Affinity DataKi: 0.00800nMAssay Description:Potency of inhibition against human leukocyte elastase (HLE) expressed as an apparent binding constantMore data for this Ligand-Target Pair
Affinity DataKi: 0.0110nMAssay Description:Potency of inhibition against human leukocyte elastase (HLE) expressed as an apparent binding constantMore data for this Ligand-Target Pair
Affinity DataKi: 0.0110nMAssay Description:Potency of inhibition against human leukocyte elastase (HLE) expressed as an apparent binding constantMore data for this Ligand-Target Pair
Affinity DataKi: 0.0130nMAssay Description:Potency of inhibition against human leukocyte elastase (HLE) expressed as an apparent binding constantMore data for this Ligand-Target Pair
Affinity DataKi: 0.0130nMAssay Description:Potency of inhibition against human leukocyte elastase (HLE) expressed as an apparent binding constantMore data for this Ligand-Target Pair
Affinity DataKi: 0.0140nMAssay Description:Potency of inhibition against human leukocyte elastase (HLE) expressed as an apparent binding constantMore data for this Ligand-Target Pair
Affinity DataKi: 0.200nMAssay Description:Potency of inhibition against human leukocyte elastase (HLE) expressed as an apparent binding constantMore data for this Ligand-Target Pair
Affinity DataKi: 15nMAssay Description:Potency of inhibition against human leukocyte elastase (HLE) expressed as an apparent binding constantMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Sterling Winthrop Research
Curated by ChEMBL
Sterling Winthrop Research
Curated by ChEMBL
Affinity DataIC50: 2.10E+4nMAssay Description:Blockade of the delayed rectifier K+ current (IKr) of guinea pig myocytesMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Sterling Winthrop Research
Curated by ChEMBL
Sterling Winthrop Research
Curated by ChEMBL
Affinity DataIC50: 2.90E+4nMAssay Description:Blockade of the delayed rectifier K+ current (IKr) of guinea pig myocytesMore data for this Ligand-Target Pair
TargetSodium channel protein type 5 subunit alpha(Homo sapiens (Human))
Sterling Winthrop Research
Curated by ChEMBL
Sterling Winthrop Research
Curated by ChEMBL
Affinity DataIC50: >3.00E+4nMAssay Description:Blockade of Na+ current in frog oocytes expressing human cardiac sodium channel (HH1)More data for this Ligand-Target Pair
TargetSodium channel protein type 5 subunit alpha(Homo sapiens (Human))
Sterling Winthrop Research
Curated by ChEMBL
Sterling Winthrop Research
Curated by ChEMBL
Affinity DataIC50: >3.00E+4nMAssay Description:Blockade of Na+ current in frog oocytes expressing human cardiac sodium channel (HH1)More data for this Ligand-Target Pair
TargetSodium channel protein type 5 subunit alpha(Homo sapiens (Human))
Sterling Winthrop Research
Curated by ChEMBL
Sterling Winthrop Research
Curated by ChEMBL
Affinity DataIC50: >3.00E+4nMAssay Description:Blockade of Na+ current in frog oocytes expressing human cardiac sodium channel (HH1)More data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Sterling Winthrop Research
Curated by ChEMBL
Sterling Winthrop Research
Curated by ChEMBL
Affinity DataIC50: 3.80E+4nMAssay Description:Blockade of the delayed rectifier K+ current (IKr) of guinea pig myocytesMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Sterling Winthrop Research
Curated by ChEMBL
Sterling Winthrop Research
Curated by ChEMBL
Affinity DataIC50: 3.80E+4nMAssay Description:Blockade of the delayed rectifier K+ current (IKr) of guinea pig myocytesMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Sterling Winthrop Research
Curated by ChEMBL
Sterling Winthrop Research
Curated by ChEMBL
Affinity DataIC50: 4.40E+4nMAssay Description:Blockade of the delayed rectifier K+ current (IKr) of guinea pig myocytesMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Sterling Winthrop Research
Curated by ChEMBL
Sterling Winthrop Research
Curated by ChEMBL
Affinity DataIC50: 8.50E+4nMAssay Description:Blockade of the delayed rectifier K+ current (IKr) of guinea pig myocytesMore data for this Ligand-Target Pair
TargetSodium channel protein type 5 subunit alpha(Homo sapiens (Human))
Sterling Winthrop Research
Curated by ChEMBL
Sterling Winthrop Research
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Blockade of Na+ current in frog oocytes expressing human cardiac sodium channel (HH1)More data for this Ligand-Target Pair
TargetSodium channel protein type 5 subunit alpha(Homo sapiens (Human))
Sterling Winthrop Research
Curated by ChEMBL
Sterling Winthrop Research
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Blockade of Na+ current in frog oocytes expressing human cardiac sodium channel (HH1)More data for this Ligand-Target Pair
TargetSodium channel protein type 5 subunit alpha(Homo sapiens (Human))
Sterling Winthrop Research
Curated by ChEMBL
Sterling Winthrop Research
Curated by ChEMBL
Affinity DataIC50: 1.26E+5nMAssay Description:Blockade of Na+ current in frog oocytes expressing human cardiac sodium channel (HH1)More data for this Ligand-Target Pair
TargetSodium channel protein type 5 subunit alpha(Homo sapiens (Human))
Sterling Winthrop Research
Curated by ChEMBL
Sterling Winthrop Research
Curated by ChEMBL
Affinity DataIC50: >3.00E+5nMAssay Description:Blockade of Na+ current in frog oocytes expressing human cardiac sodium channel (HH1)More data for this Ligand-Target Pair