Compile Data Set for Download or QSAR
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Found 2 Enz. Inhib. hit(s) with Target = 'Adenosine receptor A1' and Ligand = 'BDBM50150078'
TargetAdenosine receptor A1(Homo sapiens (Human))
University Of Leiden

Curated by ChEMBL
LigandPNGBDBM50150078(2-Amino-4-(3-hydroxy-phenyl)-6-(1H-imidazol-2-ylme...)
Affinity DataKi:  4.40nMAssay Description:Binding affinity against human adenosine A1 receptor expressed in CHO cells using [3H]DPCPXMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
University Of Leiden

Curated by ChEMBL
LigandPNGBDBM50150078(2-Amino-4-(3-hydroxy-phenyl)-6-(1H-imidazol-2-ylme...)
Affinity DataKi:  4.40nMAssay Description:Displacement of [3H]DPCPX from recombinant human adenosine A1 receptor expressed in CHO cell membrane by by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed