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Found 97 with Last Name = 'brand' and Initial = 'gd'
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
University Of Bras£Lia

Curated by ChEMBL
LigandPNGBDBM50198338(CHEMBL3938038)
Affinity DataKi:  0.389nMAssay Description:Displacement of [3H]prazosin from human alpha1A-adrenoceptor expressed in CHO cell membranes measured after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
University Of Bras£Lia

Curated by ChEMBL
LigandPNGBDBM50200566(CHEMBL3902626)
Affinity DataKi:  0.603nMAssay Description:Displacement of [3H]prazosin from human alpha1D-adrenoceptor expressed in CHO cell membranes measured after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
University Of Bras£Lia

Curated by ChEMBL
LigandPNGBDBM50201790(CHEMBL3917716)
Affinity DataKi:  1.10nMAssay Description:Displacement of [3H]prazosin from human alpha1A-adrenoceptor expressed in CHO cell membranes measured after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
University Of Bras£Lia

Curated by ChEMBL
LigandPNGBDBM50200441(CHEMBL3930616)
Affinity DataKi:  1.10nMAssay Description:Displacement of [3H]prazosin from human alpha1A-adrenoceptor expressed in CHO cell membranes measured after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
University Of Bras£Lia

Curated by ChEMBL
LigandPNGBDBM50201789(CHEMBL3946843)
Affinity DataKi:  1.30nMAssay Description:Displacement of [3H]prazosin from human alpha1D-adrenoceptor expressed in CHO cell membranes measured after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
University Of Bras£Lia

Curated by ChEMBL
LigandPNGBDBM50201791(CHEMBL3920110)
Affinity DataKi:  1.30nMAssay Description:Displacement of [3H]prazosin from human alpha1D-adrenoceptor expressed in CHO cell membranes measured after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
University Of Bras£Lia

Curated by ChEMBL
LigandPNGBDBM50200441(CHEMBL3930616)
Affinity DataKi:  1.30nMAssay Description:Displacement of [3H]prazosin from human alpha1D-adrenoceptor expressed in CHO cell membranes measured after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
University Of Bras£Lia

Curated by ChEMBL
LigandPNGBDBM50393116(CHEMBL2153423)
Affinity DataKi:  1.30nMAssay Description:Displacement of [3H]prazosin from human alpha1D-adrenoceptor expressed in CHO cell membranes measured after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
University Of Bras£Lia

Curated by ChEMBL
LigandPNGBDBM50201790(CHEMBL3917716)
Affinity DataKi:  1.5nMAssay Description:Displacement of [3H]prazosin from human alpha1D-adrenoceptor expressed in CHO cell membranes measured after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
University Of Bras£Lia

Curated by ChEMBL
LigandPNGBDBM50198338(CHEMBL3938038)
Affinity DataKi:  1.70nMAssay Description:Displacement of [3H]prazosin from human alpha1D-adrenoceptor expressed in CHO cell membranes measured after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
University Of Bras£Lia

Curated by ChEMBL
LigandPNGBDBM50201791(CHEMBL3920110)
Affinity DataKi:  2nMAssay Description:Displacement of [3H]prazosin from human alpha1A-adrenoceptor expressed in CHO cell membranes measured after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
University Of Bras£Lia

Curated by ChEMBL
LigandPNGBDBM50200566(CHEMBL3902626)
Affinity DataKi:  2.10nMAssay Description:Displacement of [3H]prazosin from human alpha1A-adrenoceptor expressed in CHO cell membranes measured after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
University Of Bras£Lia

Curated by ChEMBL
LigandPNGBDBM50197059(CHEMBL3976144)
Affinity DataKi:  2.20nMAssay Description:Displacement of [3H]prazosin from human alpha1A-adrenoceptor expressed in CHO cell membranes measured after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
University Of Bras£Lia

Curated by ChEMBL
LigandPNGBDBM50197548(CHEMBL3947302)
Affinity DataKi:  2.60nMAssay Description:Displacement of [3H]prazosin from human alpha1D-adrenoceptor expressed in CHO cell membranes measured after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
University Of Bras£Lia

Curated by ChEMBL
LigandPNGBDBM50201789(CHEMBL3946843)
Affinity DataKi:  2.80nMAssay Description:Displacement of [3H]prazosin from human alpha1A-adrenoceptor expressed in CHO cell membranes measured after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
University Of Bras£Lia

Curated by ChEMBL
LigandPNGBDBM50197548(CHEMBL3947302)
Affinity DataKi:  3nMAssay Description:Displacement of [3H]prazosin from human alpha1A-adrenoceptor expressed in CHO cell membranes measured after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
University Of Bras£Lia

Curated by ChEMBL
LigandPNGBDBM50197059(CHEMBL3976144)
Affinity DataKi:  3.10nMAssay Description:Displacement of [3H]prazosin from human alpha1D-adrenoceptor expressed in CHO cell membranes measured after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
University Of Bras£Lia

