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Found 38 with Last Name = 'burno' and Initial = 'm'
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50156061(CHEMBL365797 | CHEMBL556609 | N-(4-chloro-2-((1,3-...)
Affinity DataEC50:  245nMAssay Description:Effective concentration against metabotropic glutamate receptor 5 of human transfected into CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 5(Rattus norvegicus (Rat))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50156075(CHEMBL372002 | Pyridine-2-carboxylic acid (2,5-dip...)
Affinity DataEC50:  585nMAssay Description:Effective concentration against metabotropic glutamate receptor 5 of ratMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50156063(3-Chloro-N-(2,5-diphenyl-2H-pyrazol-3-yl)-benzamid...)
Affinity DataEC50:  40nMAssay Description:Effective concentration against metabotropic glutamate receptor 5 of human transfected into CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 5(Rattus norvegicus (Rat))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50156064(CHEMBL362527 | N-(2,5-Diphenyl-2H-pyrazol-3-yl)-4-...)
Affinity DataEC50:  50nMAssay Description:Effective concentration against metabotropic glutamate receptor 5 of ratMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 5(Rattus norvegicus (Rat))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50156065(CHEMBL191039 | N-(1,3-diphenyl-1H-pyrazol-5-yl)ben...)
Affinity DataEC50:  300nMAssay Description:Effective concentration against metabotropic glutamate receptor 5 of ratMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 5(Rattus norvegicus (Rat))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50156066(CHEMBL360813 | N-(2,5-Diphenyl-2H-pyrazol-3-yl)-3-...)
Affinity DataEC50:  100nMAssay Description:Effective concentration against metabotropic glutamate receptor 5 of ratMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 5(Rattus norvegicus (Rat))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50156067(CHEMBL188871 | Thiophene-2-carboxylic acid (2,5-di...)
Affinity DataEC50:  400nMAssay Description:Effective concentration against metabotropic glutamate receptor 5 of ratMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 5(Rattus norvegicus (Rat))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50156068(CHEMBL190326 | N-(1,3-diphenyl-1H-pyrazol-5-yl)-4-...)
Affinity DataEC50:  20nMAssay Description:Effective concentration against metabotropic glutamate receptor 5 of ratMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 5(Rattus norvegicus (Rat))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50156069(CHEMBL365409 | N-(1,3-diphenyl-1H-pyrazol-5-yl)-4-...)
Affinity DataEC50:  40nMAssay Description:Effective concentration against metabotropic glutamate receptor 5 of ratMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50156070(CHEMBL366217 | N-(4-Chloro-2-[(1,3-dioxo-1,3-dihyd...)
Affinity DataEC50:  300nMAssay Description:Effective concentration against metabotropic glutamate receptor 5 of human transfected into CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50156071(3-Cyano-N-(2,5-diphenyl-2H-pyrazol-3-yl)-benzamide...)
Affinity DataEC50:  10nMAssay Description:Effective concentration against metabotropic glutamate receptor 5 of human transfected into CHO cellsMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50156072(2-Chloro-N-(2,5-diphenyl-2H-pyrazol-3-yl)-benzamid...)
Affinity DataEC50:  2.50E+3nMAssay Description:Effective concentration against metabotropic glutamate receptor 5 of human transfected into CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 5(Rattus norvegicus (Rat))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50156073(CHEMBL194051 | N-(2,5-Diphenyl-2H-pyrazol-3-yl)-3-...)
Affinity DataEC50:  65nMAssay Description:Effective concentration against metabotropic glutamate receptor 5 of ratMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50156074(1,2-bis(3-fluorobenzylidene)hydrazine | CHEMBL3718...)
Affinity DataEC50:  2.36nMAssay Description:Effective concentration against metabotropic glutamate receptor 5 of human transfected into CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50156075(CHEMBL372002 | Pyridine-2-carboxylic acid (2,5-dip...)
Affinity DataEC50:  290nMAssay Description:Effective concentration against metabotropic glutamate receptor 5 of human transfected into CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50156076(CHEMBL191147 | N-(2,5-Diphenyl-2H-pyrazol-3-yl)-3,...)
Affinity DataEC50:  10nMAssay Description:Effective concentration against metabotropic glutamate receptor 5 of human transfected into CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50156065(CHEMBL191039 | N-(1,3-diphenyl-1H-pyrazol-5-yl)ben...)
Affinity DataEC50:  40nMAssay Description:Effective concentration against metabotropic glutamate receptor 5 of human transfected into CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50156073(CHEMBL194051 | N-(2,5-Diphenyl-2H-pyrazol-3-yl)-3-...)
Affinity DataEC50:  20nMAssay Description:Effective concentration against metabotropic glutamate receptor 5 of human transfected into CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 5(Rattus norvegicus (Rat))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50156077(4-Chloro-N-(2,5-diphenyl-2H-pyrazol-3-yl)-benzamid...)
