Affinity DataKi: 0.790nMAssay Description:Displacement of [125I]ABA from human recombinant adenosine A3 receptor by rapid filtration techniqueMore data for this Ligand-Target Pair
Affinity DataKi: 2.22nMAssay Description:Displacement of [125I]ABA from human recombinant adenosine A3 receptor by rapid filtration techniqueMore data for this Ligand-Target Pair
Affinity DataKi: 2.25nMAssay Description:Displacement of [125I]ABA from human recombinant adenosine A3 receptor by rapid filtration techniqueMore data for this Ligand-Target Pair
Affinity DataKi: 4.26nMAssay Description:Displacement of [125I]ABA from human recombinant adenosine A3 receptor by rapid filtration techniqueMore data for this Ligand-Target Pair
TargetGlycine receptor subunit alpha-1(Homo sapiens (Human))
The German University In Cairo
Curated by ChEMBL
The German University In Cairo
Curated by ChEMBL
Affinity DataKi: 5nMAssay Description:Displacement of [3H]strychnine from human glycine receptor subunit alpha-1 expressed in HEK293 cell membranes preincubated for 30 mins followed by [3...More data for this Ligand-Target Pair
Affinity DataKi: 5.04nMAssay Description:Displacement of [125I]ABA from human recombinant adenosine A3 receptor by rapid filtration techniqueMore data for this Ligand-Target Pair
Affinity DataKi: 5.63nMAssay Description:Displacement of [125I]ABA from human recombinant adenosine A3 receptor by rapid filtration techniqueMore data for this Ligand-Target Pair
Affinity DataKi: 7nMAssay Description:Binding affinity to adenosine A3 receptorMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Homo sapiens (Human))
Monash University (Parkville Campus)
Curated by ChEMBL
Monash University (Parkville Campus)
Curated by ChEMBL
Affinity DataKi: 7nMAssay Description:Binding affinity to adenosine A1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 9nMAssay Description:Displacement of [125I]ABA from human recombinant adenosine A3 receptor by rapid filtration techniqueMore data for this Ligand-Target Pair
Affinity DataKi: 9.02nMAssay Description:Displacement of [125I]ABA from human recombinant adenosine A3 receptor by rapid filtration techniqueMore data for this Ligand-Target Pair
Affinity DataKi: 12nMAssay Description:Antagonist potency against adenosine A2B receptor of guinea pig thoracic aortic smooth muscleMore data for this Ligand-Target Pair
Affinity DataKi: 14nMAssay Description:Binding affinity to adenosine A3 receptorMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Homo sapiens (Human))
Monash University (Parkville Campus)
Curated by ChEMBL
Monash University (Parkville Campus)
Curated by ChEMBL
Affinity DataKi: 15nMAssay Description:Binding affinity to adenosine A1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 25nMAssay Description:Displacement of [125I]ABA from human recombinant adenosine A3 receptor by rapid filtration techniqueMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Homo sapiens (Human))
Monash University (Parkville Campus)
Curated by ChEMBL
Monash University (Parkville Campus)
Curated by ChEMBL
Affinity DataKi: 26.2nMAssay Description:Displacement of [125I]ABA from human recombinant adenosine A1 receptor by rapid filtration techniqueMore data for this Ligand-Target Pair
Affinity DataKi: 30nMAssay Description:Displacement of [125I]ABA from human recombinant adenosine A3 receptor by rapid filtration techniqueMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Homo sapiens (Human))
Monash University (Parkville Campus)
Curated by ChEMBL
Monash University (Parkville Campus)
Curated by ChEMBL
Affinity DataKi: 32nMAssay Description:Binding affinity to adenosine A1 receptorMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Homo sapiens (Human))
Monash University (Parkville Campus)
Curated by ChEMBL
Monash University (Parkville Campus)
Curated by ChEMBL
Affinity DataKi: 40nMAssay Description:Binding affinity to adenosine A1 receptorMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Homo sapiens (Human))
Monash University (Parkville Campus)
Curated by ChEMBL
Monash University (Parkville Campus)
Curated by ChEMBL
Affinity DataKi: 42.1nMAssay Description:Displacement of [125I]ABA from human recombinant adenosine A1 receptor by rapid filtration techniqueMore data for this Ligand-Target Pair
Affinity DataKi: 45nMAssay Description:Displacement of [125I]ABA from human recombinant adenosine A3 receptor by rapid filtration techniqueMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Homo sapiens (Human))
Monash University (Parkville Campus)
Curated by ChEMBL
Monash University (Parkville Campus)
Curated by ChEMBL
Affinity DataKi: 50nMAssay Description:Displacement of [125I]ABA from human recombinant adenosine A1 receptor by rapid filtration techniqueMore data for this Ligand-Target Pair
Affinity DataKi: 50nMAssay Description:Binding affinity to adenosine A3 receptorMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Homo sapiens (Human))
Monash University (Parkville Campus)
Curated by ChEMBL
Monash University (Parkville Campus)
Curated by ChEMBL
Affinity DataKi: 50nMAssay Description:Displacement of [125I]ABA from human recombinant adenosine A1 receptor by rapid filtration techniqueMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Homo sapiens (Human))
Monash University (Parkville Campus)
Curated by ChEMBL
Monash University (Parkville Campus)
Curated by ChEMBL
Affinity DataKi: 50nMAssay Description:Binding affinity to adenosine A1 receptorMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Homo sapiens (Human))
Monash University (Parkville Campus)
Curated by ChEMBL
Monash University (Parkville Campus)
Curated by ChEMBL
Affinity DataKi: 50nMAssay Description:Binding affinity to adenosine A1 receptorMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Homo sapiens (Human))
Monash University (Parkville Campus)
Curated by ChEMBL
Monash University (Parkville Campus)
Curated by ChEMBL
Affinity DataKi: 53.1nMAssay Description:Displacement of [125I]ABA from human recombinant adenosine A1 receptor by rapid filtration techniqueMore data for this Ligand-Target Pair
Affinity DataKi: 70nMAssay Description:Displacement of [125I]ABA from human recombinant adenosine A3 receptor by rapid filtration techniqueMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Homo sapiens (Human))
Monash University (Parkville Campus)
Curated by ChEMBL
Monash University (Parkville Campus)
Curated by ChEMBL
Affinity DataKi: 76.8nMAssay Description:Displacement of [125I]ABA from human recombinant adenosine A1 receptor by rapid filtration techniqueMore data for this Ligand-Target Pair
TargetGlycine receptor subunit alpha-1(Homo sapiens (Human))
The German University In Cairo
Curated by ChEMBL
The German University In Cairo
Curated by ChEMBL
Affinity DataKi: 81nMAssay Description:Displacement of [3H]strychnine from human glycine receptor subunit alpha-1 expressed in HEK293 cell membranes preincubated for 30 mins followed by [3...More data for this Ligand-Target Pair
Affinity DataKi: 84nMAssay Description:Binding affinity to adenosine A3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 89nMAssay Description:Binding affinity to adenosine A3 receptorMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Homo sapiens (Human))
Monash University (Parkville Campus)
Curated by ChEMBL
Monash University (Parkville Campus)
Curated by ChEMBL
Affinity DataKi: 100nMAssay Description:Displacement of [125I]ABA from human recombinant adenosine A1 receptor by rapid filtration techniqueMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Homo sapiens (Human))
Monash University (Parkville Campus)
Curated by ChEMBL
Monash University (Parkville Campus)
Curated by ChEMBL
Affinity DataKi: 100nMAssay Description:Binding affinity to adenosine A1 receptorMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Homo sapiens (Human))
Monash University (Parkville Campus)
Curated by ChEMBL
Monash University (Parkville Campus)
Curated by ChEMBL
Affinity DataKi: 105nMAssay Description:Displacement of [125I]ABA from human recombinant adenosine A1 receptor by rapid filtration techniqueMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Homo sapiens (Human))
Monash University (Parkville Campus)
Curated by ChEMBL
Monash University (Parkville Campus)
Curated by ChEMBL
Affinity DataKi: 128nMAssay Description:Displacement of [125I]ABA from human recombinant adenosine A1 receptor by rapid filtration techniqueMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Homo sapiens (Human))
Monash University (Parkville Campus)
Curated by ChEMBL
Monash University (Parkville Campus)
Curated by ChEMBL
Affinity DataKi: 150nMAssay Description:Displacement of [125I]ABA from human recombinant adenosine A1 receptor by rapid filtration techniqueMore data for this Ligand-Target Pair
TargetGlycine receptor subunit alpha-1(Homo sapiens (Human))
The German University In Cairo
Curated by ChEMBL
The German University In Cairo
Curated by ChEMBL
Affinity DataKi: 204nMAssay Description:Displacement of [3H]strychnine from human glycine receptor subunit alpha-1 expressed in HEK293 cell membranes preincubated for 30 mins followed by [3...More data for this Ligand-Target Pair
Affinity DataKi: 230nMAssay Description:Binding affinity to adenosine A3 receptorMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Homo sapiens (Human))
Monash University (Parkville Campus)
Curated by ChEMBL
Monash University (Parkville Campus)
Curated by ChEMBL
Affinity DataKi: 243nMAssay Description:Displacement of [125I]ABA from human recombinant adenosine A1 receptor by rapid filtration techniqueMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Homo sapiens (Human))
Monash University (Parkville Campus)
Curated by ChEMBL
Monash University (Parkville Campus)
Curated by ChEMBL
Affinity DataKi: 245nMAssay Description:Displacement of [125I]ABA from human recombinant adenosine A1 receptor by rapid filtration techniqueMore data for this Ligand-Target Pair
Affinity DataKi: 280nMAssay Description:Binding affinity to adenosine A3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 280nMAssay Description:Displacement of [125I]ABA from human recombinant adenosine A3 receptor by rapid filtration techniqueMore data for this Ligand-Target Pair
Affinity DataKi: 280nMAssay Description:Displacement of [125I]ABA from human recombinant adenosine A3 receptor by rapid filtration techniqueMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Homo sapiens (Human))
Monash University (Parkville Campus)
Curated by ChEMBL
Monash University (Parkville Campus)
Curated by ChEMBL
Affinity DataKi: 290nMAssay Description:Displacement of [125I]ABA from human recombinant adenosine A1 receptor by rapid filtration techniqueMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Homo sapiens (Human))
Monash University (Parkville Campus)
Curated by ChEMBL
Monash University (Parkville Campus)
Curated by ChEMBL
Affinity DataKi: 290nMAssay Description:Binding affinity to adenosine A1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 320nMAssay Description:Displacement of [125I]ABA from human recombinant adenosine A3 receptor by rapid filtration techniqueMore data for this Ligand-Target Pair
TargetGlycine receptor subunit alpha-1(Homo sapiens (Human))
The German University In Cairo
Curated by ChEMBL
The German University In Cairo
Curated by ChEMBL
Affinity DataKi: 436nMAssay Description:Displacement of [3H]strychnine from human glycine receptor subunit alpha-1 expressed in HEK293 cell membranes preincubated for 30 mins followed by [3...More data for this Ligand-Target Pair
Affinity DataKi: 530nMAssay Description:Displacement of [125I]ABA from human recombinant adenosine A3 receptor by rapid filtration techniqueMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Homo sapiens (Human))
Monash University (Parkville Campus)
Curated by ChEMBL
Monash University (Parkville Campus)
Curated by ChEMBL
Affinity DataKi: 570nMAssay Description:Displacement of [125I]ABA from human recombinant adenosine A1 receptor by rapid filtration techniqueMore data for this Ligand-Target Pair