Reaction Details Report a problem with these data
Target
Heme ligase
Ligand
BDBM558639
Substrate
n/a
Meas. Tech.
TBD
IC50
>100000±n/a nM
Citation
Bhattacharya, AK; Aratikatla, EK; Malhotra, P; Mohmmed, A Antimalarial compounds, process for preparation and their use for drug resistant malaria US Patent US11365202 Publication Date 6/21/2022
More Info.:
Target
Name:
Heme ligase
Synonyms:
4.99.1.8 | HDP | HDP_PLAF7
Type:
PROTEIN
Mol. Mass.:
24349.37
Organism:
Plasmodium falciparum (isolate 3D7)
Description:
ChEMBL_117325
Residue:
205
Sequence:
MKNRFYYNLIIKRLYTRSGGLRKPQKVTNDPESINRKVYWCFEHKPVKRTIINLIYSHNELKIFSNLLNHPTVGSSLIHELSLDGPYTAFFPSNEAMQLINIESFNKLYNDENKLSEFVLNHVTKEYWLYRDLYGSSYQPWLMYNEKREAPEKLRNLLNNDLIVKIEGEFKHCNHSIYLNGSKIIRPNMKCHNGVVHIVDKPIIF