:  2.01E+4nMAssay Description:Inhibition of rabbit liver guanaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMannose-6-phosphate isomerase(Homo sapiens (Human))
Affymax Research Institute

Curated by ChEMBL
LigandPNGBDBM50071516(2-[4-(3,4-Dichloro-phenylsulfanyl)-butyrylamino]-i...)
Affinity DataKi:  2.60E+4nMAssay Description:Compound was evaluated for the inhibition constant against phosphomannose isomerase enzyme of Candida albicans (CaPMI)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGuanine deaminase(Homo sapiens (Human))
University Of Maryland

Curated by ChEMBL
LigandPNGBDBM50193756(4,5,7,8-tetrahydro-6-hydroxymethyl-6H-imidazo[4,5-...)
Affinity DataKi:  5.36E+4nMAssay Description:Inhibition of rabbit liver guanaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-secretase 1(Homo sapiens (Human))
Tehran University Of Medical Sciences

Curated by ChEMBL
LigandPNGBDBM16047((4S)-4-[(2S)-2-[(2R,4S,5S)-5-[(2S)-2-[(2S)-2-[(4S)...)
Affinity DataIC50:  3nMAssay Description:Inhibition of BACE1 (unknown origin) expressed in baculovirus expression system using Rh-EVNLDAEFK-Quencher as substrate after 90 mins by FRET assayMore data for this Ligand-Target Pair
TargetDihydrofolate reductase(Homo sapiens (Human))
Guru Nanak Dev University

Curated by ChEMBL
LigandPNGBDBM50515758(CHEMBL4453575)
Affinity DataIC50:  10nMAssay Description:Inhibition of human dihydrofolate reductase using dihydrofolic acid as substrate preincubated for 1 hr in presence of NADPH followed by substrate add...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDihydrofolate reductase(Homo sapiens (Human))
Guru Nanak Dev University

Curated by ChEMBL
LigandPNGBDBM50515763(CHEMBL4458303)
Affinity DataIC50:  20nMAssay Description:Inhibition of human dihydrofolate reductase using dihydrofolic acid as substrate preincubated for 1 hr in presence of NADPH followed by substrate add...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Affymax

Curated by ChEMBL
LigandPNGBDBM50171117(2-(4-(N-(3-bromo-4-(difluoro(phosphono)methyl)benz...)
Affinity DataIC50:  28nMAssay Description:Inhibitory activity against protein tyrosine phosphatase 1B using O-methyl fluorescein monophosphateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Affymax

Curated by ChEMBL
LigandPNGBDBM50171106((4-{[(Benzyl-methyl-carbamoyl)-methyl]-[3-bromo-4-...)
Affinity DataIC50:  31nMAssay Description:Inhibitory activity against protein tyrosine phosphatase 1B using O-methyl fluorescein monophosphateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Affymax

Curated by ChEMBL
LigandPNGBDBM50171096(CHEMBL371929 | {4-[[3-Bromo-4-(difluoro-phosphono-...)
Affinity DataIC50:  35nMAssay Description:Inhibitory activity against protein tyrosine phosphatase 1B using O-methyl fluorescein monophosphateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Affymax

Curated by ChEMBL
LigandPNGBDBM50171091(CHEMBL198939 | {4-[[4-(Difluoro-phosphono-methyl)-...)
Affinity DataIC50:  60nMAssay Description:Inhibitory activity against protein tyrosine phosphatase 1B using O-methyl fluorescein monophosphateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Affymax

Curated by ChEMBL
LigandPNGBDBM50171100(CHEMBL198882 | {4-[[4-(Difluoro-phosphono-methyl)-...)
Affinity DataIC50:  74nMAssay Description:Inhibitory activity against protein tyrosine phosphatase 1B using O-methyl fluorescein monophosphateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Affymax

Curated by ChEMBL
LigandPNGBDBM50171100(CHEMBL198882 | {4-[[4-(Difluoro-phosphono-methyl)-...)
Affinity DataIC50:  74nMAssay Description:Inhibition of PTP1BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-secretase 1(Homo sapiens (Human))
Tehran University Of Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50432316(CHEMBL2347874)
Affinity DataIC50:  98nMAssay Description:Inhibition of BACE1 (unknown origin) expressed in baculovirus expression system using Rh-EVNLDAEFK-Quencher as substrate after 90 mins by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDihydrofolate reductase(Homo sapiens (Human))
Guru Nanak Dev University

