Affinity DataKi: 1.10nMAssay Description:Binding affinity for adenosine A3 receptor as inhibition of [125I]-AB-MECA binding to human receptor expressed in HEK 293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 7.80nMAssay Description:Binding affinity for adenosine A3 receptor as inhibition of [125I]-AB-MECA binding to human receptor expressed in HEK 293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 20nMAssay Description:Binding affinity for adenosine A3 receptor as inhibition of [125I]-AB-MECA binding to human receptor expressed in HEK 293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 26nMAssay Description:Binding affinity for adenosine A3 receptor as inhibition of [125I]-AB-MECA binding to human receptor expressed in HEK 293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 31nMAssay Description:Binding affinity for adenosine A3 receptor as inhibition of [125I]-AB-MECA binding to human receptor expressed in HEK 293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 41nMAssay Description:Binding affinity for adenosine A3 receptor as inhibition of [125I]-AB-MECA binding to human receptor expressed in HEK 293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 54nMAssay Description:Binding affinity for adenosine A1 receptor as inhibition of 3[H]-R-PIA binding in rat brainMore data for this Ligand-Target Pair
Affinity DataKi: 56nMAssay Description:Binding affinity for adenosine A2a receptor as inhibition of 3[H]-CGS 21680 binding in rat striatumMore data for this Ligand-Target Pair
Affinity DataKi: 74nMAssay Description:Binding affinity for adenosine A1 receptor as inhibition of 3[H]-R-PIA binding in rat brainMore data for this Ligand-Target Pair
Affinity DataKi: 620nMAssay Description:Binding affinity for adenosine A1 receptor as inhibition of 3[H]-R-PIA binding in rat brainMore data for this Ligand-Target Pair
Affinity DataKi: 1.23E+3nMAssay Description:Binding affinity for adenosine A1 receptor as inhibition of 3[H]-R-PIA binding in rat brainMore data for this Ligand-Target Pair
Affinity DataKi: 1.90E+3nMAssay Description:Binding affinity for adenosine A2a receptor as inhibition of 3[H]-CGS 21680 binding in rat striatumMore data for this Ligand-Target Pair
Affinity DataKi: 1.90E+3nMAssay Description:Binding affinity for adenosine A1 receptor as inhibition of 3[H]-R-PIA binding in rat brainMore data for this Ligand-Target Pair
Affinity DataKi: 2.10E+3nMAssay Description:Binding affinity for adenosine A2a receptor as inhibition of 3[H]-CGS 21680 binding in rat striatumMore data for this Ligand-Target Pair
Affinity DataKi: 2.40E+3nMAssay Description:Binding affinity for adenosine A1 receptor as inhibition of 3[H]-R-PIA binding in rat brainMore data for this Ligand-Target Pair
Affinity DataKi: 4.65E+3nMAssay Description:Binding affinity for adenosine A2a receptor as inhibition of 3[H]-CGS 21680 binding in rat striatumMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity for adenosine A2a receptor as inhibition of 3[H]-CGS 21680 binding in rat striatumMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity for adenosine A2a receptor as inhibition of 3[H]-CGS 21680 binding in rat striatumMore data for this Ligand-Target Pair
Affinity DataIC50: 100nMAssay Description:Inhibitory activity against human glycogen synthase kinase-3beta (GSK3-beta) at 100 uM ATPMore data for this Ligand-Target Pair
Affinity DataIC50: 100nMAssay Description:Inhibitory activity against human glycogen synthase kinase-3beta (GSK3-beta) at 100 uM ATPMore data for this Ligand-Target Pair
Affinity DataIC50: 160nMAssay Description:Inhibitory activity against human glycogen synthase kinase-3beta (GSK3-beta) at 100 uM ATPMore data for this Ligand-Target Pair
Affinity DataIC50: 240nMAssay Description:Inhibitory activity against human glycogen synthase kinase-3beta (GSK3-beta) at 100 uM ATPMore data for this Ligand-Target Pair
Affinity DataIC50: 280nMAssay Description:Inhibitory activity against human glycogen synthase kinase-3beta (GSK3-beta) at 100 uM ATPMore data for this Ligand-Target Pair
TargetCyclin-A1/Cyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
Novo Nordisk
Curated by ChEMBL
Novo Nordisk
Curated by ChEMBL
Affinity DataIC50: 380nMAssay Description:Inhibition of Cyclin-dependent kinase 2-cyclin AMore data for this Ligand-Target Pair
Affinity DataIC50: 380nMAssay Description:Inhibitory activity against human glycogen synthase kinase-3beta (GSK3-beta) at 100 uM ATPMore data for this Ligand-Target Pair
Affinity DataIC50: 410nMAssay Description:Inhibitory activity against human glycogen synthase kinase-3beta (GSK3-beta) at 100 uM ATPMore data for this Ligand-Target Pair
Affinity DataIC50: 1.16E+3nMAssay Description:Inhibitory activity against human glycogen synthase kinase-3beta (GSK3-beta) at 100 uM ATPMore data for this Ligand-Target Pair
Affinity DataIC50: 2.10E+3nMAssay Description:Inhibitory activity against human glycogen synthase kinase-3beta (GSK3-beta) at 100 uM ATPMore data for this Ligand-Target Pair
Affinity DataIC50: 6.92E+3nMAssay Description:Inhibitory activity against human glycogen synthase kinase-3beta (GSK3-beta) at 100 uM ATPMore data for this Ligand-Target Pair
Affinity DataIC50: 9.30E+3nMAssay Description:Inhibitory activity against human glycogen synthase kinase-3beta (GSK3-beta) at 100 uM ATPMore data for this Ligand-Target Pair
Affinity DataIC50: 9.60E+3nMAssay Description:Inhibitory activity against human glycogen synthase kinase-3beta (GSK3-beta) at 100 uM ATPMore data for this Ligand-Target Pair
Affinity DataIC50: 1.17E+4nMAssay Description:Inhibitory activity against human glycogen synthase kinase-3beta (GSK3-beta) at 100 uM ATPMore data for this Ligand-Target Pair
Affinity DataIC50: 1.70E+4nMAssay Description:Inhibition of human Glycogen synthase kinase-3 beta (GSK3-beta) at 100 uM ATPMore data for this Ligand-Target Pair
TargetCyclin-A1/Cyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
Novo Nordisk
Curated by ChEMBL
Novo Nordisk
Curated by ChEMBL
Affinity DataIC50: 9.60E+4nMAssay Description:Inhibition of Cyclin-dependent kinase 2-cyclin AMore data for this Ligand-Target Pair
TargetCyclin-A1/Cyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
Novo Nordisk
Curated by ChEMBL
Novo Nordisk
Curated by ChEMBL
Affinity DataIC50: 1.19E+5nMAssay Description:Inhibition of Cyclin-dependent kinase 2-cyclin AMore data for this Ligand-Target Pair
Affinity DataIC50: >2.50E+5nMAssay Description:Inhibitory activity against human glycogen synthase kinase-3beta (GSK3-beta) at 100 uM ATPMore data for this Ligand-Target Pair
TargetCyclin-A1/Cyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
Novo Nordisk
Curated by ChEMBL
Novo Nordisk
Curated by ChEMBL
Affinity DataIC50: >2.50E+5nMAssay Description:Inhibition of Cyclin-dependent kinase 2-cyclin AMore data for this Ligand-Target Pair
Affinity DataIC50: >2.50E+5nMAssay Description:Inhibitory activity against human glycogen synthase kinase-3beta (GSK3-beta) at 100 uM ATPMore data for this Ligand-Target Pair