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Found 137 with Last Name = 'bormans' and Initial = 'g'
TargetCannabinoid receptor 2(Homo sapiens (Human))
Helmholtz-Zentrum Dresden-Rossendorf (Hzdr)

Curated by ChEMBL
LigandPNGBDBM50600964(CHEMBL5181335)
Affinity DataKi:  0.400nMAssay Description:Displacement of [3H]-WIN55212-2 from human CB2 receptor transfected in CHO cells membrane incubated for 90 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Helmholtz-Zentrum Dresden-Rossendorf (Hzdr)

Curated by ChEMBL
LigandPNGBDBM50600966(CHEMBL5205138)
Affinity DataKi:  0.600nMAssay Description:Inhibition of human CB2 receptor assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Helmholtz-Zentrum Dresden-Rossendorf (Hzdr)

Curated by ChEMBL
LigandPNGBDBM50600961(CHEMBL5198892)
Affinity DataKi:  0.600nMAssay Description:Displacement of [3H]-SR141716A from recombinant human CB1 receptor expressed in CHO cells membrane incubated for 90 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Helmholtz-Zentrum Dresden-Rossendorf (Hzdr)

Curated by ChEMBL
LigandPNGBDBM50600965(CHEMBL5182619)
Affinity DataKi:  0.900nMAssay Description:Displacement of [3H]-WIN55212-2 from human CB2 receptor transfected in CHO-K1 cell membrane incubated for 90 mins by Liquid scintillation counter ana...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Helmholtz-Zentrum Dresden-Rossendorf (Hzdr)

Curated by ChEMBL
LigandPNGBDBM50600962(CHEMBL5186632)
Affinity DataKi:  1.5nMAssay Description:Displacement of [3H]-SR141716A from recombinant human CB1 receptor expressed in CHO cells membrane incubated for 90 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Helmholtz-Zentrum Dresden-Rossendorf (Hzdr)

Curated by ChEMBL
LigandPNGBDBM50029958(CHEMBL3353439)
Affinity DataKi:  1.70nMAssay Description:Displacement of [3H]-SR141716A from recombinant human CB1 receptor expressed in CHO cells membrane incubated for 90 minsMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Katholieke Universiteit Leuven

Curated by ChEMBL
LigandPNGBDBM50293110(2-(4-Fluorophenyl)-6-methoxybenzo[d]thiazole | 6-M...)
Affinity DataKi:  2.20nMAssay Description:Displacement of [125I]IMPY from beta-amyloid plaques in Alzheimer's disease patient brain homogenateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Katholieke Universiteit Leuven

Curated by ChEMBL
LigandPNGBDBM50129793(2-(4''-methylaminophenyl)-6-hydroxybenzothiazole |...)
Affinity DataKi:  2.80nMAssay Description:Displacement of [125I]IMPY from beta-amyloid plaques in Alzheimer's disease patient brain homogenateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Katholieke Universiteit Leuven

Curated by ChEMBL
LigandPNGBDBM50129793(2-(4''-methylaminophenyl)-6-hydroxybenzothiazole |...)
Affinity DataKi:  2.80nMAssay Description:Displacement of [125I]IMPY from beta-amyloid plaques in Alzheimer's disease patient brain homogenateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Katholieke Universiteit Leuven

Curated by ChEMBL
LigandPNGBDBM50129793(2-(4''-methylaminophenyl)-6-hydroxybenzothiazole |...)
Affinity DataKi:  2.80nMAssay Description:Displacement of [125I]IMPY from beta-amyloid plaques in Alzheimer's disease patient brain homogenateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Katholieke Universiteit Leuven

Curated by ChEMBL
LigandPNGBDBM50129793(2-(4''-methylaminophenyl)-6-hydroxybenzothiazole |...)
Affinity DataKi:  2.80nMAssay Description:Displacement of [125I]IMPY from beta-amyloid plaques in brain homogenate of patient with Alzheimer's disease by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Helmholtz-Zentrum Dresden-Rossendorf (Hzdr)

