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Found 121 with Last Name = 'binet' and Initial = 'j'
TargetLanosterol synthase(Rattus norvegicus)
Laboratoires Fournier

Curated by ChEMBL
LigandPNGBDBM50051375((6S,8aS)-5,5,8a-Trimethyl-2-((E)-1,5,9-trimethyl-d...)
Affinity DataKi:  300nMAssay Description:Binding affinity towards competitive inhibition against rat microsomal Oxidosqualene-lanosterol cyclaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLanosterol synthase(Rattus norvegicus)
Laboratoires Fournier

Curated by ChEMBL
LigandPNGBDBM50051375((6S,8aS)-5,5,8a-Trimethyl-2-((E)-1,5,9-trimethyl-d...)
Affinity DataKi:  400nMAssay Description:Binding affinity towards noncompetetive inhibition against rat microsomal Oxidosqualene-lanosterol cyclaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLanosterol synthase(Rattus norvegicus)
Laboratoires Fournier

Curated by ChEMBL
LigandPNGBDBM50051383((4aR,6S,8aS)-2-((E)-5,9-Dimethyl-deca-4,8-dienyl)-...)
Affinity DataIC50:  100nMAssay Description:Inhibitory activity against Oxidosqualene-lanosterol cyclase from Rat liver microsomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLanosterol synthase(Rattus norvegicus)
Laboratoires Fournier

Curated by ChEMBL
LigandPNGBDBM50051372((6R,8aR)-2-((E)-5,9-Dimethyl-deca-4,8-dienyl)-5,5,...)
Affinity DataIC50:  600nMAssay Description:Inhibitory activity against Oxidosqualene-lanosterol cyclase from Rat liver microsomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLanosterol synthase(Rattus norvegicus)
Laboratoires Fournier

Curated by ChEMBL
LigandPNGBDBM50051375((6S,8aS)-5,5,8a-Trimethyl-2-((E)-1,5,9-trimethyl-d...)
Affinity DataIC50:  600nMAssay Description:Inhibitory activity against Oxidosqualene-lanosterol cyclase from Rat liver microsomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLanosterol synthase(Rattus norvegicus)
Laboratoires Fournier

Curated by ChEMBL
LigandPNGBDBM50051372((6R,8aR)-2-((E)-5,9-Dimethyl-deca-4,8-dienyl)-5,5,...)
Affinity DataIC50:  600nMAssay Description:Inhibitory activity against Oxidosqualene-lanosterol cyclase from Rat liver microsomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLanosterol synthase(Rattus norvegicus)
Laboratoires Fournier

Curated by ChEMBL
LigandPNGBDBM50051371(1,1,4a-Trimethyl-5-(4,8,12-trimethyl-trideca-3,7,1...)
Affinity DataIC50:  600nMAssay Description:Inhibitory activity against Oxidosqualene-lanosterol cyclase from Rat liver microsomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLanosterol synthase(Rattus norvegicus)
Laboratoires Fournier

Curated by ChEMBL
LigandPNGBDBM50051366((E)-1-((6S,8aS)-6-Hydroxy-5,5,8a-trimethyl-3,5,6,7...)
Affinity DataIC50:  680nMAssay Description:Inhibitory activity against Oxidosqualene-lanosterol cyclase from Rat liver microsomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLanosterol synthase(Rattus norvegicus)
Laboratoires Fournier

Curated by ChEMBL
LigandPNGBDBM50051380((4aS,6S,8aS)-2-((E)-5,9-Dimethyl-deca-4,8-dienyl)-...)
Affinity DataIC50:  700nMAssay Description:Inhibitory activity against Oxidosqualene-lanosterol cyclase from Rat liver microsomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLanosterol synthase(Rattus norvegicus)
Laboratoires Fournier

Curated by ChEMBL
LigandPNGBDBM50051376((4aR,6S,8aS)-2-((E)-5,9-Dimethyl-deca-4,8-dienyl)-...)
Affinity DataIC50:  900nMAssay Description:Inhibitory activity against Oxidosqualene-lanosterol cyclase from Rat liver microsomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLanosterol synthase(Rattus norvegicus)
Laboratoires Fournier

Curated by ChEMBL
LigandPNGBDBM50051368((6S,8aS)-2-((E)-5,9-Dimethyl-deca-4,8-dienyl)-5,5,...)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibitory activity against Oxidosqualene-lanosterol cyclase from Rat liver microsomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLanosterol synthase(Rattus norvegicus)
Laboratoires Fournier

Curated by ChEMBL
LigandPNGBDBM50051373((6S,8aS)-2-Dodecyl-5,5,8a-trimethyl-1,2,3,5,6,7,8,...)
Affinity DataIC50:  1.10E+3nMAssay Description:Inhibitory activity against Oxidosqualene-lanosterol cyclase from Rat liver microsomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLanosterol synthase(Rattus norvegicus)
Laboratoires Fournier

Curated by ChEMBL
LigandPNGBDBM50051379((6S,8aS)-5,5,8a-Trimethyl-2-tetradecyl-1,2,3,5,6,7...)
Affinity DataIC50:  2.90E+3nMAssay Description:Inhibitory activity against Oxidosqualene-lanosterol cyclase from Rat liver microsomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLanosterol synthase(Rattus norvegicus)
Laboratoires Fournier

Curated by ChEMBL
LigandPNGBDBM50051370((6S,8aS)-5,5,8a-Trimethyl-2-((Z)-1,5,9-trimethyl-d...)
Affinity DataIC50:  6.80E+3nMAssay Description:Inhibitory activity against Oxidosqualene-lanosterol cyclase from Rat liver microsomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLanosterol synthase(Rattus norvegicus)
Laboratoires Fournier

Curated by ChEMBL
LigandPNGBDBM50051382((6S,8aS)-2-Dodecyl-8a-methyl-1,2,3,5,6,7,8,8a-octa...)
Affinity DataIC50:  1.64E+4nMAssay Description:Inhibitory activity against Oxidosqualene-lanosterol cyclase from Rat liver microsomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLanosterol synthase(Rattus norvegicus)
Laboratoires Fournier

Curated by ChEMBL
LigandPNGBDBM50051367((6S,8aS)-2-(1,5-Dimethyl-hex-4-enyl)-5,5,8a-trimet...)
Affinity DataIC50:  1.70E+4nMAssay Description:Inhibitory activity against Oxidosqualene-lanosterol cyclase from Rat liver microsomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLanosterol synthase(Rattus norvegicus)
Laboratoires Fournier

Curated by ChEMBL
LigandPNGBDBM50051381((6R,8aS)-2-((E)-5,9-Dimethyl-deca-4,8-dienyl)-5,5,...)
Affinity DataIC50:  2.00E+4nMAssay Description:Inhibitory activity against Oxidosqualene-lanosterol cyclase from Rat liver microsomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLanosterol synthase(Rattus norvegicus)
Laboratoires Fournier

Curated by ChEMBL
LigandPNGBDBM50051378((6S,8aS)-2-Benzyl-5,5,8a-trimethyl-1,2,3,5,6,7,8,8...)
Affinity DataIC50:  2.50E+4nMAssay Description:Inhibitory activity against Oxidosqualene-lanosterol cyclase from Rat liver microsomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLanosterol synthase(Rattus norvegicus)
Laboratoires Fournier

Curated by ChEMBL
LigandPNGBDBM50051365((6S,8aS)-5,5,8a-Trimethyl-2-(3-phenyl-propyl)-1,2,...)
Affinity DataIC50: >2.50E+4nMAssay Description:Inhibitory activity against Oxidosqualene-lanosterol cyclase from Rat liver microsomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLanosterol synthase(Rattus norvegicus)
Laboratoires Fournier

Curated by ChEMBL
LigandPNGBDBM50003030((2S,4aS,8aR)-1,1,4a-Trimethyl-decahydro-naphthalen...)
Affinity DataIC50: >2.50E+4nMAssay Description:Inhibitory activity against Oxidosqualene-lanosterol cyclase from Rat liver microsomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLanosterol synthase(Rattus norvegicus)
Laboratoires Fournier

Curated by ChEMBL
LigandPNGBDBM50051377((4aR,8aS)-2-Dodecyl-5,5-dimethyl-decahydro-isoquin...)
Affinity DataIC50: >2.50E+4nMAssay Description:Inhibitory activity against Oxidosqualene-lanosterol cyclase from Rat liver microsomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLanosterol synthase(Rattus norvegicus)
Laboratoires Fournier

Curated by ChEMBL
LigandPNGBDBM50051374((6S,8aS)-5,5,8a-Trimethyl-1,2,3,5,6,7,8,8a-octahyd...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibitory activity against Oxidosqualene-lanosterol cyclase from Rat liver microsomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLanosterol synthase(Rattus norvegicus)
Laboratoires Fournier

Curated by ChEMBL
LigandPNGBDBM50051369((6S,8aS)-5,5,8a-Trimethyl-2-octadecyl-1,2,3,5,6,7,...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibitory activity against Oxidosqualene-lanosterol cyclase from Rat liver microsomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Inventiva

