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Found 39 with Last Name = 'binderup' and Initial = 'l'
TargetVitamin D3 receptor(Gallus gallus)
TBA

Curated by ChEMBL
LigandPNGBDBM50212896(CHEMBL293146)
Affinity DataKi: <0.00100nMAssay Description:Displacement from vitamin D receptor in chick intestine: 50% displacementMore data for this Ligand-Target Pair
In DepthDetails Article
TargetVitamin D3 receptor(Gallus gallus)
TBA

Curated by ChEMBL
LigandPNGBDBM50200182((1S,3R,5Z,7E)-9,10-secocholesta-5,7,10(19)-triene-...)
Affinity DataKi:  0.0250nMAssay Description:Displacement from vitamin D receptor in chick intestine : 50% displacementMore data for this Ligand-Target Pair
In DepthDetails Article
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Leo Pharma

Curated by ChEMBL
LigandPNGBDBM50136890(CHEMBL152208 | [2-Chloro-4-(4-fluoro-2-methyl-phen...)
Affinity DataIC50:  4nMAssay Description:In vitro inhibitory activity determined against human mitogen-activated protein kinase p38 alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Leo Pharma

Curated by ChEMBL
LigandPNGBDBM50136887(CHEMBL356455 | [4-(2-Amino-phenylamino)-2-chloro-p...)
Affinity DataIC50:  5nMAssay Description:In vitro inhibitory activity determined against human mitogen-activated protein kinase p38 alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Leo Pharma

Curated by ChEMBL
LigandPNGBDBM50136897((2-Chloro-4-phenylamino-phenyl)-o-tolyl-methanone ...)
Affinity DataIC50:  7nMAssay Description:In vitro inhibitory activity determined against human mitogen-activated protein kinase p38 alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Leo Pharma

Curated by ChEMBL
LigandPNGBDBM50136886(CHEMBL152767 | [4-(2-Amino-phenylamino)-2-chloro-p...)
Affinity DataIC50:  10nMAssay Description:In vitro inhibitory activity determined against human mitogen-activated protein kinase p38 alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Leo Pharma

Curated by ChEMBL
LigandPNGBDBM50136884((2-Chloro-4-o-tolylamino-phenyl)-o-tolyl-methanone...)
Affinity DataIC50:  12nMAssay Description:In vitro inhibitory activity determined against human mitogen-activated protein kinase p38 alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Leo Pharma

Curated by ChEMBL
LigandPNGBDBM50136898(CHEMBL152820 | [4-(2-Amino-phenylamino)-2-methyl-p...)
Affinity DataIC50:  13nMAssay Description:In vitro inhibitory activity determined against human mitogen-activated protein kinase p38 alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Leo Pharma

Curated by ChEMBL
LigandPNGBDBM50136900(1-{2-[3-Chloro-4-(2-methyl-benzoyl)-phenylamino]-p...)
Affinity DataIC50:  21nMAssay Description:In vitro inhibitory activity determined against human mitogen-activated protein kinase p38 alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Leo Pharma

Curated by ChEMBL
LigandPNGBDBM50136903(CHEMBL357732 | [4-(2-Amino-phenylamino)-phenyl]-o-...)
Affinity DataIC50:  29nMAssay Description:In vitro inhibitory activity determined against human mitogen-activated protein kinase p38 alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Leo Pharma

Curated by ChEMBL
LigandPNGBDBM15244(5-(2,6-dichlorophenyl)-2-(2,4-difluorophenyl)sulfa...)
Affinity DataIC50:  29nMAssay Description:In vitro inhibitory activity determined against human mitogen-activated protein kinase p38 alphaMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Leo Pharma

Curated by ChEMBL
LigandPNGBDBM50099331(4-(4-(4-fluorophenyl)-1-(piperidin-4-yl)-1H-imidaz...)
Affinity DataIC50:  38nMAssay Description:In vitro inhibitory activity determined against human mitogen-activated protein kinase p38 alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Leo Pharma

Curated by ChEMBL
LigandPNGBDBM50136885(CHEMBL347496 | [4-(2-Amino-4-bromo-phenylamino)-2-...)
Affinity DataIC50:  39nMAssay Description:In vitro inhibitory activity determined against human mitogen-activated protein kinase p38 alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Leo Pharma

Curated by ChEMBL
LigandPNGBDBM50136888(CHEMBL153012 | {2-[3-Chloro-4-(2-methyl-benzoyl)-p...)
Affinity DataIC50:  42nMAssay Description:In vitro inhibitory activity determined against human mitogen-activated protein kinase p38 alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Leo Pharma

Curated by ChEMBL
LigandPNGBDBM50136899(CHEMBL152440 | [4-(2-Amino-phenylamino)-phenyl]-(2...)
Affinity DataIC50:  54nMAssay Description:In vitro inhibitory activity determined against human mitogen-activated protein kinase p38 alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Leo Pharma

Curated by ChEMBL
LigandPNGBDBM50136901(CHEMBL422510 | N-{2-[3-Chloro-4-(2-methyl-benzoyl)...)
Affinity DataIC50:  63nMAssay Description:In vitro inhibitory activity determined against human mitogen-activated protein kinase p38 alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Leo Pharma

Curated by ChEMBL
LigandPNGBDBM50136895(CHEMBL347770 | {4-[(2-Amino-phenyl)-methyl-amino]-...)
Affinity DataIC50:  101nMAssay Description:In vitro inhibitory activity determined against human mitogen-activated protein kinase p38 alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Leo Pharma

Curated by ChEMBL
LigandPNGBDBM50136902(CHEMBL155448 | [4-(2-Amino-phenylamino)-2-chloro-p...)
Affinity DataIC50:  139nMAssay Description:In vitro inhibitory activity determined against human mitogen-activated protein kinase p38 alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Leo Pharma

Curated by ChEMBL
LigandPNGBDBM50136896(CHEMBL356157 | [4-(2-Amino-phenylamino)-3-methyl-p...)
Affinity DataIC50:  143nMAssay Description:In vitro inhibitory activity determined against human mitogen-activated protein kinase p38 alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Leo Pharma

Curated by ChEMBL
LigandPNGBDBM50136882(CHEMBL152596 | [4-(2-Amino-phenylamino)-phenyl]-ph...)
Affinity DataIC50:  145nMAssay Description:In vitro inhibitory activity determined against human mitogen-activated protein kinase p38 alphaMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Leo Pharma

Curated by ChEMBL
LigandPNGBDBM50136891(CHEMBL152349 | Phenyl-(4-phenylamino-phenyl)-metha...)
Affinity DataIC50:  193nMAssay Description:In vitro inhibitory activity determined against human mitogen-activated protein kinase p38 alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Technical University Of Denmark

Curated by ChEMBL
LigandPNGBDBM50001013(CHEMBL93959 | Phosphoric acid 4-(4,5-dihydroxy-3-m...)
Affinity DataIC50:  220nMAssay Description:Inhibitory concentration against Clostridium histolyticum CollagenaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Technical University Of Denmark

Curated by ChEMBL
LigandPNGBDBM50001007((Aranciamycin) 4-(4,5-Dihydroxy-3-methoxy-6-methyl...)
Affinity DataIC50:  370nMAssay Description:Inhibitory concentration against Clostridium histolyticum CollagenaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Technical University Of Denmark

Curated by ChEMBL
LigandPNGBDBM50001006((10-(p-tolylsulfonyl)hydrazone)-Aranciamycin | CHE...)
Affinity DataIC50:  420nMAssay Description:Inhibitory concentration against Clostridium histolyticum CollagenaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Leo Pharma

Curated by ChEMBL
LigandPNGBDBM50136883(CHEMBL347576 | [2-Chloro-4-(2-nitro-phenylamino)-p...)
Affinity DataIC50:  437nMAssay Description:In vitro inhibitory activity determined against human mitogen-activated protein kinase p38 alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Leo Pharma

Curated by ChEMBL
LigandPNGBDBM50136893(CHEMBL152209 | [4-(2-Amino-phenylamino)-phenyl]-m-...)
Affinity DataIC50:  574nMAssay Description:In vitro inhibitory activity determined against human mitogen-activated protein kinase p38 alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Technical University Of Denmark

Curated by ChEMBL
LigandPNGBDBM50001017(2,5,7-Trihydroxy-3-methoxy-2-methyl-4-(3,4,5-trime...)
Affinity DataIC50:  670nMAssay Description:Inhibitory concentration against Clostridium histolyticum CollagenaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Leo Pharma

Curated by ChEMBL
LigandPNGBDBM50136892(CHEMBL356809 | [4-(2-Amino-phenylamino)-phenyl]-bi...)
Affinity DataIC50:  811nMAssay Description:In vitro inhibitory activity determined against human mitogen-activated protein kinase p38 alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Technical University Of Denmark

Curated by ChEMBL
LigandPNGBDBM22984((8S,10S)-10-{[(2R,4S,5S,6S)-4-amino-5-hydroxy-6-me...)
Affinity DataIC50:  1.10E+3nMAssay Description:Inhibitory concentration against Clostridium histolyticum CollagenaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Leo Pharma

Curated by ChEMBL
LigandPNGBDBM50136889(CHEMBL152403 | N-[3-Chloro-4-(1-o-tolyl-vinyl)-phe...)
Affinity DataIC50:  1.55E+3nMAssay Description:In vitro inhibitory activity determined against human mitogen-activated protein kinase p38 alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Technical University Of Denmark

Curated by ChEMBL
LigandPNGBDBM50368352(Cerubidine | DAUNORUBICIN)
Affinity DataIC50:  1.90E+3nMAssay Description:Inhibitory concentration against Clostridium histolyticum CollagenaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Technical University Of Denmark

Curated by ChEMBL
LigandPNGBDBM50001011(4-(4,5-Dihydroxy-3-methoxy-6-methyl-tetrahydro-pyr...)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibitory concentration against Clostridium histolyticum CollagenaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Technical University Of Denmark

Curated by ChEMBL
LigandPNGBDBM50001009(4-(4,5-Dihydroxy-3-methoxy-6-methyl-tetrahydro-pyr...)
Affinity DataIC50:  3.00E+3nMAssay Description:Inhibitory concentration against Clostridium histolyticum CollagenaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Technical University Of Denmark

Curated by ChEMBL
LigandPNGBDBM50368351(ACLACINOMYCIN A | ACLARUBICIN)
Affinity DataIC50:  9.90E+3nMAssay Description:Concentration inhibiting Clostridium histolyticum collagenase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Technical University Of Denmark

Curated by ChEMBL
LigandPNGBDBM50001010(4-[4-(tert-Butyl-dimethyl-silanyloxy)-5-hydroxy-3-...)
Affinity DataIC50:  1.70E+4nMAssay Description:Inhibitory concentration against Clostridium histolyticum CollagenaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Technical University Of Denmark

Curated by ChEMBL
LigandPNGBDBM50001012(2,4,5,7-Tetrahydroxy-3-methoxy-2-methyl-3,4-dihydr...)
Affinity DataIC50:  1.90E+4nMAssay Description:Inhibitory concentration against Clostridium histolyticum CollagenaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Technical University Of Denmark

Curated by ChEMBL
LigandPNGBDBM50001016(Acetic acid 3-acetoxy-5-methoxy-2-methyl-6-(3,10,1...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibitory concentration against Clostridium histolyticum CollagenaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Technical University Of Denmark

Curated by ChEMBL
LigandPNGBDBM50001008(4-(4,5-Dihydroxy-3-methoxy-6-methyl-tetrahydro-pyr...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibitory concentration against Clostridium histolyticum CollagenaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Leo Pharma

Curated by ChEMBL
LigandPNGBDBM50136894(CHEMBL153795 | N*1*-[3-Chloro-4-(2-methyl-benzyl)-...)
Affinity DataIC50: >1.00E+5nMAssay Description:In vitro inhibitory activity determined against human mitogen-activated protein kinase p38 alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed