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Found 3 Enz. Inhib. hit(s) with Target = 'Alpha-1A adrenergic receptor' and Ligand = 'BDBM50393116'
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Universidade Federal Do Rio De Janeiro

Curated by ChEMBL
LigandPNGBDBM50393116(CHEMBL2153423)
Affinity DataKi:  0.140nMAssay Description:Displacement of [3H]prazosin from rat salivary gland adrenergic alpha 1A receptor after 45 mins by liquid scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
University Of Bras£Lia

Curated by ChEMBL
LigandPNGBDBM50393116(CHEMBL2153423)
Affinity DataKi:  3.5nMAssay Description:Displacement of [3H]prazosin from human alpha1A-adrenoceptor expressed in CHO cell membranes measured after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Universidade Federal Do Rio De Janeiro

Curated by ChEMBL
LigandPNGBDBM50393116(CHEMBL2153423)
Affinity DataIC50:  0.269nMAssay Description:Displacement of [3H]prazosin from rat salivary gland adrenergic alpha 1A receptor after 45 mins by liquid scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed