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Found 113 with Last Name = 'brady' and Initial = 't'
TargetTaste receptor type 2 member 8(Homo sapiens (Human))
Firmenich

Curated by ChEMBL
LigandPNGBDBM211262(US9247759, 10-10)
Affinity DataIC50:  20nMAssay Description:Antagonist activity at recombinant human TAS2R8 stably expressed in cells co-expressing Galpha16gust44 assessed as inhibition of andrographolide-indu...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTaste receptor type 2 member 8(Homo sapiens (Human))
Firmenich

Curated by ChEMBL
LigandPNGBDBM211356(US9247759, 12-7)
Affinity DataIC50:  20nMAssay Description:Antagonist activity at recombinant human TAS2R8 stably expressed in cells co-expressing Galpha16gust44 assessed as inhibition of andrographolide-indu...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTaste receptor type 2 member 8(Homo sapiens (Human))
Firmenich

Curated by ChEMBL
LigandPNGBDBM211364(US9247759, 12-15)
Affinity DataIC50:  20nMAssay Description:Antagonist activity at recombinant human TAS2R8 stably expressed in cells co-expressing Galpha16gust44 assessed as inhibition of andrographolide-indu...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTaste receptor type 2 member 8(Homo sapiens (Human))
Firmenich

Curated by ChEMBL
LigandPNGBDBM211355(US9247759, 12-6)
Affinity DataIC50:  20nMAssay Description:Antagonist activity at recombinant human TAS2R8 stably expressed in cells co-expressing Galpha16gust44 assessed as inhibition of andrographolide-indu...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTaste receptor type 2 member 8(Homo sapiens (Human))
Firmenich

Curated by ChEMBL
LigandPNGBDBM211358(US9247759, 12-9)
Affinity DataIC50:  40nMAssay Description:Antagonist activity at recombinant human TAS2R8 stably expressed in cells co-expressing Galpha16gust44 assessed as inhibition of andrographolide-indu...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTaste receptor type 2 member 8(Homo sapiens (Human))
Firmenich

Curated by ChEMBL
LigandPNGBDBM211353(US9247759, 12-4)
Affinity DataIC50:  40nMAssay Description:Antagonist activity at recombinant human TAS2R8 stably expressed in cells co-expressing Galpha16gust44 assessed as inhibition of andrographolide-indu...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTaste receptor type 2 member 8(Homo sapiens (Human))
Firmenich

Curated by ChEMBL
LigandPNGBDBM211264(US9247759, 10-12)
Affinity DataIC50:  40nMAssay Description:Antagonist activity at recombinant human TAS2R8 stably expressed in cells co-expressing Galpha16gust44 assessed as inhibition of andrographolide-indu...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTaste receptor type 2 member 8(Homo sapiens (Human))
Firmenich

Curated by ChEMBL
LigandPNGBDBM211350(US9247759, 12-1)
Affinity DataIC50:  60nMAssay Description:Antagonist activity at recombinant human TAS2R8 stably expressed in cells co-expressing Galpha16gust44 assessed as inhibition of andrographolide-indu...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTaste receptor type 2 member 8(Homo sapiens (Human))
Firmenich

Curated by ChEMBL
LigandPNGBDBM211359(US9247759, 12-10)
Affinity DataIC50:  100nMAssay Description:Antagonist activity at recombinant human TAS2R8 stably expressed in cells co-expressing Galpha16gust44 assessed as inhibition of andrographolide-indu...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTaste receptor type 2 member 8(Homo sapiens (Human))
Firmenich

Curated by ChEMBL
LigandPNGBDBM211273(US9247759, 10-21)
Affinity DataIC50:  100nMAssay Description:Antagonist activity at recombinant human TAS2R8 stably expressed in cells co-expressing Galpha16gust44 assessed as inhibition of andrographolide-indu...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTaste receptor type 2 member 8(Homo sapiens (Human))
Firmenich

Curated by ChEMBL
LigandPNGBDBM211272(US9247759, 10-20)
Affinity DataIC50:  100nMAssay Description:Antagonist activity at recombinant human TAS2R8 stably expressed in cells co-expressing Galpha16gust44 assessed as inhibition of andrographolide-indu...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTaste receptor type 2 member 8(Homo sapiens (Human))
Firmenich

Curated by ChEMBL
LigandPNGBDBM211270(US9247759, 10-18)
Affinity DataIC50:  100nMAssay Description:Antagonist activity at recombinant human TAS2R8 stably expressed in cells co-expressing Galpha16gust44 assessed as inhibition of andrographolide-indu...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTaste receptor type 2 member 8(Homo sapiens (Human))
Firmenich