Curated by ChEMBL
LigandPNGBDBM50515761(CHEMBL4533705)
Affinity DataIC50:  100nMAssay Description:Inhibition of human dihydrofolate reductase using dihydrofolic acid as substrate preincubated for 1 hr in presence of NADPH followed by substrate add...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBreakpoint cluster region protein/Tyrosine-protein kinase ABL1(Homo sapiens (Human))
The University Of Texas M.D. Anderson Cancer Center

Curated by ChEMBL
LigandPNGBDBM13530(4-[(4-methylpiperazin-1-yl)methyl]-N-[4-methyl-3-[...)
Affinity DataIC50:  116nMAssay Description:Inhibition of Bcr-Abl (unknown origin) phosphorylation by spectrophotometric assayMore data for this Ligand-Target Pair
TargetBeta-secretase 1(Homo sapiens (Human))
Tehran University Of Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50432318(CHEMBL2347872)
Affinity DataIC50:  119nMAssay Description:Inhibition of BACE1 (unknown origin) expressed in baculovirus expression system using Rh-EVNLDAEFK-Quencher as substrate after 90 mins by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Affymax

Curated by ChEMBL
LigandPNGBDBM50171109(CHEMBL196268 | {4-[[4-(Difluoro-phosphono-methyl)-...)
Affinity DataIC50:  180nMAssay Description:Inhibitory activity against protein tyrosine phosphatase 1B using O-methyl fluorescein monophosphateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Affymax

Curated by ChEMBL
LigandPNGBDBM50171099((4-((N-(4-(1,2,3-thiadiazol-4-yl)benzyl)phenylsulf...)
Affinity DataIC50:  200nMAssay Description:Inhibition of PTP1BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Affymax

Curated by ChEMBL
LigandPNGBDBM50171099((4-((N-(4-(1,2,3-thiadiazol-4-yl)benzyl)phenylsulf...)
Affinity DataIC50:  210nMAssay Description:Inhibitory activity against protein tyrosine phosphatase 1B using O-methyl fluorescein monophosphateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDihydrofolate reductase(Homo sapiens (Human))
Guru Nanak Dev University

Curated by ChEMBL
LigandPNGBDBM50515760(CHEMBL4544130)
Affinity DataIC50:  210nMAssay Description:Inhibition of human dihydrofolate reductase using dihydrofolic acid as substrate preincubated for 1 hr in presence of NADPH followed by substrate add...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Affymax

Curated by ChEMBL
LigandPNGBDBM50171097(CHEMBL197681 | {4-[[4-(Difluoro-phosphono-methyl)-...)
Affinity DataIC50:  220nMAssay Description:Inhibitory activity against protein tyrosine phosphatase 1B using O-methyl fluorescein monophosphateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-secretase 1(Homo sapiens (Human))
Tehran University Of Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50432315(CHEMBL2347875)
Affinity DataIC50:  326nMAssay Description:Inhibition of BACE1 (unknown origin) expressed in baculovirus expression system using Rh-EVNLDAEFK-Quencher as substrate after 90 mins by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-secretase 1(Homo sapiens (Human))
Tehran University Of Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50432324(CHEMBL2347867)
Affinity DataIC50:  503nMAssay Description:Inhibition of BACE1 (unknown origin) expressed in baculovirus expression system using Rh-EVNLDAEFK-Quencher as substrate after 90 mins by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-secretase 1(Homo sapiens (Human))
Tehran University Of Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50432317(CHEMBL2347873)
Affinity DataIC50:  578nMAssay Description:Inhibition of BACE1 (unknown origin) expressed in baculovirus expression system using Rh-EVNLDAEFK-Quencher as substrate after 90 mins by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Affymax

Curated by ChEMBL
LigandPNGBDBM50171118((4-{[(Benzyl-methyl-carbamoyl)-methyl]-[4-(difluor...)
Affinity DataIC50:  600nMAssay Description:Inhibitory activity against protein tyrosine phosphatase 1B using O-methyl fluorescein monophosphateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Affymax

Curated by ChEMBL
LigandPNGBDBM50171101((4-{Benzyl-[4-(difluoro-phosphono-methyl)-benzyl]-...)
Affinity DataIC50:  600nMAssay Description:Inhibitory activity against protein tyrosine phosphatase 1B using O-methyl fluorescein monophosphateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Affymax

