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Found 18 with Last Name = 'bouaziz' and Initial = 's'
TargetNAD-dependent protein deacetylase sirtuin-1(Homo sapiens (Human))
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50190131(Oblongifolin C)
Affinity DataIC50:  9.00E+3nMAssay Description:Inhibition of human recombinant GST-fused SIRT1 expressed in Escherichia coli DH5-alpha using [3H]acetic acid labeled MPSDKTIGG as substrate after ov...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 1(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50223445(CHEMBL410408 | c[homoPhe-Hca-Glu-Gly-Leu-Glu-Glu]-...)
Affinity DataIC50:  1.93E+4nMAssay Description:Displacement of biotinylated VEGF165 from human recombinant VEGFR1 by chemiluminescent assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 1(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50221338(CHEMBL251540 | N3-GHQMFYYPra-NH2)
Affinity DataIC50:  1.94E+4nMAssay Description:Displacement of biotinylated VEGF165 from human recombinant VEGFR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNAD-dependent protein deacetylase sirtuin-2(Homo sapiens (Human))
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50190131(Oblongifolin C)
Affinity DataIC50:  2.20E+4nMAssay Description:Inhibition of human recombinant GST-fused SIRT2 expressed in Escherichia coli DH5-alpha using [3H]acetic acid labeled MPSDKTIGG as substrate after ov...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 1(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50221337(CHEMBL399724 | N3-GLDNKMIFWYPra-NH2)
Affinity DataIC50:  2.29E+4nMAssay Description:Displacement of biotinylated VEGF165 from human recombinant VEGFR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 1(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50223447(CHEMBL438299 | NGYEIEWYSWVTHGMY-NH2)
Affinity DataIC50:  2.80E+4nMAssay Description:Displacement of biotinylated VEGF165 from human recombinant VEGFR1 by chemiluminescent assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 1(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50221339(CHEMBL430206 | NGYEIEWYSWVTHGMY-NH2)
Affinity DataIC50:  2.80E+4nMAssay Description:Displacement of biotinylated VEGF165 from human recombinant VEGFR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNAD-dependent protein deacetylase sirtuin-1(Homo sapiens (Human))
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50195222(CHEMBL3894424)
Affinity DataIC50:  3.00E+4nMAssay Description:Inhibition of human SIRT1 preincubated with enzyme followed by Fluor de Lys substrate addition by fluorescence-based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 1(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50221335(CHEMBL398243 | Cyclo[GLDNKMIFWYbtA]-NH2)
Affinity DataIC50:  3.11E+4nMAssay Description:Displacement of biotinylated VEGF165 from human recombinant VEGFR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 1(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50223446(CHEMBL389147 | c[Tyr-Tyr-Asp-Glu-Gly-Leu-Glu-Glu]-...)
Affinity DataIC50:  3.99E+4nMAssay Description:Displacement of biotinylated VEGF165 from human recombinant VEGFR1 by chemiluminescent assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 1(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50221333(CHEMBL399914 | Cyclo[FYDEPLEbtA]-NH2)
Affinity DataIC50:  9.30E+4nMAssay Description:Displacement of biotinylated VEGF165 from human recombinant VEGFR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 1(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50221340(CHEMBL399500 | N3-FYDEPLEPra-NH2)
Affinity DataIC50:  9.60E+4nMAssay Description:Displacement of biotinylated VEGF165 from human recombinant VEGFR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 1(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50221336(CHEMBL249743 | Cyclo[GHQMFYYbtA]-NH2)
Affinity DataIC50:  1.21E+5nMAssay Description:Displacement of biotinylated VEGF165 from human recombinant VEGFR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNAD-dependent protein deacetylase sirtuin-2(Homo sapiens (Human))
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50195222(CHEMBL3894424)
Affinity DataIC50:  1.50E+5nMAssay Description:Inhibition of human SIRT2 preincubated with enzyme followed by Fluor de Lys substrate addition by fluorescence-based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 1(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50221332(CHEMBL248926 | N3-KYDEPLEPra-NH2)
Affinity DataIC50:  1.51E+5nMAssay Description:Displacement of biotinylated VEGF165 from human recombinant VEGFR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 1(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50221334(CHEMBL399245 | Cyclo[KYDEPLEbtA]-NH2)
Affinity DataIC50:  1.62E+5nMAssay Description:Displacement of biotinylated VEGF165 from human recombinant VEGFR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 1(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50521337(CHEMBL4592007)
Affinity DataIC50:  1.96E+5nMAssay Description:Displacement of biotinylated VEGF-A165 from human VEGFR-1 ECD incubated for 1 hr by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 1(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50521337(CHEMBL4592007)
Affinity DataKd:  6.21E+5nMAssay Description:Binding affinity to 15N-labeled VEGFR1 domain 2 (unknown origin) at 26 mM by TROSY [1H-15N] spectroscopic analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed