Affinity DataIC50: 3nMAssay Description:Inhibition of human recombinant HDAC1 using fluor de Lys as substrate by fluorometric analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 4nMAssay Description:Inhibition of human recombinant HDAC2 using fluor de Lys as substrate by fluorometric analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 6nMAssay Description:Inhibition of human recombinant HDAC1 using fluor de Lys as substrate by fluorometric analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 7nMAssay Description:Inhibition of human recombinant HDAC3 using fluor de Lys as substrate by fluorometric analysisMore data for this Ligand-Target Pair
TargetCell division cycle 7-related protein kinase(Homo sapiens (Human))
Nerviano Medical Sciences Oncology
Curated by ChEMBL
Nerviano Medical Sciences Oncology
Curated by ChEMBL
Affinity DataIC50: 10nMAssay Description:Inhibition of human recombinant HDAC3 using fluor de Lys as substrate by fluorometric analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 14nMAssay Description:Inhibition of human recombinant HDAC2 using fluor de Lys as substrate by fluorometric analysisMore data for this Ligand-Target Pair
TargetCyclin-dependent kinase 9(Homo sapiens (Human))
Nerviano Medical Sciences Oncology
Curated by ChEMBL
Nerviano Medical Sciences Oncology
Curated by ChEMBL
Affinity DataIC50: 24nMAssay Description:Inhibition of human recombinant HDAC2 using fluor de Lys as substrate by fluorometric analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 30nMAssay Description:Inhibition of human recombinant HDAC1 using fluor de Lys as substrate by fluorometric analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 30nMAssay Description:Inhibition of human recombinant HDAC6 using fluor de Lys as substrate by fluorometric analysisMore data for this Ligand-Target Pair
TargetCyclin-dependent kinase 1(Homo sapiens (Human))
Nerviano Medical Sciences Oncology
Curated by ChEMBL
Nerviano Medical Sciences Oncology
Curated by ChEMBL
TargetCyclin-dependent kinase 9(Homo sapiens (Human))
Nerviano Medical Sciences Oncology
Curated by ChEMBL
Nerviano Medical Sciences Oncology
Curated by ChEMBL
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
Nerviano Medical Sciences Oncology
Curated by ChEMBL
Nerviano Medical Sciences Oncology
Curated by ChEMBL
Affinity DataIC50: 150nMAssay Description:Inhibition of human recombinant HDAC3 using fluor de Lys as substrate by fluorometric analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 200nMAssay Description:Inhibition of human recombinant HDAC5 using fluor de Lys as substrate by fluorometric analysisMore data for this Ligand-Target Pair
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Nerviano Medical Sciences Oncology
Curated by ChEMBL
Nerviano Medical Sciences Oncology
Curated by ChEMBL
Affinity DataIC50: 220nMAssay Description:Inhibition of GSK3-betaMore data for this Ligand-Target Pair
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
Nerviano Medical Sciences Oncology
Curated by ChEMBL
Nerviano Medical Sciences Oncology
Curated by ChEMBL
TargetCyclin-dependent kinase 1(Homo sapiens (Human))
Nerviano Medical Sciences Oncology
Curated by ChEMBL
Nerviano Medical Sciences Oncology
Curated by ChEMBL
TargetCyclin-dependent kinase 5(Homo sapiens (Human))
Nerviano Medical Sciences Oncology
Curated by ChEMBL
Nerviano Medical Sciences Oncology
Curated by ChEMBL
TargetMAP kinase-activated protein kinase 2(Homo sapiens (Human))
Nerviano Medical Sciences Oncology
Curated by ChEMBL
Nerviano Medical Sciences Oncology
Curated by ChEMBL
Affinity DataIC50: 500nMAssay Description:Inhibition of human recombinant HDAC5 using fluor de Lys as substrate by fluorometric analysisMore data for this Ligand-Target Pair
TargetCyclin-dependent kinase 7(Homo sapiens (Human))
Nerviano Medical Sciences Oncology
Curated by ChEMBL
Nerviano Medical Sciences Oncology
Curated by ChEMBL
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
Nerviano Medical Sciences Oncology
Curated by ChEMBL
Nerviano Medical Sciences Oncology
Curated by ChEMBL
TargetSerine/threonine-protein kinase Chk2(Homo sapiens (Human))
Nerviano Medical Sciences Oncology
Curated by ChEMBL
Nerviano Medical Sciences Oncology
Curated by ChEMBL
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of chk2More data for this Ligand-Target Pair
Affinity DataIC50: 2.10E+3nMAssay Description:Inhibition of human recombinant HDAC6 using fluor de Lys as substrate by fluorometric analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of human recombinant HDAC5 using fluor de Lys as substrate by fluorometric analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 3.30E+3nMAssay Description:Inhibition of human recombinant HDAC6 using fluor de Lys as substrate by fluorometric analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of CYP2C19More data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of CYP2D6More data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of CYP2D6More data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of CYP3A4More data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of CYP3A4More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Nerviano Medical Sciences Oncology
Curated by ChEMBL
Nerviano Medical Sciences Oncology
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of chk1More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of Aurora-BMore data for this Ligand-Target Pair
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Nerviano Medical Sciences Oncology
Curated by ChEMBL
Nerviano Medical Sciences Oncology
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of AKT1More data for this Ligand-Target Pair
TargetVascular endothelial growth factor receptor 3(Homo sapiens (Human))
Nerviano Medical Sciences Oncology
Curated by ChEMBL
Nerviano Medical Sciences Oncology
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of VEGFR3More data for this Ligand-Target Pair
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Nerviano Medical Sciences Oncology
Curated by ChEMBL
Nerviano Medical Sciences Oncology
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of VEGFR2More data for this Ligand-Target Pair
TargetHigh affinity nerve growth factor receptor(Homo sapiens (Human))
Nerviano Medical Sciences Oncology
Curated by ChEMBL
Nerviano Medical Sciences Oncology
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of TRKAMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase TAO3(Homo sapiens (Human))
Nerviano Medical Sciences Oncology
Curated by ChEMBL
Nerviano Medical Sciences Oncology
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of TAO3More data for this Ligand-Target Pair
TargetSTE20-like serine/threonine-protein kinase(Homo sapiens (Human))
Nerviano Medical Sciences Oncology
Curated by ChEMBL
Nerviano Medical Sciences Oncology
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of STLK2More data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase receptor Ret(Homo sapiens (Human))
Nerviano Medical Sciences Oncology
Curated by ChEMBL
Nerviano Medical Sciences Oncology
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of RetMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Nerviano Medical Sciences Oncology
Curated by ChEMBL
Nerviano Medical Sciences Oncology
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of c-AblMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase ZAP-70(Homo sapiens (Human))
Nerviano Medical Sciences Oncology
Curated by ChEMBL
Nerviano Medical Sciences Oncology
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of ZAP70More data for this Ligand-Target Pair
TargetALK tyrosine kinase receptor(Homo sapiens (Human))
Nerviano Medical Sciences Oncology
Curated by ChEMBL
Nerviano Medical Sciences Oncology
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of AlkMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of Aurora-AMore data for this Ligand-Target Pair
TargetCyclin-dependent kinase 7(Homo sapiens (Human))
Nerviano Medical Sciences Oncology
Curated by ChEMBL
Nerviano Medical Sciences Oncology
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of Cdk7More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Nerviano Medical Sciences Oncology
Curated by ChEMBL
Nerviano Medical Sciences Oncology
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of ERK2More data for this Ligand-Target Pair
TargetFibroblast growth factor receptor 1(Homo sapiens (Human))
Nerviano Medical Sciences Oncology
Curated by ChEMBL
Nerviano Medical Sciences Oncology
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of FGFR1More data for this Ligand-Target Pair
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Nerviano Medical Sciences Oncology
Curated by ChEMBL
Nerviano Medical Sciences Oncology
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of IKK2More data for this Ligand-Target Pair