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Found 57 with Last Name = 'carmo carreiras' and Initial = 'm'
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Lisbon

Curated by ChEMBL
LigandPNGBDBM50384793(CHEMBL2037384)
Affinity DataKi:  155nMAssay Description:Mixed type inhibition of electric eel AChE using acetylthiocholine as substrate by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Lisbon

Curated by ChEMBL
LigandPNGBDBM50541071(CHEMBL4528766)
Affinity DataIC50:  1.10nMAssay Description:Inhibition of electric eel AChE by Ellman's methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
Universidade De Lisboa

Curated by ChEMBL
LigandPNGBDBM50541069(CHEMBL4635389)
Affinity DataIC50:  2.80nMAssay Description:Inhibition of rat MAO B using kynuramine as substrate preincubated for 30 mins followed by substrate additionMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
University Of Lisbon

Curated by ChEMBL
LigandPNGBDBM8961(1,2,3,4-tetrahydro-9-acridinamine | 1,2,3,4-tetrah...)
Affinity DataIC50:  5.20nMAssay Description:Inhibition of Equus caballus BChE preincubated for 10 mins measured after 15 mins by Ellman's methodMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Universidade De Lisboa

Curated by ChEMBL
LigandPNGBDBM50359391(CHEMBL1929421)
Affinity DataIC50:  5.40nMAssay Description:Inhibition of human MAO AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Universidade De Lisboa

Curated by ChEMBL
LigandPNGBDBM50541052(CHEMBL4632951)
Affinity DataIC50:  9.40nMAssay Description:Inhibition of human AChE using acetylthiocholine chloride as substrate peincubated for 15 mins followed by substrate addition measured at 1 min inter...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Lisbon

Curated by ChEMBL
LigandPNGBDBM50541052(CHEMBL4632951)
Affinity DataIC50:  11nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine chloride as substrate peincubated for 15 mins followed by substrate addition measured at 1 mi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Lisbon

Curated by ChEMBL
LigandPNGBDBM8987(6-chloro-1,2,3,4-tetrahydroacridin-9-amine | 6-chl...)
Affinity DataIC50:  24nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine chloride as substrate peincubated for 15 mins followed by substrate addition measured at 1 mi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Lisbon

Curated by ChEMBL
LigandPNGBDBM8961(1,2,3,4-tetrahydro-9-acridinamine | 1,2,3,4-tetrah...)
Affinity DataIC50:  27nMAssay Description:Inhibition of electric eel AChE preincubated for 10 mins measured after 15 mins by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Universidade De Lisboa

Curated by ChEMBL
LigandPNGBDBM50541051(CHEMBL4633540)
Affinity DataIC50:  51nMAssay Description:Inhibition of human AChE using acetylthiocholine chloride as substrate peincubated for 15 mins followed by substrate addition measured at 1 min inter...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Lisbon

Curated by ChEMBL
LigandPNGBDBM8961(1,2,3,4-tetrahydro-9-acridinamine | 1,2,3,4-tetrah...)
Affinity DataIC50:  51nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine chloride as substrate peincubated for 15 mins followed by substrate addition measured at 1 mi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Lisbon

Curated by ChEMBL
LigandPNGBDBM50541051(CHEMBL4633540)
Affinity DataIC50:  51nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine chloride as substrate peincubated for 15 mins followed by substrate addition measured at 1 mi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Lisbon

Curated by ChEMBL
LigandPNGBDBM50384793(CHEMBL2037384)
Affinity DataIC50:  69nMAssay Description:Inhibition of electric eel AChE preincubated for 10 mins measured after 15 mins by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
University Of Lisbon

Curated by ChEMBL
LigandPNGBDBM50541051(CHEMBL4633540)
Affinity DataIC50:  78nMAssay Description:Inhibition of equine serum BuChE using butylthiocholine chloride as substrate peincubated for 15 mins followed by substrate addition measured at 1 mi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
University Of Lisbon

Curated by ChEMBL
LigandPNGBDBM50541052(CHEMBL4632951)
Affinity DataIC50:  84nMAssay Description:Inhibition of equine serum BuChE using butylthiocholine chloride as substrate peincubated for 15 mins followed by substrate addition measured at 1 mi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Universidade De Lisboa

Curated by ChEMBL
LigandPNGBDBM50359391(CHEMBL1929421)
Affinity DataIC50:  177nMAssay Description:Inhibition of human MAO BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
Universidade De Lisboa

Curated by ChEMBL
LigandPNGBDBM8961(1,2,3,4-tetrahydro-9-acridinamine | 1,2,3,4-tetrah...)
Affinity DataIC50:  190nMAssay Description:Inhibition of Torpedo californica AChE using acetylthiocholine chloride as substrate peincubated for 15 mins followed by substrate addition measured ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
Universidade De Lisboa

Curated by ChEMBL
LigandPNGBDBM50541068(CHEMBL4648667)
Affinity DataIC50:  214nMAssay Description:Inhibition of rat MAO B using kynuramine as substrate preincubated for 30 mins followed by substrate additionMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Lisbon

Curated by ChEMBL
LigandPNGBDBM50541054(CHEMBL4637721)
Affinity DataIC50:  226nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine chloride as substrate peincubated for 15 mins followed by substrate addition measured at 1 mi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Lisbon

Curated by ChEMBL
LigandPNGBDBM50384792(CHEMBL2037385)
Affinity DataIC50:  230nMAssay Description:Inhibition of electric eel AChE preincubated for 10 mins measured after 15 mins by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
Universidade De Lisboa

Curated by ChEMBL
LigandPNGBDBM50541064(CHEMBL4635698)
Affinity DataIC50:  250nMAssay Description:Inhibition of Torpedo californica AChE using acetylthiocholine chloride as substrate peincubated for 15 mins followed by substrate addition measured ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
Universidade De Lisboa

Curated by ChEMBL
LigandPNGBDBM50541065(CHEMBL4633417)
Affinity DataIC50:  250nMAssay Description:Inhibition of Torpedo californica AChE using acetylthiocholine chloride as substrate peincubated for 15 mins followed by substrate addition measured ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
Universidade De Lisboa

Curated by ChEMBL
LigandPNGBDBM50541061(CHEMBL4635342)
Affinity DataIC50:  250nMAssay Description:Inhibition of Torpedo californica AChE using acetylthiocholine chloride as substrate peincubated for 15 mins followed by substrate addition measured ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
Universidade De Lisboa

Curated by ChEMBL
LigandPNGBDBM50541063(CHEMBL4637185)
Affinity DataIC50:  250nMAssay Description:Inhibition of Torpedo californica AChE using acetylthiocholine chloride as substrate peincubated for 15 mins followed by substrate addition measured ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
Universidade De Lisboa

Curated by ChEMBL
LigandPNGBDBM50541066(CHEMBL4641182)
Affinity DataIC50:  250nMAssay Description:Inhibition of Torpedo californica AChE using acetylthiocholine chloride as substrate peincubated for 15 mins followed by substrate addition measured ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
Universidade De Lisboa

Curated by ChEMBL
LigandPNGBDBM50541059(CHEMBL4648566)
Affinity DataIC50:  250nMAssay Description:Inhibition of Torpedo californica AChE using acetylthiocholine chloride as substrate peincubated for 15 mins followed by substrate addition measured ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
Universidade De Lisboa

Curated by ChEMBL
LigandPNGBDBM50541060(CHEMBL4642573)
Affinity DataIC50:  250nMAssay Description:Inhibition of Torpedo californica AChE using acetylthiocholine chloride as substrate peincubated for 15 mins followed by substrate addition measured ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
Universidade De Lisboa

Curated by ChEMBL
LigandPNGBDBM50541062(CHEMBL4640059)
Affinity DataIC50:  280nMAssay Description:Inhibition of Torpedo californica AChE using acetylthiocholine chloride as substrate peincubated for 15 mins followed by substrate addition measured ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
Universidade De Lisboa

Curated by ChEMBL
LigandPNGBDBM50541057(CHEMBL4639993)
Affinity DataIC50:  300nMAssay Description:Inhibition of Torpedo californica AChE using acetylthiocholine chloride as substrate peincubated for 15 mins followed by substrate addition measured ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Lisbon

Curated by ChEMBL
LigandPNGBDBM50541055(CHEMBL4647462)
Affinity DataIC50:  339nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine chloride as substrate peincubated for 15 mins followed by substrate addition measured at 1 mi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
University Of Lisbon

Curated by ChEMBL
LigandPNGBDBM50541055(CHEMBL4647462)
Affinity DataIC50:  353nMAssay Description:Inhibition of equine serum BuChE using butylthiocholine chloride as substrate peincubated for 15 mins followed by substrate addition measured at 1 mi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
Universidade De Lisboa

Curated by ChEMBL
LigandPNGBDBM50541067(CHEMBL4638612)
Affinity DataIC50:  377nMAssay Description:Inhibition of rat MAO B using kynuramine as substrate preincubated for 30 mins followed by substrate additionMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
Universidade De Lisboa