Curated by ChEMBL
LigandPNGBDBM50171098((4-{(4-Benzoylamino-benzyl)-[4-(difluoro-phosphono...)
Affinity DataIC50:  630nMAssay Description:Inhibitory activity against protein tyrosine phosphatase 1B using O-methyl fluorescein monophosphateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDihydrofolate reductase(Homo sapiens (Human))
Guru Nanak Dev University

Curated by ChEMBL
LigandPNGBDBM50515762(CHEMBL4581410)
Affinity DataIC50:  670nMAssay Description:Inhibition of human dihydrofolate reductase using dihydrofolic acid as substrate preincubated for 1 hr in presence of NADPH followed by substrate add...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBreakpoint cluster region protein/Tyrosine-protein kinase ABL1(Homo sapiens (Human))
The University Of Texas M.D. Anderson Cancer Center

Curated by ChEMBL
LigandPNGBDBM50444656(CHEMBL3098614)
Affinity DataIC50:  740nMAssay Description:Inhibition of Bcr-Abl (unknown origin) phosphorylation by spectrophotometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-secretase 1(Homo sapiens (Human))
Tehran University Of Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50432308(CHEMBL2347882)
Affinity DataIC50:  741nMAssay Description:Inhibition of BACE1 (unknown origin) expressed in baculovirus expression system using Rh-EVNLDAEFK-Quencher as substrate after 90 mins by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Affymax

Curated by ChEMBL
LigandPNGBDBM50171103((4-{(3-Acetyl-benzyl)-[4-(difluoro-phosphono-methy...)
Affinity DataIC50:  770nMAssay Description:Inhibitory activity against protein tyrosine phosphatase 1B using O-methyl fluorescein monophosphateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-secretase 1(Homo sapiens (Human))
Tehran University Of Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50432320(CHEMBL2347870)
Affinity DataIC50:  849nMAssay Description:Inhibition of BACE1 (unknown origin) expressed in baculovirus expression system using Rh-EVNLDAEFK-Quencher as substrate after 90 mins by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-secretase 1(Homo sapiens (Human))
Tehran University Of Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50432314(CHEMBL2347876)
Affinity DataIC50:  854nMAssay Description:Inhibition of BACE1 (unknown origin) expressed in baculovirus expression system using Rh-EVNLDAEFK-Quencher as substrate after 90 mins by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-secretase 1(Homo sapiens (Human))
Tehran University Of Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50432313(CHEMBL2347877)
Affinity DataIC50:  928nMAssay Description:Inhibition of BACE1 (unknown origin) expressed in baculovirus expression system using Rh-EVNLDAEFK-Quencher as substrate after 90 mins by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDihydrofolate reductase(Homo sapiens (Human))
Guru Nanak Dev University

Curated by ChEMBL
LigandPNGBDBM66082((2S)-2-[[4-[(2,4-diaminopteridin-6-yl)methyl-methy...)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of human dihydrofolate reductase using dihydrofolic acid as substrate preincubated for 1 hr in presence of NADPH followed by substrate add...More data for this Ligand-Target Pair
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Affymax

Curated by ChEMBL
LigandPNGBDBM50171105((4-{[4-(Difluoro-phosphono-methyl)-benzyl]-thiophe...)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibitory activity against protein tyrosine phosphatase 1B using O-methyl fluorescein monophosphateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Affymax

Curated by ChEMBL
LigandPNGBDBM50171094((4-{Benzyl-[4-(difluoro-phosphono-methyl)-benzyl]-...)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibitory activity against protein tyrosine phosphatase 1B using O-methyl fluorescein monophosphateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Affymax

Curated by ChEMBL
LigandPNGBDBM50171123(CHEMBL197720 | {4-[[4-(Difluoro-phosphono-methyl)-...)
Affinity DataIC50:  1.10E+3nMAssay Description:Inhibitory activity against protein tyrosine phosphatase 1B using O-methyl fluorescein monophosphateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Affymax

Curated by ChEMBL
LigandPNGBDBM50171124(CHEMBL383163 | {4-[[4-(Difluoro-phosphono-methyl)-...)
Affinity DataIC50:  1.10E+3nMAssay Description:Inhibitory activity against protein tyrosine phosphatase 1B using O-methyl fluorescein monophosphateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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