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Found 52 with Last Name = 'buonerba' and Initial = 'f'
TargetQuinolone resistance protein NorA(Staphylococcus aureus)
University Of Perugia

Curated by ChEMBL
LigandPNGBDBM50211232(CHEMBL3929187)
Affinity DataIC50:  1.80E+3nMAssay Description:Inhibition of Staphylococcus aureus 1199B NorA assessed as inhibition of ethidium bromide efflux measured after 5 mins by fluorometric methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetQuinolone resistance protein NorA(Staphylococcus aureus)
University Of Perugia

Curated by ChEMBL
LigandPNGBDBM50211228(CHEMBL3956740)
Affinity DataIC50:  2.02E+3nMAssay Description:Inhibition of Staphylococcus aureus 1199B NorA assessed as inhibition of ethidium bromide efflux measured after 5 mins by fluorometric methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetQuinolone resistance protein NorA(Staphylococcus aureus)
University Of Perugia

Curated by ChEMBL
LigandPNGBDBM50211230(CHEMBL3948087)
Affinity DataIC50:  3.83E+3nMAssay Description:Inhibition of Staphylococcus aureus 1199B NorA assessed as inhibition of ethidium bromide efflux measured after 5 mins by fluorometric methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetQuinolone resistance protein NorA(Staphylococcus aureus)
University Of Perugia

Curated by ChEMBL
LigandPNGBDBM50153269(CHEMBL3775575)
Affinity DataIC50:  4.40E+3nMAssay Description:Inhibition of NorA efflux pump in Staphylococcus aureus 1199B assessed as reduction in EtBr efflux incubated for 20 mins measured for 5 mins by real-...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetQuinolone resistance protein NorA(Staphylococcus aureus)
University Of Perugia

Curated by ChEMBL
LigandPNGBDBM50153186(CHEMBL3774520)
Affinity DataIC50:  4.80E+3nMAssay Description:Inhibition of NorA efflux pump in Staphylococcus aureus 1199B assessed as reduction in EtBr efflux incubated for 20 mins measured for 5 mins by real-...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetQuinolone resistance protein NorA(Staphylococcus aureus)
University Of Perugia

Curated by ChEMBL
LigandPNGBDBM50153316(CHEMBL3775207)
Affinity DataIC50:  4.80E+3nMAssay Description:Inhibition of NorA efflux pump in Staphylococcus aureus 1199B assessed as reduction in EtBr efflux incubated for 20 mins measured for 5 mins by real-...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetQuinolone resistance protein NorA(Staphylococcus aureus)
University Of Perugia

Curated by ChEMBL
LigandPNGBDBM50211229(CHEMBL3955315)
Affinity DataIC50:  4.93E+3nMAssay Description:Inhibition of Staphylococcus aureus 1199B NorA assessed as inhibition of ethidium bromide efflux measured after 5 mins by fluorometric methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetQuinolone resistance protein NorA(Staphylococcus aureus)
University Of Perugia

Curated by ChEMBL
LigandPNGBDBM50153183(CHEMBL3774548)
Affinity DataIC50:  5.00E+3nMAssay Description:Inhibition of NorA efflux pump in Staphylococcus aureus 1199B assessed as reduction in EtBr efflux incubated for 20 mins measured for 5 mins by real-...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetQuinolone resistance protein NorA(Staphylococcus aureus)
University Of Perugia

Curated by ChEMBL
LigandPNGBDBM50153314(CHEMBL3774689)
Affinity DataIC50:  5.10E+3nMAssay Description:Inhibition of NorA efflux pump in Staphylococcus aureus 1199B assessed as reduction in EtBr efflux incubated for 20 mins measured for 5 mins by real-...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetQuinolone resistance protein NorA(Staphylococcus aureus)
University Of Perugia

Curated by ChEMBL
LigandPNGBDBM50153284(CHEMBL3775852)
Affinity DataIC50:  5.80E+3nMAssay Description:Inhibition of NorA efflux pump in Staphylococcus aureus 1199B assessed as reduction in EtBr efflux incubated for 20 mins measured for 5 mins by real-...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetQuinolone resistance protein NorA(Staphylococcus aureus)
University Of Perugia

Curated by ChEMBL
LigandPNGBDBM50153278(CHEMBL3775105)
Affinity DataIC50:  6.00E+3nMAssay Description:Inhibition of Staphylococcus aureus 1199B NorA assessed as inhibition of ethidium bromide efflux measured after 5 mins by fluorometric methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetQuinolone resistance protein NorA(Staphylococcus aureus)
University Of Perugia

Curated by ChEMBL
LigandPNGBDBM50153278(CHEMBL3775105)
Affinity DataIC50:  6.00E+3nMAssay Description:Inhibition of NorA efflux pump in Staphylococcus aureus 1199B assessed as reduction in EtBr efflux incubated for 20 mins measured for 5 mins by real-...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetQuinolone resistance protein NorA(Staphylococcus aureus)
University Of Perugia

Curated by ChEMBL
LigandPNGBDBM50153271(CHEMBL3774968)
Affinity DataIC50:  6.10E+3nMAssay Description:Inhibition of NorA efflux pump in Staphylococcus aureus 1199B assessed as reduction in EtBr efflux incubated for 20 mins measured for 5 mins by real-...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetQuinolone resistance protein NorA(Staphylococcus aureus)
University Of Perugia

Curated by ChEMBL
LigandPNGBDBM50153187(CHEMBL3775401)
Affinity DataIC50:  6.10E+3nMAssay Description:Inhibition of NorA efflux pump in Staphylococcus aureus 1199B assessed as reduction in EtBr efflux incubated for 20 mins measured for 5 mins by real-...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetQuinolone resistance protein NorA(Staphylococcus aureus)
University Of Perugia

Curated by ChEMBL
LigandPNGBDBM50153317(CHEMBL3774886)
Affinity DataIC50:  6.10E+3nMAssay Description:Inhibition of NorA efflux pump in Staphylococcus aureus 1199B assessed as reduction in EtBr efflux incubated for 20 mins measured for 5 mins by real-...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetQuinolone resistance protein NorA(Staphylococcus aureus)
University Of Perugia

Curated by ChEMBL
LigandPNGBDBM50153268(CHEMBL3775173)
Affinity DataIC50:  6.30E+3nMAssay Description:Inhibition of NorA efflux pump in Staphylococcus aureus 1199B assessed as reduction in EtBr efflux incubated for 20 mins measured for 5 mins by real-...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetQuinolone resistance protein NorA(Staphylococcus aureus)
University Of Perugia

Curated by ChEMBL
LigandPNGBDBM50153270(CHEMBL3775819)
Affinity DataIC50:  6.50E+3nMAssay Description:Inhibition of NorA efflux pump in Staphylococcus aureus 1199B assessed as reduction in EtBr efflux incubated for 20 mins measured for 5 mins by real-...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetQuinolone resistance protein NorA(Staphylococcus aureus)
University Of Perugia

Curated by ChEMBL
LigandPNGBDBM50153272(CHEMBL3775722)
Affinity DataIC50:  6.60E+3nMAssay Description:Inhibition of NorA efflux pump in Staphylococcus aureus 1199B assessed as reduction in EtBr efflux incubated for 20 mins measured for 5 mins by real-...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetQuinolone resistance protein NorA(Staphylococcus aureus)
University Of Perugia

Curated by ChEMBL
LigandPNGBDBM50153283(CHEMBL3774445)
Affinity DataIC50:  6.70E+3nMAssay Description:Inhibition of NorA efflux pump in Staphylococcus aureus 1199B assessed as reduction in EtBr efflux incubated for 20 mins measured for 5 mins by real-...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetQuinolone resistance protein NorA(Staphylococcus aureus)
University Of Perugia

Curated by ChEMBL
LigandPNGBDBM50153182(CHEMBL3775053)
Affinity DataIC50:  6.70E+3nMAssay Description:Inhibition of NorA efflux pump in Staphylococcus aureus 1199B assessed as reduction in EtBr efflux incubated for 20 mins measured for 5 mins by real-...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetQuinolone resistance protein NorA(Staphylococcus aureus)
University Of Perugia

Curated by ChEMBL
LigandPNGBDBM50153285(CHEMBL3774995)
Affinity DataIC50:  6.80E+3nMAssay Description:Inhibition of NorA efflux pump in Staphylococcus aureus 1199B assessed as reduction in EtBr efflux incubated for 20 mins measured for 5 mins by real-...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetQuinolone resistance protein NorA(Staphylococcus aureus)
University Of Perugia

Curated by ChEMBL
LigandPNGBDBM50153185(CHEMBL3775726)
Affinity DataIC50:  7.10E+3nMAssay Description:Inhibition of NorA efflux pump in Staphylococcus aureus 1199B assessed as reduction in EtBr efflux incubated for 20 mins measured for 5 mins by real-...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetQuinolone resistance protein NorA(Staphylococcus aureus)
University Of Perugia

Curated by ChEMBL
LigandPNGBDBM50153184(CHEMBL3774891)
Affinity DataIC50:  7.30E+3nMAssay Description:Inhibition of NorA efflux pump in Staphylococcus aureus 1199B assessed as reduction in EtBr efflux incubated for 20 mins measured for 5 mins by real-...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetQuinolone resistance protein NorA(Staphylococcus aureus)
University Of Perugia

Curated by ChEMBL
LigandPNGBDBM50153192(CHEMBL3775789)
Affinity DataIC50:  8.70E+3nMAssay Description:Inhibition of NorA efflux pump in Staphylococcus aureus 1199B assessed as reduction in EtBr efflux incubated for 20 mins measured for 5 mins by real-...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetQuinolone resistance protein NorA(Staphylococcus aureus)
University Of Perugia

Curated by ChEMBL
LigandPNGBDBM50153277(CHEMBL3774527)
Affinity DataIC50:  1.01E+4nMAssay Description:Inhibition of NorA efflux pump in Staphylococcus aureus 1199B assessed as reduction in EtBr efflux incubated for 20 mins measured for 5 mins by real-...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetQuinolone resistance protein NorA(Staphylococcus aureus)
University Of Perugia

Curated by ChEMBL
LigandPNGBDBM50153288(CHEMBL3775693)
Affinity DataIC50:  1.04E+4nMAssay Description:Inhibition of NorA efflux pump in Staphylococcus aureus 1199B assessed as reduction in EtBr efflux incubated for 20 mins measured for 5 mins by real-...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetQuinolone resistance protein NorA(Staphylococcus aureus)
University Of Perugia

Curated by ChEMBL
LigandPNGBDBM50153279(CHEMBL3775483)
Affinity DataIC50:  1.06E+4nMAssay Description:Inhibition of NorA efflux pump in Staphylococcus aureus 1199B assessed as reduction in EtBr efflux incubated for 20 mins measured for 5 mins by real-...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetQuinolone resistance protein NorA(Staphylococcus aureus)
University Of Perugia

Curated by ChEMBL
LigandPNGBDBM50153274(CHEMBL3775322)
Affinity DataIC50:  1.16E+4nMAssay Description:Inhibition of NorA efflux pump in Staphylococcus aureus 1199B assessed as reduction in EtBr efflux incubated for 20 mins measured for 5 mins by real-...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetQuinolone resistance protein NorA(Staphylococcus aureus)
University Of Perugia

Curated by ChEMBL
LigandPNGBDBM50153280(CHEMBL3774675)
Affinity DataIC50:  1.19E+4nMAssay Description:Inhibition of NorA efflux pump in Staphylococcus aureus 1199B assessed as reduction in EtBr efflux incubated for 20 mins measured for 5 mins by real-...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetQuinolone resistance protein NorA(Staphylococcus aureus)
University Of Perugia

Curated by ChEMBL
LigandPNGBDBM50153282(CHEMBL3775841)
Affinity DataIC50:  1.25E+4nMAssay Description:Inhibition of NorA efflux pump in Staphylococcus aureus 1199B assessed as reduction in EtBr efflux incubated for 20 mins measured for 5 mins by real-...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetQuinolone resistance protein NorA(Staphylococcus aureus)
University Of Perugia

Curated by ChEMBL
LigandPNGBDBM50153281(CHEMBL3775062)
Affinity DataIC50:  1.25E+4nMAssay Description:Inhibition of NorA efflux pump in Staphylococcus aureus 1199B assessed as reduction in EtBr efflux incubated for 20 mins measured for 5 mins by real-...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetQuinolone resistance protein NorA(Staphylococcus aureus)
University Of Perugia

Curated by ChEMBL
LigandPNGBDBM50153282(CHEMBL3775841)
Affinity DataIC50:  1.25E+4nMAssay Description:Inhibition of Staphylococcus aureus 1199B NorA assessed as inhibition of ethidium bromide efflux measured after 5 mins by fluorometric methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetQuinolone resistance protein NorA(Staphylococcus aureus)
University Of Perugia

Curated by ChEMBL
LigandPNGBDBM50153315(CHEMBL3774582)
Affinity DataIC50:  1.37E+4nMAssay Description:Inhibition of NorA efflux pump in Staphylococcus aureus 1199B assessed as reduction in EtBr efflux incubated for 20 mins measured for 5 mins by real-...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetQuinolone resistance protein NorA(Staphylococcus aureus)
University Of Perugia

Curated by ChEMBL
LigandPNGBDBM50153249(CHEMBL3775871)
Affinity DataIC50:  1.41E+4nMAssay Description:Inhibition of NorA efflux pump in Staphylococcus aureus 1199B assessed as reduction in EtBr efflux incubated for 20 mins measured for 5 mins by real-...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetQuinolone resistance protein NorA(Staphylococcus aureus)
University Of Perugia

Curated by ChEMBL
LigandPNGBDBM50153247(CHEMBL3775857)
Affinity DataIC50:  1.42E+4nMAssay Description:Inhibition of NorA efflux pump in Staphylococcus aureus 1199B assessed as reduction in EtBr efflux incubated for 20 mins measured for 5 mins by real-...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetQuinolone resistance protein NorA(Staphylococcus aureus)
University Of Perugia