Curated by ChEMBL
LigandPNGBDBM50244312(CHEMBL4074391)
Affinity DataEC50:  1.91E+3nMAssay Description:Transactivation of human GAL4-fused PPARdelta LBD expressed in African green monkey COS7 cells co-expressing 5Gal4 pGL3 TK Luc after overnight incuba...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Inventiva

Curated by ChEMBL
LigandPNGBDBM50244314(CHEMBL4079308)
Affinity DataEC50: >5.00E+3nMAssay Description:Transactivation of human GAL4-fused PPARdelta LBD expressed in African green monkey COS7 cells co-expressing 5Gal4 pGL3 TK Luc after overnight incuba...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Inventiva

Curated by ChEMBL
LigandPNGBDBM50244315(CHEMBL4095821)
Affinity DataEC50: >5.00E+3nMAssay Description:Transactivation of human GAL4-fused PPARdelta LBD expressed in African green monkey COS7 cells co-expressing 5Gal4 pGL3 TK Luc after overnight incuba...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Inventiva

Curated by ChEMBL
LigandPNGBDBM50244324(CHEMBL4081907)
Affinity DataEC50:  1.61E+3nMAssay Description:Transactivation of human GAL4-fused PPARdelta LBD expressed in African green monkey COS7 cells co-expressing 5Gal4 pGL3 TK Luc after overnight incuba...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Inventiva

Curated by ChEMBL
LigandPNGBDBM50244325(CHEMBL4067479)
Affinity DataEC50:  2.03E+3nMAssay Description:Transactivation of human GAL4-fused PPARdelta LBD expressed in African green monkey COS7 cells co-expressing 5Gal4 pGL3 TK Luc after overnight incuba...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Inventiva

Curated by ChEMBL
LigandPNGBDBM50244326(CHEMBL4062724)
Affinity DataEC50:  1.65E+3nMAssay Description:Transactivation of human GAL4-fused PPARdelta LBD expressed in African green monkey COS7 cells co-expressing 5Gal4 pGL3 TK Luc after overnight incuba...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Inventiva

Curated by ChEMBL
LigandPNGBDBM50244345(CHEMBL4098415)
Affinity DataEC50:  2.10E+3nMAssay Description:Transactivation of human GAL4-fused PPARdelta LBD expressed in African green monkey COS7 cells co-expressing 5Gal4 pGL3 TK Luc after overnight incuba...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Inventiva

Curated by ChEMBL
LigandPNGBDBM50244346(CHEMBL4093146)
Affinity DataEC50:  1.23E+3nMAssay Description:Transactivation of human GAL4-fused PPARdelta LBD expressed in African green monkey COS7 cells co-expressing 5Gal4 pGL3 TK Luc after overnight incuba...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Inventiva

Curated by ChEMBL
LigandPNGBDBM50244347(CHEMBL4073181)
Affinity DataEC50:  1.35E+3nMAssay Description:Transactivation of human GAL4-fused PPARdelta LBD expressed in African green monkey COS7 cells co-expressing 5Gal4 pGL3 TK Luc after overnight incuba...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Inventiva

Curated by ChEMBL
LigandPNGBDBM50244348(CHEMBL4083589)
Affinity DataEC50:  697nMAssay Description:Transactivation of human GAL4-fused PPARdelta LBD expressed in African green monkey COS7 cells co-expressing 5Gal4 pGL3 TK Luc after overnight incuba...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Inventiva

Curated by ChEMBL
LigandPNGBDBM50244349(CHEMBL4101596)
Affinity DataEC50:  977nMAssay Description:Transactivation of human GAL4-fused PPARdelta LBD expressed in African green monkey COS7 cells co-expressing 5Gal4 pGL3 TK Luc after overnight incuba...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Inventiva

Curated by ChEMBL
LigandPNGBDBM50244350(CHEMBL4091374)
Affinity DataEC50:  866nMAssay Description:Transactivation of human GAL4-fused PPARdelta LBD expressed in African green monkey COS7 cells co-expressing 5Gal4 pGL3 TK Luc after overnight incuba...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Inventiva

Curated by ChEMBL
LigandPNGBDBM50244312(CHEMBL4074391)
Affinity DataEC50:  1.56E+3nMAssay Description:Transactivation of human GAL4-fused PPARgamma LBD expressed in African green monkey COS7 cells co-expressing 5Gal4 pGL3 TK Luc after overnight incuba...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Inventiva

Curated by ChEMBL
LigandPNGBDBM50244361(CHEMBL4094877)
Affinity DataEC50:  284nMAssay Description:Transactivation of human GAL4-fused PPARgamma LBD expressed in African green monkey COS7 cells co-expressing 5Gal4 pGL3 TK Luc after overnight incuba...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Inventiva

Curated by ChEMBL
LigandPNGBDBM50244314(CHEMBL4079308)
Affinity DataEC50:  417nMAssay Description:Transactivation of human GAL4-fused PPARgamma LBD expressed in African green monkey COS7 cells co-expressing 5Gal4 pGL3 TK Luc after overnight incuba...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Inventiva

Curated by ChEMBL
LigandPNGBDBM50244315(CHEMBL4095821)
Affinity DataEC50:  284nMAssay Description:Transactivation of human GAL4-fused PPARgamma LBD expressed in African green monkey COS7 cells co-expressing 5Gal4 pGL3 TK Luc after overnight incuba...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Inventiva

Curated by ChEMBL
LigandPNGBDBM50244324(CHEMBL4081907)
Affinity DataEC50:  65nMAssay Description:Transactivation of human GAL4-fused PPARgamma LBD expressed in African green monkey COS7 cells co-expressing 5Gal4 pGL3 TK Luc after overnight incuba...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Inventiva

Curated by ChEMBL
LigandPNGBDBM50244362(CHEMBL4089775)
Affinity DataEC50:  1.25E+3nMAssay Description:Transactivation of human GAL4-fused PPARgamma LBD expressed in African green monkey COS7 cells co-expressing 5Gal4 pGL3 TK Luc after overnight incuba...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Inventiva

Curated by ChEMBL
LigandPNGBDBM50244325(CHEMBL4067479)
Affinity DataEC50:  256nMAssay Description:Transactivation of human GAL4-fused PPARgamma LBD expressed in African green monkey COS7 cells co-expressing 5Gal4 pGL3 TK Luc after overnight incuba...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Inventiva

Curated by ChEMBL
LigandPNGBDBM50244363(CHEMBL4090691)
Affinity DataEC50: >5.00E+3nMAssay Description:Transactivation of human GAL4-fused PPARgamma LBD expressed in African green monkey COS7 cells co-expressing 5Gal4 pGL3 TK Luc after overnight incuba...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Inventiva

Curated by ChEMBL
LigandPNGBDBM50244364(CHEMBL4071373)
Affinity DataEC50:  201nMAssay Description:Transactivation of human GAL4-fused PPARgamma LBD expressed in African green monkey COS7 cells co-expressing 5Gal4 pGL3 TK Luc after overnight incuba...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Inventiva

Curated by ChEMBL
LigandPNGBDBM50244345(CHEMBL4098415)
Affinity DataEC50:  573nMAssay Description:Transactivation of human GAL4-fused PPARgamma LBD expressed in African green monkey COS7 cells co-expressing 5Gal4 pGL3 TK Luc after overnight incuba...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Inventiva

Curated by ChEMBL
LigandPNGBDBM50244392(CHEMBL4072395)
Affinity DataEC50:  72nMAssay Description:Transactivation of human GAL4-fused PPARgamma LBD expressed in African green monkey COS7 cells co-expressing 5Gal4 pGL3 TK Luc after overnight incuba...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Inventiva

Curated by ChEMBL
LigandPNGBDBM50244347(CHEMBL4073181)
Affinity DataEC50:  75nMAssay Description:Transactivation of human GAL4-fused PPARgamma LBD expressed in African green monkey COS7 cells co-expressing 5Gal4 pGL3 TK Luc after overnight incuba...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Inventiva

Curated by ChEMBL
LigandPNGBDBM50244393(CHEMBL4093864)
Affinity DataEC50:  277nMAssay Description:Transactivation of human GAL4-fused PPARgamma LBD expressed in African green monkey COS7 cells co-expressing 5Gal4 pGL3 TK Luc after overnight incuba...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Inventiva

Curated by ChEMBL
LigandPNGBDBM50244349(CHEMBL4101596)
Affinity DataEC50:  71nMAssay Description:Transactivation of human GAL4-fused PPARgamma LBD expressed in African green monkey COS7 cells co-expressing 5Gal4 pGL3 TK Luc after overnight incuba...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Inventiva

Curated by ChEMBL
LigandPNGBDBM50244350(CHEMBL4091374)
Affinity DataEC50:  206nMAssay Description:Transactivation of human GAL4-fused PPARgamma LBD expressed in African green monkey COS7 cells co-expressing 5Gal4 pGL3 TK Luc after overnight incuba...More data for this Ligand-Target Pair
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