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Found 84 with Last Name = 'boucher' and Initial = 'jl'
TargetNitric oxide synthase, brain(Rattus norvegicus (rat))
Université

Curated by ChEMBL
LigandPNGBDBM50271277(1H-Indazole-7-carbonitrile | CHEMBL484298)
Affinity DataKi:  1.30E+4nMAssay Description:Activity of rat brain recombinant nNOS assessed as L-arginine oxidation in presence of 10 uM (6R)-5,6,7,8-tetrahydro-L-biopterinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, inducible(Mus musculus (mouse))
Christian-Albrechts-University Of Kiel

Curated by ChEMBL
LigandPNGBDBM50295565(3-[4'-(4''-Bromophenyl)benzoyl]-3,4-dihydro-8-meth...)
Affinity DataKi:  1.40E+4nMAssay Description:Inhibition of mouse iNOS expressed in insect Sf9 cells by competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, inducible(Mus musculus (mouse))
Christian-Albrechts-University Of Kiel

Curated by ChEMBL
LigandPNGBDBM50295567(3-[4'-(4''-Methoxyphenyl)benzoyl]-3,4-dihydro-8-me...)
Affinity DataKi:  1.50E+4nMAssay Description:Inhibition of mouse iNOS expressed in insect Sf9 cells by competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, inducible(Mus musculus (mouse))
Christian-Albrechts-University Of Kiel

Curated by ChEMBL
LigandPNGBDBM50295568(3,4-Dihydro-8-methyl-3-[2-(6-methylnaphthoyl)]-2H-...)
Affinity DataKi:  2.30E+4nMAssay Description:Inhibition of mouse iNOS expressed in insect Sf9 cells by competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, brain(Rattus norvegicus (rat))
Université

Curated by ChEMBL
LigandPNGBDBM50270528(3-BROMO-7-NITROINDAZOLE | 3-bromo-7-nitro-1H-indaz...)
Affinity DataIC50:  1.80E+3nMAssay Description:Inhibition of rat brain recombinant nNOSMore data for this Ligand-Target Pair
TargetNitric oxide synthase, endothelial(Bos taurus (bovine))
Université

Curated by ChEMBL
LigandPNGBDBM50270528(3-BROMO-7-NITROINDAZOLE | 3-bromo-7-nitro-1H-indaz...)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of bovine recombinant eNOSMore data for this Ligand-Target Pair
TargetNitric oxide synthase, inducible(Mus musculus (mouse))
Christian-Albrechts-University Of Kiel

Curated by ChEMBL
LigandPNGBDBM50270528(3-BROMO-7-NITROINDAZOLE | 3-bromo-7-nitro-1H-indaz...)
Affinity DataIC50:  2.20E+3nMAssay Description:Inhibition of mouse recombinant iNOSMore data for this Ligand-Target Pair
TargetNitric oxide synthase, brain(Rattus norvegicus (rat))
Université

Curated by ChEMBL
LigandPNGBDBM50270530(3-Bromo-1H-indazole-7-carbonitrile | CHEMBL451541)
Affinity DataIC50:  2.50E+3nMAssay Description:Inhibition of rat brain recombinant nNOSMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, inducible(Mus musculus (mouse))
Christian-Albrechts-University Of Kiel

Curated by ChEMBL
LigandPNGBDBM50270530(3-Bromo-1H-indazole-7-carbonitrile | CHEMBL451541)
Affinity DataIC50:  5.70E+3nMAssay Description:Inhibition of mouse recombinant iNOSMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
University Of The Mediterranean

Curated by ChEMBL
LigandPNGBDBM50157216(2-Bromomethyl-8-nitro-benzo[c]chromen-6-one | CHEM...)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibitory concentration against HIV aspartyl proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, inducible(Mus musculus (mouse))
Christian-Albrechts-University Of Kiel

Curated by ChEMBL
LigandPNGBDBM50295566(3-[4'-(4''-Cyanophenyl)benzoyl]-3,4-dihydro-8-meth...)
Affinity DataIC50:  1.10E+4nMAssay Description:Inhibition of mouse recombinant iNOS expressed in Escherichia coli assessed as NADPH consumption after 2 mins by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, endothelial(Bos taurus (bovine))
Université

Curated by ChEMBL
LigandPNGBDBM50295571(3-[4'-(4''-Chlorobenzyloxy)benzoyl]-3,4-dihydro-8-...)
Affinity DataIC50:  1.20E+4nMAssay Description:Inhibition of bovine recombinant eNOS expressed in Escherichia coli assessed as conversion of [gamma-14C]L-arginine to [14C]L-citrulline by radioacti...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, endothelial(Bos taurus (bovine))
Université

Curated by ChEMBL
LigandPNGBDBM50295566(3-[4'-(4''-Cyanophenyl)benzoyl]-3,4-dihydro-8-meth...)
Affinity DataIC50:  1.20E+4nMAssay Description:Inhibition of bovine recombinant eNOS expressed in Escherichia coli assessed as conversion of [gamma-14C]L-arginine to [14C]L-citrulline by radioacti...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, endothelial(Bos taurus (bovine))
Université

Curated by ChEMBL
LigandPNGBDBM50270530(3-Bromo-1H-indazole-7-carbonitrile | CHEMBL451541)
Affinity DataIC50:  1.30E+4nMAssay Description:Inhibition of bovine recombinant eNOSMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, inducible(Mus musculus (mouse))
Christian-Albrechts-University Of Kiel

Curated by ChEMBL
LigandPNGBDBM50295567(3-[4'-(4''-Methoxyphenyl)benzoyl]-3,4-dihydro-8-me...)
Affinity DataIC50:  1.80E+4nMAssay Description:Inhibition of mouse recombinant iNOS expressed in Escherichia coli assessed as conversion of [gamma-14C]L-arginine to [14C]L-citrulline by radioactiv...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, brain(Rattus norvegicus (rat))
Université

Curated by ChEMBL
LigandPNGBDBM50209245(CHEMBL247378)
Affinity DataIC50:  2.50E+4nMAssay Description:Inhibition of rat brain recombinant nNOSMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, brain(Rattus norvegicus (rat))
Université

Curated by ChEMBL
LigandPNGBDBM50271277(1H-Indazole-7-carbonitrile | CHEMBL484298)
Affinity DataIC50:  2.50E+4nMAssay Description:Inhibition of rat brain recombinant nNOSMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, brain(Rattus norvegicus (rat))
Université

Curated by ChEMBL
LigandPNGBDBM50209245(CHEMBL247378)
Affinity DataIC50:  2.70E+4nMAssay Description:Inhibition of rat recombinant nNOS expressed in Saccharomyces cerevisiae assessed as conversion of [gamma-14C]L-arginine to [14C]L-citrulline by radi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, inducible(Mus musculus (mouse))
Christian-Albrechts-University Of Kiel

Curated by ChEMBL
LigandPNGBDBM50295565(3-[4'-(4''-Bromophenyl)benzoyl]-3,4-dihydro-8-meth...)
Affinity DataIC50:  2.80E+4nMAssay Description:Inhibition of mouse recombinant iNOS expressed in Escherichia coli assessed as conversion of [gamma-14C]L-arginine to [14C]L-citrulline by radioactiv...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, inducible(Mus musculus (mouse))
Christian-Albrechts-University Of Kiel

Curated by ChEMBL
LigandPNGBDBM50295568(3,4-Dihydro-8-methyl-3-[2-(6-methylnaphthoyl)]-2H-...)
Affinity DataIC50:  2.90E+4nMAssay Description:Inhibition of mouse recombinant iNOS expressed in Escherichia coli assessed as conversion of [gamma-14C]L-arginine to [14C]L-citrulline by radioactiv...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, endothelial(Bos taurus (bovine))
Université

Curated by ChEMBL
LigandPNGBDBM50271277(1H-Indazole-7-carbonitrile | CHEMBL484298)
Affinity DataIC50:  3.00E+4nMAssay Description:Inhibition of bovine recombinant eNOSMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, endothelial(Bos taurus (bovine))
Université

Curated by ChEMBL
LigandPNGBDBM50209245(CHEMBL247378)
Affinity DataIC50:  3.50E+4nMAssay Description:Inhibition of bovine recombinant eNOSMore data for this Ligand-Target Pair
TargetNitric oxide synthase, inducible(Mus musculus (mouse))
Christian-Albrechts-University Of Kiel

Curated by ChEMBL
LigandPNGBDBM50295570(3,4-Dihydro-6,8-dimethyl-3-[2-(6-methylnaphthoyl)]...)
Affinity DataIC50:  3.50E+4nMAssay Description:Inhibition of mouse recombinant iNOS expressed in Escherichia coli assessed as conversion of [gamma-14C]L-arginine to [14C]L-citrulline by radioactiv...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, inducible(Mus musculus (mouse))
Christian-Albrechts-University Of Kiel

Curated by ChEMBL
LigandPNGBDBM50295565(3-[4'-(4''-Bromophenyl)benzoyl]-3,4-dihydro-8-meth...)
Affinity DataIC50:  3.50E+4nMAssay Description:Inhibition of mouse recombinant iNOS expressed in Escherichia coli assessed as NADPH consumption after 2 mins by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, inducible(Mus musculus (mouse))
Christian-Albrechts-University Of Kiel

Curated by ChEMBL
LigandPNGBDBM50209245(CHEMBL247378)
Affinity DataIC50:  4.00E+4nMAssay Description:Inhibition of mouse recombinant iNOS expressed in Escherichia coli assessed as conversion of [gamma-14C]L-arginine to [14C]L-citrulline by radioactiv...More data for this Ligand-Target Pair
TargetNitric oxide synthase, endothelial(Bos taurus (bovine))
Université

Curated by ChEMBL
LigandPNGBDBM50209245(CHEMBL247378)
Affinity DataIC50:  4.10E+4nMAssay Description:Inhibition of bovine recombinant eNOS expressed in Escherichia coli assessed as conversion of [gamma-14C]L-arginine to [14C]L-citrulline by radioacti...More data for this Ligand-Target Pair
TargetNitric oxide synthase, inducible(Mus musculus (mouse))
Christian-Albrechts-University Of Kiel

Curated by ChEMBL
LigandPNGBDBM50209245(CHEMBL247378)
Affinity DataIC50:  5.00E+4nMAssay Description:Inhibition of mouse recombinant iNOSMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
University Of The Mediterranean

Curated by ChEMBL
LigandPNGBDBM50157215(8-Amino-2-bromomethyl-benzo[c]chromen-6-one | CHEM...)
Affinity DataIC50:  5.00E+4nMAssay Description:Inhibitory concentration against HIV aspartyl proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, brain(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50071730(BORONIC ACID ANALOG OF L-ARGININE | CHEMBL2448330)
Affinity DataIC50:  5.00E+4nMAssay Description:Compound was tested for inhibitory activity against inducible nitric oxide synthaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
University Of The Mediterranean

Curated by ChEMBL
LigandPNGBDBM50157217(2-Methyl-8-nitro-benzo[c]chromen-6-one | CHEMBL182...)
Affinity DataIC50:  5.00E+4nMAssay Description:Inhibitory concentration against HIV aspartyl proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, inducible(Mus musculus (mouse))
Christian-Albrechts-University Of Kiel

Curated by ChEMBL
LigandPNGBDBM50295566(3-[4'-(4''-Cyanophenyl)benzoyl]-3,4-dihydro-8-meth...)
Affinity DataIC50:  5.00E+4nMAssay Description:Inhibition of mouse recombinant iNOS expressed in Escherichia coli assessed as conversion of [gamma-14C]L-arginine to [14C]L-citrulline by radioactiv...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, endothelial(Bos taurus (bovine))
Université

Curated by ChEMBL
LigandPNGBDBM50295570(3,4-Dihydro-6,8-dimethyl-3-[2-(6-methylnaphthoyl)]...)
Affinity DataIC50:  5.30E+4nMAssay Description:Inhibition of bovine recombinant eNOS expressed in Escherichia coli assessed as conversion of [gamma-14C]L-arginine to [14C]L-citrulline by radioacti...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, brain(Rattus norvegicus (rat))
Université

Curated by ChEMBL
LigandPNGBDBM50271279(1H-Indazole-7-carboxamide | CHEMBL451401)
Affinity DataIC50:  5.50E+4nMAssay Description:Inhibition of rat brain recombinant nNOSMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, endothelial(Bos taurus (bovine))
Université

Curated by ChEMBL
LigandPNGBDBM50295567(3-[4'-(4''-Methoxyphenyl)benzoyl]-3,4-dihydro-8-me...)
Affinity DataIC50:  6.00E+4nMAssay Description:Inhibition of bovine recombinant eNOS expressed in Escherichia coli assessed as conversion of [gamma-14C]L-arginine to [14C]L-citrulline by radioacti...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, brain(Rattus norvegicus (rat))
Université

Curated by ChEMBL
LigandPNGBDBM50295570(3,4-Dihydro-6,8-dimethyl-3-[2-(6-methylnaphthoyl)]...)
Affinity DataIC50:  6.00E+4nMAssay Description:Inhibition of rat recombinant nNOS expressed in Saccharomyces cerevisiae assessed as conversion of [gamma-14C]L-arginine to [14C]L-citrulline by radi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, brain(Rattus norvegicus (rat))
Université

Curated by ChEMBL
LigandPNGBDBM50295567(3-[4'-(4''-Methoxyphenyl)benzoyl]-3,4-dihydro-8-me...)
Affinity DataIC50:  8.70E+4nMAssay Description:Inhibition of rat recombinant nNOS expressed in Saccharomyces cerevisiae assessed as conversion of [gamma-14C]L-arginine to [14C]L-citrulline by radi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, inducible(Mus musculus (mouse))
Christian-Albrechts-University Of Kiel

Curated by ChEMBL
LigandPNGBDBM50271277(1H-Indazole-7-carbonitrile | CHEMBL484298)
Affinity DataIC50:  1.10E+5nMAssay Description:Inhibition of mouse recombinant iNOSMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, inducible(Mus musculus (mouse))
Christian-Albrechts-University Of Kiel

Curated by ChEMBL
LigandPNGBDBM50271275(1H-Indazol-7-amine | 1H-indazol-7-amine, 1 | CHEMB...)
Affinity DataIC50:  1.10E+5nMAssay Description:Inhibition of mouse recombinant iNOSMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, inducible(Mus musculus (mouse))
Christian-Albrechts-University Of Kiel

Curated by ChEMBL
LigandPNGBDBM50295569(3-[4'-(4''-Bromophenyl)benzoyl]-3,4-dihydro-6,8-di...)
Affinity DataIC50:  1.20E+5nMAssay Description:Inhibition of mouse recombinant iNOS expressed in Escherichia coli assessed as conversion of [gamma-14C]L-arginine to [14C]L-citrulline by radioactiv...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, endothelial(Bos taurus (bovine))
Université

Curated by ChEMBL
LigandPNGBDBM50271276(7-Iodo-1H-indazole | CHEMBL510569)
Affinity DataIC50:  1.25E+5nMAssay Description:Inhibition of bovine recombinant eNOSMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, brain(Rattus norvegicus (rat))
Université

Curated by ChEMBL
LigandPNGBDBM50295566(3-[4'-(4''-Cyanophenyl)benzoyl]-3,4-dihydro-8-meth...)
Affinity DataIC50:  1.28E+5nMAssay Description:Inhibition of rat recombinant nNOS expressed in Saccharomyces cerevisiae assessed as conversion of [gamma-14C]L-arginine to [14C]L-citrulline by radi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, endothelial(Bos taurus (bovine))
Université

Curated by ChEMBL
LigandPNGBDBM50295569(3-[4'-(4''-Bromophenyl)benzoyl]-3,4-dihydro-6,8-di...)
Affinity DataIC50:  1.88E+5nMAssay Description:Inhibition of bovine recombinant eNOS expressed in Escherichia coli assessed as conversion of [gamma-14C]L-arginine to [14C]L-citrulline by radioacti...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, brain(Rattus norvegicus (rat))
Université

Curated by ChEMBL
LigandPNGBDBM50271276(7-Iodo-1H-indazole | CHEMBL510569)
Affinity DataIC50:  2.00E+5nMAssay Description:Inhibition of rat brain recombinant nNOSMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, endothelial(Bos taurus (bovine))
Université

Curated by ChEMBL
LigandPNGBDBM50270526(7-Ethynyl-1H-indazole | CHEMBL452956)
Affinity DataIC50:  2.25E+5nMAssay Description:Inhibition of bovine recombinant eNOSMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, endothelial(Bos taurus (bovine))
Université

Curated by ChEMBL
LigandPNGBDBM50240903(1-methyl-7-nitro-1H-indazole | CHEMBL354723)
Affinity DataIC50:  2.50E+5nMAssay Description:Inhibition of bovine recombinant eNOSMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, inducible(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50071730(BORONIC ACID ANALOG OF L-ARGININE | CHEMBL2448330)
Affinity DataIC50:  3.00E+5nMAssay Description:Compound was tested for inhibitory activity against inducible nitric oxide synthaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, inducible(Mus musculus (mouse))
Christian-Albrechts-University Of Kiel

Curated by ChEMBL
LigandPNGBDBM50271276(7-Iodo-1H-indazole | CHEMBL510569)
Affinity DataIC50:  3.70E+5nMAssay Description:Inhibition of mouse recombinant iNOSMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, endothelial(Bos taurus (bovine))
Université

Curated by ChEMBL
LigandPNGBDBM50271275(1H-Indazol-7-amine | 1H-indazol-7-amine, 1 | CHEMB...)
Affinity DataIC50:  4.00E+5nMAssay Description:Inhibition of bovine recombinant eNOSMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, inducible(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50071731(BORONIC ACID ANALOG OF L-ARGININE | CHEMBL2448331)
Affinity DataIC50: >5.00E+5nMAssay Description:Compound was tested for inhibitory activity against neuronal nitric oxide synthaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, brain(Rattus norvegicus (rat))
Université

Curated by ChEMBL
LigandPNGBDBM50270533(3-Bromo-1-methyl-7-nitro-1H-indazole | CHEMBL50488...)
Affinity DataIC50: >5.00E+5nMAssay Description:Inhibition of rat brain recombinant nNOSMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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