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Found 219 with Last Name = 'brodeur' and Initial = 'am'
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50249516(CHEMBL514011 | cis-2-(4-((3S,5S)-5-(3,3-difluoropy...)
Affinity DataIC50:  4.80nMAssay Description:Inhibition of human plasma DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM15494(3-{6-[(3R,4S)-3-amino-4-(2,4,5-trifluorophenyl)pyr...)
Affinity DataIC50:  5nMAssay Description:Inhibition of human recombinant DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50249548(CHEMBL475586 | cis-(3,3-difluoropyrrolidin-1-yl)((...)
Affinity DataIC50:  5.20nMAssay Description:Inhibition of human plasma DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50249515(CHEMBL474410 | cis-(3,3-difluoropyrrolidin-1-yl)((...)
Affinity DataIC50:  5.20nMAssay Description:Inhibition of human plasma DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50249514(CHEMBL474409 | cis-(3,3-difluoropyrrolidin-1-yl)((...)
Affinity DataIC50:  5.60nMAssay Description:Inhibition of human plasma DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50249513(CHEMBL475574 | cis-(3,3-difluoropyrrolidin-1-yl)((...)
Affinity DataIC50:  5.80nMAssay Description:Inhibition of human plasma DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50249512(CHEMBL475573 | cis-(3,3-difluoropyrrolidin-1-yl)((...)
Affinity DataIC50:  7.40nMAssay Description:Inhibition of human plasma DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50249481(CHEMBL515597 | cis-((2S,4S)-4-(4-(benzo[d]oxazol-2...)
Affinity DataIC50:  8.20nMAssay Description:Inhibition of human plasma DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50249480(CHEMBL475246 | cis-((2S,4S)-4-(4-(benzo[d]isoxazol...)
Affinity DataIC50:  8.70nMAssay Description:Inhibition of human plasma DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50249479(2-(4-{(3S,5S)-5-[(3,3-difluoropyrrolidin-1-yl)carb...)
Affinity DataIC50:  11nMAssay Description:Inhibition of human plasma DPP4More data for this Ligand-Target Pair
TargetDipeptidyl peptidase 4(Rattus norvegicus (rat))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50249479(2-(4-{(3S,5S)-5-[(3,3-difluoropyrrolidin-1-yl)carb...)
Affinity DataIC50:  13nMAssay Description:Inhibition of rat plasma DPP4More data for this Ligand-Target Pair
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50249479(2-(4-{(3S,5S)-5-[(3,3-difluoropyrrolidin-1-yl)carb...)
Affinity DataIC50:  13nMAssay Description:Inhibition of human recombinant DPP4More data for this Ligand-Target Pair
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50249552(CHEMBL474421 | cis-((3S,4R)-3,4-difluoropyrrolidin...)
Affinity DataIC50:  13nMAssay Description:Inhibition of human plasma DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50221102(CHEMBL236719 | N-(3-(6-((3R,4S)-3-amino-4-(2,4,5-t...)
Affinity DataIC50:  14nMAssay Description:Inhibition of human recombinant DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50221075(1-(3-(6-((3R,4S)-3-amino-4-(2,4,5-trifluorophenyl)...)
Affinity DataIC50:  19nMAssay Description:Inhibition of human recombinant DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM15492((3R,4S)-1-(6-phenylpyrimidin-4-yl)-4-(2,4,5-triflu...)
Affinity DataIC50:  21nMAssay Description:Inhibition of human recombinant DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM15492((3R,4S)-1-(6-phenylpyrimidin-4-yl)-4-(2,4,5-triflu...)
Affinity DataIC50:  21nMAssay Description:Inhibition of human recombinant DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50249098(CHEMBL515869 | cis-((2S,4S)-4-(4-(pyrimidin-2-yl)p...)
Affinity DataIC50:  25nMAssay Description:Inhibition of human plasma DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50249551(CHEMBL514623 | cis-((S)-3-fluoropyrrolidin-1-yl)((...)
Affinity DataIC50:  31nMAssay Description:Inhibition of human plasma DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50249549(CHEMBL473418 | cis-((2S,4S)-4-(4-(pyrimidin-2-yl)p...)
Affinity DataIC50:  31nMAssay Description:Inhibition of human plasma DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50221083((3R,4S)-1-(6-(pyridin-3-yl)pyrimidin-4-yl)-4-(2,4,...)
Affinity DataIC50:  31nMAssay Description:Inhibition of human recombinant DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50221094((3-(6-((3R,4S)-3-amino-4-(2,4,5-trifluorophenyl)py...)
Affinity DataIC50:  32nMAssay Description:Inhibition of human recombinant DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50221080(3-(6-((3R,4S)-3-amino-4-(2,4,5-trifluorophenyl)pyr...)
Affinity DataIC50:  37nMAssay Description:Inhibition of human recombinant DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50221073((3R,4S)-1-(6-(6-methoxypyridin-3-yl)pyrimidin-4-yl...)
Affinity DataIC50:  37nMAssay Description:Inhibition of human recombinant DPP4More data for this Ligand-Target Pair
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50221073((3R,4S)-1-(6-(6-methoxypyridin-3-yl)pyrimidin-4-yl...)
Affinity DataIC50:  37nMAssay Description:Inhibition of human recombinant DPP4More data for this Ligand-Target Pair
TargetDipeptidyl peptidase 4(Rattus norvegicus (rat))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50187266((2R,5S)-1-(2-(1-(hydroxymethyl)cyclopentylamino)ac...)
Affinity DataIC50:  38nMAssay Description:Inhibition of DPP4 in Sprague-Dawley rat plasmaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50249100(CHEMBL473188 | cis-(3-fluoroazetidin-1-yl)((2S,4S)...)
Affinity DataIC50:  41nMAssay Description:Inhibition of human plasma DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50221104((3R,4S)-1-(6-(3-methoxyphenyl)pyrimidin-4-yl)-4-(2...)
Affinity DataIC50:  47nMAssay Description:Inhibition of human recombinant DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50249550(CHEMBL473419 | cis-((R)-3-fluoropyrrolidin-1-yl)((...)
Affinity DataIC50:  51nMAssay Description:Inhibition of human plasma DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50221101((3R,4S)-1-(6-(4-fluorophenyl)pyrimidin-4-yl)-4-(2,...)
Affinity DataIC50:  51nMAssay Description:Inhibition of human recombinant DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50221085((3R,4S)-1-(6-(3-fluorophenyl)pyrimidin-4-yl)-4-(2,...)
Affinity DataIC50:  51nMAssay Description:Inhibition of human recombinant DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50221085((3R,4S)-1-(6-(3-fluorophenyl)pyrimidin-4-yl)-4-(2,...)
Affinity DataIC50:  51nMAssay Description:Inhibition of human recombinant DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50221088((3R,4S)-1-(6-(2-fluorophenyl)pyrimidin-4-yl)-4-(2,...)
Affinity DataIC50:  57nMAssay Description:Inhibition of human recombinant DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50187283((2R,5S)-1-(2-(1-(ethoxymethyl)cyclopentylamino)ace...)
Affinity DataIC50:  64nMAssay Description:Inhibition of human recombinant DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50221074(3-(6-((3R,4S)-3-amino-4-(2,4,5-trifluorophenyl)pyr...)
Affinity DataIC50:  70nMAssay Description:Inhibition of human recombinant DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50221082((3R,4S)-1-(6-(3-(trifluoromethyl)phenyl)pyrimidin-...)
Affinity DataIC50:  71nMAssay Description:Inhibition of human recombinant DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50187258((2S,5R)-1-[2-(hexahydro-2,5-methano-pentalen-3a-yl...)
Affinity DataIC50:  72nMAssay Description:Inhibition of human recombinant DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50187263((2S,5R)-1-[2-(3-hydroxy-adamantan-1-ylamino)-acety...)
Affinity DataIC50:  74nMAssay Description:Inhibition of human recombinant DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50187275((2R,5S)-1-(2-(1-(methoxymethyl)cyclopentylamino)ac...)
Affinity DataIC50:  84nMAssay Description:Inhibition of human recombinant DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50187261((2R,5S)-1-(2-(1-(butoxymethyl)cyclopentylamino)ace...)
Affinity DataIC50:  91nMAssay Description:Inhibition of human recombinant DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50187266((2R,5S)-1-(2-(1-(hydroxymethyl)cyclopentylamino)ac...)
Affinity DataIC50:  92nMAssay Description:Inhibition of DPP4 in cynomolgus monkey plasmaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50221098(2-(6-((3R,4S)-3-amino-4-(2,4,5-trifluorophenyl)pyr...)
Affinity DataIC50:  93nMAssay Description:Inhibition of human recombinant DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50187266((2R,5S)-1-(2-(1-(hydroxymethyl)cyclopentylamino)ac...)
Affinity DataIC50:  104nMAssay Description:Inhibition of human recombinant DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50187268((2S,5R)-1-[2-(adamantan-1-ylamino)-acetyl]-pyrroli...)
Affinity DataIC50:  106nMAssay Description:Inhibition of human recombinant DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50187266((2R,5S)-1-(2-(1-(hydroxymethyl)cyclopentylamino)ac...)
Affinity DataIC50:  109nMAssay Description:Inhibition of DPP4 in beagle dog plasmaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50187266((2R,5S)-1-(2-(1-(hydroxymethyl)cyclopentylamino)ac...)
Affinity DataIC50:  109nMAssay Description:Inhibition of DPP4 in beagle dog plasmaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50221099((3R,4S)-1-(6-(3-nitrophenyl)pyrimidin-4-yl)-4-(2,4...)
Affinity DataIC50:  120nMAssay Description:Inhibition of human recombinant DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50221086((3R,4S)-1-(6-(4-methoxyphenyl)pyrimidin-4-yl)-4-(2...)
Affinity DataIC50:  120nMAssay Description:Inhibition of human recombinant DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50187294((2R,5S)-1-(2-(1-(propoxymethyl)cyclopentylamino)ac...)
Affinity DataIC50:  123nMAssay Description:Inhibition of human recombinant DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50221077(4-(6-((3R,4S)-3-amino-4-(2,4,5-trifluorophenyl)pyr...)
Affinity DataIC50:  130nMAssay Description:Inhibition of human recombinant DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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