Affinity DataKi: 0.400nMAssay Description:Binding affinity against human Dopamine receptor D4 by [3H]-spiperone displacement.More data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Displacement of [3H]R214127 from mGluR1 in rat cerebellum membranesMore data for this Ligand-Target Pair
Affinity DataKi: 1.5nMAssay Description:In vitro binding affinity tested on HEK293 cells co-transfected with human D4.4 receptor using [3H]spiperone as a radioligand in FLIPR assayMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Displacement of [3H]R214127 from mGluR1 in rat cerebellum membranesMore data for this Ligand-Target Pair
Affinity DataKi: 2.70nMAssay Description:Binding affinity against human Dopamine receptor D4 by [3H]-spiperone displacement.More data for this Ligand-Target Pair
Affinity DataKi: 3.60nMAssay Description:Binding affinity towards human D4.4 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 3.80nMAssay Description:In vitro binding affinity towards alpha-2B adrenergic receptor of rat neonatal lung in radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 3.80nMAssay Description:In vitro binding affinity tested on HEK293 cells co-transfected with human D4.4 receptor using [3H]spiperone as a radioligand in FLIPR assayMore data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:Displacement of [3H]R214127 from mGluR1 in rat cerebellum membranesMore data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:Displacement of [3H]R214127 from mGluR1 in rat cerebellum membranesMore data for this Ligand-Target Pair
Affinity DataKi: 4.30nMAssay Description:Binding affinity against human Dopamine receptor D4 by [3H]-spiperone displacement.More data for this Ligand-Target Pair
Affinity DataKi: 5nMAssay Description:Displacement of [3H]R214127 from mGluR1 in rat cerebellum membranesMore data for this Ligand-Target Pair
Affinity DataKi: 6nMAssay Description:Displacement of [3H]R214127 from mGluR1 in rat cerebellum membranesMore data for this Ligand-Target Pair
Affinity DataKi: 6.30nMAssay Description:Displacement of [3H]A-369508 from human recombinant D4.4 receptor expressed in HEK293 cell membraneMore data for this Ligand-Target Pair
Affinity DataKi: 6.40nMAssay Description:Displacement of [3H]A-369508 from human recombinant D4.4 receptor expressed in HEK293 cell membraneMore data for this Ligand-Target Pair
Affinity DataKi: 6.40nMAssay Description:Displacement of [3H]A-369508 from human recombinant D4.4 receptor expressed in HEK293 cell membraneMore data for this Ligand-Target Pair
Affinity DataKi: 8nMAssay Description:Displacement of [3H]A-369508 from human recombinant D4.4 receptor expressed in HEK293 cell membraneMore data for this Ligand-Target Pair
Affinity DataKi: 8nMAssay Description:Displacement of [3H]R214127 from mGluR1 in rat cerebellum membranesMore data for this Ligand-Target Pair
Affinity DataKi: 8nMAssay Description:Displacement of [3H]R214127 from mGluR1 in rat cerebellum membranesMore data for this Ligand-Target Pair
Affinity DataKi: 8.5nMAssay Description:Binding affinity against human Dopamine receptor D4 by [3H]-spiperone displacement.More data for this Ligand-Target Pair
Affinity DataKi: 8.5nMAssay Description:Binding affinity against human Dopamine receptor D4 by [3H]-spiperone displacement.More data for this Ligand-Target Pair
Affinity DataKi: 8.70nMAssay Description:In vitro binding affinity towards alpha-2A adrenergic receptor of human clone in radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 9.60nMAssay Description:Binding affinity against human Dopamine receptor D4 by [3H]-spiperone displacement.More data for this Ligand-Target Pair
Affinity DataKi: 9.60nMAssay Description:Binding affinity against human Dopamine receptor D4 by [3H]-spiperone displacement.More data for this Ligand-Target Pair
Affinity DataKi: 11nMAssay Description:Displacement of [3H]R214127 from mGluR1 in rat cerebellum membranesMore data for this Ligand-Target Pair
Affinity DataKi: 11.4nMAssay Description:Displacement of [3H]A-369508 from human recombinant D4.4 receptor expressed in HEK293 cell membraneMore data for this Ligand-Target Pair
Affinity DataKi: 11.6nMAssay Description:Displacement of [3H]A-369508 from human recombinant D4.4 receptor expressed in HEK293 cell membraneMore data for this Ligand-Target Pair
Affinity DataKi: 12nMAssay Description:In vitro binding affinity towards alpha-1A adrenergic receptor of rat submaxillary gland in radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 13.5nMAssay Description:Displacement of [3H]A-369508 from human recombinant D4.4 receptor expressed in HEK293 cell membraneMore data for this Ligand-Target Pair
Affinity DataKi: 13.9nMAssay Description:Displacement of [3H]A-369508 from human recombinant D4.4 receptor expressed in HEK293 cell membraneMore data for this Ligand-Target Pair
Affinity DataKi: 14.2nMAssay Description:Displacement of [3H]A-369508 from human recombinant D4.4 receptor expressed in HEK293 cell membraneMore data for this Ligand-Target Pair
Affinity DataKi: 14.8nMAssay Description:Binding affinity against human Dopamine receptor D4 by [3H]-spiperone displacement.More data for this Ligand-Target Pair
Affinity DataKi: 14.8nMAssay Description:Binding affinity against human Dopamine receptor D4 by [3H]-spiperone displacement.More data for this Ligand-Target Pair
Affinity DataKi: 19.4nMAssay Description:Displacement of [3H]PIPAT from human recombinant D2L receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 20.1nMAssay Description:Displacement of [3H]A-369508 from human recombinant D4.4 receptor expressed in HEK293 cell membraneMore data for this Ligand-Target Pair
Affinity DataKi: 20.4nMAssay Description:Binding affinity against human Dopamine receptor D4 by [3H]-spiperone displacement.More data for this Ligand-Target Pair
Affinity DataKi: 22nMAssay Description:In vitro binding affinity towards alpha-1A adrenergic receptor of rat submaxillary gland in radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 22nMAssay Description:In vitro binding affinity towards alpha-2B adrenergic receptor of rat neonatal lung in radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 22.8nMAssay Description:Displacement of [3H]A-369508 from human recombinant D4.4 receptor expressed in HEK293 cell membraneMore data for this Ligand-Target Pair
Affinity DataKi: 23nMAssay Description:In vitro binding affinity towards alpha-2A adrenergic receptor of human clone in radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 25.3nMAssay Description:Displacement of [3H]PIPAT from human recombinant D2L receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 25.4nMAssay Description:Displacement of [3H]A-369508 from human recombinant D4.4 receptor expressed in HEK293 cell membraneMore data for this Ligand-Target Pair
Affinity DataKi: 26.5nMAssay Description:Binding affinity against human Dopamine receptor D4 by [3H]-spiperone displacement.More data for this Ligand-Target Pair
Affinity DataKi: 27.5nMAssay Description:Displacement of [3H]A-369508 from human recombinant D4.4 receptor expressed in HEK293 cell membraneMore data for this Ligand-Target Pair
Affinity DataKi: 31nMAssay Description:In vitro binding affinity towards alpha-1D adrenergic receptor of rat clone in radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 32.1nMAssay Description:Displacement of [3H]A-369508 from human recombinant D4.4 receptor expressed in HEK293 cell membraneMore data for this Ligand-Target Pair
Affinity DataKi: 33nMAssay Description:Binding affinity tested against D4.2 receptor in Chinese hamster ovary cell line (CHO cells) using [3H]spiperone as a radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 33nMAssay Description:In vitro binding affinity towards alpha-2A adrenergic receptor of human clone in radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 36nMAssay Description:In vitro binding affinity towards alpha-1A adrenergic receptor of rat submaxillary gland in radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 38nMAssay Description:Displacement of [3H]A-369508 from human recombinant D4.4 receptor expressed in HEK293 cell membraneMore data for this Ligand-Target Pair