Affinity DataKi: 300nMAssay Description:Binding affinity towards competitive inhibition against rat microsomal Oxidosqualene-lanosterol cyclaseMore data for this Ligand-Target Pair
Affinity DataKi: 400nMAssay Description:Binding affinity towards noncompetetive inhibition against rat microsomal Oxidosqualene-lanosterol cyclaseMore data for this Ligand-Target Pair
Affinity DataIC50: 100nMAssay Description:Inhibitory activity against Oxidosqualene-lanosterol cyclase from Rat liver microsomesMore data for this Ligand-Target Pair
Affinity DataIC50: 600nMAssay Description:Inhibitory activity against Oxidosqualene-lanosterol cyclase from Rat liver microsomesMore data for this Ligand-Target Pair
Affinity DataIC50: 600nMAssay Description:Inhibitory activity against Oxidosqualene-lanosterol cyclase from Rat liver microsomesMore data for this Ligand-Target Pair
Affinity DataIC50: 600nMAssay Description:Inhibitory activity against Oxidosqualene-lanosterol cyclase from Rat liver microsomesMore data for this Ligand-Target Pair
Affinity DataIC50: 600nMAssay Description:Inhibitory activity against Oxidosqualene-lanosterol cyclase from Rat liver microsomesMore data for this Ligand-Target Pair
Affinity DataIC50: 680nMAssay Description:Inhibitory activity against Oxidosqualene-lanosterol cyclase from Rat liver microsomesMore data for this Ligand-Target Pair
Affinity DataIC50: 700nMAssay Description:Inhibitory activity against Oxidosqualene-lanosterol cyclase from Rat liver microsomesMore data for this Ligand-Target Pair
Affinity DataIC50: 900nMAssay Description:Inhibitory activity against Oxidosqualene-lanosterol cyclase from Rat liver microsomesMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibitory activity against Oxidosqualene-lanosterol cyclase from Rat liver microsomesMore data for this Ligand-Target Pair
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibitory activity against Oxidosqualene-lanosterol cyclase from Rat liver microsomesMore data for this Ligand-Target Pair
Affinity DataIC50: 2.90E+3nMAssay Description:Inhibitory activity against Oxidosqualene-lanosterol cyclase from Rat liver microsomesMore data for this Ligand-Target Pair
Affinity DataIC50: 6.80E+3nMAssay Description:Inhibitory activity against Oxidosqualene-lanosterol cyclase from Rat liver microsomesMore data for this Ligand-Target Pair
Affinity DataIC50: 1.64E+4nMAssay Description:Inhibitory activity against Oxidosqualene-lanosterol cyclase from Rat liver microsomesMore data for this Ligand-Target Pair
Affinity DataIC50: 1.70E+4nMAssay Description:Inhibitory activity against Oxidosqualene-lanosterol cyclase from Rat liver microsomesMore data for this Ligand-Target Pair
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibitory activity against Oxidosqualene-lanosterol cyclase from Rat liver microsomesMore data for this Ligand-Target Pair
Affinity DataIC50: 2.50E+4nMAssay Description:Inhibitory activity against Oxidosqualene-lanosterol cyclase from Rat liver microsomesMore data for this Ligand-Target Pair
Affinity DataIC50: >2.50E+4nMAssay Description:Inhibitory activity against Oxidosqualene-lanosterol cyclase from Rat liver microsomesMore data for this Ligand-Target Pair
Affinity DataIC50: >2.50E+4nMAssay Description:Inhibitory activity against Oxidosqualene-lanosterol cyclase from Rat liver microsomesMore data for this Ligand-Target Pair
Affinity DataIC50: >2.50E+4nMAssay Description:Inhibitory activity against Oxidosqualene-lanosterol cyclase from Rat liver microsomesMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibitory activity against Oxidosqualene-lanosterol cyclase from Rat liver microsomesMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibitory activity against Oxidosqualene-lanosterol cyclase from Rat liver microsomesMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Inventiva
Curated by ChEMBL
Inventiva
Curated by ChEMBL
Affinity DataEC50: 1.91E+3nMAssay Description:Transactivation of human GAL4-fused PPARdelta LBD expressed in African green monkey COS7 cells co-expressing 5Gal4 pGL3 TK Luc after overnight incuba...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Inventiva
Curated by ChEMBL
Inventiva
Curated by ChEMBL
Affinity DataEC50: >5.00E+3nMAssay Description:Transactivation of human GAL4-fused PPARdelta LBD expressed in African green monkey COS7 cells co-expressing 5Gal4 pGL3 TK Luc after overnight incuba...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Inventiva
Curated by ChEMBL
Inventiva
Curated by ChEMBL
Affinity DataEC50: >5.00E+3nMAssay Description:Transactivation of human GAL4-fused PPARdelta LBD expressed in African green monkey COS7 cells co-expressing 5Gal4 pGL3 TK Luc after overnight incuba...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Inventiva
Curated by ChEMBL
Inventiva
Curated by ChEMBL
Affinity DataEC50: 1.61E+3nMAssay Description:Transactivation of human GAL4-fused PPARdelta LBD expressed in African green monkey COS7 cells co-expressing 5Gal4 pGL3 TK Luc after overnight incuba...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Inventiva
Curated by ChEMBL
Inventiva
Curated by ChEMBL
Affinity DataEC50: 2.03E+3nMAssay Description:Transactivation of human GAL4-fused PPARdelta LBD expressed in African green monkey COS7 cells co-expressing 5Gal4 pGL3 TK Luc after overnight incuba...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Inventiva
Curated by ChEMBL
Inventiva
Curated by ChEMBL
Affinity DataEC50: 1.65E+3nMAssay Description:Transactivation of human GAL4-fused PPARdelta LBD expressed in African green monkey COS7 cells co-expressing 5Gal4 pGL3 TK Luc after overnight incuba...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Inventiva
Curated by ChEMBL
Inventiva
Curated by ChEMBL
Affinity DataEC50: 2.10E+3nMAssay Description:Transactivation of human GAL4-fused PPARdelta LBD expressed in African green monkey COS7 cells co-expressing 5Gal4 pGL3 TK Luc after overnight incuba...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Inventiva
Curated by ChEMBL
Inventiva
Curated by ChEMBL
Affinity DataEC50: 1.23E+3nMAssay Description:Transactivation of human GAL4-fused PPARdelta LBD expressed in African green monkey COS7 cells co-expressing 5Gal4 pGL3 TK Luc after overnight incuba...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Inventiva
Curated by ChEMBL
Inventiva
Curated by ChEMBL
Affinity DataEC50: 1.35E+3nMAssay Description:Transactivation of human GAL4-fused PPARdelta LBD expressed in African green monkey COS7 cells co-expressing 5Gal4 pGL3 TK Luc after overnight incuba...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Inventiva
Curated by ChEMBL
Inventiva
Curated by ChEMBL
Affinity DataEC50: 697nMAssay Description:Transactivation of human GAL4-fused PPARdelta LBD expressed in African green monkey COS7 cells co-expressing 5Gal4 pGL3 TK Luc after overnight incuba...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Inventiva
Curated by ChEMBL
Inventiva
Curated by ChEMBL
Affinity DataEC50: 977nMAssay Description:Transactivation of human GAL4-fused PPARdelta LBD expressed in African green monkey COS7 cells co-expressing 5Gal4 pGL3 TK Luc after overnight incuba...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Inventiva
Curated by ChEMBL
Inventiva
Curated by ChEMBL
Affinity DataEC50: 866nMAssay Description:Transactivation of human GAL4-fused PPARdelta LBD expressed in African green monkey COS7 cells co-expressing 5Gal4 pGL3 TK Luc after overnight incuba...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Inventiva
Curated by ChEMBL
Inventiva
Curated by ChEMBL
Affinity DataEC50: 1.56E+3nMAssay Description:Transactivation of human GAL4-fused PPARgamma LBD expressed in African green monkey COS7 cells co-expressing 5Gal4 pGL3 TK Luc after overnight incuba...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Inventiva
Curated by ChEMBL
Inventiva
Curated by ChEMBL
Affinity DataEC50: 284nMAssay Description:Transactivation of human GAL4-fused PPARgamma LBD expressed in African green monkey COS7 cells co-expressing 5Gal4 pGL3 TK Luc after overnight incuba...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Inventiva