Curated by ChEMBL
LigandPNGBDBM50600942(CHEMBL5173419)
Affinity DataKi:  2.90nMAssay Description:Displacement of [3H]-SR141716A from recombinant human CB1 receptor expressed in CHO cells membrane incubated for 90 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Helmholtz-Zentrum Dresden-Rossendorf (Hzdr)

Curated by ChEMBL
LigandPNGBDBM50600948(CHEMBL5199801)
Affinity DataKi:  3.30nMAssay Description:Displacement of [3H]-SR141716A from recombinant human CB1 receptor expressed in CHO cells membrane incubated for 90 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Katholieke Universiteit Leuven

Curated by ChEMBL
LigandPNGBDBM50480917(CHEMBL566354)
Affinity DataKi:  3.80nMAssay Description:Displacement of [125I]IMPY from beta-amyloid plaques in Alzheimer's disease patient brain homogenateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Helmholtz-Zentrum Dresden-Rossendorf (Hzdr)

Curated by ChEMBL
LigandPNGBDBM50600963(CHEMBL5183565)
Affinity DataKi:  3.90nMAssay Description:Displacement of [3H]-SR141716A from recombinant human CB1 receptor expressed in CHO cells membrane incubated for 90 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Katholieke Universiteit Leuven

Curated by ChEMBL
LigandPNGBDBM50480918(CHEMBL578982)
Affinity DataKi:  4.10nMAssay Description:Displacement of [125I]IMPY from beta-amyloid plaques in Alzheimer's disease patient brain homogenateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Helmholtz-Zentrum Dresden-Rossendorf (Hzdr)

Curated by ChEMBL
LigandPNGBDBM50600950(CHEMBL5195027)
Affinity DataKi:  4.80nMAssay Description:Displacement of [3H]-SR141716A from recombinant human CB1 receptor expressed in CHO cells membrane incubated for 90 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Helmholtz-Zentrum Dresden-Rossendorf (Hzdr)

Curated by ChEMBL
LigandPNGBDBM50029962(CHEMBL3353450)
Affinity DataKi:  5nMAssay Description:Displacement of [3H]-SR141716A from recombinant human CB1 receptor expressed in CHO cells membrane incubated for 90 minsMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Katholieke Universiteit Leuven

Curated by ChEMBL
LigandPNGBDBM50479543(CHEMBL510384)
Affinity DataKi:  5.70nMAssay Description:Displacement of [125I]IMPY from beta-amyloid plaques in Alzheimer's disease patient brain homogenateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Katholieke Universiteit Leuven

Curated by ChEMBL
LigandPNGBDBM50479543(CHEMBL510384)
Affinity DataKi:  5.70nMAssay Description:Displacement of [125I]IMPY from beta-amyloid plaques in Alzheimer's disease patient brain homogenateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Helmholtz-Zentrum Dresden-Rossendorf (Hzdr)

Curated by ChEMBL
LigandPNGBDBM50600941(CHEMBL5173890)
Affinity DataKi:  6nMAssay Description:Displacement of [3H]-SR141716A from recombinant human CB1 receptor expressed in CHO cells membrane incubated for 90 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Katholieke Universiteit Leuven

Curated by ChEMBL
LigandPNGBDBM50479682(2-(4-Nitrophenyl)Benzo[D]Thiazole | CHEMBL477841)
Affinity DataKi:  9nMAssay Description:Displacement of [125I]IMPY from beta-amyloid plaques in Alzheimer's disease patient brain homogenateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Helmholtz-Zentrum Dresden-Rossendorf (Hzdr)

Curated by ChEMBL
LigandPNGBDBM50312837(CHEMBL1081610 | [11C]8-butoxy-N-cyclohexyl-7-metho...)
Affinity DataKi:  9.60nMAssay Description:Inhibition of human CB2 receptor assessed as inhibition constantMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Katholieke Universiteit Leuven

Curated by ChEMBL
LigandPNGBDBM50480919(CHEMBL568061)
Affinity DataKi:  10nMAssay Description:Displacement of [125I]IMPY from beta-amyloid plaques in Alzheimer's disease patient brain homogenateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Katholieke Universiteit Leuven

Curated by ChEMBL
LigandPNGBDBM50480215(CHEMBL486529)
Affinity DataKi:  11nMAssay Description:Displacement of [125I]IMPY from beta-amyloid plaques in brain homogenate of patient with Alzheimer's disease by gamma countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Katholieke Universiteit Leuven

Curated by ChEMBL
LigandPNGBDBM50480216(CHEMBL503833)
Affinity DataKi:  12nMAssay Description:Displacement of [125I]IMPY from beta-amyloid plaques in brain homogenate of patient with Alzheimer's disease by gamma countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Helmholtz-Zentrum Dresden-Rossendorf (Hzdr)

Curated by ChEMBL
LigandPNGBDBM50600953(CHEMBL5181324)
Affinity DataKi:  13nMAssay Description:Displacement of [3H]-SR141716A from recombinant human CB1 receptor expressed in CHO cells membrane incubated for 90 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Katholieke Universiteit Leuven

Curated by ChEMBL
LigandPNGBDBM50480217(CHEMBL524651)
Affinity DataKi:  19nMAssay Description:Displacement of [125I]IMPY from beta-amyloid plaques in brain homogenate of patient with Alzheimer's disease by gamma countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Katholieke Universiteit Leuven

Curated by ChEMBL
LigandPNGBDBM50479545(CHEMBL490084)
Affinity DataKi:  23nMAssay Description:Displacement of [125I]IMPY from beta-amyloid plaques in Alzheimer's disease patient brain homogenateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Helmholtz-Zentrum Dresden-Rossendorf (Hzdr)

Curated by ChEMBL
LigandPNGBDBM50349311(CHEMBL1807841)
Affinity DataKi:  27nMAssay Description:Displacement of [3H]-CP55940 from human CB2 receptor expressed in CHO cells after 1 hrs by beta countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Helmholtz-Zentrum Dresden-Rossendorf (Hzdr)

Curated by ChEMBL
LigandPNGBDBM50600946(CHEMBL5185306)
Affinity DataKi:  28nMAssay Description:Displacement of [3H]-SR141716A from recombinant human CB1 receptor expressed in CHO cells membrane incubated for 90 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Helmholtz-Zentrum Dresden-Rossendorf (Hzdr)

Curated by ChEMBL
LigandPNGBDBM50600949(CHEMBL5181748)
Affinity DataKi:  49nMAssay Description:Displacement of [3H]-SR141716A from recombinant human CB1 receptor expressed in CHO cells membrane incubated for 90 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Helmholtz-Zentrum Dresden-Rossendorf (Hzdr)

Curated by ChEMBL
LigandPNGBDBM50600944(CHEMBL5169843)
Affinity DataKi:  65nMAssay Description:Displacement of [3H]-SR141716A from recombinant human CB1 receptor expressed in CHO cells membrane incubated for 90 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Helmholtz-Zentrum Dresden-Rossendorf (Hzdr)

Curated by ChEMBL
LigandPNGBDBM50029961(CHEMBL3353449)
Affinity DataKi:  86nMAssay Description:Displacement of [3H]-SR141716A from recombinant human CB1 receptor expressed in CHO cells membrane incubated for 90 minsMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Helmholtz-Zentrum Dresden-Rossendorf (Hzdr)

Curated by ChEMBL
LigandPNGBDBM50600951(CHEMBL5184679)
Affinity DataKi:  115nMAssay Description:Displacement of [3H]-SR141716A from recombinant human CB1 receptor expressed in CHO cells membrane incubated for 90 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Helmholtz-Zentrum Dresden-Rossendorf (Hzdr)

Curated by ChEMBL
LigandPNGBDBM50029958(CHEMBL3353439)
Affinity DataKi: >155nMAssay Description:Displacement of [3H]-WIN55212-2 from human CB2 receptor transfected in CHO cells membrane incubated for 90 minsMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Katholieke Universiteit Leuven

Curated by ChEMBL
LigandPNGBDBM50479546(CHEMBL490085)
Affinity DataKi:  776nMAssay Description:Displacement of [125I]IMPY from beta-amyloid plaques in Alzheimer's disease patient brain homogenateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Helmholtz-Zentrum Dresden-Rossendorf (Hzdr)

Curated by ChEMBL
LigandPNGBDBM50600954(CHEMBL5177464)
Affinity DataKi:  780nMAssay Description:Displacement of [3H]-SR141716A from recombinant human CB1 receptor expressed in CHO cells membrane incubated for 90 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Helmholtz-Zentrum Dresden-Rossendorf (Hzdr)

Curated by ChEMBL
LigandPNGBDBM50029962(CHEMBL3353450)
Affinity DataKi:  915nMAssay Description:Displacement of [3H]-WIN55212-2 from human CB2 receptor transfected in CHO cells membrane incubated for 90 minsMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Helmholtz-Zentrum Dresden-Rossendorf (Hzdr)

Curated by ChEMBL
LigandPNGBDBM50600962(CHEMBL5186632)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]-WIN55212-2 from human CB2 receptor transfected in CHO cells membrane incubated for 90 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Helmholtz-Zentrum Dresden-Rossendorf (Hzdr)

Curated by ChEMBL
LigandPNGBDBM50600963(CHEMBL5183565)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]-WIN55212-2 from human CB2 receptor transfected in CHO cells membrane incubated for 90 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Helmholtz-Zentrum Dresden-Rossendorf (Hzdr)

Curated by ChEMBL
LigandPNGBDBM50600957(CHEMBL5170046)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]-SR141716A from recombinant human CB1 receptor expressed in CHO cells membrane incubated for 90 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Helmholtz-Zentrum Dresden-Rossendorf (Hzdr)

Curated by ChEMBL
LigandPNGBDBM50600959(CHEMBL5177747)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]-SR141716A from recombinant human CB1 receptor expressed in CHO cells membrane incubated for 90 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Helmholtz-Zentrum Dresden-Rossendorf (Hzdr)

Curated by ChEMBL
LigandPNGBDBM50600960(CHEMBL5208223)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]-SR141716A from recombinant human CB1 receptor expressed in CHO cells membrane incubated for 90 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Helmholtz-Zentrum Dresden-Rossendorf (Hzdr)

Curated by ChEMBL
LigandPNGBDBM50600941(CHEMBL5173890)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]-WIN55212-2 from human CB2 receptor transfected in CHO cells membrane incubated for 90 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Helmholtz-Zentrum Dresden-Rossendorf (Hzdr)

Curated by ChEMBL
LigandPNGBDBM50600961(CHEMBL5198892)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]-WIN55212-2 from human CB2 receptor transfected in CHO cells membrane incubated for 90 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Helmholtz-Zentrum Dresden-Rossendorf (Hzdr)

Curated by ChEMBL
LigandPNGBDBM50600958(CHEMBL5186106)
Affinity DataKi:  1.10E+3nMAssay Description:Displacement of [3H]-SR141716A from recombinant human CB1 receptor expressed in CHO cells membrane incubated for 90 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Helmholtz-Zentrum Dresden-Rossendorf (Hzdr)

Curated by ChEMBL
LigandPNGBDBM50600955(CHEMBL5192937)
Affinity DataKi:  2.20E+3nMAssay Description:Displacement of [3H]-SR141716A from recombinant human CB1 receptor expressed in CHO cells membrane incubated for 90 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Helmholtz-Zentrum Dresden-Rossendorf (Hzdr)

Curated by ChEMBL
LigandPNGBDBM50600956(CHEMBL5172791)
Affinity DataKi:  3.90E+3nMAssay Description:Displacement of [3H]-SR141716A from recombinant human CB1 receptor expressed in CHO cells membrane incubated for 90 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Katholieke Universiteit Leuven

Curated by ChEMBL
LigandPNGBDBM50479544(CHEMBL501127)
Affinity DataKi: >4.00E+3nMAssay Description:Displacement of [125I]IMPY from beta-amyloid plaques in Alzheimer's disease patient brain homogenateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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