TargetAlpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor(RAT)
Reckitt & Colman
Curated by ChEMBL
Reckitt & Colman
Curated by ChEMBL
Affinity DataIC50: 78nMAssay Description:Inhibitory activity against Alpha-2 adrenergic receptor in rat vas deferensMore data for this Ligand-Target Pair
Affinity DataKd: 14nMAssay Description:In vitro presynaptic agonist potency at alpha-2 adrenergic receptor in rat or mouse vas deferens relative to clonidineMore data for this Ligand-Target Pair
Affinity DataKd: 13.8nMAssay Description:In vitro presynaptic agonist potency at alpha-2 adrenergic receptor in rat or mouse vas deferens relative to clonidineMore data for this Ligand-Target Pair