TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Csir-Indian Institute Of Integrative Medicine
Curated by ChEMBL
Csir-Indian Institute Of Integrative Medicine
Curated by ChEMBL
Affinity DataKi: 0.160nMAssay Description:Binding affinity to AKT1 (unknown origin)More data for this Ligand-Target Pair
TargetAdenosine receptor A1(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Affinity DataKi: 4.40nMAssay Description:Displacement of [3H]DPCPX from recombinant human adenosine A1 receptor expressed in CHO cell membrane by by scintillation counting methodMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Affinity DataKi: 4.40nMAssay Description:Displacement of [3H]DPCPX from recombinant human adenosine A1 receptor expressed in CHO cell membrane by by scintillation counting methodMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Affinity DataKi: 21nMAssay Description:Displacement of [3H]ZM241385 from recombinant human adenosine A2A receptor expressed in HEK293 cell membrane by scintillation counting methodMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Affinity DataKi: 21nMAssay Description:Displacement of [3H]ZM241385 from recombinant human adenosine A2A receptor expressed in HEK293 cell membrane by scintillation counting methodMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Affinity DataKi: 102nMAssay Description:Displacement of [3H]NECA from recombinant human adenosine A2A receptor expressed in CHO cell membrane after 3 hrs by microbeta scintillation counting...More data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Affinity DataKi: 102nMAssay Description:Displacement of [3H]NECA from recombinant human adenosine A2A receptor expressed in CHO cell membrane after 3 hrs by microbeta scintillation counting...More data for this Ligand-Target Pair
TargetAdenosine receptor A3(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Affinity DataKi: 104nMAssay Description:Displacement of [125I]I-ABMECA from recombinant human adenosine A3 receptor expressed in HEK293 cell membrane by scintillation counting methodMore data for this Ligand-Target Pair
TargetAdenosine receptor A3(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Affinity DataKi: 104nMAssay Description:Displacement of [125I]I-ABMECA from recombinant human adenosine A3 receptor expressed in HEK293 cell membrane by scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 150nMAssay Description:Mixed type inhibition of equine serum BChE assessed as decrease in Vmax and increase in Km using varying level of S-butyrylthiocholine iodide as subs...More data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Affinity DataKi: 153nMAssay Description:Displacement of [3H]NECA from recombinant human adenosine A2A receptor expressed in CHO cell membrane after 3 hrs by microbeta scintillation counting...More data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Affinity DataKi: 153nMAssay Description:Displacement of [3H]NECA from recombinant human adenosine A2A receptor expressed in CHO cell membrane after 3 hrs by microbeta scintillation counting...More data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Affinity DataKi: 200nMAssay Description:Displacement of [3H]NECA from recombinant human adenosine A2A receptor expressed in CHO cell membrane after 3 hrs by microbeta scintillation counting...More data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Affinity DataKi: 200nMAssay Description:Displacement of [3H]NECA from recombinant human adenosine A2A receptor expressed in CHO cell membrane after 3 hrs by microbeta scintillation counting...More data for this Ligand-Target Pair
Affinity DataKi: 210nMAssay Description:Non-competitive inhibition of recombinant human AChE assessed as decrease in Vmax with constant Km using varying level of acetylthiocholine iodide as...More data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Affinity DataKi: 245nMAssay Description:Displacement of [3H]NECA from recombinant human adenosine A2A receptor expressed in CHO cell membrane after 3 hrs by microbeta scintillation counting...More data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Affinity DataKi: 245nMAssay Description:Displacement of [3H]NECA from recombinant human adenosine A2A receptor expressed in CHO cell membrane after 3 hrs by microbeta scintillation counting...More data for this Ligand-Target Pair
Affinity DataKi: 280nMAssay Description:Competitive inhibition of human CYP1A1 using 7-ethoxyresorufin as substrateMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Affinity DataKi: 313nMAssay Description:Displacement of [3H]NECA from recombinant human adenosine A2A receptor expressed in CHO cell membrane after 3 hrs by microbeta scintillation counting...More data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Affinity DataKi: 313nMAssay Description:Displacement of [3H]NECA from recombinant human adenosine A2A receptor expressed in CHO cell membrane after 3 hrs by microbeta scintillation counting...More data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Affinity DataKi: 330nMAssay Description:Displacement of [3H]NECA from recombinant human adenosine A2A receptor expressed in CHO cell membrane after 3 hrs by microbeta scintillation counting...More data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Affinity DataKi: 330nMAssay Description:Displacement of [3H]NECA from recombinant human adenosine A2A receptor expressed in CHO cell membrane after 3 hrs by microbeta scintillation counting...More data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Affinity DataKi: 333nMAssay Description:Displacement of [3H]NECA from recombinant human adenosine A2A receptor expressed in CHO cell membrane after 3 hrs by microbeta scintillation counting...More data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Affinity DataKi: 333nMAssay Description:Displacement of [3H]NECA from recombinant human adenosine A2A receptor expressed in CHO cell membrane after 3 hrs by microbeta scintillation counting...More data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Affinity DataKi: 351nMAssay Description:Displacement of [3H]NECA from recombinant human adenosine A2A receptor expressed in CHO cell membrane after 3 hrs by microbeta scintillation counting...More data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Affinity DataKi: 351nMAssay Description:Displacement of [3H]NECA from recombinant human adenosine A2A receptor expressed in CHO cell membrane after 3 hrs by microbeta scintillation counting...More data for this Ligand-Target Pair
TargetAdenosine receptor A1(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Affinity DataKi: 399nMAssay Description:Displacement of [3H]CCPA from recombinant human adenosine A1 receptor expressed in CHO cell membrane after 3 hrs by microbeta scintillation counting ...More data for this Ligand-Target Pair
TargetAdenosine receptor A1(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Affinity DataKi: 399nMAssay Description:Displacement of [3H]CCPA from recombinant human adenosine A1 receptor expressed in CHO cell membrane after 3 hrs by microbeta scintillation counting ...More data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Affinity DataKi: 466nMAssay Description:Displacement of [3H]NECA from recombinant human adenosine A2A receptor expressed in CHO cell membrane after 3 hrs by microbeta scintillation counting...More data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Affinity DataKi: 466nMAssay Description:Displacement of [3H]NECA from recombinant human adenosine A2A receptor expressed in CHO cell membrane after 3 hrs by microbeta scintillation counting...More data for this Ligand-Target Pair
TargetAdenosine receptor A1(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Affinity DataKi: 530nMAssay Description:Displacement of [3H]CCPA from recombinant human adenosine A1 receptor expressed in CHO cell membrane after 3 hrs by microbeta scintillation counting ...More data for this Ligand-Target Pair
TargetAdenosine receptor A1(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Affinity DataKi: 530nMAssay Description:Displacement of [3H]CCPA from recombinant human adenosine A1 receptor expressed in CHO cell membrane after 3 hrs by microbeta scintillation counting ...More data for this Ligand-Target Pair
TargetAdenosine receptor A1(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Affinity DataKi: 555nMAssay Description:Displacement of [3H]CCPA from recombinant human adenosine A1 receptor expressed in CHO cell membrane after 3 hrs by microbeta scintillation counting ...More data for this Ligand-Target Pair
TargetAdenosine receptor A1(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Affinity DataKi: 555nMAssay Description:Displacement of [3H]CCPA from recombinant human adenosine A1 receptor expressed in CHO cell membrane after 3 hrs by microbeta scintillation counting ...More data for this Ligand-Target Pair
TargetAdenosine receptor A3(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Affinity DataKi: 563nMAssay Description:Displacement of [3H]HEMADO from recombinant human adenosine A3 receptor expressed in CHO cell membrane after 3 hrs by microbeta scintillation countin...More data for this Ligand-Target Pair