Curated by ChEMBL
Inventiva
Curated by ChEMBL
Affinity DataEC50: 417nMAssay Description:Transactivation of human GAL4-fused PPARgamma LBD expressed in African green monkey COS7 cells co-expressing 5Gal4 pGL3 TK Luc after overnight incuba...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Inventiva
Curated by ChEMBL
Inventiva
Curated by ChEMBL
Affinity DataEC50: 284nMAssay Description:Transactivation of human GAL4-fused PPARgamma LBD expressed in African green monkey COS7 cells co-expressing 5Gal4 pGL3 TK Luc after overnight incuba...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Inventiva
Curated by ChEMBL
Inventiva
Curated by ChEMBL
Affinity DataEC50: 65nMAssay Description:Transactivation of human GAL4-fused PPARgamma LBD expressed in African green monkey COS7 cells co-expressing 5Gal4 pGL3 TK Luc after overnight incuba...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Inventiva
Curated by ChEMBL
Inventiva
Curated by ChEMBL
Affinity DataEC50: 1.25E+3nMAssay Description:Transactivation of human GAL4-fused PPARgamma LBD expressed in African green monkey COS7 cells co-expressing 5Gal4 pGL3 TK Luc after overnight incuba...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Inventiva
Curated by ChEMBL
Inventiva
Curated by ChEMBL
Affinity DataEC50: 256nMAssay Description:Transactivation of human GAL4-fused PPARgamma LBD expressed in African green monkey COS7 cells co-expressing 5Gal4 pGL3 TK Luc after overnight incuba...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Inventiva
Curated by ChEMBL
Inventiva
Curated by ChEMBL
Affinity DataEC50: >5.00E+3nMAssay Description:Transactivation of human GAL4-fused PPARgamma LBD expressed in African green monkey COS7 cells co-expressing 5Gal4 pGL3 TK Luc after overnight incuba...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Inventiva
Curated by ChEMBL
Inventiva
Curated by ChEMBL
Affinity DataEC50: 201nMAssay Description:Transactivation of human GAL4-fused PPARgamma LBD expressed in African green monkey COS7 cells co-expressing 5Gal4 pGL3 TK Luc after overnight incuba...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Inventiva
Curated by ChEMBL
Inventiva
Curated by ChEMBL
Affinity DataEC50: 573nMAssay Description:Transactivation of human GAL4-fused PPARgamma LBD expressed in African green monkey COS7 cells co-expressing 5Gal4 pGL3 TK Luc after overnight incuba...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Inventiva
Curated by ChEMBL
Inventiva
Curated by ChEMBL
Affinity DataEC50: 72nMAssay Description:Transactivation of human GAL4-fused PPARgamma LBD expressed in African green monkey COS7 cells co-expressing 5Gal4 pGL3 TK Luc after overnight incuba...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Inventiva
Curated by ChEMBL
Inventiva
Curated by ChEMBL
Affinity DataEC50: 75nMAssay Description:Transactivation of human GAL4-fused PPARgamma LBD expressed in African green monkey COS7 cells co-expressing 5Gal4 pGL3 TK Luc after overnight incuba...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Inventiva
Curated by ChEMBL
Inventiva
Curated by ChEMBL
Affinity DataEC50: 277nMAssay Description:Transactivation of human GAL4-fused PPARgamma LBD expressed in African green monkey COS7 cells co-expressing 5Gal4 pGL3 TK Luc after overnight incuba...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Inventiva
Curated by ChEMBL
Inventiva
Curated by ChEMBL
Affinity DataEC50: 71nMAssay Description:Transactivation of human GAL4-fused PPARgamma LBD expressed in African green monkey COS7 cells co-expressing 5Gal4 pGL3 TK Luc after overnight incuba...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Inventiva
Curated by ChEMBL
Inventiva
Curated by ChEMBL
Affinity DataEC50: 206nMAssay Description:Transactivation of human GAL4-fused PPARgamma LBD expressed in African green monkey COS7 cells co-expressing 5Gal4 pGL3 TK Luc after overnight incuba...More data for this Ligand-Target Pair