Curated by ChEMBL
LigandPNGBDBM50153276(CHEMBL3775445)
Affinity DataIC50:  1.55E+4nMAssay Description:Inhibition of NorA efflux pump in Staphylococcus aureus 1199B assessed as reduction in EtBr efflux incubated for 20 mins measured for 5 mins by real-...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetQuinolone resistance protein NorA(Staphylococcus aureus)
University Of Perugia

Curated by ChEMBL
LigandPNGBDBM50153275(CHEMBL3775842)
Affinity DataIC50:  1.68E+4nMAssay Description:Inhibition of NorA efflux pump in Staphylococcus aureus 1199B assessed as reduction in EtBr efflux incubated for 20 mins measured for 5 mins by real-...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetQuinolone resistance protein NorA(Staphylococcus aureus)
University Of Perugia

Curated by ChEMBL
LigandPNGBDBM50153286(CHEMBL3775271)
Affinity DataIC50:  1.70E+4nMAssay Description:Inhibition of NorA efflux pump in Staphylococcus aureus 1199B assessed as reduction in EtBr efflux incubated for 20 mins measured for 5 mins by real-...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetQuinolone resistance protein NorA(Staphylococcus aureus)
University Of Perugia

Curated by ChEMBL
LigandPNGBDBM50153287(CHEMBL3775507)
Affinity DataIC50:  1.71E+4nMAssay Description:Inhibition of Staphylococcus aureus 1199B NorA assessed as inhibition of ethidium bromide efflux measured after 5 mins by fluorometric methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetQuinolone resistance protein NorA(Staphylococcus aureus)
University Of Perugia

Curated by ChEMBL
LigandPNGBDBM50153287(CHEMBL3775507)
Affinity DataIC50:  1.71E+4nMAssay Description:Inhibition of NorA efflux pump in Staphylococcus aureus 1199B assessed as reduction in EtBr efflux incubated for 20 mins measured for 5 mins by real-...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetQuinolone resistance protein NorA(Staphylococcus aureus)
University Of Perugia

Curated by ChEMBL
LigandPNGBDBM50211231(CHEMBL3945575)
Affinity DataIC50:  1.99E+4nMAssay Description:Inhibition of Staphylococcus aureus 1199B NorA assessed as inhibition of ethidium bromide efflux measured after 5 mins by fluorometric methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetQuinolone resistance protein NorA(Staphylococcus aureus)
University Of Perugia

Curated by ChEMBL
LigandPNGBDBM50153273(CHEMBL3775114)
Affinity DataIC50:  2.25E+4nMAssay Description:Inhibition of NorA efflux pump in Staphylococcus aureus 1199B assessed as reduction in EtBr efflux incubated for 20 mins measured for 5 mins by real-...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBile acid receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50385214(CHEMBL2037313)
Affinity DataEC50:  3.00E+3nMAssay Description:Agonist activity at GST-tagged human FXR LBD assessed as recruitment of biotinylated SRC-1 peptide after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBile acid receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50436148(CHEMBL2398211)
Affinity DataEC50: >1.50E+5nMAssay Description:Agonist activity at GST-tagged human FXR LBD assessed as recruitment of biotinylated SRC-1 peptide after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBile acid receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50436141(CHEMBL2398210)
Affinity DataEC50: >1.50E+5nMAssay Description:Agonist activity at GST-tagged human FXR LBD assessed as recruitment of biotinylated SRC-1 peptide after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBile acid receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50436147(CHEMBL2398204)
Affinity DataEC50: >1.50E+5nMAssay Description:Agonist activity at GST-tagged human FXR LBD assessed as recruitment of biotinylated SRC-1 peptide after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBile acid receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50436146(CHEMBL2398205)
Affinity DataEC50: >1.50E+5nMAssay Description:Agonist activity at GST-tagged human FXR LBD assessed as recruitment of biotinylated SRC-1 peptide after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBile acid receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50385214(CHEMBL2037313)
Affinity DataEC50:  3.00E+3nMAssay Description:Agonist activity at GST-tagged human FXR LBD assessed as recruitment of biotinylated SRC-1 peptide after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBile acid receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50436145(CHEMBL2398206)
Affinity DataEC50: >1.50E+5nMAssay Description:Agonist activity at GST-tagged human FXR LBD assessed as recruitment of biotinylated SRC-1 peptide after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBile acid receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50436142(CHEMBL2398209)
Affinity DataEC50:  3.00E+3nMAssay Description:Agonist activity at GST-tagged human FXR LBD assessed as recruitment of biotinylated SRC-1 peptide after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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