TargetAdenosine receptor A3(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Affinity DataKi: 563nMAssay Description:Displacement of [3H]HEMADO from recombinant human adenosine A3 receptor expressed in CHO cell membrane after 3 hrs by microbeta scintillation countin...More data for this Ligand-Target Pair
TargetAdenosine receptor A3(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Affinity DataKi: 594nMAssay Description:Displacement of [3H]HEMADO from recombinant human adenosine A3 receptor expressed in CHO cell membrane after 3 hrs by microbeta scintillation countin...More data for this Ligand-Target Pair
TargetAdenosine receptor A3(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Affinity DataKi: 594nMAssay Description:Displacement of [3H]HEMADO from recombinant human adenosine A3 receptor expressed in CHO cell membrane after 3 hrs by microbeta scintillation countin...More data for this Ligand-Target Pair
TargetAdenosine receptor A1(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Affinity DataKi: 629nMAssay Description:Displacement of [3H]CCPA from recombinant human adenosine A1 receptor expressed in CHO cell membrane after 3 hrs by microbeta scintillation counting ...More data for this Ligand-Target Pair
TargetAdenosine receptor A1(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Affinity DataKi: 629nMAssay Description:Displacement of [3H]CCPA from recombinant human adenosine A1 receptor expressed in CHO cell membrane after 3 hrs by microbeta scintillation counting ...More data for this Ligand-Target Pair
TargetAdenosine receptor A1(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Affinity DataKi: 713nMAssay Description:Displacement of [3H]CCPA from recombinant human adenosine A1 receptor expressed in CHO cell membrane after 3 hrs by microbeta scintillation counting ...More data for this Ligand-Target Pair
TargetAdenosine receptor A1(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Affinity DataKi: 713nMAssay Description:Displacement of [3H]CCPA from recombinant human adenosine A1 receptor expressed in CHO cell membrane after 3 hrs by microbeta scintillation counting ...More data for this Ligand-Target Pair
TargetAdenosine receptor A3(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Affinity DataKi: 843nMAssay Description:Displacement of [3H]HEMADO from recombinant human adenosine A3 receptor expressed in CHO cell membrane after 3 hrs by microbeta scintillation countin...More data for this Ligand-Target Pair
TargetAdenosine receptor A3(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Affinity DataKi: 843nMAssay Description:Displacement of [3H]HEMADO from recombinant human adenosine A3 receptor expressed in CHO cell membrane after 3 hrs by microbeta scintillation countin...More data for this Ligand-Target Pair
TargetAdenosine receptor A3(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Affinity DataKi: 934nMAssay Description:Displacement of [3H]HEMADO from recombinant human adenosine A3 receptor expressed in CHO cell membrane after 3 hrs by microbeta scintillation countin...More data for this Ligand-Target Pair
TargetAdenosine receptor A3(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Affinity DataKi: 934nMAssay Description:Displacement of [3H]HEMADO from recombinant human adenosine A3 receptor expressed in CHO cell membrane after 3 hrs by microbeta scintillation countin...More data for this Ligand-Target Pair
TargetAdenosine receptor A1(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Affinity DataKi: 974nMAssay Description:Displacement of [3H]CCPA from recombinant human adenosine A1 receptor expressed in CHO cell membrane after 3 hrs by microbeta scintillation counting ...More data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Affinity DataKi: 974nMAssay Description:Displacement of [3H]NECA from recombinant human adenosine A2A receptor expressed in CHO cell membrane after 3 hrs by microbeta scintillation counting...More data for this Ligand-Target Pair
TargetAdenosine receptor A1(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Affinity DataKi: 974nMAssay Description:Displacement of [3H]CCPA from recombinant human adenosine A1 receptor expressed in CHO cell membrane after 3 hrs by microbeta scintillation counting ...More data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Julius-Maximilians-Universit£T W£Rzburg
Curated by ChEMBL
Affinity DataKi: 974nMAssay Description:Displacement of [3H]NECA from recombinant human adenosine A2A receptor expressed in CHO cell membrane after 3 hrs by microbeta scintillation counting...More data for this Ligand-Target Pair