Curated by ChEMBL
LigandPNGBDBM50541058(CHEMBL4639503)
Affinity DataIC50:  560nMAssay Description:Inhibition of Torpedo californica AChE using acetylthiocholine chloride as substrate peincubated for 15 mins followed by substrate addition measured ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Lisbon

Curated by ChEMBL
LigandPNGBDBM50384794(CHEMBL2037380)
Affinity DataIC50:  570nMAssay Description:Inhibition of electric eel AChE preincubated for 10 mins measured after 15 mins by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
University Of Lisbon

Curated by ChEMBL
LigandPNGBDBM50541071(CHEMBL4528766)
Affinity DataIC50:  600nMAssay Description:Inhibition of equine serum BuChE by Ellman's methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Lisbon

Curated by ChEMBL
LigandPNGBDBM50384796(CHEMBL2037382)
Affinity DataIC50:  600nMAssay Description:Inhibition of electric eel AChE preincubated for 10 mins measured after 15 mins by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
Universidade De Lisboa

Curated by ChEMBL
LigandPNGBDBM50541068(CHEMBL4648667)
Affinity DataIC50:  669nMAssay Description:Inhibition of rat MAO A using kynuramine as substrate preincubated for 30 mins followed by substrate additionMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Universidade De Lisboa

Curated by ChEMBL
LigandPNGBDBM50359391(CHEMBL1929421)
Affinity DataIC50:  810nMAssay Description:Inhibition of human AChEMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
Universidade De Lisboa

Curated by ChEMBL
LigandPNGBDBM50541056(CHEMBL4633036)
Affinity DataIC50:  880nMAssay Description:Inhibition of Torpedo californica AChE using acetylthiocholine chloride as substrate peincubated for 15 mins followed by substrate addition measured ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Lisbon

Curated by ChEMBL
LigandPNGBDBM50541053(CHEMBL4642125)
Affinity DataIC50:  884nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine chloride as substrate peincubated for 15 mins followed by substrate addition measured at 1 mi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
Universidade De Lisboa

Curated by ChEMBL
LigandPNGBDBM50541050(CHEMBL4647757)
Affinity DataIC50:  1.21E+3nMAssay Description:Inhibition of Torpedo californica AChE using acetylthiocholine chloride as substrate peincubated for 15 mins followed by substrate addition measured ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Lisbon

Curated by ChEMBL
LigandPNGBDBM50384795(CHEMBL2037381)
Affinity DataIC50:  1.70E+3nMAssay Description:Inhibition of electric eel AChE preincubated for 10 mins measured after 15 mins by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Homo sapiens (Human))
Universidade De Lisboa

Curated by ChEMBL
LigandPNGBDBM50359391(CHEMBL1929421)
Affinity DataIC50:  1.82E+3nMAssay Description:Inhibition of human BuChEMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Lisbon

Curated by ChEMBL
LigandPNGBDBM50541070(CHEMBL4647954)
Affinity DataIC50:  2.78E+3nMAssay Description:Inhibition of electric eel AChE by Ellman's methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Lisbon

Curated by ChEMBL
LigandPNGBDBM50541068(CHEMBL4648667)
Affinity DataIC50:  2.78E+3nMAssay Description:Inhibition of electric eel AChE by Ellman's methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Lisbon

Curated by ChEMBL
LigandPNGBDBM50541067(CHEMBL4638612)
Affinity DataIC50:  2.78E+3nMAssay Description:Inhibition of electric eel AChE by Ellman's methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Universidade De Lisboa

Curated by ChEMBL
LigandPNGBDBM50541071(CHEMBL4528766)
Affinity DataIC50:  3.95E+3nMAssay Description:Inhibition of human MAO BMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
University Of Lisbon

Curated by ChEMBL
LigandPNGBDBM50541053(CHEMBL4642125)
Affinity DataIC50:  5.38E+3nMAssay Description:Inhibition of equine serum BuChE using butylthiocholine chloride as substrate peincubated for 15 mins followed by substrate addition measured at 1 mi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
University Of Lisbon

Curated by ChEMBL
LigandPNGBDBM50384796(CHEMBL2037382)
Affinity DataIC50:  5.40E+3nMAssay Description:Inhibition of Equus caballus BChE preincubated for 10 mins measured after 15 mins by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
University Of Lisbon

Curated by ChEMBL
LigandPNGBDBM50384793(CHEMBL2037384)
Affinity DataIC50:  6.30E+3nMAssay Description:Inhibition of Equus caballus BChE preincubated for 10 mins measured after 15 mins by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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