Affinity DataEC50:  100nMAssay Description:Effective concentration against metabotropic glutamate receptor 5 of ratMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 5(Rattus norvegicus (Rat))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50156078(CHEMBL361478 | N-(2,5-Diphenyl-2H-pyrazol-3-yl)-2-...)
Affinity DataEC50:  100nMAssay Description:Effective concentration against metabotropic glutamate receptor 5 of ratMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 5(Rattus norvegicus (Rat))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50156079(CHEMBL365767 | N-(2,5-Diphenyl-2H-pyrazol-3-yl)-2-...)
Affinity DataEC50: >1.00E+4nMAssay Description:Effective concentration against metabotropic glutamate receptor 5 of ratMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 5(Rattus norvegicus (Rat))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50156076(CHEMBL191147 | N-(2,5-Diphenyl-2H-pyrazol-3-yl)-3,...)
Affinity DataEC50:  20nMAssay Description:Effective concentration against metabotropic glutamate receptor 5 of ratMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50156078(CHEMBL361478 | N-(2,5-Diphenyl-2H-pyrazol-3-yl)-2-...)
Affinity DataEC50:  75nMAssay Description:Effective concentration against metabotropic glutamate receptor 5 of human transfected into CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 5(Rattus norvegicus (Rat))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50156063(3-Chloro-N-(2,5-diphenyl-2H-pyrazol-3-yl)-benzamid...)
Affinity DataEC50:  200nMAssay Description:Effective concentration against metabotropic glutamate receptor 5 of ratMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 5(Rattus norvegicus (Rat))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50156062(CHEMBL188911 | Pyrazine-2-carboxylic acid (2,5-dip...)
Affinity DataEC50:  400nMAssay Description:Effective concentration against metabotropic glutamate receptor 5 of ratMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50156081(CHEMBL190084 | N-(2,5-Diphenyl-2H-pyrazol-3-yl)-2-...)
Affinity DataEC50: >1.00E+4nMAssay Description:Effective concentration against metabotropic glutamate receptor 5 of human transfected into CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 5(Rattus norvegicus (Rat))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50156071(3-Cyano-N-(2,5-diphenyl-2H-pyrazol-3-yl)-benzamide...)
Affinity DataEC50:  20nMAssay Description:Effective concentration against metabotropic glutamate receptor 5 of ratMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50156068(CHEMBL190326 | N-(1,3-diphenyl-1H-pyrazol-5-yl)-4-...)
Affinity DataEC50:  19nMAssay Description:Effective concentration against metabotropic glutamate receptor 5 of human transfected into CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50156066(CHEMBL360813 | N-(2,5-Diphenyl-2H-pyrazol-3-yl)-3-...)
Affinity DataEC50:  90nMAssay Description:Effective concentration against metabotropic glutamate receptor 5 of human transfected into CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50156079(CHEMBL365767 | N-(2,5-Diphenyl-2H-pyrazol-3-yl)-2-...)
Affinity DataEC50: >1.00E+4nMAssay Description:Effective concentration against metabotropic glutamate receptor 5 of human transfected into CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50156080(CHEMBL366326 | Thiophene-3-carboxylic acid (2,5-di...)
Affinity DataEC50:  1.80E+3nMAssay Description:Effective concentration against metabotropic glutamate receptor 5 of human transfected into CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50156064(CHEMBL362527 | N-(2,5-Diphenyl-2H-pyrazol-3-yl)-4-...)
Affinity DataEC50:  30nMAssay Description:Effective concentration against metabotropic glutamate receptor 5 of human transfected into CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 5(Rattus norvegicus (Rat))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50156080(CHEMBL366326 | Thiophene-3-carboxylic acid (2,5-di...)
Affinity DataEC50:  2.90E+3nMAssay Description:Effective concentration against metabotropic glutamate receptor 5 of ratMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50156077(4-Chloro-N-(2,5-diphenyl-2H-pyrazol-3-yl)-benzamid...)
Affinity DataEC50:  20nMAssay Description:Effective concentration against metabotropic glutamate receptor 5 of human transfected into CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50156069(CHEMBL365409 | N-(1,3-diphenyl-1H-pyrazol-5-yl)-4-...)
Affinity DataEC50:  30nMAssay Description:Effective concentration against metabotropic glutamate receptor 5 of human transfected into CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50156067(CHEMBL188871 | Thiophene-2-carboxylic acid (2,5-di...)
Affinity DataEC50:  200nMAssay Description:Effective concentration against metabotropic glutamate receptor 5 of human transfected into CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50156082(CHEMBL362969 | N-(4-bromo-2-((1,3-dioxoisoindolin-...)
Affinity DataEC50:  740nMAssay Description:Effective concentration against metabotropic glutamate receptor 5 of human transfected into CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50156062(CHEMBL188911 | Pyrazine-2-carboxylic acid (2,5-dip...)
Affinity DataEC50:  200nMAssay Description:Effective concentration against metabotropic glutamate receptor 5 of human transfected into CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed