Affinity DataIC50: 1.20nMAssay Description:Binding affinity for rat brain Opioid receptor mu 1More data for this Ligand-Target Pair
Affinity DataIC50: 1.39nMAssay Description:Binding affinity for rat brain Opioid receptor mu 1More data for this Ligand-Target Pair
Affinity DataIC50: 12.1nMAssay Description:Binding affinity for rat brain Opioid receptor mu 1More data for this Ligand-Target Pair
Affinity DataIC50: 18.7nMAssay Description:Binding affinity for rat brain Opioid receptor mu 1More data for this Ligand-Target Pair
Affinity DataIC50: 20nMAssay Description:Binding affinity for rat brain Opioid receptor mu 1More data for this Ligand-Target Pair
Affinity DataIC50: 21nMAssay Description:Binding affinity for rat brain Opioid receptor mu 1More data for this Ligand-Target Pair
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
University Of Arizona
Curated by ChEMBL
University Of Arizona
Curated by ChEMBL
Affinity DataIC50: 100nMAssay Description:Inhibition of 1 nM alpha melanocortin stimulating hormone (MSH) from frog skinMore data for this Ligand-Target Pair
Affinity DataIC50: 173nMAssay Description:Binding affinity for rat brain Opioid receptor mu 1More data for this Ligand-Target Pair
Affinity DataIC50: 211nMAssay Description:Binding affinity for rat brain Opioid receptor delta 1More data for this Ligand-Target Pair
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
University Of Arizona
Curated by ChEMBL
University Of Arizona
Curated by ChEMBL
Affinity DataIC50: 500nMAssay Description:Inhibition of 1 nM alpha melanocortin stimulating hormone (MSH) from frog skinMore data for this Ligand-Target Pair
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
University Of Arizona
Curated by ChEMBL
University Of Arizona
Curated by ChEMBL
Affinity DataIC50: 500nMAssay Description:Inhibition of 1 nM alpha melanocortin stimulating hormone (MSH) from frog skinMore data for this Ligand-Target Pair
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
University Of Arizona
Curated by ChEMBL
University Of Arizona
Curated by ChEMBL
Affinity DataIC50: 500nMAssay Description:Inhibition of 1 nM alpha melanocortin stimulating hormone (MSH) from frog skinMore data for this Ligand-Target Pair
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
University Of Arizona
Curated by ChEMBL
University Of Arizona
Curated by ChEMBL
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of 1 nM alpha melanocortin stimulating hormone (MSH) from frog skinMore data for this Ligand-Target Pair
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
University Of Arizona
Curated by ChEMBL
University Of Arizona
Curated by ChEMBL
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of 1 nM alpha melanocortin stimulating hormone (MSH) from frog skinMore data for this Ligand-Target Pair
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
University Of Arizona
Curated by ChEMBL
University Of Arizona
Curated by ChEMBL
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of 1 nM alpha melanocortin stimulating hormone (MSH) from frog skinMore data for this Ligand-Target Pair
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
University Of Arizona
Curated by ChEMBL
University Of Arizona
Curated by ChEMBL
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of 1 nM alpha melanocortin stimulating hormone (MSH) from frog skinMore data for this Ligand-Target Pair
Affinity DataIC50: 1.19E+3nMAssay Description:Binding affinity for rat brain Opioid receptor delta 1More data for this Ligand-Target Pair
Affinity DataIC50: 1.27E+3nMAssay Description:Binding affinity for rat brain Opioid receptor delta 1More data for this Ligand-Target Pair
Affinity DataIC50: 1.32E+3nMAssay Description:Binding affinity for rat brain Opioid receptor delta 1More data for this Ligand-Target Pair
Affinity DataIC50: 1.36E+3nMAssay Description:Binding affinity for rat brain Opioid receptor mu 1More data for this Ligand-Target Pair
Affinity DataIC50: 1.50E+3nMAssay Description:Binding affinity for rat brain Opioid receptor mu 1More data for this Ligand-Target Pair
Affinity DataIC50: 3.40E+3nMAssay Description:Binding affinity for rat brain Opioid receptor mu 1More data for this Ligand-Target Pair
Affinity DataIC50: 3.53E+3nMAssay Description:Binding affinity for rat brain Opioid receptor delta 1More data for this Ligand-Target Pair
Affinity DataIC50: 3.64E+3nMAssay Description:Binding affinity for rat brain Opioid receptor delta 1More data for this Ligand-Target Pair
Affinity DataIC50: 5.42E+3nMAssay Description:Binding affinity for rat brain Opioid receptor mu 1More data for this Ligand-Target Pair
Affinity DataIC50: 7.46E+3nMAssay Description:Binding affinity for rat brain Opioid receptor delta 1More data for this Ligand-Target Pair
Affinity DataIC50: 7.48E+3nMAssay Description:Binding affinity for rat brain Opioid receptor delta 1More data for this Ligand-Target Pair
Affinity DataIC50: 9.18E+3nMAssay Description:Binding affinity for rat brain Opioid receptor delta 1More data for this Ligand-Target Pair
Affinity DataIC50: 1.32E+4nMAssay Description:Binding affinity for rat brain Opioid receptor delta 1More data for this Ligand-Target Pair
Affinity DataIC50: >1.50E+4nMAssay Description:Binding affinity for rat brain Opioid receptor delta 1More data for this Ligand-Target Pair
Affinity DataEC50: 0.0460nMAssay Description:Maximal agonist response of mouse melanocortin 1 receptor (MC1R)More data for this Ligand-Target Pair
Affinity DataEC50: 0.290nMAssay Description:Effective concentration for maximum agonist response towards mouse melanocortin 4 receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 0.100nMAssay Description:Maximal agonist response at rat melanocortin 3 receptor (MC3R)More data for this Ligand-Target Pair
Affinity DataEC50: 0.0640nMAssay Description:Maximum agonist response for mouse melanocortin 5 receptor (MC5R)More data for this Ligand-Target Pair
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
University Of Arizona
Curated by ChEMBL
University Of Arizona
Curated by ChEMBL
Affinity DataEC50: 100nMAssay Description:Effective concentration required for maximum agonist response at melanocortin 1 receptor from frog skin.More data for this Ligand-Target Pair
Affinity DataEC50: 0.0470nMAssay Description:Maximal agonist response of mouse melanocortin 1 receptor (MC1R)More data for this Ligand-Target Pair
Affinity DataEC50: 0.140nMAssay Description:Maximum agonist response for mouse melanocortin 5 receptor (MC5R)More data for this Ligand-Target Pair
Affinity DataEC50: 64nMAssay Description:Maximal agonist response at rat melanocortin 3 receptor (MC3R)More data for this Ligand-Target Pair
Affinity DataEC50: 0.380nMAssay Description:Effective concentration for maximum agonist response towards mouse melanocortin 4 receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 59nMAssay Description:Maximal agonist response of mouse melanocortin 1 receptor (MC1R)More data for this Ligand-Target Pair
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
University Of Arizona
Curated by ChEMBL
University Of Arizona
Curated by ChEMBL
Affinity DataEC50: 1nMAssay Description:Effective concentration required for maximum agonist response at melanocortin 1 receptor from frog skin.More data for this Ligand-Target Pair
Affinity DataEC50: 0.230nMAssay Description:Maximal agonist response of mouse melanocortin 1 receptor (MC1R)More data for this Ligand-Target Pair
Affinity DataEC50: 0.230nMAssay Description:Maximal agonist response at rat melanocortin 3 receptor (MC3R)More data for this Ligand-Target Pair
Affinity DataEC50: 0.200nMAssay Description:Effective concentration for maximum agonist response towards mouse melanocortin 4 receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 75nMAssay Description:Maximal agonist response at rat melanocortin 3 receptor (MC3R)More data for this Ligand-Target Pair
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
University Of Arizona
Curated by ChEMBL
University Of Arizona
Curated by ChEMBL
Affinity DataEC50: 30nMAssay Description:Effective concentration required for maximum agonist response at melanocortin 1 receptor from frog skin.More data for this Ligand-Target Pair
Affinity DataEC50: 3nMAssay Description:Maximal agonist response at rat melanocortin 3 receptor (MC3R)More data for this Ligand-Target Pair
Affinity DataEC50: 0.0740nMAssay Description:Maximum agonist response for mouse melanocortin 5 receptor (MC5R)More data for this Ligand-Target Pair
Affinity DataEC50: 0.230nMAssay Description:Maximal agonist response at rat melanocortin 3 receptor (MC3R)More data for this Ligand-Target Pair
Affinity DataEC50: 35nMAssay Description:Maximal agonist response of mouse melanocortin 1 receptor (MC1R)More data for this Ligand-Target Pair