Curated by ChEMBL
LigandPNGBDBM211263(US9247759, 10-11)
Affinity DataIC50:  100nMAssay Description:Antagonist activity at recombinant human TAS2R8 stably expressed in cells co-expressing Galpha16gust44 assessed as inhibition of andrographolide-indu...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTaste receptor type 2 member 8(Homo sapiens (Human))
Firmenich

Curated by ChEMBL
LigandPNGBDBM211259(US9247759, 10-7)
Affinity DataIC50:  100nMAssay Description:Antagonist activity at recombinant human TAS2R8 stably expressed in cells co-expressing Galpha16gust44 assessed as inhibition of andrographolide-indu...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTaste receptor type 2 member 8(Homo sapiens (Human))
Firmenich

Curated by ChEMBL
LigandPNGBDBM211261(US9247759, 10-9)
Affinity DataIC50:  100nMAssay Description:Antagonist activity at recombinant human TAS2R8 stably expressed in cells co-expressing Galpha16gust44 assessed as inhibition of andrographolide-indu...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTaste receptor type 2 member 8(Homo sapiens (Human))
Firmenich

Curated by ChEMBL
LigandPNGBDBM210974(US9247759, 4-8)
Affinity DataIC50:  200nMAssay Description:Antagonist activity at recombinant human TAS2R8 stably expressed in cells co-expressing Galpha16gust44 assessed as inhibition of andrographolide-indu...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTaste receptor type 2 member 8(Homo sapiens (Human))
Firmenich

Curated by ChEMBL
LigandPNGBDBM211305(US9247759, 10-53 | US9247759, 10-88)
Affinity DataIC50:  200nMAssay Description:Antagonist activity at recombinant human TAS2R8 stably expressed in cells co-expressing Galpha16gust44 assessed as inhibition of andrographolide-indu...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTaste receptor type 2 member 8(Homo sapiens (Human))
Firmenich

Curated by ChEMBL
LigandPNGBDBM50511890(CHEMBL4514970)
Affinity DataIC50:  200nMAssay Description:Antagonist activity at recombinant human TAS2R8 stably expressed in cells co-expressing Galpha16gust44 assessed as inhibition of andrographolide-indu...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTaste receptor type 2 member 8(Homo sapiens (Human))
Firmenich

Curated by ChEMBL
LigandPNGBDBM211244(US9247759, 9-1)
Affinity DataIC50:  200nMAssay Description:Antagonist activity at recombinant human TAS2R8 stably expressed in cells co-expressing Galpha16gust44 assessed as inhibition of andrographolide-indu...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTaste receptor type 2 member 8(Homo sapiens (Human))
Firmenich

Curated by ChEMBL
LigandPNGBDBM211285(US9247759, 10-33)
Affinity DataIC50:  300nMAssay Description:Antagonist activity at recombinant human TAS2R8 stably expressed in cells co-expressing Galpha16gust44 assessed as inhibition of andrographolide-indu...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTaste receptor type 2 member 8(Homo sapiens (Human))
Firmenich

Curated by ChEMBL
LigandPNGBDBM211326(US9247759, 10-74)
Affinity DataIC50:  300nMAssay Description:Antagonist activity at recombinant human TAS2R8 stably expressed in cells co-expressing Galpha16gust44 assessed as inhibition of andrographolide-indu...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTaste receptor type 2 member 8(Homo sapiens (Human))
Firmenich

Curated by ChEMBL
LigandPNGBDBM210975(US9247759, 4-9)
Affinity DataIC50:  300nMAssay Description:Antagonist activity at recombinant human TAS2R8 stably expressed in cells co-expressing Galpha16gust44 assessed as inhibition of andrographolide-indu...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTaste receptor type 2 member 8(Homo sapiens (Human))
Firmenich

Curated by ChEMBL
LigandPNGBDBM50511886(CHEMBL4452065)
Affinity DataIC50:  300nMAssay Description:Antagonist activity at recombinant human TAS2R8 stably expressed in cells co-expressing Galpha16gust44 assessed as inhibition of andrographolide-indu...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTaste receptor type 2 member 8(Homo sapiens (Human))
Firmenich

Curated by ChEMBL
LigandPNGBDBM50511892(CHEMBL4469393)
Affinity DataIC50:  400nMAssay Description:Antagonist activity at recombinant human TAS2R8 stably expressed in cells co-expressing Galpha16gust44 assessed as inhibition of andrographolide-indu...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTaste receptor type 2 member 8(Homo sapiens (Human))
Firmenich

Curated by ChEMBL
LigandPNGBDBM211020(US9247759, 4-55)
Affinity DataIC50:  400nMAssay Description:Antagonist activity at recombinant human TAS2R8 stably expressed in cells co-expressing Galpha16gust44 assessed as inhibition of andrographolide-indu...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTaste receptor type 2 member 8(Homo sapiens (Human))
Firmenich

Curated by ChEMBL
LigandPNGBDBM211307(US9247759, 10-55)
Affinity DataIC50:  400nMAssay Description:Antagonist activity at recombinant human TAS2R8 stably expressed in cells co-expressing Galpha16gust44 assessed as inhibition of andrographolide-indu...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTaste receptor type 2 member 8(Homo sapiens (Human))
Firmenich

Curated by ChEMBL
LigandPNGBDBM211052(US9247759, 4-88)
Affinity DataIC50:  400nMAssay Description:Antagonist activity at recombinant human TAS2R8 stably expressed in cells co-expressing Galpha16gust44 assessed as inhibition of andrographolide-indu...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTaste receptor type 2 member 8(Homo sapiens (Human))
Firmenich

Curated by ChEMBL
LigandPNGBDBM211271(US9247759, 10-19)
Affinity DataIC50:  500nMAssay Description:Antagonist activity at recombinant human TAS2R8 stably expressed in cells co-expressing Galpha16gust44 assessed as inhibition of andrographolide-indu...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTaste receptor type 2 member 8(Homo sapiens (Human))
Firmenich

Curated by ChEMBL
LigandPNGBDBM50511893(CHEMBL4567380)
Affinity DataIC50:  500nMAssay Description:Antagonist activity at recombinant human TAS2R8 stably expressed in cells co-expressing Galpha16gust44 assessed as inhibition of andrographolide-indu...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTaste receptor type 2 member 8(Homo sapiens (Human))
Firmenich

Curated by ChEMBL
LigandPNGBDBM210983(US9247759, 4-17)
Affinity DataIC50:  700nMAssay Description:Antagonist activity at recombinant human TAS2R8 stably expressed in cells co-expressing Galpha16gust44 assessed as inhibition of andrographolide-indu...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTaste receptor type 2 member 8(Homo sapiens (Human))
Firmenich

Curated by ChEMBL
LigandPNGBDBM50511894(CHEMBL4447100)
Affinity DataIC50:  700nMAssay Description:Antagonist activity at recombinant human TAS2R8 stably expressed in cells co-expressing Galpha16gust44 assessed as inhibition of andrographolide-indu...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTaste receptor type 2 member 8(Homo sapiens (Human))
Firmenich

Curated by ChEMBL
LigandPNGBDBM210973(US9247759, 4-7 | US9247759, compound B)
Affinity DataIC50:  700nMAssay Description:Antagonist activity at recombinant human TAS2R8 stably expressed in cells co-expressing Galpha16gust44 assessed as inhibition of andrographolide-indu...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTaste receptor type 2 member 8(Homo sapiens (Human))
Firmenich

Curated by ChEMBL
LigandPNGBDBM211021(US9247759, 4-56)
Affinity DataIC50:  800nMAssay Description:Antagonist activity at recombinant human TAS2R8 stably expressed in cells co-expressing Galpha16gust44 assessed as inhibition of andrographolide-indu...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTaste receptor type 2 member 8(Homo sapiens (Human))
Firmenich

Curated by ChEMBL
LigandPNGBDBM210972(US9247759, 4-6)
Affinity DataIC50:  800nMAssay Description:Antagonist activity at recombinant human TAS2R8 stably expressed in cells co-expressing Galpha16gust44 assessed as inhibition of andrographolide-indu...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTaste receptor type 2 member 8(Homo sapiens (Human))
Firmenich

Curated by ChEMBL
LigandPNGBDBM50511888(CHEMBL4456506)
Affinity DataIC50:  800nMAssay Description:Antagonist activity at recombinant human TAS2R8 stably expressed in cells co-expressing Galpha16gust44 assessed as inhibition of andrographolide-indu...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTaste receptor type 2 member 8(Homo sapiens (Human))
Firmenich

Curated by ChEMBL
LigandPNGBDBM211253(US9247759, 10-1)
Affinity DataIC50:  900nMAssay Description:Antagonist activity at recombinant human TAS2R8 stably expressed in cells co-expressing Galpha16gust44 assessed as inhibition of andrographolide-indu...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTaste receptor type 2 member 8(Homo sapiens (Human))
Firmenich

Curated by ChEMBL
LigandPNGBDBM211306(US9247759, 10-54)
Affinity DataIC50:  1.00E+3nMAssay Description:Antagonist activity at recombinant human TAS2R8 stably expressed in cells co-expressing Galpha16gust44 assessed as inhibition of andrographolide-indu...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTaste receptor type 2 member 8(Homo sapiens (Human))
Firmenich

Curated by ChEMBL
LigandPNGBDBM50511896(CHEMBL4526144)
Affinity DataIC50:  1.00E+3nMAssay Description:Antagonist activity at recombinant human TAS2R8 stably expressed in cells co-expressing Galpha16gust44 assessed as inhibition of andrographolide-indu...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTaste receptor type 2 member 8(Homo sapiens (Human))
Firmenich

Curated by ChEMBL
LigandPNGBDBM50511891(CHEMBL4530528)
Affinity DataIC50:  1.00E+3nMAssay Description:Antagonist activity at recombinant human TAS2R8 stably expressed in cells co-expressing Galpha16gust44 assessed as inhibition of andrographolide-indu...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTaste receptor type 2 member 8(Homo sapiens (Human))
Firmenich

Curated by ChEMBL
LigandPNGBDBM210987(US9247759, 4-21)
Affinity DataIC50:  1.00E+3nMAssay Description:Antagonist activity at recombinant human TAS2R8 stably expressed in cells co-expressing Galpha16gust44 assessed as inhibition of andrographolide-indu...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTaste receptor type 2 member 8(Homo sapiens (Human))
Firmenich

Curated by ChEMBL
LigandPNGBDBM211325(US9247759, 10-73)
Affinity DataIC50:  1.00E+3nMAssay Description:Antagonist activity at recombinant human TAS2R8 stably expressed in cells co-expressing Galpha16gust44 assessed as inhibition of andrographolide-indu...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTaste receptor type 2 member 8(Homo sapiens (Human))
Firmenich

Curated by ChEMBL
LigandPNGBDBM50511887(CHEMBL4588973)
Affinity DataIC50:  1.00E+3nMAssay Description:Antagonist activity at recombinant human TAS2R8 stably expressed in cells co-expressing Galpha16gust44 assessed as inhibition of andrographolide-indu...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTaste receptor type 2 member 8(Homo sapiens (Human))
Firmenich

Curated by ChEMBL
LigandPNGBDBM50511889(CHEMBL4579065)
Affinity DataIC50:  1.10E+3nMAssay Description:Antagonist activity at recombinant human TAS2R8 stably expressed in cells co-expressing Galpha16gust44 assessed as inhibition of andrographolide-indu...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTaste receptor type 2 member 8(Homo sapiens (Human))
Firmenich

Curated by ChEMBL
LigandPNGBDBM211011(US9247759, 4-46)
Affinity DataIC50:  1.10E+3nMAssay Description:Antagonist activity at recombinant human TAS2R8 stably expressed in cells co-expressing Galpha16gust44 assessed as inhibition of andrographolide-indu...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTaste receptor type 2 member 8(Homo sapiens (Human))
Firmenich

Curated by ChEMBL
LigandPNGBDBM210989(US9247759, 4-24)
Affinity DataIC50:  1.70E+3nMAssay Description:Antagonist activity at recombinant human TAS2R8 stably expressed in cells co-expressing Galpha16gust44 assessed as inhibition of andrographolide-indu...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTaste receptor type 2 member 8(Homo sapiens (Human))
Firmenich

Curated by ChEMBL
LigandPNGBDBM210985(US9247759, 4-19)
Affinity DataIC50:  1.90E+3nMAssay Description:Antagonist activity at recombinant human TAS2R8 stably expressed in cells co-expressing Galpha16gust44 assessed as inhibition of andrographolide-indu...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTaste receptor type 2 member 8(Homo sapiens (Human))
Firmenich

Curated by ChEMBL
LigandPNGBDBM211260(US9247759, 10-8)
Affinity DataIC50:  2.00E+3nMAssay Description:Antagonist activity at recombinant human TAS2R8 stably expressed in cells co-expressing Galpha16gust44 assessed as inhibition of andrographolide-indu...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTaste receptor type 2 member 8(Homo sapiens (Human))
Firmenich

Curated by ChEMBL
LigandPNGBDBM50511884(CHEMBL4471870)
Affinity DataIC50:  2.00E+3nMAssay Description:Antagonist activity at recombinant human TAS2R8 stably expressed in cells co-expressing Galpha16gust44 assessed as inhibition of andrographolide-indu...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTaste receptor type 2 member 8(Homo sapiens (Human))
Firmenich

Curated by ChEMBL
LigandPNGBDBM50511885(CHEMBL4443466)
Affinity DataIC50:  2.00E+3nMAssay Description:Antagonist activity at recombinant human TAS2R8 stably expressed in cells co-expressing Galpha16gust44 assessed as inhibition of andrographolide-indu...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTaste receptor type 2 member 8(Homo sapiens (Human))
Firmenich

Curated by ChEMBL
LigandPNGBDBM210967(US9247759, 4-1)
Affinity DataIC50:  2.30E+3nMAssay Description:Antagonist activity at recombinant human TAS2R8 stably expressed in cells co-expressing Galpha16gust44 assessed as inhibition of andrographolide-indu...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
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