Curated by ChEMBL
LigandPNGBDBM50393116(CHEMBL2153423)
Affinity DataKi:  3.5nMAssay Description:Displacement of [3H]prazosin from human alpha1A-adrenoceptor expressed in CHO cell membranes measured after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
University Of Bras£Lia

Curated by ChEMBL
LigandPNGBDBM50198439(CHEMBL3967641)
Affinity DataKi:  4.60nMAssay Description:Displacement of [3H]prazosin from human alpha1D-adrenoceptor expressed in CHO cell membranes measured after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
University Of Bras£Lia

Curated by ChEMBL
LigandPNGBDBM50198439(CHEMBL3967641)
Affinity DataKi:  5nMAssay Description:Displacement of [3H]prazosin from human alpha1A-adrenoceptor expressed in CHO cell membranes measured after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
University Of Bras£Lia

Curated by ChEMBL
LigandPNGBDBM50393116(CHEMBL2153423)
Affinity DataKi:  5.20nMAssay Description:Displacement of [3H]prazosin from human alpha1B-adrenoceptor expressed in CHO cell membranes measured after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
University Of Bras£Lia

Curated by ChEMBL
LigandPNGBDBM50201790(CHEMBL3917716)
Affinity DataKi:  5.40nMAssay Description:Displacement of [3H]prazosin from human alpha1B-adrenoceptor expressed in CHO cell membranes measured after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
University Of Bras£Lia

Curated by ChEMBL
LigandPNGBDBM50200441(CHEMBL3930616)
Affinity DataKi:  10nMAssay Description:Displacement of [3H]prazosin from human alpha1B-adrenoceptor expressed in CHO cell membranes measured after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
University Of Bras£Lia

Curated by ChEMBL
LigandPNGBDBM50201791(CHEMBL3920110)
Affinity DataKi:  10nMAssay Description:Displacement of [3H]prazosin from human alpha1B-adrenoceptor expressed in CHO cell membranes measured after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
University Of Bras£Lia

Curated by ChEMBL
LigandPNGBDBM50198338(CHEMBL3938038)
Affinity DataKi:  13nMAssay Description:Displacement of [3H]prazosin from human alpha1B-adrenoceptor expressed in CHO cell membranes measured after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
University Of Bras£Lia

Curated by ChEMBL
LigandPNGBDBM50201789(CHEMBL3946843)
Affinity DataKi:  14nMAssay Description:Displacement of [3H]prazosin from human alpha1B-adrenoceptor expressed in CHO cell membranes measured after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
University Of Bras£Lia

Curated by ChEMBL
LigandPNGBDBM50197059(CHEMBL3976144)
Affinity DataKi:  15nMAssay Description:Displacement of [3H]prazosin from human alpha1B-adrenoceptor expressed in CHO cell membranes measured after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
University Of Bras£Lia

Curated by ChEMBL
LigandPNGBDBM50200566(CHEMBL3902626)
Affinity DataKi:  16nMAssay Description:Displacement of [3H]prazosin from human alpha1B-adrenoceptor expressed in CHO cell membranes measured after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
University Of Bras£Lia

Curated by ChEMBL
LigandPNGBDBM50201787(CHEMBL27021)
Affinity DataKi:  17nMAssay Description:Displacement of [3H]prazosin from human alpha1D-adrenoceptor expressed in CHO cell membranes measured after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
University Of Bras£Lia

Curated by ChEMBL
LigandPNGBDBM50197548(CHEMBL3947302)
Affinity DataKi:  25nMAssay Description:Displacement of [3H]prazosin from human alpha1B-adrenoceptor expressed in CHO cell membranes measured after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
University Of Bras£Lia

Curated by ChEMBL
LigandPNGBDBM50201787(CHEMBL27021)
Affinity DataKi:  32nMAssay Description:Displacement of [3H]prazosin from human alpha1A-adrenoceptor expressed in CHO cell membranes measured after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
University Of Bras£Lia

Curated by ChEMBL
LigandPNGBDBM50198439(CHEMBL3967641)
Affinity DataKi:  78nMAssay Description:Displacement of [3H]prazosin from human alpha1B-adrenoceptor expressed in CHO cell membranes measured after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
University Of Bras£Lia

Curated by ChEMBL
LigandPNGBDBM50201787(CHEMBL27021)
Affinity DataKi:  91nMAssay Description:Displacement of [3H]prazosin from human alpha1B-adrenoceptor expressed in CHO cell membranes measured after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Bras£Lia

Curated by ChEMBL
LigandPNGBDBM50139050(CHEMBL3753906)
Affinity DataKi:  8.60E+3nMAssay Description:Non-competitive inhibition of electric eel acetylcholine esterase using acetylcholine iodide as substrate by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Bras£Lia

Curated by ChEMBL
LigandPNGBDBM50139006(CHEMBL3753607)
Affinity DataKi:  1.04E+4nMAssay Description:Non-competitive inhibition of electric eel acetylcholine esterase using acetylcholine iodide as substrate by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Bras£Lia

Curated by ChEMBL
LigandPNGBDBM50139052(CHEMBL3754700)
Affinity DataKi:  1.70E+4nMAssay Description:Non-competitive inhibition of electric eel acetylcholine esterase using acetylcholine iodide as substrate by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Bras£Lia

Curated by ChEMBL
LigandPNGBDBM50139049(CHEMBL3753732)
Affinity DataKi:  1.90E+4nMAssay Description:Non-competitive inhibition of electric eel acetylcholine esterase using acetylcholine iodide as substrate by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Bras£Lia

Curated by ChEMBL
LigandPNGBDBM50139051(CHEMBL3753070)
Affinity DataKi:  2.24E+4nMAssay Description:Non-competitive inhibition of electric eel acetylcholine esterase using acetylcholine iodide as substrate by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Bras£Lia

Curated by ChEMBL
LigandPNGBDBM50139007(CHEMBL3754287)
Affinity DataKi:  2.24E+4nMAssay Description:Mixed inhibition of electric eel acetylcholine esterase using acetylcholine iodide as substrate by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Bras£Lia

Curated by ChEMBL
LigandPNGBDBM50139053(CHEMBL3752227)
Affinity DataKi:  2.44E+4nMAssay Description:Non-competitive inhibition of electric eel acetylcholine esterase using acetylcholine iodide as substrate by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
University Of Bras£Lia

Curated by ChEMBL
LigandPNGBDBM10404((1S,12S,14R)-9-methoxy-4-methyl-11-oxa-4-azatetrac...)
Affinity DataIC50:  2.01E+3nMAssay Description:Inhibition of human acetylcholine esterase preincubated for 10 mins followed by the addition of 550 uM of acetylcholine iodide as substrate measured ...More data for this Ligand-Target Pair
TargetCholinesterase(Equus caballus (Horse))
University Of Bras£Lia

Curated by ChEMBL
LigandPNGBDBM50139052(CHEMBL3754700)
Affinity DataIC50:  3.10E+3nMAssay Description:Inhibition of horse butyrylcholine esterase preincubated for 10 mins followed by the addition of butyrylcholine iodide as substrate measured after 5 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Homo sapiens (Human))
University Of Bras£Lia

Curated by ChEMBL
LigandPNGBDBM50597595(CHEMBL5190179)
Affinity DataIC50:  4.62E+3nMAssay Description:Inhibition of BChE in human serum by Ellman's methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCholinesterase(Equus caballus (Horse))
University Of Bras£Lia

Curated by ChEMBL
LigandPNGBDBM50139053(CHEMBL3752227)
Affinity DataIC50:  5.00E+3nMAssay Description:Inhibition of horse butyrylcholine esterase preincubated for 10 mins followed by the addition of butyrylcholine iodide as substrate measured after 5 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
University Of Bras£Lia

Curated by ChEMBL
LigandPNGBDBM50139053(CHEMBL3752227)
Affinity DataIC50:  5.65E+3nMAssay Description:Inhibition of human acetylcholine esterase preincubated for 10 mins followed by the addition of 550 uM of acetylcholine iodide as substrate measured ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
University Of Bras£Lia

Curated by ChEMBL
LigandPNGBDBM50139053(CHEMBL3752227)
Affinity DataIC50:  5.65E+3nMAssay Description:Inhibition of AChE in human serum by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCholinesterase(Homo sapiens (Human))
University Of Bras£Lia

Curated by ChEMBL
LigandPNGBDBM50597594(CHEMBL5183866)
Affinity DataIC50:  6.12E+3nMAssay Description:Inhibition of BChE in human serum by Ellman's methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Bras£Lia

Curated by ChEMBL
LigandPNGBDBM50139053(CHEMBL3752227)
Affinity DataIC50:  6.60E+3nMAssay Description:Inhibition of electric eel acetylcholine esterase preincubated for 10 mins followed by the addition of acetylcholine iodide as substrate measured aft...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Homo sapiens (Human))
University Of Bras£Lia

Curated by ChEMBL
LigandPNGBDBM50597596(CHEMBL5195029)
Affinity DataIC50:  6.74E+3nMAssay Description:Inhibition of BChE in human serum by Ellman's methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCholinesterase(Equus caballus (Horse))
University Of Bras£Lia

Curated by ChEMBL
LigandPNGBDBM50139006(CHEMBL3753607)
Affinity DataIC50:  8.00E+3nMAssay Description:Inhibition of horse butyrylcholine esterase preincubated for 10 mins followed by the addition of butyrylcholine iodide as substrate measured after 5 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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