Affinity DataKi: 3.36nMAssay Description:Inhibition of cathepsin BMore data for this Ligand-Target Pair
Affinity DataKi: 23nMAssay Description:Inhibition of papaya papainMore data for this Ligand-Target Pair
Affinity DataKi: 500nMAssay Description:Inhibition of cathepsin BMore data for this Ligand-Target Pair
TargetHeme ligase(Plasmodium falciparum (isolate 3D7))
Council of Scientific and Industrial Research
US Patent
Council of Scientific and Industrial Research
US Patent
Affinity DataKi: 2.49E+3nMAssay Description:Inhibition of recombinant Plasmodium falciparum falcipain-2 expressed in Escherichia coli M15 assessed as reduction in free AMC release using Z-FR-AM...More data for this Ligand-Target Pair
Affinity DataKi: 2.60E+3nMAssay Description:Inhibition of recombinant Plasmodium falciparum falcipain-2 expressed in Escherichia coli M15 assessed as reduction in free AMC release using Z-FR-AM...More data for this Ligand-Target Pair
TargetHeme ligase(Plasmodium falciparum (isolate 3D7))
Council of Scientific and Industrial Research
US Patent
Council of Scientific and Industrial Research
US Patent
TargetHeme ligase(Plasmodium falciparum (isolate 3D7))
Council of Scientific and Industrial Research
US Patent
Council of Scientific and Industrial Research
US Patent
Affinity DataKi: 2.78E+3nMAssay Description:Inhibition of recombinant Plasmodium falciparum falcipain-2 expressed in Escherichia coli M15 assessed as reduction in free AMC release using Z-FR-AM...More data for this Ligand-Target Pair
Affinity DataKi: 3.32E+3nMAssay Description:Inhibition of recombinant Plasmodium falciparum falcipain-2 expressed in Escherichia coli M15 assessed as reduction in free AMC release using Z-FR-AM...More data for this Ligand-Target Pair
TargetHeme ligase(Plasmodium falciparum (isolate 3D7))
Council of Scientific and Industrial Research
US Patent
Council of Scientific and Industrial Research
US Patent
TargetHeme ligase(Plasmodium falciparum (isolate 3D7))
Council of Scientific and Industrial Research
US Patent
Council of Scientific and Industrial Research
US Patent
Affinity DataKi: 3.49E+3nMAssay Description:Inhibition of recombinant Plasmodium falciparum falcipain-2 expressed in Escherichia coli M15 assessed as reduction in free AMC release using Z-FR-AM...More data for this Ligand-Target Pair
TargetHeme ligase(Plasmodium falciparum (isolate 3D7))
Council of Scientific and Industrial Research
US Patent
Council of Scientific and Industrial Research
US Patent
Affinity DataKi: 4.54E+3nMAssay Description:Inhibition of recombinant Plasmodium falciparum falcipain-2 expressed in Escherichia coli M15 assessed as reduction in free AMC release using Z-FR-AM...More data for this Ligand-Target Pair
Affinity DataKi: 6.91E+3nMAssay Description:Inhibition of recombinant Plasmodium falciparum falcipain-2 expressed in Escherichia coli M15 assessed as reduction in free AMC release using Z-FR-AM...More data for this Ligand-Target Pair
TargetHeme ligase(Plasmodium falciparum (isolate 3D7))
Council of Scientific and Industrial Research
US Patent
Council of Scientific and Industrial Research
US Patent
TargetHeme ligase(Plasmodium falciparum (isolate 3D7))
Council of Scientific and Industrial Research
US Patent
Council of Scientific and Industrial Research
US Patent
Affinity DataKi: 9.92E+3nMAssay Description:Inhibition of recombinant Plasmodium falciparum falcipain-2 expressed in Escherichia coli M15 assessed as reduction in free AMC release using Z-FR-AM...More data for this Ligand-Target Pair
TargetHeme ligase(Plasmodium falciparum (isolate 3D7))
Council of Scientific and Industrial Research
US Patent
Council of Scientific and Industrial Research
US Patent
Affinity DataIC50: 3.38E+3nMAssay Description:Inhibition of recombinant Plasmodium falciparum falcipain-2 expressed in Escherichia coli M15 assessed as reduction in free AMC release using Z-FR-AM...More data for this Ligand-Target Pair
Affinity DataIC50: 3.53E+3nMAssay Description:Inhibition of recombinant Plasmodium falciparum falcipain-2 expressed in Escherichia coli M15 assessed as reduction in free AMC release using Z-FR-AM...More data for this Ligand-Target Pair
TargetHeme ligase(Plasmodium falciparum (isolate 3D7))
Council of Scientific and Industrial Research
US Patent
Council of Scientific and Industrial Research
US Patent
Affinity DataIC50: 3.78E+3nMAssay Description:Inhibition of recombinant Plasmodium falciparum falcipain-2 expressed in Escherichia coli M15 assessed as reduction in free AMC release using Z-FR-AM...More data for this Ligand-Target Pair
TargetHeme ligase(Plasmodium falciparum (isolate 3D7))
Council of Scientific and Industrial Research
US Patent
Council of Scientific and Industrial Research
US Patent
Affinity DataIC50: 5.62E+3nMAssay Description:Inhibition of recombinant Plasmodium falciparum falcipain-2 expressed in Escherichia coli M15 assessed as reduction in free AMC release using Z-FR-AM...More data for this Ligand-Target Pair
TargetHeme ligase(Plasmodium falciparum (isolate 3D7))
Council of Scientific and Industrial Research
US Patent
Council of Scientific and Industrial Research
US Patent
Affinity DataIC50: 5.90E+3nMAssay Description:Inhibition of recombinant Plasmodium falciparum falcipain-2 expressed in Escherichia coli M15 assessed as reduction in free AMC release using Z-FR-AM...More data for this Ligand-Target Pair
TargetHeme ligase(Plasmodium falciparum (isolate 3D7))
Council of Scientific and Industrial Research
US Patent
Council of Scientific and Industrial Research
US Patent
Affinity DataIC50: 7.67E+3nMAssay Description:Inhibition of recombinant Plasmodium falciparum falcipain-2 expressed in Escherichia coli M15 assessed as reduction in free AMC release using Z-FR-AM...More data for this Ligand-Target Pair
TargetHeme ligase(Plasmodium falciparum (isolate 3D7))
Council of Scientific and Industrial Research
US Patent
Council of Scientific and Industrial Research
US Patent
Affinity DataIC50: 9.38E+3nMAssay Description:Inhibition of recombinant Plasmodium falciparum falcipain-2 expressed in Escherichia coli M15 assessed as reduction in free AMC release using Z-FR-AM...More data for this Ligand-Target Pair
TargetHeme ligase(Plasmodium falciparum (isolate 3D7))
Council of Scientific and Industrial Research
US Patent
Council of Scientific and Industrial Research
US Patent
TargetHeme ligase(Plasmodium falciparum (isolate 3D7))
Council of Scientific and Industrial Research
US Patent
Council of Scientific and Industrial Research
US Patent
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of recombinant Plasmodium falciparum falcipain-2 expressed in Escherichia coli M15 assessed as reduction in free AMC release using Z-FR-AM...More data for this Ligand-Target Pair
Affinity DataIC50: 1.35E+4nMAssay Description:Inhibition of recombinant Plasmodium falciparum falcipain-2 expressed in Escherichia coli M15 assessed as reduction in free AMC release using Z-FR-AM...More data for this Ligand-Target Pair
TargetHeme ligase(Plasmodium falciparum (isolate 3D7))
Council of Scientific and Industrial Research
US Patent
Council of Scientific and Industrial Research
US Patent
Affinity DataIC50: >2.50E+4nMAssay Description:Inhibition of recombinant Plasmodium falciparum falcipain-2 expressed in Escherichia coli M15 assessed as reduction in free AMC release using Z-FR-AM...More data for this Ligand-Target Pair
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of papaya papain using BAPNA as substrate assessed as p-nitroaniline release by spectrophotometric analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 4.00E+4nMAssay Description:Inhibition of papaya papain using BAPNA as substrate assessed as p-nitroaniline release by spectrophotometric analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 5.40E+4nMAssay Description:Inhibition of papaya papain using BAPNA as substrate assessed as p-nitroaniline release by spectrophotometric analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 8.30E+4nMAssay Description:Inhibition of papaya papain using BAPNA as substrate assessed as p-nitroaniline release by spectrophotometric analysisMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of recombinant Plasmodium falciparum falcipain-2 expressed in Escherichia coli M15 assessed as reduction in free AMC release using Z-FR-AM...More data for this Ligand-Target Pair
TargetHeme ligase(Plasmodium falciparum (isolate 3D7))
Council of Scientific and Industrial Research
US Patent
Council of Scientific and Industrial Research
US Patent
TargetHeme ligase(Plasmodium falciparum (isolate 3D7))
Council of Scientific and Industrial Research
US Patent
Council of Scientific and Industrial Research
US Patent
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of recombinant Plasmodium falciparum falcipain-2 expressed in Escherichia coli M15 assessed as reduction in free AMC release using Z-FR-AM...More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of recombinant Plasmodium falciparum falcipain-2 expressed in Escherichia coli M15 assessed as reduction in free AMC release using Z-FR-AM...More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of recombinant Plasmodium falciparum falcipain-2 expressed in Escherichia coli M15 assessed as reduction in free AMC release using Z-FR-AM...More data for this Ligand-Target Pair
TargetHeme ligase(Plasmodium falciparum (isolate 3D7))
Council of Scientific and Industrial Research
US Patent
Council of Scientific and Industrial Research
US Patent
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of recombinant Plasmodium falciparum falcipain-2 expressed in Escherichia coli M15 assessed as reduction in free AMC release using Z-FR-AM...More data for this Ligand-Target Pair