Affinity DataKi: 16nMAssay Description:Antagonist activity at human CXCR3 expressed in CHO cells by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 28nMAssay Description:Antagonist activity at human CXCR3 expressed in CHO cells by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 29nMAssay Description:Antagonist activity at human CXCR3 expressed in CHO cells by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 31nMAssay Description:Antagonist activity at human CXCR3 expressed in CHO cells by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 36nMAssay Description:Antagonist activity at human CXCR3 expressed in CHO cells by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 39nMAssay Description:Antagonist activity at human CXCR3 expressed in CHO cells by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 41nMAssay Description:Antagonist activity at human CXCR3 expressed in CHO cells by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 46nMAssay Description:Antagonist activity at human CXCR3 expressed in CHO cells by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 47nMAssay Description:Antagonist activity at human CXCR3 expressed in CHO cells by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 70nMAssay Description:Antagonist activity at human CXCR3 expressed in CHO cells by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 73nMAssay Description:Antagonist activity at human CXCR3 expressed in CHO cells by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 81nMAssay Description:Antagonist activity at human CXCR3 expressed in CHO cells by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 83nMAssay Description:Antagonist activity at human CXCR3 expressed in CHO cells by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 88nMAssay Description:Antagonist activity at human CXCR3 expressed in CHO cells by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 104nMAssay Description:Antagonist activity at human CXCR3 expressed in CHO cells by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 107nMAssay Description:Antagonist activity at human CXCR3 expressed in CHO cells by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 108nMAssay Description:Antagonist activity at human CXCR3 expressed in CHO cells by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 110nMAssay Description:Antagonist activity at human CXCR3 expressed in CHO cells by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 141nMAssay Description:Antagonist activity at human CXCR3 expressed in CHO cells by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 171nMAssay Description:Antagonist activity at human CXCR3 expressed in CHO cells by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 171nMAssay Description:Antagonist activity at human CXCR3 expressed in CHO cells by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 175nMAssay Description:Antagonist activity at human CXCR3 expressed in CHO cells by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 191nMAssay Description:Antagonist activity at human CXCR3 expressed in CHO cells by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 191nMAssay Description:Antagonist activity at human CXCR3 expressed in CHO cells by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 201nMAssay Description:Antagonist activity at human CXCR3 expressed in CHO cells by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 229nMAssay Description:Antagonist activity at human CXCR3 expressed in CHO cells by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 258nMAssay Description:Antagonist activity at human CXCR3 expressed in CHO cells by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 290nMAssay Description:Antagonist activity at human CXCR3 expressed in CHO cells by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 306nMAssay Description:Antagonist activity at human CXCR3 expressed in CHO cells by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 376nMAssay Description:Antagonist activity at human CXCR3 expressed in CHO cells by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 400nMAssay Description:Antagonist activity at mouse CXCR3 by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 429nMAssay Description:Antagonist activity at human CXCR3 expressed in CHO cells by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 600nMAssay Description:Inhibition at human CYP2D6More data for this Ligand-Target Pair
Affinity DataKi: 637nMAssay Description:Antagonist activity at human CXCR3 expressed in CHO cells by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 660nMAssay Description:Antagonist activity at human CXCR3 expressed in CHO cells by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 1.04E+3nMAssay Description:Antagonist activity at human CXCR3 expressed in CHO cells by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 1.30E+3nMAssay Description:Antagonist activity at human CXCR3 expressed in CHO cells by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 2.00E+3nMAssay Description:Antagonist activity at human CXCR3 expressed in CHO cells by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 2.20E+3nMAssay Description:Antagonist activity at human CXCR3 expressed in CHO cells by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 3.40E+3nMAssay Description:Antagonist activity at human CXCR3 expressed in CHO cells by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
TargetSeed linoleate 13S-lipoxygenase-1(Glycine max (soybean))
Groningen Research Institute Of Pharmacy
Curated by ChEMBL
Groningen Research Institute Of Pharmacy
Curated by ChEMBL
Affinity DataKi: 9.80E+3nMAssay Description:Inhibition of soyabean lipoxygenase-1 assessed as inhibition constant for enzyme-inhibitor complex by Lineweaver-Burk plotMore data for this Ligand-Target Pair
TargetSeed linoleate 13S-lipoxygenase-1(Glycine max (soybean))
Groningen Research Institute Of Pharmacy
Curated by ChEMBL
Groningen Research Institute Of Pharmacy
Curated by ChEMBL
Affinity DataKi: 1.57E+4nMAssay Description:Inhibition of soyabean lipoxygenase-1 assessed as inhibition constant for enzyme-substrate-inhibitor complex by Lineweaver-Burk plotMore data for this Ligand-Target Pair
TargetTryptase delta(Homo sapiens (Human))
The Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by ChEMBL
The Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by ChEMBL
Affinity DataIC50: 0.400nMAssay Description:In vitro inhibition of human tryptase.More data for this Ligand-Target Pair
TargetTryptase delta(Homo sapiens (Human))
The Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by ChEMBL
The Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by ChEMBL
Affinity DataIC50: 0.700nMAssay Description:In vitro inhibition of human tryptase.More data for this Ligand-Target Pair
TargetTryptase delta(Homo sapiens (Human))
The Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by ChEMBL
The Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by ChEMBL
Affinity DataIC50: 0.700nMAssay Description:In vitro inhibition of human tryptase.More data for this Ligand-Target Pair
TargetTryptase beta-2/delta/gamma(Homo sapiens (Human))
The Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by ChEMBL
The Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by ChEMBL
Affinity DataIC50: 1nMAssay Description:Inhibitory activity against human tryptaseMore data for this Ligand-Target Pair
TargetTryptase delta(Homo sapiens (Human))
The Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by ChEMBL
The Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by ChEMBL
Affinity DataIC50: 1nMAssay Description:In vitro inhibition of human tryptase.More data for this Ligand-Target Pair
TargetTryptase beta-2/delta/gamma(Homo sapiens (Human))
The Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by ChEMBL
The Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by ChEMBL
Affinity DataIC50: 1nMAssay Description:Inhibitory activity against human tryptaseMore data for this Ligand-Target Pair
TargetTryptase beta-2/delta/gamma(Homo sapiens (Human))
The Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by ChEMBL
The Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by ChEMBL
Affinity DataIC50: 1nMAssay Description:Inhibitory activity against human tryptaseMore data for this Ligand-Target Pair
TargetTryptase beta-2/delta/gamma(Homo sapiens (Human))
The Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by ChEMBL
The Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by ChEMBL
Affinity DataIC50: 1nMAssay Description:Inhibitory activity against human tryptaseMore data for this Ligand-Target Pair