TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Lisbon
Curated by ChEMBL
University Of Lisbon
Curated by ChEMBL
Affinity DataKi: 155nMAssay Description:Mixed type inhibition of electric eel AChE using acetylthiocholine as substrate by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Lisbon
Curated by ChEMBL
University Of Lisbon
Curated by ChEMBL
Affinity DataIC50: 1.10nMAssay Description:Inhibition of electric eel AChE by Ellman's methodMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
Universidade De Lisboa
Curated by ChEMBL
Universidade De Lisboa
Curated by ChEMBL
Affinity DataIC50: 2.80nMAssay Description:Inhibition of rat MAO B using kynuramine as substrate preincubated for 30 mins followed by substrate additionMore data for this Ligand-Target Pair
Affinity DataIC50: 5.20nMAssay Description:Inhibition of Equus caballus BChE preincubated for 10 mins measured after 15 mins by Ellman's methodMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Universidade De Lisboa
Curated by ChEMBL
Universidade De Lisboa
Curated by ChEMBL
Affinity DataIC50: 5.40nMAssay Description:Inhibition of human MAO AMore data for this Ligand-Target Pair
Affinity DataIC50: 9.40nMAssay Description:Inhibition of human AChE using acetylthiocholine chloride as substrate peincubated for 15 mins followed by substrate addition measured at 1 min inter...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Lisbon
Curated by ChEMBL
University Of Lisbon
Curated by ChEMBL
Affinity DataIC50: 11nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine chloride as substrate peincubated for 15 mins followed by substrate addition measured at 1 mi...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Lisbon
Curated by ChEMBL
University Of Lisbon
Curated by ChEMBL
Affinity DataIC50: 24nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine chloride as substrate peincubated for 15 mins followed by substrate addition measured at 1 mi...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Lisbon
Curated by ChEMBL
University Of Lisbon
Curated by ChEMBL
Affinity DataIC50: 27nMAssay Description:Inhibition of electric eel AChE preincubated for 10 mins measured after 15 mins by Ellman's methodMore data for this Ligand-Target Pair
Affinity DataIC50: 51nMAssay Description:Inhibition of human AChE using acetylthiocholine chloride as substrate peincubated for 15 mins followed by substrate addition measured at 1 min inter...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Lisbon
Curated by ChEMBL
University Of Lisbon
Curated by ChEMBL
Affinity DataIC50: 51nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine chloride as substrate peincubated for 15 mins followed by substrate addition measured at 1 mi...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Lisbon
Curated by ChEMBL
University Of Lisbon
Curated by ChEMBL
Affinity DataIC50: 51nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine chloride as substrate peincubated for 15 mins followed by substrate addition measured at 1 mi...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Lisbon
Curated by ChEMBL
University Of Lisbon
Curated by ChEMBL
Affinity DataIC50: 69nMAssay Description:Inhibition of electric eel AChE preincubated for 10 mins measured after 15 mins by Ellman's methodMore data for this Ligand-Target Pair
Affinity DataIC50: 78nMAssay Description:Inhibition of equine serum BuChE using butylthiocholine chloride as substrate peincubated for 15 mins followed by substrate addition measured at 1 mi...More data for this Ligand-Target Pair
Affinity DataIC50: 84nMAssay Description:Inhibition of equine serum BuChE using butylthiocholine chloride as substrate peincubated for 15 mins followed by substrate addition measured at 1 mi...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Universidade De Lisboa
Curated by ChEMBL
Universidade De Lisboa
Curated by ChEMBL
Affinity DataIC50: 177nMAssay Description:Inhibition of human MAO BMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
Universidade De Lisboa
Curated by ChEMBL
Universidade De Lisboa
Curated by ChEMBL
Affinity DataIC50: 190nMAssay Description:Inhibition of Torpedo californica AChE using acetylthiocholine chloride as substrate peincubated for 15 mins followed by substrate addition measured ...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
Universidade De Lisboa
Curated by ChEMBL
Universidade De Lisboa
Curated by ChEMBL
Affinity DataIC50: 214nMAssay Description:Inhibition of rat MAO B using kynuramine as substrate preincubated for 30 mins followed by substrate additionMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Lisbon
Curated by ChEMBL
University Of Lisbon
Curated by ChEMBL
Affinity DataIC50: 226nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine chloride as substrate peincubated for 15 mins followed by substrate addition measured at 1 mi...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Lisbon
Curated by ChEMBL
University Of Lisbon
Curated by ChEMBL
Affinity DataIC50: 230nMAssay Description:Inhibition of electric eel AChE preincubated for 10 mins measured after 15 mins by Ellman's methodMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
Universidade De Lisboa
Curated by ChEMBL
Universidade De Lisboa
Curated by ChEMBL
Affinity DataIC50: 250nMAssay Description:Inhibition of Torpedo californica AChE using acetylthiocholine chloride as substrate peincubated for 15 mins followed by substrate addition measured ...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
Universidade De Lisboa
Curated by ChEMBL
Universidade De Lisboa
Curated by ChEMBL
Affinity DataIC50: 250nMAssay Description:Inhibition of Torpedo californica AChE using acetylthiocholine chloride as substrate peincubated for 15 mins followed by substrate addition measured ...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
Universidade De Lisboa
Curated by ChEMBL
Universidade De Lisboa
Curated by ChEMBL
Affinity DataIC50: 250nMAssay Description:Inhibition of Torpedo californica AChE using acetylthiocholine chloride as substrate peincubated for 15 mins followed by substrate addition measured ...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
Universidade De Lisboa
Curated by ChEMBL
Universidade De Lisboa
Curated by ChEMBL
Affinity DataIC50: 250nMAssay Description:Inhibition of Torpedo californica AChE using acetylthiocholine chloride as substrate peincubated for 15 mins followed by substrate addition measured ...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
Universidade De Lisboa
Curated by ChEMBL
Universidade De Lisboa
Curated by ChEMBL
Affinity DataIC50: 250nMAssay Description:Inhibition of Torpedo californica AChE using acetylthiocholine chloride as substrate peincubated for 15 mins followed by substrate addition measured ...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
Universidade De Lisboa
Curated by ChEMBL
Universidade De Lisboa
Curated by ChEMBL
Affinity DataIC50: 250nMAssay Description:Inhibition of Torpedo californica AChE using acetylthiocholine chloride as substrate peincubated for 15 mins followed by substrate addition measured ...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
Universidade De Lisboa
Curated by ChEMBL
Universidade De Lisboa
Curated by ChEMBL
Affinity DataIC50: 250nMAssay Description:Inhibition of Torpedo californica AChE using acetylthiocholine chloride as substrate peincubated for 15 mins followed by substrate addition measured ...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
Universidade De Lisboa
Curated by ChEMBL
Universidade De Lisboa
Curated by ChEMBL
Affinity DataIC50: 280nMAssay Description:Inhibition of Torpedo californica AChE using acetylthiocholine chloride as substrate peincubated for 15 mins followed by substrate addition measured ...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
Universidade De Lisboa
Curated by ChEMBL
Universidade De Lisboa
Curated by ChEMBL
Affinity DataIC50: 300nMAssay Description:Inhibition of Torpedo californica AChE using acetylthiocholine chloride as substrate peincubated for 15 mins followed by substrate addition measured ...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Lisbon
Curated by ChEMBL
University Of Lisbon
Curated by ChEMBL
Affinity DataIC50: 339nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine chloride as substrate peincubated for 15 mins followed by substrate addition measured at 1 mi...More data for this Ligand-Target Pair
Affinity DataIC50: 353nMAssay Description:Inhibition of equine serum BuChE using butylthiocholine chloride as substrate peincubated for 15 mins followed by substrate addition measured at 1 mi...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
Universidade De Lisboa
Curated by ChEMBL
Universidade De Lisboa
Curated by ChEMBL
Affinity DataIC50: 377nMAssay Description:Inhibition of rat MAO B using kynuramine as substrate preincubated for 30 mins followed by substrate additionMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
Universidade De Lisboa
Curated by ChEMBL
Universidade De Lisboa
Curated by ChEMBL
Affinity DataIC50: 560nMAssay Description:Inhibition of Torpedo californica AChE using acetylthiocholine chloride as substrate peincubated for 15 mins followed by substrate addition measured ...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Lisbon
Curated by ChEMBL
University Of Lisbon
Curated by ChEMBL
Affinity DataIC50: 570nMAssay Description:Inhibition of electric eel AChE preincubated for 10 mins measured after 15 mins by Ellman's methodMore data for this Ligand-Target Pair
Affinity DataIC50: 600nMAssay Description:Inhibition of equine serum BuChE by Ellman's methodMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Lisbon
Curated by ChEMBL
University Of Lisbon
Curated by ChEMBL
Affinity DataIC50: 600nMAssay Description:Inhibition of electric eel AChE preincubated for 10 mins measured after 15 mins by Ellman's methodMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
Universidade De Lisboa
Curated by ChEMBL
Universidade De Lisboa
Curated by ChEMBL
Affinity DataIC50: 669nMAssay Description:Inhibition of rat MAO A using kynuramine as substrate preincubated for 30 mins followed by substrate additionMore data for this Ligand-Target Pair
Affinity DataIC50: 810nMAssay Description:Inhibition of human AChEMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
Universidade De Lisboa
Curated by ChEMBL
Universidade De Lisboa
Curated by ChEMBL
Affinity DataIC50: 880nMAssay Description:Inhibition of Torpedo californica AChE using acetylthiocholine chloride as substrate peincubated for 15 mins followed by substrate addition measured ...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Lisbon
Curated by ChEMBL
University Of Lisbon
Curated by ChEMBL
Affinity DataIC50: 884nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine chloride as substrate peincubated for 15 mins followed by substrate addition measured at 1 mi...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
Universidade De Lisboa
Curated by ChEMBL
Universidade De Lisboa
Curated by ChEMBL
Affinity DataIC50: 1.21E+3nMAssay Description:Inhibition of Torpedo californica AChE using acetylthiocholine chloride as substrate peincubated for 15 mins followed by substrate addition measured ...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Lisbon
Curated by ChEMBL
University Of Lisbon
Curated by ChEMBL
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of electric eel AChE preincubated for 10 mins measured after 15 mins by Ellman's methodMore data for this Ligand-Target Pair
Affinity DataIC50: 1.82E+3nMAssay Description:Inhibition of human BuChEMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Lisbon
Curated by ChEMBL
University Of Lisbon
Curated by ChEMBL
Affinity DataIC50: 2.78E+3nMAssay Description:Inhibition of electric eel AChE by Ellman's methodMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Lisbon
Curated by ChEMBL
University Of Lisbon
Curated by ChEMBL
Affinity DataIC50: 2.78E+3nMAssay Description:Inhibition of electric eel AChE by Ellman's methodMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Lisbon
Curated by ChEMBL
University Of Lisbon
Curated by ChEMBL
Affinity DataIC50: 2.78E+3nMAssay Description:Inhibition of electric eel AChE by Ellman's methodMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Universidade De Lisboa
Curated by ChEMBL
Universidade De Lisboa
Curated by ChEMBL
Affinity DataIC50: 3.95E+3nMAssay Description:Inhibition of human MAO BMore data for this Ligand-Target Pair
Affinity DataIC50: 5.38E+3nMAssay Description:Inhibition of equine serum BuChE using butylthiocholine chloride as substrate peincubated for 15 mins followed by substrate addition measured at 1 mi...More data for this Ligand-Target Pair
Affinity DataIC50: 5.40E+3nMAssay Description:Inhibition of Equus caballus BChE preincubated for 10 mins measured after 15 mins by Ellman's methodMore data for this Ligand-Target Pair
Affinity DataIC50: 6.30E+3nMAssay Description:Inhibition of Equus caballus BChE preincubated for 10 mins measured after 15 mins by Ellman's methodMore data for this Ligand-Target Pair